Page last updated: 2024-08-16

tiopronin and naloxone

tiopronin has been researched along with naloxone in 31 studies

Research

Studies (31)

TimeframeStudies, this research(%)All Research%
pre-199029 (93.55)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (6.45)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Kehl, LJ1
Benoliel, JJ; Berthier, JL; Bourgoin, S; Cesselin, F; Hamon, M; Hirsch, M; Mauborgne, A1
Dzoljic, MR; Haffmans, J; van Amsterdam, JC; Walsum, MV1
Buéno, L; Fioramonti, J1
Costentin, J; Giros, B; Michael-Titus, A; Preterre, P1
Dzoljic, MR1
Livingston, SJ; Rooney, KF; Sewell, RD; Smith, HJ1
Hill, RG; Hughes, J; Pittaway, KM1
Kameyama, T; Katoh, A; Nabeshima, T1
Fukaya, H; Furukawa, H; Hiramatsu, M; Kameyama, T; Nabeshima, T1
Kuraishi, Y; Satoh, M; Sugimoto, M; Takagi, H1
Dickenson, AH; Fournie-Zaluski, MC; Roques, BP; Sullivan, AF1
Costentin, J; Lecomte, JM; Marçais-Collado, H; Schwartz, JC; Uchida, G1
Han, JS; Jin, WQ; Zhou, ZF1
Chaillet, P; Costentin, J; Leboyer, M; Lecomte, JM; Llorens-Cortes, C; Marcais-Collado, H; Schwartz, JC; Vlaiculescu, A1
Coquerel, A; Costentin, J; Dubuc, I; Kitabgi, P; Menard, JF1
Dzoljic, MR; Haffmans, J1
Anadón, A; Martinez-Larrañaga, MR1
Beckman, AL; Sartin, NF; Stanton, TL1
Chaillet, P; Costentin, J; Coulaud, A; Fournie-Zaluski, MC; Roques, BP; Zajac, JM1
Bean, AJ; Vaught, JL1
Guilbaud, G; Kayser, V1
Chaillet, P; Costentin, J; Lecomte, JM; Marçais, H; Natan, LB; Uchida, G1
Giovino, AA; Glimcher, PW; Hoebel, BG; Margolin, DH1
de Groat, WC; Hisamitsu, T1
Chipkin, RE; O'Connor, P1
Llorens-Cortes, C; Schwartz, JC1
Barnett, A; Berger, J; Billard, W; Chipkin, RE; Iorio, LC1
Barnett, A; Chipkin, RE; Iorio, LC; Latranyi, MZ1

Reviews

2 review(s) available for tiopronin and naloxone

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Enkephalins, other endogenous opioids and colonic motility in dog and man.
    Gastroenterologie clinique et biologique, 1987, Volume: 11, Issue:3 Pt 2

    Topics: Animals; Central Nervous System; Colon; Dogs; Endorphins; Enkephalins; Gastrointestinal Motility; Humans; In Vitro Techniques; Morphine; Muscle Contraction; Naloxone; Receptors, Opioid; Species Specificity; Thiorphan; Tiopronin

1987

Other Studies

29 other study(ies) available for tiopronin and naloxone

ArticleYear
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Analgesia after inhibition of enkephalin degradation.
    Journal of the American Dental Association (1939), 1986, Volume: 112, Issue:2

    Topics: Amino Acids, Sulfur; Analgesia; Animals; Enkephalins; Injections, Spinal; Male; Mice; Mice, Inbred Strains; Naloxone; Neprilysin; Protease Inhibitors; Spinal Cord; Substance P; Thiorphan; Tiopronin

1986
Enkephalinase is involved in the degradation of endogenous substance P released from slices of rat substantia nigra.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 243, Issue:2

    Topics: Animals; Captopril; Dipeptides; In Vitro Techniques; Leucine; Male; Metalloendopeptidases; Naloxone; Neprilysin; Oligopeptides; Peptidyl-Dipeptidase A; Potassium; Protease Inhibitors; Rats; Rats, Inbred Strains; Substance P; Substantia Nigra; Thiorphan; Tiopronin

1987
Phelorphan, an inhibitor of enzymes involved in the biodegradation of enkephalins, affected the withdrawal symptoms in chronic morphine-dependent rats.
    Neuroscience, 1987, Volume: 22, Issue:1

    Topics: Aminopeptidases; Animals; Brain; CD13 Antigens; Dipeptides; Dipeptidyl-Peptidases and Tripeptidyl-Peptidases; Endopeptidases; Enkephalins; Male; Morphine Dependence; Naloxone; Neprilysin; Protease Inhibitors; Rats; Rats, Inbred Strains; Receptors, Opioid; Substance Withdrawal Syndrome; Thiorphan; Tiopronin

1987
Role of endogenous enkephalins in locomotion evidenced by acetorphan, an "enkephalinase" inhibitor.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 243, Issue:3

    Topics: Amino Acids, Sulfur; Animals; Dose-Response Relationship, Drug; Enkephalins; Hydroxydopamines; Male; Metalloendopeptidases; Mice; Motor Activity; Naloxone; Neprilysin; Oxidopamine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Thiorphan; Tiopronin

1987
Enkephalinase inhibitors attenuate naloxone-precipitated withdrawal syndrome.
    NIDA research monograph, 1986, Volume: 75

    Topics: Amino Acids, Sulfur; Animals; Cerebral Ventricles; Cerebrospinal Fluid; Dipeptides; Glycopeptides; Male; Metalloendopeptidases; Mice; Mice, Inbred Strains; Morphine Dependence; Naloxone; Neprilysin; Rats; Rats, Inbred Strains; Stereotyped Behavior; Substance Withdrawal Syndrome; Thiorphan; Tiopronin

1986
Amelioration of naloxone-precipitated opioid withdrawal symptoms by peripheral administration of the enkephalinase inhibitor acetorphan.
    Psychopharmacology, 1988, Volume: 94, Issue:4

    Topics: Amino Acids, Sulfur; Analgesics; Animals; Body Temperature; Body Weight; Male; Metalloendopeptidases; Mice; Mice, Inbred Strains; Morphine; Morphine Dependence; Naloxone; Neprilysin; Rats; Rats, Inbred Strains; Substance Withdrawal Syndrome; Thiorphan; Tiopronin

1988
Antinociceptive action of cholecystokinin octapeptide (CCK 8) and related peptides in rats and mice: effects of naloxone and peptidase inhibitors.
    Neuropharmacology, 1987, Volume: 26, Issue:4

    Topics: Animals; Captopril; FMRFamide; Gastrins; Leucine; Male; Mice; Naloxone; Neuropeptides; Pain; Protease Inhibitors; Rats; Rats, Inbred Strains; Reaction Time; Sincalide; Tetragastrin; Thiorphan; Tiopronin

1987
Inhibition of enkephalin degradation attenuated stress-induced motor suppression (conditioned suppression of motility).
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:1

    Topics: Amino Acids, Sulfur; Aminopeptidases; Animals; Corpus Striatum; Dopamine; Enkephalin, Methionine; Enkephalins; Leucine; Male; Metalloendopeptidases; Mice; Motor Activity; Naloxone; Neprilysin; Pimozide; Stress, Physiological; Thiorphan; Tiopronin

1988
Potentiation of phencyclidine-induced stereotyped behaviors in rats by thiorphan and bestatin.
    European journal of pharmacology, 1986, Jan-14, Volume: 120, Issue:1

    Topics: Amino Acids, Sulfur; Animals; Drug Synergism; Leucine; Male; Naloxone; Phencyclidine; Rats; Rats, Inbred Strains; Stereotyped Behavior; Thiorphan; Time Factors; Tiopronin

1986
Involvement of medullary opioid-peptidergic and spinal noradrenergic systems in the regulation of formalin-induced persistent pain.
    Neuropharmacology, 1986, Volume: 25, Issue:5

    Topics: Animals; Endorphins; Formaldehyde; Injections, Spinal; Leucine; Male; Medulla Oblongata; Naloxone; Norepinephrine; Pain; Rats; Rats, Inbred Strains; Spinal Cord; Thiorphan; Time Factors; Tiopronin

1986
Prevention of degradation of endogenous enkephalins produces inhibition of nociceptive neurones in rat spinal cord.
    Brain research, 1987, Apr-07, Volume: 408, Issue:1-2

    Topics: Action Potentials; Animals; Dipeptides; Enkephalins; Leucine; Male; Naloxone; Nerve Fibers; Neural Inhibition; Neurons, Afferent; Pain; Protease Inhibitors; Rats; Rats, Inbred Strains; Spinal Cord; Thiorphan; Tiopronin

1987
Naloxone-reversible antidiarrheal effects of enkephalinase inhibitors.
    European journal of pharmacology, 1987, Dec-01, Volume: 144, Issue:2

    Topics: Amino Acids, Sulfur; Animals; Castor Oil; Diarrhea; Drug Interactions; Gastrointestinal Transit; Loperamide; Male; Metalloendopeptidases; Mice; Naloxone; Neprilysin; Rats; Rats, Inbred Strains; Thiorphan; Tiopronin

1987
Electroacupuncture and morphine analgesia potentiated by bestatin and thiorphan administered to the nucleus accumbens of the rabbit.
    Brain research, 1986, Aug-20, Volume: 380, Issue:2

    Topics: Amino Acids, Sulfur; Analgesia; Animals; Dose-Response Relationship, Drug; Enkephalin, Methionine; Immune Sera; Leucine; Male; Microinjections; Morphine; Naloxone; Nucleus Accumbens; Rabbits; Septal Nuclei; Thiorphan; Time Factors; Tiopronin; Transcutaneous Electric Nerve Stimulation

1986
Pharmacological properties of acetorphan, a parenterally active "enkephalinase" inhibitor.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:3

    Topics: Amino Acids, Sulfur; Analgesics; Animals; Antidiarrheals; Biogenic Amines; Brain Chemistry; Dose-Response Relationship, Drug; Endopeptidases; Enkephalin, Methionine; Injections; Kinetics; Male; Mice; Naloxone; Neprilysin; Protease Inhibitors; Rats; Rats, Inbred Strains; Thiorphan; Tiopronin

1986
Naloxone-insensitive potentiation of neurotensin hypothermic effect by the enkephalinase inhibitor thiorphan.
    Brain research, 1986, Nov-29, Volume: 398, Issue:2

    Topics: Amino Acids, Sulfur; Animals; Body Temperature; Captopril; Drug Synergism; Endopeptidases; Injections, Intraventricular; Leucine; Male; Mice; Naloxone; Neprilysin; Neurotensin; Thiorphan; Tiopronin

1986
Inhibition of enkephalinase activity attenuates naloxone-precipitated withdrawal symptoms.
    General pharmacology, 1987, Volume: 18, Issue:1

    Topics: Amino Acids, Sulfur; Animals; Behavior, Animal; Endopeptidases; Injections; Injections, Intraventricular; Male; Morphine Dependence; Naloxone; Neprilysin; Periaqueductal Gray; Protease Inhibitors; Rats; Rats, Inbred Strains; Substance Withdrawal Syndrome; Thiorphan; Tiopronin

1987
An inhibitory action of tetracyclines on guinea-pig myenteric plexus.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 335, Issue:2

    Topics: Animals; Captopril; Drug Interactions; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Leucine; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Naloxone; Protease Inhibitors; Tetracyclines; Thiorphan; Tiopronin

1987
Changes in body temperature and metabolic rate following microinjection of Met-enkephalinamide in the preoptic/anterior hypothalamus of rats.
    Regulatory peptides, 1985, Nov-28, Volume: 12, Issue:4

    Topics: Animals; Behavior, Animal; Body Temperature; Dose-Response Relationship, Drug; Enkephalin, Methionine; Male; Metabolic Clearance Rate; Microinjections; Naloxone; Preoptic Area; Rats; Rats, Inbred Strains; Thiorphan; Tiopronin

1985
The mu rather than the delta subtype of opioid receptors appears to be involved in enkephalin-induced analgesia.
    European journal of pharmacology, 1984, May-18, Volume: 101, Issue:1-2

    Topics: Analgesics; Animals; Enkephalin, Leucine; Enkephalins; Guinea Pigs; In Vitro Techniques; Leucine; Male; Mice; Morphine; Muscle Contraction; Muscle, Smooth; Nalorphine; Naloxone; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Thiorphan; Tiopronin

1984
Physical dependence produced by chronic intracerebroventricular infusion of [D-Arg]kyotorphin or thiorphan to rats.
    European journal of pharmacology, 1984, Oct-15, Volume: 105, Issue:3-4

    Topics: Amino Acids, Sulfur; Analgesics; Animals; Cerebral Ventricles; Endorphins; Humans; Male; Morphine; Naloxone; Neprilysin; Opioid-Related Disorders; Protease Inhibitors; Rats; Rats, Inbred Strains; Receptors, Opioid; Substance Withdrawal Syndrome; Thiorphan; Tiopronin

1984
The analgesic effects of morphine, but not those of the enkephalinase inhibitor thiorphan, are enhanced in arthritic rats.
    Brain research, 1983, May-09, Volume: 267, Issue:1

    Topics: Amino Acids, Sulfur; Analgesia; Animals; Arthritis; Arthritis, Experimental; Male; Morphine; Naloxone; Pain; Protease Inhibitors; Rats; Rats, Inbred Strains; Sensory Thresholds; Thiorphan; Tiopronin; Vocalization, Animal

1983
Involvement of endogenous enkephalins in the mouse 'behavioral despair' test.
    European journal of pharmacology, 1984, Jan-27, Volume: 97, Issue:3-4

    Topics: Aminopeptidases; Animals; Behavior, Animal; Enkephalin, Methionine; Enkephalins; Leucine; Male; Mice; Motor Activity; Naloxone; Protease Inhibitors; Thiorphan; Tiopronin

1984
Endogenous opiate reward induced by an enkephalinase inhibitor, thiorphan, injected into the ventral midbrain.
    Behavioral neuroscience, 1984, Volume: 98, Issue:2

    Topics: Amino Acids, Sulfur; Animals; Endorphins; Enkephalin, Methionine; Female; Mesencephalon; Naloxone; Rats; Rats, Inbred Strains; Reward; Tegmentum Mesencephali; Thiorphan; Tiopronin

1984
The inhibitory effect of opioid peptides and morphine applied intrathecally and intracerebroventricularly on the micturition reflex in the cat.
    Brain research, 1984, Apr-23, Volume: 298, Issue:1

    Topics: Animals; Cats; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Enkephalins; Female; Morphine; Naloxone; Oligopeptides; Reflex; Thiorphan; Tiopronin; Urination

1984
Comparisons between warm and cold water swim stress in mice.
    Life sciences, 1984, Aug-06, Volume: 35, Issue:6

    Topics: Analgesia; Animals; Cold Temperature; Hot Temperature; Male; Mice; Naloxone; Protease Inhibitors; Stress, Physiological; Swimming; Thiorphan; Time Factors; Tiopronin

1984
Changes in turnover of cerebral monoamines following inhibition of enkephalin metabolism by thiorphan and bestatin.
    European journal of pharmacology, 1984, Sep-17, Volume: 104, Issue:3-4

    Topics: alpha-Methyltyrosine; Amino Acids, Sulfur; Aminopeptidases; Animals; Biogenic Amines; Brain; Enkephalins; Leucine; Male; Methyltyrosines; Mice; Naloxone; Protease Inhibitors; Thiorphan; Tiopronin

1984
In vitro and in vivo effects of thiorphan: an inhibitor of enkephalinase A.
    Advances in biochemical psychopharmacology, 1982, Volume: 33

    Topics: Amino Acids, Sulfur; Aminopeptidases; Analgesics; Animals; Captopril; Drug Synergism; Enkephalins; In Vitro Techniques; Male; Mice; Naloxone; Neprilysin; Protease Inhibitors; Thiorphan; Tiopronin

1982
Potentiation of [D-ala2]enkephalinamide analgesia in rats by thiorphan.
    European journal of pharmacology, 1982, Sep-24, Volume: 83, Issue:3-4

    Topics: Amino Acids, Sulfur; Analgesics; Animals; Drug Synergism; Enkephalin, Methionine; Male; Naloxone; Neprilysin; Nociceptors; Protease Inhibitors; Rats; Rats, Inbred Strains; Thiorphan; Time Factors; Tiopronin

1982