tiagabine has been researched along with piperidines in 7 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (14.29) | 18.2507 |
2000's | 3 (42.86) | 29.6817 |
2010's | 3 (42.86) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Egebjerg, J; Sørensen, PO; Thomsen, C | 1 |
Dalby, NO | 1 |
Berger, P; Bloch, DA; Coleman, FS; Elkashef, A; Goldsmith, RJ; Harrer, JM; Leiderman, DB; Mezinskis, JP; Montgomery, MA; Singal, BM; Somoza, EC; Winhusen, TM | 1 |
Fang, K; Lin, G; Liu, X; Zhang, J; Zhang, P | 1 |
Bräuner-Osborne, H; Clausen, RP; Jensen, AA; Jørgensen, L; Kragholm, B; Kvist, T; Madsen, KK; Schousboe, A; Vogensen, SB | 1 |
Amador-Arjona, A; D'Amico, D; Dierssen, M; Santos, M; Spadoni, O; Stork, O | 1 |
Hiramatsu, M | 1 |
1 review(s) available for tiagabine and piperidines
Article | Year |
---|---|
[Functional role for GABA transporters in the CNS].
Topics: Animals; Brain; Camphanes; Carbazoles; Carrier Proteins; Central Nervous System Diseases; Drug Discovery; GABA Plasma Membrane Transport Proteins; GABA Uptake Inhibitors; Humans; Isoxazoles; Mental Disorders; Molecular Targeted Therapy; Nipecotic Acids; Piperidines; Tiagabine | 2014 |
1 trial(s) available for tiagabine and piperidines
Article | Year |
---|---|
A placebo-controlled screening trial of tiagabine, sertraline and donepezil as cocaine dependence treatments.
Topics: Adult; Anticonvulsants; Cocaine-Related Disorders; Donepezil; Female; Humans; Indans; Male; Middle Aged; Nipecotic Acids; Piperidines; Selective Serotonin Reuptake Inhibitors; Sertraline; Tiagabine | 2005 |
5 other study(ies) available for tiagabine and piperidines
Article | Year |
---|---|
1-(3-(9H-carbazol-9-yl)-1-propyl)-4-(2-methoxyphenyl)-4-piperidinol, a novel subtype selective inhibitor of the mouse type II GABA-transporter.
Topics: Animals; Carrier Proteins; Cell Line; Cricetinae; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Membrane Proteins; Membrane Transport Proteins; Mice; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Organic Anion Transporters; Piperidines; Proline; Tiagabine | 1997 |
GABA-level increasing and anticonvulsant effects of three different GABA uptake inhibitors.
Topics: Acoustic Stimulation; Anesthesia; Animals; Anisoles; Anticonvulsants; Carbazoles; Chromatography, High Pressure Liquid; Convulsants; Electroshock; Female; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Male; Mice; Mice, Inbred DBA; Microdialysis; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Pentylenetetrazole; Piperidines; Seizures; Substantia Nigra; Thalamus; Tiagabine | 2000 |
Synthesis and biological evaluation of (R)-N-(diarylmethylthio/sulfinyl)ethyl/propyl-piperidine-3-carboxylic acid hydrochlorides as novel GABA uptake inhibitors.
Topics: Animals; Anticonvulsants; Carboxylic Acids; Chemistry, Pharmaceutical; Drug Design; GABA Antagonists; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Imidazoles; Inhibitory Concentration 50; Mice; Models, Chemical; Nipecotic Acids; Piperidines; Structure-Activity Relationship; Temperature; Tiagabine | 2007 |
Discovery of a subtype selective inhibitor of the human betaine/GABA transporter 1 (BGT-1) with a non-competitive pharmacological profile.
Topics: Animals; Benzamides; Betaine; Carrier Proteins; CHO Cells; Cricetinae; Databases, Factual; GABA Plasma Membrane Transport Proteins; HEK293 Cells; High-Throughput Screening Assays; Humans; Membrane Potentials; Mice; Nipecotic Acids; Piperidines; Small Molecule Libraries; Tiagabine | 2013 |
Hippocampal hyperexcitability underlies enhanced fear memories in TgNTRK3, a panic disorder mouse model.
Topics: Analysis of Variance; Animals; Bacterial Proteins; Conditioning, Classical; Disease Models, Animal; Disks Large Homolog 4 Protein; Excitatory Amino Acid Antagonists; Exploratory Behavior; Extinction, Psychological; Fear; GABA Agonists; Generalization, Psychological; Glutamate Decarboxylase; Guanylate Kinases; Hippocampus; Luminescent Proteins; Maze Learning; Membrane Proteins; Memory; Mice; Mice, Transgenic; Nipecotic Acids; Panic Disorder; Piperidines; Proto-Oncogene Proteins c-fos; Receptor, trkC; Tiagabine; Vesicular Glutamate Transport Proteins | 2013 |