Page last updated: 2024-08-24

tiagabine and diazepam

tiagabine has been researched along with diazepam in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (26.67)18.2507
2000's6 (40.00)29.6817
2010's5 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andricopulo, AD; Moda, TL; Montanari, CA1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Choi, SS; Contrera, JF; Hastings, KL; Kruhlak, NL; Sancilio, LF; Weaver, JL; Willard, JM1
Campillo, NE; Guerra, A; Páez, JA1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Alelyunas, YW; Bui, K; Empfield, JR; McCarthy, D; Pelosi-Kilby, L; Shen, C; Spreen, RC1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Brown, GB; DeLorey, TM1
Diemer, NH; Johansen, FF1
Andersen, KE; Braestrup, C; Knutsen, LJ; Nielsen, EB; Sonnewald, U; Suzdak, PD1
Bazil, CW; Pedley, TA1
Heilig, M; Rimondini, R; Sommer, W1
Hiemke, C; Lüddens, H; Schmitt, U1
Lee, CY; Liou, HH1

Reviews

2 review(s) available for tiagabine and diazepam

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Advances in the medical treatment of epilepsy.
    Annual review of medicine, 1998, Volume: 49

    Topics: Acetates; Amines; Anticonvulsants; Carbamazepine; Cyclohexanecarboxylic Acids; Diazepam; Drug Approval; Drug Design; Drug Interactions; Drug Resistance; Epilepsy; Felbamate; Fructose; Gabapentin; gamma-Aminobutyric Acid; Humans; Injections, Intravenous; Ketones; Lamotrigine; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Phenylcarbamates; Phenytoin; Prodrugs; Propylene Glycols; Tiagabine; Topiramate; Triazines; United States; Valproic Acid; Vigabatrin

1998

Other Studies

13 other study(ies) available for tiagabine and diazepam

ArticleYear
Hologram QSAR model for the prediction of human oral bioavailability.
    Bioorganic & medicinal chemistry, 2007, Dec-15, Volume: 15, Issue:24

    Topics: Administration, Oral; Biological Availability; Holography; Humans; Models, Biological; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2007
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Development of a phospholipidosis database and predictive quantitative structure-activity relationship (QSAR) models.
    Toxicology mechanisms and methods, 2008, Volume: 18, Issue:2-3

    Topics:

2008
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Experimental solubility profiling of marketed CNS drugs, exploring solubility limit of CNS discovery candidate.
    Bioorganic & medicinal chemistry letters, 2010, Dec-15, Volume: 20, Issue:24

    Topics: Central Nervous System Agents; Drug Evaluation, Preclinical; Hydrogen-Ion Concentration; Pharmaceutical Preparations; Solubility

2010
gamma-Aminobutyric acidA receptor pharmacology in rat cerebral cortical synaptoneurosomes.
    Journal of neurochemistry, 1992, Volume: 58, Issue:6

    Topics: Animals; Benzodiazepines; Cerebral Cortex; Diazepam; Male; Muscimol; Nipecotic Acids; Rats; Rats, Inbred Strains; Receptors, GABA-A; Synaptosomes; Tiagabine; Tritium

1992
Enhancement of GABA neurotransmission after cerebral ischemia in the rat reduces loss of hippocampal CA1 pyramidal cells.
    Acta neurologica Scandinavica, 1991, Volume: 84, Issue:1

    Topics: Animals; Arousal; Brain Ischemia; Cell Count; Cell Survival; Diazepam; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Hippocampus; Isoxazoles; Male; Motor Activity; Nerve Degeneration; Neurons; Nipecotic Acids; Rats; Rats, Inbred Strains; Synaptic Transmission; Tiagabine

1991
Characterization of tiagabine (NO-328), a new potent and selective GABA uptake inhibitor.
    European journal of pharmacology, 1991, Apr-24, Volume: 196, Issue:3

    Topics: Animals; Anticonvulsants; Carbolines; Clonazepam; Convulsants; Diazepam; Female; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred DBA; Neurotransmitter Uptake Inhibitors; Nicotinic Acids; Nipecotic Acids; Pentylenetetrazole; Rats; Rats, Inbred Strains; Seizures; Tiagabine

1991
Effects of tiagabine and diazepam on operant ethanol self-administration in the rat.
    Journal of studies on alcohol, 2002, Volume: 63, Issue:1

    Topics: Animals; Central Nervous System Depressants; Conditioning, Operant; Diazepam; Dose-Response Relationship, Drug; Ethanol; GABA Agonists; GABA Modulators; Injections, Intraperitoneal; Male; Motor Activity; Nipecotic Acids; Rats; Rats, Wistar; Self Administration; Tiagabine

2002
Anxiolytic-like effects of acute and chronic GABA transporter inhibition in rats.
    Journal of neural transmission (Vienna, Austria : 1996), 2002, Volume: 109, Issue:5-6

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Carrier Proteins; Diazepam; Drug Administration Schedule; Drug Synergism; GABA Plasma Membrane Transport Proteins; Male; Maze Learning; Membrane Proteins; Membrane Transport Proteins; Nipecotic Acids; Organic Anion Transporters; Pyridines; Rats; Rats, Inbred Strains; Tiagabine; Time Factors; Zolpidem

2002
GABAergic tonic inhibition is regulated by developmental age and epilepsy in the dentate gyrus.
    Neuroreport, 2013, Jul-10, Volume: 24, Issue:10

    Topics: Aging; Animals; Anticonvulsants; Data Interpretation, Statistical; Dentate Gyrus; Diazepam; Electrophysiological Phenomena; Epilepsy; GABA Agonists; GABA Modulators; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Nipecotic Acids; Patch-Clamp Techniques; Rats; Rats, Wistar; Status Epilepticus; Tiagabine

2013