Page last updated: 2024-08-24

tiagabine and nnc 711

tiagabine has been researched along with nnc 711 in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (50.00)18.2507
2000's4 (40.00)29.6817
2010's1 (10.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andrade e Silva, ML; Cunha, WR; Fontana, AC; Magalhães, LG; Mortensen, OV; Pereira, AC; Souza Rezende, KC; Timple, JM1
Andersen, KE; Frederiksen, K; Knutsen, LJ; Nielsen, EB; Suzdak, PD; Sørensen, PO1
Chapman, AG; Meldrum, BS; Parvez, NS; Smith, SE1
Borden, LA; Branchek, TA; Gluchowski, C; Murali Dhar, TG; Smith, KE; Weinshank, RL1
Bowery, NG; Richards, DA1
Bowery, NG; Davies, CC; Sutch, RJ1
Peng, W; Simantov, R1
Kreil, A; Richter, A1
Clausen, RP; Frølund, B; Krogsgaard-Larsen, P; Larsson, OM; Madsen, K; Schousboe, A1
Cai, GQ; Cai, YQ; Fei, J; Jiang, J; Sheng, ZJ; Wang, ZG; Xu, YF1

Reviews

1 review(s) available for tiagabine and nnc 711

ArticleYear
Structure-activity relationship and pharmacology of gamma-aminobutyric acid (GABA) transport inhibitors.
    Advances in pharmacology (San Diego, Calif.), 2006, Volume: 54

    Topics: Animals; GABA Agonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; GABA Uptake Inhibitors; Humans; Molecular Structure; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Oximes; Structure-Activity Relationship; Tiagabine

2006

Other Studies

9 other study(ies) available for tiagabine and nnc 711

ArticleYear
The lignan (-)-hinokinin displays modulatory effects on human monoamine and GABA transporter activities.
    Journal of natural products, 2013, Oct-25, Volume: 76, Issue:10

    Topics: 4-Butyrolactone; Attention Deficit Disorder with Hyperactivity; Benzodioxoles; Dioxoles; Dopamine; Dose-Response Relationship, Drug; GABA Plasma Membrane Transport Proteins; Humans; Lignans; Molecular Structure; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Serotonin Plasma Membrane Transport Proteins; Stereoisomerism

2013
NNC-711, a novel potent and selective gamma-aminobutyric acid uptake inhibitor: pharmacological characterization.
    European journal of pharmacology, 1992, Dec-02, Volume: 224, Issue:2-3

    Topics: Animals; Anticonvulsants; Astrocytes; Behavior, Animal; Brain; Carbolines; Cells, Cultured; Convulsants; Female; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Motor Activity; Neurons; Nicotinic Acids; Nipecotic Acids; Oximes; Pentylenetetrazole; Rats; Seizures; Synaptosomes; Tiagabine

1992
The gamma-aminobutyric acid uptake inhibitor, tiagabine, is anticonvulsant in two animal models of reflex epilepsy.
    European journal of pharmacology, 1995, Feb-06, Volume: 273, Issue:3

    Topics: Acoustic Stimulation; Animals; Anticonvulsants; Behavior, Animal; Carbamazepine; Epilepsy; Female; GABA Agents; Male; Motor Activity; Myoclonus; Neurotransmitter Uptake Inhibitors; Nicotinic Acids; Nipecotic Acids; Oximes; Papio; Photic Stimulation; Proline; Rats; Rats, Inbred Strains; Tiagabine

1995
Tiagabine, SK&F 89976-A, CI-966, and NNC-711 are selective for the cloned GABA transporter GAT-1.
    European journal of pharmacology, 1994, Oct-14, Volume: 269, Issue:2

    Topics: Animals; Anticonvulsants; Carrier Proteins; Cell Line; Cloning, Molecular; GABA Antagonists; GABA Plasma Membrane Transport Proteins; Humans; Membrane Proteins; Membrane Transport Proteins; Nerve Tissue Proteins; Nicotinic Acids; Nipecotic Acids; Organic Anion Transporters; Oximes; Pyridines; Rats; Recombinant Proteins; Structure-Activity Relationship; Tiagabine; Transfection

1994
Comparative effects of the GABA uptake inhibitors, tiagabine and NNC-711, on extracellular GABA levels in the rat ventrolateral thalamus.
    Neurochemical research, 1996, Volume: 21, Issue:2

    Topics: Analysis of Variance; Animals; Anticonvulsants; Basal Metabolism; Drug Evaluation, Preclinical; Epilepsy; gamma-Aminobutyric Acid; Male; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Oximes; Rats; Rats, Wistar; Thalamus; Tiagabine

1996
GABA release and uptake measured in crude synaptosomes from Genetic Absence Epilepsy Rats from Strasbourg (GAERS).
    Neurochemistry international, 1999, Volume: 34, Issue:5

    Topics: Aminooxyacetic Acid; Animals; Autoradiography; beta-Alanine; Cerebral Cortex; Epilepsy; GABA Agents; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Kinetics; Nipecotic Acids; Oximes; Rats; Rats, Mutant Strains; Synaptosomes; Thalamus; Tiagabine; Tritium

1999
Altered gene expression in frontal cortex and midbrain of 3,4-methylenedioxymethamphetamine (MDMA) treated mice: differential regulation of GABA transporter subtypes.
    Journal of neuroscience research, 2003, Apr-15, Volume: 72, Issue:2

    Topics: Animals; Carrier Proteins; Cloning, Molecular; Frontal Lobe; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Gene Expression Regulation; Male; Membrane Proteins; Membrane Transport Proteins; Mesencephalon; Mice; Mice, Knockout; N-Methyl-3,4-methylenedioxyamphetamine; Nerve Tissue Proteins; Nipecotic Acids; Organic Anion Transporters; Oximes; Protein Isoforms; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Tiagabine

2003
Antidystonic efficacy of gamma-aminobutyric acid uptake inhibitors in the dtsz mutant.
    European journal of pharmacology, 2005, Oct-03, Volume: 521, Issue:1-3

    Topics: Animals; Cricetinae; Disease Progression; Dose-Response Relationship, Drug; Dystonia; Female; GABA Antagonists; Injections, Intraperitoneal; Male; Mutation; Nipecotic Acids; Oximes; Random Allocation; Severity of Illness Index; Tiagabine; Time Factors; Treatment Outcome

2005
Hypoalgesia in mice lacking GABA transporter subtype 1.
    Journal of neuroscience research, 2008, Feb-01, Volume: 86, Issue:2

    Topics: Animals; GABA Antagonists; GABA Plasma Membrane Transport Proteins; Mice; Mice, Knockout; Nipecotic Acids; Oximes; Pain; Pain Threshold; Tiagabine

2008