Page last updated: 2024-09-03

tifluadom and mr 2266

tifluadom has been researched along with mr 2266 in 8 studies

Compound Research Comparison

Studies
(tifluadom)
Trials
(tifluadom)
Recent Studies (post-2010)
(tifluadom)
Studies
(mr 2266)
Trials
(mr 2266)
Recent Studies (post-2010) (mr 2266)
780017600

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19907 (87.50)18.7374
1990's1 (12.50)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Caliezi, A; Drack, E; Halter, F; Scheurer, U; Varga, L; Wenger, F1
Dykstra, LA; Picker, MJ1
Frey, HH1
Bueno, L; Fioramonti, J; Gué, M; Junien, JL1
Boeck, G; Ciaramelli, F; Freye, E; Schaal, M1
Freye, E; Schaal, M; Windelschmidt, R1
Bueno, L; Fioramonti, J; Gue, M; Honde, C; Junien, JL; Pascaud, X1
Jackson, HC; Sewell, RD1

Other Studies

8 other study(ies) available for tifluadom and mr 2266

ArticleYear
Different motor actions of dynorphins and nonpeptide kappa opioid receptor agonists in the isolated rat colon.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 252, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Antihypertensive Agents; Benzeneacetamides; Benzodiazepines; Benzomorphans; Colon; Diuretics; Dynorphins; Gastrointestinal Motility; In Vitro Techniques; Male; Muscle, Smooth; Naloxone; Narcotic Antagonists; Pressure; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1990
Discriminative stimulus effects of mu and kappa opioids in the pigeon: analysis of the effects of full and partial mu and kappa agonists.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 249, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzomorphans; Columbidae; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Fentanyl; Morphinans; Naloxone; Narcotics; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1989
Effect of mu- and kappa-opioid agonists on the electroconvulsive seizure threshold in mice and antagonism by naloxone and MR 2266.
    Pharmacology & toxicology, 1988, Volume: 62, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzeneacetamides; Benzodiazepines; Benzomorphans; Electroshock; Fentanyl; Male; Mice; Morphinans; Morphine; Nalbuphine; Naloxone; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Seizures

1988
Orally administered kappa but not mu opiate agonists enhance gastric emptying of a solid canned food meal in dogs.
    The Journal of pharmacy and pharmacology, 1988, Volume: 40, Issue:12

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animal Feed; Animals; Benzodiazepines; Benzomorphans; Diuretics; Dogs; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Female; Gastric Emptying; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1988
The benzodiazepine (+)-tifluadom (KC-6128), but not its optical isomer (KC-5911) induces opioid kappa receptor-related EEG power spectra and evoked potential changes.
    Pharmacology, 1986, Volume: 33, Issue:5

    Topics: Animals; Benzodiazepines; Benzomorphans; Dogs; Electroencephalography; Evoked Potentials; Flumazenil; Naloxone; Receptors, Opioid; Receptors, Opioid, kappa; Stereoisomerism

1986
[Tifluadom, a benzodiazepine with opioid-like activity: study of its central mechanism of action in conscious dogs].
    EEG-EMG Zeitschrift fur Elektroenzephalographie, Elektromyographie und verwandte Gebiete, 1986, Volume: 17, Issue:1

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Benzomorphans; Brain; Dogs; Dose-Response Relationship, Drug; Electroencephalography; Evoked Potentials, Somatosensory; Flumazenil; Naloxone

1986
Opposite effects of kappa-opioid agonists on gastric emptying of liquids and solids in dogs.
    Gastroenterology, 1988, Volume: 95, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Administration, Oral; Animal Feed; Animals; Benzodiazepines; Benzomorphans; Dogs; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Female; Gastric Emptying; Injections, Intravenous; Morphinans; Morphine; Naloxone; Pyrrolidines

1988
The role of opioid receptor sub-types in tifluadom-induced feeding.
    The Journal of pharmacy and pharmacology, 1984, Volume: 36, Issue:10

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Benzomorphans; Convulsants; Eating; Enkephalin, Leucine; Flumazenil; Male; Naloxone; Naltrexone; Narcotic Antagonists; Rats; Rats, Inbred Strains; Receptors, Opioid; Stereoisomerism

1984