thiorphan and piperidines

thiorphan has been researched along with piperidines in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's7 (53.85)18.2507
2000's4 (30.77)29.6817
2010's2 (15.38)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bryce, DK; Desai, MC; Heym, J; Longo, KP; McLean, S; Rosen, T; Schmidt, AW; Snider, RM1
Advenier, C; Emonds-Alt, X; Girard, V; Yavo, JC1
Chan, CC; Rodger, IW; Savoie, C; Tousignant, C1
Giuliani, S; Maggi, CA1
Costa, C; Cozzolino, A; Esposito, C; Falciani, M; Filippelli, A; Porta, R; Rossi, F1
Dean, PM; Mills, JE; Perkins, TD1
Carter, JD; Devlin, RB; Oortgiesen, M; Simon, SA; Veronesi, B1
Coupar, IM; Kerr, KP; Thai, B1
Craib, SJ; Ellington, HC; Pertwee, RG; Ross, RA1
D'Orléans-Juste, P; Honoré, JC; Neugebauer, W; Plante, M1
De Lima, TC; Duarte, FS; Testolin, R1
Kamata, K; Kobayashi, T; Matsumoto, T; Ozawa, Y; Taguchi, K1
Batenburg, WW; Bhaggoe, UM; Clahsen-van Groningen, MC; de Vries, R; Domenig, O; Friesema, EC; Garrelds, IM; Hoorn, EJ; Jan Danser, AH; Leijten, FP; Poglitsch, M; Roksnoer, LC; van Veghel, R1

Other Studies

13 other study(ies) available for thiorphan and piperidines

ArticleYear
CP-99,994, a nonpeptide antagonist of the tachykinin NK1 receptor.
    Regulatory peptides, 1993, Jul-02, Volume: 46, Issue:1-2

    Topics: Albuterol; Animals; Binding, Competitive; Calcium Channels; Capsaicin; Dose-Response Relationship, Drug; Guinea Pigs; Kinetics; Lung; Neurokinin A; Neurokinin-1 Receptor Antagonists; Piperidines; Receptors, Neurokinin-1; Thiorphan; Verapamil

1993
The tachykinin NK2 receptor antagonist SR 48968 inhibits citric acid-induced airway hyperresponsiveness in guinea pigs.
    American journal of respiratory and critical care medicine, 1996, Volume: 153, Issue:5

    Topics: Acetylcholine; Aerosols; Animals; Benzamides; Bronchial Hyperreactivity; Bronchoconstriction; Capsaicin; Citrates; Citric Acid; Codeine; Disease Models, Animal; Dose-Response Relationship, Drug; Female; Guinea Pigs; Injections, Intraperitoneal; Injections, Intravenous; Male; Narcotics; Piperidines; Protease Inhibitors; Quinuclidines; Receptors, Neurokinin-2; Receptors, Tachykinin; Stereoisomerism; Tachykinins; Thiorphan

1996
Involvement of NK1 and NK2 receptors in pulmonary responses elicited by non-adrenergic, non-cholinergic vagal stimulation in guinea-pigs.
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:11

    Topics: Animals; Benzamides; Bronchi; Bronchoconstriction; Capillary Permeability; Enalapril; Guinea Pigs; Male; Piperidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Substance P; Thiorphan; Trachea; Vagus Nerve

1995
Characterization of the apamin- and L-nitroarginine-resistant NANC inhibitory transmission to the circular muscle of guinea-pig colon.
    Journal of autonomic pharmacology, 1996, Volume: 16, Issue:3

    Topics: Adrenergic Agents; Animals; Apamin; Atropine; Autonomic Nervous System; Colon; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; Guanethidine; Guinea Pigs; Humans; Indoles; Male; Muscarinic Antagonists; Muscle Relaxation; Muscle, Smooth; Nitroarginine; Piperidines; Protease Inhibitors; Quinuclidines; Thiorphan; Vasoactive Intestinal Peptide

1996
Transglutaminase-synthesized spermine derivative of substance P recognizes rat portal vein neurokinin-3 receptors.
    Life sciences, 1997, Volume: 60, Issue:6

    Topics: Androstanes; Animals; Benzimidazoles; In Vitro Techniques; Male; Neurokinin A; Peptide Fragments; Physalaemin; Piperidines; Portal Vein; Rats; Rats, Wistar; Receptors, Neurokinin-3; Substance P; Thiorphan; Transglutaminases; Vasoconstriction

1997
An automated method for predicting the positions of hydrogen-bonding atoms in binding sites.
    Journal of computer-aided molecular design, 1997, Volume: 11, Issue:3

    Topics: Antithrombins; Binding Sites; Computer Simulation; Folic Acid; Hydrogen Bonding; Ligands; Methotrexate; Models, Molecular; Piperidines; Protein Structure, Tertiary; Software; Stereoisomerism; Thermolysin; Thiorphan; Thrombin

1997
Neuropeptides and capsaicin stimulate the release of inflammatory cytokines in a human bronchial epithelial cell line.
    Neuropeptides, 1999, Volume: 33, Issue:6

    Topics: Bronchi; Calcitonin Gene-Related Peptide; Calcium; Capsaicin; Cell Line, Transformed; Cytokines; Epithelial Cells; Gene Expression; Humans; Interleukin-6; Interleukin-8; Peptide Fragments; Piperidines; Protease Inhibitors; RNA, Messenger; Substance P; Thiorphan; Tumor Necrosis Factor-alpha

1999
Tachykinin-induced contraction of the guinea-pig isolated oesophageal mucosa is mediated by NK(2) receptors.
    British journal of pharmacology, 2000, Volume: 131, Issue:7

    Topics: Animals; Benzamides; Captopril; Dose-Response Relationship, Drug; Esophagus; Guinea Pigs; In Vitro Techniques; Mucous Membrane; Muscle Contraction; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Protease Inhibitors; Quinolines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Tachykinins; Thiorphan

2000
A possible role of lipoxygenase in the activation of vanilloid receptors by anandamide in the guinea-pig bronchus.
    British journal of pharmacology, 2001, Volume: 134, Issue:1

    Topics: 5,8,11,14-Eicosatetraynoic Acid; Animals; Arachidonic Acids; Bronchi; Calcium Channel Blockers; Capsaicin; Cyclohexanols; Dose-Response Relationship, Drug; Endocannabinoids; Fatty Acids, Unsaturated; Guinea Pigs; Hydrazines; In Vitro Techniques; Indomethacin; Lipoxygenase; Muscle Contraction; Oxazepines; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Receptors, Drug; Rimonabant; Thiorphan

2001
Endothelin-1 (1-31) induces a thiorphan-sensitive release of eicosanoids via ET(B) receptors in the guinea pig perfused lung.
    Clinical science (London, England : 1979), 2002, Volume: 103 Suppl 48

    Topics: 6-Ketoprostaglandin F1 alpha; Animals; Eicosanoids; Endothelin Receptor Antagonists; Endothelin-1; Endothelins; Enzyme Inhibitors; Guinea Pigs; Lung; Neprilysin; Oligopeptides; Peptide Fragments; Peptides, Cyclic; Perfusion; Piperidines; Protein Precursors; Receptor, Endothelin A; Receptor, Endothelin B; Receptors, Endothelin; Thiorphan; Thromboxane A2

2002
Further evidence on the anxiogenic-like effect of substance P evaluated in the elevated plus-maze in rats.
    Behavioural brain research, 2004, Oct-05, Volume: 154, Issue:2

    Topics: Analysis of Variance; Animals; Behavior, Animal; Benzamides; Dipeptides; Dose-Response Relationship, Drug; Drug Interactions; Glycopeptides; Indoles; Injections, Intraventricular; Male; Maze Learning; Microinjections; Motor Activity; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Protease Inhibitors; Pyrrolidonecarboxylic Acid; Rats; Rats, Wistar; Receptors, Neurokinin-2; Substance P; Thiorphan; Time Factors

2004
Diabetes-associated changes and role of N epsilon-(carboxymethyl)lysine in big ET-1-induced coronary vasoconstriction.
    Peptides, 2010, Volume: 31, Issue:2

    Topics: Animals; Aspartic Acid Endopeptidases; Benzofurans; Blood Glucose; Body Weight; Coronary Vessels; Diabetes Mellitus, Experimental; Endothelin A Receptor Antagonists; Endothelin B Receptor Antagonists; Endothelin-1; Endothelin-Converting Enzymes; Enzyme Inhibitors; Glycopeptides; Heart; Lipids; Lysine; Male; Metalloendopeptidases; Myocardium; Oligopeptides; Organ Size; Organophosphonates; Peptides, Cyclic; Perfusion; Piperidines; Rats; Rats, Wistar; Receptor, Endothelin A; Receptor, Endothelin B; Thiorphan; Vasoconstriction

2010
Optimum AT1 receptor-neprilysin inhibition has superior cardioprotective effects compared with AT1 receptor blockade alone in hypertensive rats.
    Kidney international, 2015, Volume: 88, Issue:1

    Topics: Angiotensin II Type 1 Receptor Blockers; Animals; Arterial Pressure; Atrial Natriuretic Factor; Biphenyl Compounds; Body Weight; Endothelin B Receptor Antagonists; Endothelin-1; Irbesartan; Kidney; Myocardium; Myocytes, Cardiac; Neprilysin; Oligopeptides; Organ Size; Piperidines; Protease Inhibitors; Rats; Receptor, Angiotensin, Type 1; Receptor, Endothelin B; Renin-Angiotensin System; Sodium-Hydrogen Exchanger 3; Sodium-Hydrogen Exchangers; Tetrazoles; Thiorphan; Up-Regulation; Vasoconstriction; Vasodilation

2015