Page last updated: 2024-08-24

tiagabine and baclofen

tiagabine has been researched along with baclofen in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19901 (6.67)18.7374
1990's7 (46.67)18.2507
2000's3 (20.00)29.6817
2010's4 (26.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Greentree, SG; Pertwee, RG; Swift, PA1
Bowery, NG; Lemos, T; Richards, DA; Whitton, PS1
Mayfield, RD; Zahniser, NR1
Draguhn, A; Heinemann, U; Meierkord, H; Pfeiffer, M1
Andreasen, M; Fueta, Y; Lambert, JD; Roepstorff, A1
Ben-Ari, Y; Caillard, O; Gaïarsa, JL; McLean, HA1
Labar, D; Solomon, GE1
Bartolini, A; Ipponi, A; Lamberti, C; Malmberg-Aiello, P; Medica, A1
Froestl, W; Griffiths, RR; Weerts, EM1
Froestl, W; Griffiths, RR; Kaminski, BJ; Weerts, EM1
Hutson, PH; McDonald, LM; Sheppard, WF; Sohal, B; Staveley, SM; Tattersall, FD1
Ma, H; Yang, K1
Bai, X; Fei, J; Huang, D; Huang, F; Huang, L; Liu, J; Ma, Y; Suo, H; Tong, J; Wang, P; Wang, Z; Xu, J; Yang, Y; Yu, M1
Abdel-Galil, AG; El-Gowilly, SM; El-Mas, MM; Sallam, MY1

Reviews

1 review(s) available for tiagabine and baclofen

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

14 other study(ies) available for tiagabine and baclofen

ArticleYear
Drugs which stimulate or facilitate central GABAergic transmission interact synergistically with delta-9-tetrahydrocannabinol to produce marked catalepsy in mice.
    Neuropharmacology, 1988, Volume: 27, Issue:12

    Topics: Aminooxyacetic Acid; Animals; Baclofen; Bicuculline; Catalepsy; Dronabinol; Drug Synergism; Flumazenil; Flupenthixol; Flurazepam; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Muscimol; Nipecotic Acids; Receptors, GABA-A; Strychnine; Taurine; Tiagabine

1988
Extracellular GABA in the ventrolateral thalamus of rats exhibiting spontaneous absence epilepsy: a microdialysis study.
    Journal of neurochemistry, 1995, Volume: 65, Issue:4

    Topics: Animals; Baclofen; Electroencephalography; Epilepsy, Absence; Extracellular Space; GABA Antagonists; gamma-Aminobutyric Acid; Microdialysis; Nipecotic Acids; Organophosphorus Compounds; Potassium; Rats; Rats, Wistar; Stereoisomerism; Thalamus; Tiagabine

1995
Endogenous GABA release from rat striatal slices: effects of the GABAB receptor antagonist 2-hydroxy-saclofen.
    Synapse (New York, N.Y.), 1993, Volume: 14, Issue:1

    Topics: Animals; Baclofen; Calcium; Chromatography, High Pressure Liquid; Corpus Striatum; Dose-Response Relationship, Drug; Electric Stimulation; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Nipecotic Acids; Osmolar Concentration; Rats; Rats, Sprague-Dawley; Tiagabine

1993
Effects of gamma-aminobutyric acid (GABA) agonists and GABA uptake inhibitors on pharmacosensitive and pharmacoresistant epileptiform activity in vitro.
    British journal of pharmacology, 1996, Volume: 119, Issue:3

    Topics: Animals; Baclofen; Dose-Response Relationship, Drug; Entorhinal Cortex; Epilepsy; Female; GABA Agonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Magnesium; Male; Membrane Potentials; Muscimol; Neurons; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Proline; Rats; Rats, Wistar; Tiagabine

1996
Analysis of the kinetics of synaptic inhibition points to a reduction in GABA release in area CA1 of the genetically epileptic mouse, El.
    Epilepsy research, 1996, Volume: 26, Issue:1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Anticonvulsants; Baclofen; Disease Models, Animal; Electric Stimulation; Epilepsy; gamma-Aminobutyric Acid; Hippocampus; Interneurons; Mice; Mice, Mutant Strains; Neural Inhibition; Nipecotic Acids; Receptors, GABA; Species Specificity; Synaptic Transmission; Tiagabine

1996
Ontogenesis of presynaptic GABAB receptor-mediated inhibition in the CA3 region of the rat hippocampus.
    Journal of neurophysiology, 1998, Volume: 79, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Aging; Animals; Animals, Newborn; Baclofen; Calcium; Electric Stimulation; Evoked Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Male; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Organophosphorus Compounds; Pyramidal Cells; Rats; Rats, Wistar; Receptors, GABA-B; Synaptic Transmission; Tiagabine

1998
Hypothesis that tiagabine-induced NCSE is associated with GABAergic hyperfunction, with GABA(B) receptors playing a critical role, is supported by a case of generalized NCSE induced by baclofen.
    Epilepsia, 1998, Volume: 39, Issue:12

    Topics: Anticonvulsants; Baclofen; Humans; Nipecotic Acids; Receptors, GABA; Status Epilepticus; Tiagabine

1998
Tiagabine antinociception in rodents depends on GABA(B) receptor activation: parallel antinociception testing and medial thalamus GABA microdialysis.
    European journal of pharmacology, 1999, Mar-05, Volume: 368, Issue:2-3

    Topics: Abdomen; Animals; Baclofen; Constriction, Pathologic; Dose-Response Relationship, Drug; Escape Reaction; Extracellular Space; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Male; Mice; Microdialysis; Naloxone; Narcotic Antagonists; Neurotransmitter Uptake Inhibitors; Nipecotic Acids; Nociceptors; Organophosphorus Compounds; Pain; Pain Measurement; Pain Threshold; Psychomotor Performance; Receptors, GABA-B; Thalamus; Tiagabine

1999
Effects of GABAergic modulators on food and cocaine self-administration in baboons.
    Drug and alcohol dependence, 2005, Dec-12, Volume: 80, Issue:3

    Topics: Alprazolam; Animals; Baclofen; Cocaine; Dopamine; Feeding Behavior; GABA Agonists; GABA Modulators; Injections, Intravenous; Male; Nipecotic Acids; Papio anubis; Reinforcement, Psychology; Self Administration; Tiagabine

2005
Attenuation of cocaine-seeking by GABA B receptor agonists baclofen and CGP44532 but not the GABA reuptake inhibitor tiagabine in baboons.
    Drug and alcohol dependence, 2007, Jul-10, Volume: 89, Issue:2-3

    Topics: Animals; Appetitive Behavior; Baclofen; Cocaine-Related Disorders; GABA Antagonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Male; Motivation; Nipecotic Acids; Organophosphonates; Papio anubis; Phosphinic Acids; Self Administration; Tiagabine

2007
Discriminative stimulus effects of tiagabine and related GABAergic drugs in rats.
    Psychopharmacology, 2008, Volume: 197, Issue:4

    Topics: Administration, Oral; Amines; Animals; Anticonvulsants; Azabicyclo Compounds; Baclofen; Benzodiazepines; Bicuculline; Brain; Cyclohexanecarboxylic Acids; Discrimination Learning; Dose-Response Relationship, Drug; GABA Agents; GABA Agonists; GABA Antagonists; GABA Plasma Membrane Transport Proteins; Gabapentin; gamma-Aminobutyric Acid; Generalization, Stimulus; Hypnotics and Sedatives; Injections, Intraperitoneal; Isoxazoles; Male; Nipecotic Acids; Piperazines; Pyridines; Rats; Thiophenes; Tiagabine; Zolpidem

2008
Blockade of GABA(B) receptors facilitates evoked neurotransmitter release at spinal dorsal horn synapse.
    Neuroscience, 2011, Oct-13, Volume: 193

    Topics: Amino Acids; Animals; Baclofen; Benzylamines; Electric Stimulation; Excitatory Amino Acid Antagonists; GABA Agonists; GABA-A Receptor Antagonists; In Vitro Techniques; Male; Neurotransmitter Agents; Nipecotic Acids; Patch-Clamp Techniques; Phosphinic Acids; Posterior Horn Cells; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Spinal Cord; Synapses; Synaptic Potentials; Tiagabine; Xanthenes

2011
Tiagabine Protects Dopaminergic Neurons against Neurotoxins by Inhibiting Microglial Activation.
    Scientific reports, 2015, Oct-26, Volume: 5

    Topics: Animals; Baclofen; Cell Line, Tumor; Disease Models, Animal; Dopaminergic Neurons; GABA Plasma Membrane Transport Proteins; Inflammation Mediators; Lipopolysaccharides; Mice; Mice, Inbred C57BL; Mice, Knockout; Microglia; MPTP Poisoning; Muscimol; Neuroprotective Agents; Neurotoxins; NF-kappa B; Nipecotic Acids; Tiagabine

2015
Central GABAA receptors are involved in inflammatory and cardiovascular consequences of endotoxemia in conscious rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 2016, Volume: 389, Issue:3

    Topics: Animals; Arterial Pressure; Baclofen; Bicuculline; Endotoxemia; GABA Agents; Heart Rate; Interleukin-6; Lipopolysaccharides; Male; Nipecotic Acids; Nitric Oxide; Rats, Wistar; Receptors, GABA-A; Tiagabine; Tumor Necrosis Factor-alpha; Vigabatrin

2016