Page last updated: 2024-08-16

thioridazine and piperidines

thioridazine has been researched along with piperidines in 29 studies

Research

Studies (29)

TimeframeStudies, this research(%)All Research%
pre-199021 (72.41)18.7374
1990's4 (13.79)18.2507
2000's4 (13.79)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Arlock, P; Gullberg, B; Olsson, SR1
Gerlach, J; Simmelsgaard, H1
Obukhov, GA1
Olsson, SO; Passwal, M; Refsum, H1
Fink, H; Morgenstern, R; Ott, T; Schremmer, C1
Cote, M; Drolet, A; Gautier, J; Jus, A; Jus, K; Pineau, R; Pires, P; Villeneuve, A; Villeneuve, R1
Zingales, IA1
Sedvall, G1
Giovannucci, M; Mastruzzo, A; Montanini, R1
Ananth, JV; Ban, TA; Deutsch, M1
Costall, B; Naylor, RJ1
Schwingenheuer, J1
Perez de Francisco, C1
Janssen, PA; Niemegeers, CJ; Verbruggen, FJ2
Hollister, LE1
Mathalone, MB1
Herzog, R; Petrilowitsch, N1
Goss, JB1
Assié, MB; Koek, W; Sleight, AJ1
Chu, KW; Damani, LA; Hawes, EM; Lin, G; Midha, KK1
Millan, MJ; Newman-Tancredi, A; Touzard, M; Verrièle, L1
DANDIYA, PC; MENON, MK1
IWAMOTO, T; SATOH, T; TOKUMITSU, Y1
HADER, M; SCHULMAN, PM1
Boyce, M; Dunn, K; Johnston, A; Ravic, M; Warrington, S1
Abe, J; Hamada, Y; Harada, T; Hashimoto, K; Horii, I; Sawada, Y; Shiotani, M1
Daniel, WA; Maurel, P; Wójcikowski, J1

Trials

5 trial(s) available for thioridazine and piperidines

ArticleYear
Tardive dyskinesia during and following treatment with haloperidol, haloperidol + biperiden, thioridazine, and clozapine.
    Psychopharmacology, 1978, Oct-31, Volume: 59, Issue:2

    Topics: Aged; Biperiden; Clinical Trials as Topic; Clozapine; Dibenzazepines; Drug Therapy, Combination; Dyskinesia, Drug-Induced; Female; Haloperidol; Humans; Male; Parkinson Disease, Secondary; Piperidines; Psychotic Disorders; Thioridazine

1978
Penfluridol: a long-acting oral neuroleptic as therapeutic agent in chronic schizophrenia.
    Current therapeutic research, clinical and experimental, 1974, Volume: 16, Issue:10

    Topics: Adult; Analysis of Variance; Basal Ganglia Diseases; Body Weight; Chlorpromazine; Chronic Disease; Clinical Trials as Topic; Electrocardiography; Electroencephalography; Female; Humans; Hydrocarbons, Halogenated; Male; Middle Aged; Piperidines; Placebos; Psychiatric Status Rating Scales; Schizophrenia; Social Behavior; Substance Withdrawal Syndrome; Thioridazine; Toluene; Tranquilizing Agents; Vision Tests

1974
A clinical study with propericiazine in chronic psychotic patients.
    Current therapeutic research, clinical and experimental, 1971, Volume: 13, Issue:6

    Topics: Adult; Chronic Disease; Clinical Trials as Topic; Female; Humans; Male; Middle Aged; Nitriles; Phenothiazines; Piperidines; Psychiatric Status Rating Scales; Psychotic Disorders; Thioridazine; Tranquilizing Agents

1971
Early clinical drug evaluation units reports.
    Psychopharmacology bulletin, 1972, Volume: 8, Issue:1

    Topics: Adult; Aged; Clinical Trials as Topic; Evaluation Studies as Topic; Female; Humans; Imipramine; Ketones; Male; Middle Aged; Phenothiazines; Piperidines; Schizophrenia; Thioridazine

1972
Repeated dosing with donepezil does not affect the safety, tolerability or pharmacokinetics of single-dose thioridazine in young volunteers.
    British journal of clinical pharmacology, 2004, Volume: 58 Suppl 1

    Topics: Adult; Antipsychotic Agents; Area Under Curve; Cholinesterase Inhibitors; Cross-Over Studies; Donepezil; Drug Interactions; Female; Humans; Indans; Male; Piperidines; Thioridazine

2004

Other Studies

24 other study(ies) available for thioridazine and piperidines

ArticleYear
Cardiac electrophysiology of four neuroleptics: melperone, haloperidol, thioridazine and chlorpromazine.
    Naunyn-Schmiedeberg's archives of pharmacology, 1978, Volume: 304, Issue:1

    Topics: Action Potentials; Animals; Antipsychotic Agents; Butyrophenones; Chlorpromazine; Guinea Pigs; Haloperidol; Heart; In Vitro Techniques; Membrane Potentials; Myocardial Contraction; Papillary Muscles; Piperidines; Refractory Period, Electrophysiological; Thioridazine

1978
[Prolonged action neuroleptics (review of the foreign literature)].
    Zhurnal nevropatologii i psikhiatrii imeni S.S. Korsakova (Moscow, Russia : 1952), 1975, Volume: 75, Issue:2

    Topics: Acute Disease; Antipsychotic Agents; Basal Ganglia Diseases; Bipolar Disorder; Child; Chronic Disease; Delayed-Action Preparations; Dibenzazepines; Dibenzothiepins; Dosage Forms; Drug Therapy, Combination; Fluphenazine; Humans; Paranoid Disorders; Perphenazine; Pimozide; Piperazines; Piperidines; Schizophrenia; Structure-Activity Relationship; Thioridazine; Thioxanthenes; Tranquilizing Agents

1975
Comparison of the electrophysiological effects of two neuroleptics, melperone and thioridazine, on isolated rat atria.
    European journal of pharmacology, 1978, Jun-01, Volume: 49, Issue:3

    Topics: Animals; Butyrophenones; Electric Stimulation; Female; Heart; Heart Rate; In Vitro Techniques; Myocardial Contraction; Piperidines; Rats; Refractory Period, Electrophysiological; Sinoatrial Node; Thioridazine; Tranquilizing Agents

1978
Atypical neuroleptics suppress dopaminergic behavioral supersensitivity.
    Psychopharmacology, 1990, Volume: 100, Issue:3

    Topics: Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Clozapine; Cyproheptadine; Haloperidol; Male; Piperidines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Ritanserin; Serotonin Antagonists; Sulpiride; Thioridazine

1990
Detection of chlorpromazine and thioridazine metabolites in human erythrocytes.
    Journal of chromatography, 1969, Nov-11, Volume: 44, Issue:3

    Topics: Chlorpromazine; Chromatography, Thin Layer; Erythrocytes; Hemolysis; Humans; Indicators and Reagents; Methods; Phenothiazines; Piperidines; Plasma; Silicon Dioxide; Sulfoxides; Thioridazine; Time Factors

1969
[Therapy of anxiety, mental anguish and sleeplessness. 3. Clinical pharmacological viewpoints].
    Lakartidningen, 1969, Mar-17, Volume: 66

    Topics: Alcoholism; Alcohols; Aldehydes; Antidepressive Agents; Azepines; Barbiturates; Bromides; Chlordiazepoxide; Chlormethiazole; Histamine H1 Antagonists; Humans; Hypnotics and Sedatives; Methaqualone; Neurotic Disorders; Phenothiazines; Piperidines; Propylene Glycols; Thioridazine; Tranquilizing Agents; Xanthenes

1969
[Clinical expressions of aggressive behavior and their treatment].
    Giornale di psichiatria e di neuropatologia, 1968, Volume: 96, Issue:3

    Topics: Aggression; Carbamazepine; Dibenzazepines; Humans; Mental Disorders; Nitriles; Phenothiazines; Piperidines; Thioridazine; Tranquilizing Agents

1968
Is there a relationship between the involvement of extrapyramidal and mesolimbic brain areas with the cataleptic action of neuroleptic agents and their clinical antipsychotic effect?
    Psychopharmacologia, 1973, Volume: 32, Issue:2

    Topics: Animals; Aporphines; Benzoates; Butyrophenones; Catalepsy; Dioxoles; Extrapyramidal Tracts; Humans; Hypothalamus; Male; Metoclopramide; Perphenazine; Piperidines; Rats; Spiro Compounds; Thioridazine; Tranquilizing Agents

1973
[Alternating use of Melleril-Sandoz (thioridazine) and its metabolite Inofal in psychiatric treatment].
    Die Medizinische Welt, 1971, Oct-22, Volume: 43

    Topics: Adolescent; Adult; Aged; Drug Synergism; Female; Humans; Male; Mental Disorders; Middle Aged; Phenothiazines; Piperidines; Sulfones; Thioridazine

1971
[Psychopharmacological treatment of anxiety].
    La Prensa medica mexicana, 1971, Volume: 36, Issue:9

    Topics: Adult; Amitriptyline; Anxiety; Benzazepines; Carbamates; Chlordiazepoxide; Diazepam; Dibenzazepines; Female; Humans; Ketones; Meprobamate; Methotrimeprazine; Nitro Compounds; Oxazepam; Piperidines; Thioridazine

1971
The influence of various neuroleptic drugs on shock avoidance responding in rats. I. Nondiscriminated Sidman avoidance procedure.
    Psychopharmacologia, 1969, Volume: 16, Issue:3

    Topics: Animals; Antidepressive Agents; Avoidance Learning; Benperidol; Benzimidazoles; Butyrophenones; Chlorpromazine; Depression, Chemical; Electroshock; Escape Reaction; Female; Fluorine; Fluphenazine; Haloperidol; Isonipecotic Acids; Perphenazine; Piperidines; Promazine; Rats; Spiro Compounds; Thioridazine; Tranquilizing Agents; Trifluoperazine

1969
Choice of antipsychotic drugs.
    The American journal of psychiatry, 1970, Volume: 127, Issue:2

    Topics: Butyrophenones; Drug Synergism; Drug Tolerance; Haloperidol; Humans; Phenothiazines; Piperazines; Piperidines; Psychopharmacology; Psychotherapy; Psychotic Disorders; Thioridazine; Thiothixene; Tranquilizing Agents; Triflupromazine; Xanthenes

1970
The influence of various neuroleptic drugs on noise escape response in rats.
    Psychopharmacologia, 1970, Volume: 18, Issue:3

    Topics: Animals; Antidepressive Agents; Avoidance Learning; Benperidol; Blepharoptosis; Butyrophenones; Catalepsy; Chlorpromazine; Escape Reaction; Female; Fluorine; Fluphenazine; Haloperidol; Humans; Noise; Perphenazine; Piperidines; Rats; Spiro Compounds; Thioridazine; Tranquilizing Agents; Trifluoperazine; Triflupromazine

1970
Ocular effects of phenothiazine derivatives and reversibility.
    Diseases of the nervous system, 1968, Volume: 29, Issue:3

    Topics: Accommodation, Ocular; Animals; Cats; Chlorpromazine; Cornea; Eye Diseases; Female; Fundus Oculi; Humans; Lens, Crystalline; Male; Penicillamine; Phenothiazines; Pigmentation Disorders; Piperazines; Piperidines; Schizophrenia; Thioridazine; Tranquilizing Agents

1968
[Complementary neurolepsy].
    Psychiatria et neurologia, 1966, Volume: 151, Issue:4

    Topics: Adult; Butyrophenones; Depression; Female; Fluphenazine; Humans; Male; Piperidines; Psychotic Disorders; Schizophrenia; Thioridazine

1966
Concomitant use of thioridazine with risperidone.
    American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists, 1995, May-01, Volume: 52, Issue:9

    Topics: Antipsychotic Agents; Drug Therapy, Combination; Humans; Isoxazoles; Piperidines; Risperidone; Schizophrenia; Thioridazine

1995
Biphasic displacement of [3H]YM-09151-2 binding in the rat brain by thioridazine, risperidone and clozapine, but not by other antipsychotics.
    European journal of pharmacology, 1993, Jun-24, Volume: 237, Issue:2-3

    Topics: Animals; Antipsychotic Agents; Benzamides; Brain; Clozapine; Corpus Striatum; Dopamine D2 Receptor Antagonists; In Vitro Techniques; Isoxazoles; Male; Olfactory Pathways; Piperidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Risperidone; Spiperone; Thioridazine

1993
Identification of lactams as in vitro metabolites of piperidine-type phenothiazine antipsychotic drugs.
    Journal of pharmaceutical and biomedical analysis, 1996, Volume: 14, Issue:6

    Topics: Animals; Antipsychotic Agents; Biotransformation; Chromatography, High Pressure Liquid; Chromatography, Ion Exchange; Dogs; Female; Humans; In Vitro Techniques; Lactams; Liver; Male; Mass Spectrometry; Mesoridazine; Phenothiazines; Piperidines; Rats; Rats, Sprague-Dawley; Thioridazine

1996
Efficacy of antipsychotic agents at human 5-HT(1A) receptors determined by [3H]WAY100,635 binding affinity ratios: relationship to efficacy for G-protein activation.
    European journal of pharmacology, 2001, Oct-05, Volume: 428, Issue:2

    Topics: Animals; Antipsychotic Agents; Binding, Competitive; Chlorpromazine; CHO Cells; Clozapine; Cricetinae; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Humans; Membranes; Piperazines; Piperidines; Pyridines; Pyrimidinones; Pyrrolidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Thiazoles; Thioridazine; Tritium

2001
Studies on central nervous system depressants. (III). Influence of some tranquillizing agents on morphine analgesia.
    Archives internationales de pharmacodynamie et de therapie, 1963, Jan-01, Volume: 141

    Topics: Amides; Analgesia; Carisoprodol; Chlorpromazine; Meprobamate; Morphine; Perphenazine; Phenothiazines; Piperidines; Prochlorperazine; Propylene Glycols; Rauwolfia; Reserpine; Thioridazine; Tranquilizing Agents

1963
EFFECTS OF SOME TRANQUILLIZING AGENTS ON BRAIN NORADRENALINE AND DOPAMINE LEVELS OF SHOCKED RATS.
    Japanese journal of pharmacology, 1964, Volume: 14

    Topics: Blood-Brain Barrier; Brain; Chlordiazepoxide; Chlorpromazine; Cyproheptadine; Dopamine; Electricity; Fluorometry; Norepinephrine; Pharmacology; Piperidines; Rats; Research; Shock; Tetrabenazine; Thioridazine; Tranquilizing Agents

1964
TANDEM PIPERIDINE AND DIMETHYL PHENOTHIAZINE TOXICITY IN A GERIATRIC PATIENT.
    New York state journal of medicine, 1965, Jul-01, Volume: 65

    Topics: Drug Therapy; Geriatrics; Patients; Phenothiazines; Piperidines; Thioridazine; Toxicology

1965
Practical application of guinea pig telemetry system for QT evaluation.
    The Journal of toxicological sciences, 2005, Volume: 30, Issue:3

    Topics: Animals; Anti-Arrhythmia Agents; Antipsychotic Agents; Bepridil; Cisapride; Disease Models, Animal; Electrocardiography; Guinea Pigs; Haloperidol; Heart; Humans; Injections, Intravenous; Long QT Syndrome; Male; Nifedipine; Pimozide; Piperidines; Pyridines; Quinidine; Reproducibility of Results; Telemetry; Terfenadine; Thioridazine

2005
Characterization of human cytochrome p450 enzymes involved in the metabolism of the piperidine-type phenothiazine neuroleptic thioridazine.
    Drug metabolism and disposition: the biological fate of chemicals, 2006, Volume: 34, Issue:3

    Topics: Animals; Antipsychotic Agents; Biotransformation; Catalysis; Cloning, Molecular; Cytochrome P-450 Enzyme System; Humans; In Vitro Techniques; Insecta; Microsomes, Liver; Piperidines; Thioridazine

2006