Page last updated: 2024-09-03

tifluadom and fentanyl

tifluadom has been researched along with fentanyl in 7 studies

Compound Research Comparison

Studies
(tifluadom)
Trials
(tifluadom)
Recent Studies (post-2010)
(tifluadom)
Studies
(fentanyl)
Trials
(fentanyl)
Recent Studies (post-2010) (fentanyl)
780015,2884,3104,483

Protein Interaction Comparison

ProteinTaxonomytifluadom (IC50)fentanyl (IC50)
ATP-dependent translocase ABCB1Homo sapiens (human)6.5
Delta-type opioid receptorMus musculus (house mouse)0.6342
Delta-type opioid receptorRattus norvegicus (Norway rat)0.0122
Mu-type opioid receptorRattus norvegicus (Norway rat)0.1888
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0122
Mu-type opioid receptorHomo sapiens (human)0.0058
Delta-type opioid receptorHomo sapiens (human)0.3092
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)5.893
Kappa-type opioid receptorHomo sapiens (human)1.58
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.0031
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.8197
Sigma non-opioid intracellular receptor 1Cavia porcellus (domestic guinea pig)4.973
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.354

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19905 (71.43)18.7374
1990's2 (28.57)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dong, XW; Headley, PM; Parsons, CG1
Dykstra, LA; Negus, SS; Picker, MJ1
Headley, PM; Parsons, CG1
Dykstra, LA; Picker, MJ1
Frey, HH1
Hayes, AG; Stewart, BR1
Hayes, AG; Skingle, M; Tyers, MB1

Other Studies

7 other study(ies) available for tifluadom and fentanyl

ArticleYear
Effects of intravenous mu and kappa opioid receptor agonists on sensory responses of convergent neurones in the dorsal horn of spinalized rats.
    British journal of pharmacology, 1991, Volume: 103, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzodiazepines; Fentanyl; Hot Temperature; Male; Morphine; Naloxone; Neurons, Afferent; Nociceptors; Physical Stimulation; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Spinal Cord

1991
Interactions between mu and kappa opioid agonists in the rat drug discrimination procedure.
    Psychopharmacology, 1990, Volume: 102, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzomorphans; Buprenorphine; Discrimination, Psychological; Dose-Response Relationship, Drug; Drug Interactions; Fentanyl; Male; Morphine; Pentobarbital; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1990
Spinal antinociceptive actions of mu- and kappa-opioids: the importance of stimulus intensity in determining 'selectivity' between reflexes to different modalities of noxious stimulus.
    British journal of pharmacology, 1989, Volume: 98, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzodiazepines; Decerebrate State; Electrophysiology; Fentanyl; Narcotics; Neurons; Nociceptors; Pain; Physical Stimulation; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Reflex

1989
Discriminative stimulus effects of mu and kappa opioids in the pigeon: analysis of the effects of full and partial mu and kappa agonists.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 249, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzomorphans; Columbidae; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Fentanyl; Morphinans; Naloxone; Narcotics; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1989
Effect of mu- and kappa-opioid agonists on the electroconvulsive seizure threshold in mice and antagonism by naloxone and MR 2266.
    Pharmacology & toxicology, 1988, Volume: 62, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzeneacetamides; Benzodiazepines; Benzomorphans; Electroshock; Fentanyl; Male; Mice; Morphinans; Morphine; Nalbuphine; Naloxone; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Seizures

1988
Effect of mu and kappa opioid receptor agonists on rat plasma corticosterone levels.
    European journal of pharmacology, 1985, Oct-08, Volume: 116, Issue:1-2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzomorphans; Corticosterone; Dose-Response Relationship, Drug; Fentanyl; Male; Morphine; Naloxone; Naltrexone; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1985
Reversal by beta-funaltrexamine of the antinociceptive effect of opioid agonists in the rat.
    British journal of pharmacology, 1986, Volume: 88, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Buprenorphine; Cyclazocine; Ethylketocyclazocine; Fentanyl; Male; Naltrexone; Pain; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1986