thiorphan and omapatrilat

thiorphan has been researched along with omapatrilat in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (25.00)29.6817
2010's2 (50.00)24.3611
2020's1 (25.00)2.80

Authors

AuthorsStudies
Berezin, AE1
Berry, C; Biggerstaff, F; Clarke, A; Dalzell, JR; Hillier, C; McMurray, JJ; Padmanabhan, N; Petrie, MC; Seed, A; Whelan, CJ1
Iqbal, S; Ul-Haq, Z; Usmani, S; Zia, SR1
Acharya, KR; Cozier, GE; Sharma, U; Sturrock, ED1

Reviews

1 review(s) available for thiorphan and omapatrilat

ArticleYear
[The new class of drugs-- metalloprotease inhibitors -- in the treatment of heart failure].
    Klinicheskaia meditsina, 2004, Volume: 82, Issue:5

    Topics: Glycopeptides; Heart Failure; Hemodynamics; Humans; Indans; Metalloproteases; Propionates; Protease Inhibitors; Pyridines; Thiazepines; Thiorphan

2004

Other Studies

3 other study(ies) available for thiorphan and omapatrilat

ArticleYear
Effects of neutral endopeptidase (neprilysin) inhibition on the response to other vasoactive peptides in small human resistance arteries: studies with thiorphan and omapatrilat.
    Cardiovascular therapeutics, 2014, Volume: 32, Issue:1

    Topics: Adrenomedullin; Aged; Angiotensin I; Arteries; Captopril; Female; Humans; Male; Middle Aged; Neprilysin; Protease Inhibitors; Pyridines; Substance P; Thiazepines; Thiorphan; Vasodilation

2014
In silico based investigation of dynamic variations in neprilysin (NEP and NEP2) proteins for extracting the point of specificity.
    Molecular bioSystems, 2016, Volume: 12, Issue:3

    Topics: Alanine; Amino Acid Sequence; Computer Simulation; Enzyme Inhibitors; Humans; Ligands; Molecular Dynamics Simulation; Molecular Sequence Data; Neprilysin; Pyridines; Sequence Alignment; Structural Homology, Protein; Thiazepines; Thiorphan

2016
Molecular Basis for Omapatrilat and Sampatrilat Binding to Neprilysin-Implications for Dual Inhibitor Design with Angiotensin-Converting Enzyme.
    Journal of medicinal chemistry, 2020, 05-28, Volume: 63, Issue:10

    Topics: Angiotensin-Converting Enzyme Inhibitors; Antihypertensive Agents; Crystallography, X-Ray; Drug Design; Mesylates; Neprilysin; Peptidyl-Dipeptidase A; Protein Binding; Protein Structure, Secondary; Pyridines; Thiazepines; Tyrosine

2020
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