Page last updated: 2024-08-24

tiagabine and piperidines

tiagabine has been researched along with piperidines in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (14.29)18.2507
2000's3 (42.86)29.6817
2010's3 (42.86)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Egebjerg, J; Sørensen, PO; Thomsen, C1
Dalby, NO1
Berger, P; Bloch, DA; Coleman, FS; Elkashef, A; Goldsmith, RJ; Harrer, JM; Leiderman, DB; Mezinskis, JP; Montgomery, MA; Singal, BM; Somoza, EC; Winhusen, TM1
Fang, K; Lin, G; Liu, X; Zhang, J; Zhang, P1
Bräuner-Osborne, H; Clausen, RP; Jensen, AA; Jørgensen, L; Kragholm, B; Kvist, T; Madsen, KK; Schousboe, A; Vogensen, SB1
Amador-Arjona, A; D'Amico, D; Dierssen, M; Santos, M; Spadoni, O; Stork, O1
Hiramatsu, M1

Reviews

1 review(s) available for tiagabine and piperidines

ArticleYear
[Functional role for GABA transporters in the CNS].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 2014, Volume: 143, Issue:4

    Topics: Animals; Brain; Camphanes; Carbazoles; Carrier Proteins; Central Nervous System Diseases; Drug Discovery; GABA Plasma Membrane Transport Proteins; GABA Uptake Inhibitors; Humans; Isoxazoles; Mental Disorders; Molecular Targeted Therapy; Nipecotic Acids; Piperidines; Tiagabine

2014

Trials

1 trial(s) available for tiagabine and piperidines

ArticleYear
A placebo-controlled screening trial of tiagabine, sertraline and donepezil as cocaine dependence treatments.
    Addiction (Abingdon, England), 2005, Volume: 100 Suppl 1

    Topics: Adult; Anticonvulsants; Cocaine-Related Disorders; Donepezil; Female; Humans; Indans; Male; Middle Aged; Nipecotic Acids; Piperidines; Selective Serotonin Reuptake Inhibitors; Sertraline; Tiagabine

2005

Other Studies

5 other study(ies) available for tiagabine and piperidines

ArticleYear
1-(3-(9H-carbazol-9-yl)-1-propyl)-4-(2-methoxyphenyl)-4-piperidinol, a novel subtype selective inhibitor of the mouse type II GABA-transporter.
    British journal of pharmacology, 1997, Volume: 120, Issue:6

    Topics: Animals; Carrier Proteins; Cell Line; Cricetinae; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Membrane Proteins; Membrane Transport Proteins; Mice; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Organic Anion Transporters; Piperidines; Proline; Tiagabine

1997
GABA-level increasing and anticonvulsant effects of three different GABA uptake inhibitors.
    Neuropharmacology, 2000, Volume: 39, Issue:12

    Topics: Acoustic Stimulation; Anesthesia; Animals; Anisoles; Anticonvulsants; Carbazoles; Chromatography, High Pressure Liquid; Convulsants; Electroshock; Female; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Male; Mice; Mice, Inbred DBA; Microdialysis; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Pentylenetetrazole; Piperidines; Seizures; Substantia Nigra; Thalamus; Tiagabine

2000
Synthesis and biological evaluation of (R)-N-(diarylmethylthio/sulfinyl)ethyl/propyl-piperidine-3-carboxylic acid hydrochlorides as novel GABA uptake inhibitors.
    Bioorganic & medicinal chemistry letters, 2007, Jul-01, Volume: 17, Issue:13

    Topics: Animals; Anticonvulsants; Carboxylic Acids; Chemistry, Pharmaceutical; Drug Design; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Imidazoles; Inhibitory Concentration 50; Mice; Models, Chemical; Nipecotic Acids; Piperidines; Structure-Activity Relationship; Temperature; Tiagabine

2007
Discovery of a subtype selective inhibitor of the human betaine/GABA transporter 1 (BGT-1) with a non-competitive pharmacological profile.
    Biochemical pharmacology, 2013, Aug-15, Volume: 86, Issue:4

    Topics: Animals; Benzamides; Betaine; Carrier Proteins; CHO Cells; Cricetinae; Databases, Factual; GABA Plasma Membrane Transport Proteins; HEK293 Cells; High-Throughput Screening Assays; Humans; Membrane Potentials; Mice; Nipecotic Acids; Piperidines; Small Molecule Libraries; Tiagabine

2013
Hippocampal hyperexcitability underlies enhanced fear memories in TgNTRK3, a panic disorder mouse model.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2013, Sep-18, Volume: 33, Issue:38

    Topics: Analysis of Variance; Animals; Bacterial Proteins; Conditioning, Classical; Disease Models, Animal; Disks Large Homolog 4 Protein; Excitatory Amino Acid Antagonists; Exploratory Behavior; Extinction, Psychological; Fear; GABA Agonists; Generalization, Psychological; Glutamate Decarboxylase; Guanylate Kinases; Hippocampus; Luminescent Proteins; Maze Learning; Membrane Proteins; Memory; Mice; Mice, Transgenic; Nipecotic Acids; Panic Disorder; Piperidines; Proto-Oncogene Proteins c-fos; Receptor, trkC; Tiagabine; Vesicular Glutamate Transport Proteins

2013