Compounds > thiophenes
Page last updated: 2024-08-18

thiophenes and sr9011

thiophenes has been researched along with sr9011 in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's8 (80.00)24.3611
2020's2 (20.00)2.80

Authors

AuthorsStudies
Banerjee, S; Burris, TP; Butler, AA; Cameron, MD; Hughes, T; Kamenecka, TM; Kojetin, DJ; Liu, J; Lundasen, T; Noel, R; Shin, Y; Solt, LA; Takahashi, JS; Wang, Y; Yoo, SH1
Bass, J1
Shea, SA1
Amador, A; Banerjee, S; Burris, TP; El-Gendy, BM; Griffett, K; Huitron-Resendiz, S; Kamenecka, TM; Kazantzis, M; Roberts, AJ; Shin, Y; Solt, LA; Wang, Y1
Burris, TP; Kojetin, D; Wang, Y1
Deventer, K; Geldof, L; Roels, K; Tudela, E; Van Eeno, P1
Kolar, MJ; Panda, S; Plikus, MV; Puca, F; Rommel, A; Saghatelian, A; Sulli, G; Verma, IM; Wang, X1
Guo, DK; Hao, ZB; Mu, CC; Ren, HG; Sun, HY; Wang, GH; Xu, XY; Zhang, S; Zhu, Y1
Gao, Y; Jiao, H; Kalsbeek, A; Sun, J; Wang, XL; Wolff, SEC; Yi, CX1
Kwak, YB; Yoo, HH; Yu, J1

Other Studies

10 other study(ies) available for thiophenes and sr9011

ArticleYear
Regulation of circadian behaviour and metabolism by synthetic REV-ERB agonists.
    Nature, 2012, Mar-29, Volume: 485, Issue:7396

    Topics: Adipose Tissue; Animals; Biological Clocks; Circadian Rhythm; Disease Models, Animal; Energy Metabolism; HEK293 Cells; Humans; Hypothalamus; Liver; Metabolome; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Muscle, Skeletal; Nuclear Receptor Subfamily 1, Group D, Member 1; Obesity; Pyrrolidines; Receptors, Cytoplasmic and Nuclear; Repressor Proteins; Thiophenes

2012
Drug discovery: Time in a bottle.
    Nature, 2012, May-02, Volume: 485, Issue:7396

    Topics: Animals; Circadian Rhythm; Energy Metabolism; Humans; Lipid Metabolism; Male; Nuclear Receptor Subfamily 1, Group D, Member 1; Pyrrolidines; Receptors, Cytoplasmic and Nuclear; Repressor Proteins; Thiophenes

2012
Obesity and pharmacologic control of the body clock.
    The New England journal of medicine, 2012, Jul-12, Volume: 367, Issue:2

    Topics: Adipose Tissue; Animals; Biological Clocks; Circadian Rhythm; Humans; Mice; Nuclear Receptor Subfamily 1, Group D, Member 1; Obesity; Pyrrolidines; Receptors, Cytoplasmic and Nuclear; Repressor Proteins; Thiophenes

2012
Pharmacological targeting of the mammalian clock regulates sleep architecture and emotional behaviour.
    Nature communications, 2014, Dec-23, Volume: 5

    Topics: Animals; Anxiety; ARNTL Transcription Factors; Behavior, Animal; Circadian Clocks; Circadian Rhythm; CLOCK Proteins; Cryptochromes; Feedback, Physiological; Gene Expression Regulation; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Nuclear Receptor Subfamily 1, Group D, Member 1; Period Circadian Proteins; Pyrrolidines; Receptors, Cytoplasmic and Nuclear; Repressor Proteins; Reward; Signal Transduction; Sleep, REM; Thiophenes

2014
Anti-proliferative actions of a synthetic REV-ERBα/β agonist in breast cancer cells.
    Biochemical pharmacology, 2015, Aug-15, Volume: 96, Issue:4

    Topics: Antineoplastic Agents; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Cyclin A; Female; Humans; Nuclear Receptor Subfamily 1, Group D, Member 1; Pyrrolidines; Receptor, ErbB-2; Receptors, Estrogen; Thiophenes; Triple Negative Breast Neoplasms

2015
In Vitro Metabolic Studies of REV-ERB Agonists SR9009 and SR9011.
    International journal of molecular sciences, 2016, Oct-03, Volume: 17, Issue:10

    Topics: Chromatography, High Pressure Liquid; Doping in Sports; Humans; Nuclear Receptor Subfamily 1, Group D, Member 1; Pyrrolidines; Retrospective Studies; Tandem Mass Spectrometry; Thiophenes

2016
Pharmacological activation of REV-ERBs is lethal in cancer and oncogene-induced senescence.
    Nature, 2018, 01-18, Volume: 553, Issue:7688

    Topics: Animals; Apoptosis; Autophagy; Cell Line, Tumor; Cell Survival; Circadian Clocks; Female; Glioblastoma; GTP Phosphohydrolases; Humans; Lipogenesis; Male; Membrane Proteins; Mice, Inbred C57BL; Neoplasms; Nevus; Nuclear Receptor Subfamily 1, Group D, Member 1; Oncogenes; Pyrrolidines; Signal Transduction; Thiophenes

2018
Pharmacological activation of REV-ERBα represses LPS-induced microglial activation through the NF-κB pathway.
    Acta pharmacologica Sinica, 2019, Volume: 40, Issue:1

    Topics: Animals; Cell Line, Tumor; Glycine; HEK293 Cells; Humans; Inflammation; Male; Mesencephalon; Mice, Inbred C57BL; Microglia; Neuroprotective Agents; Nuclear Receptor Subfamily 1, Group D, Member 1; Pyrrolidines; Signal Transduction; Thiophenes; Transcription Factor RelA

2019
The Effect of Rev-erbα Agonist SR9011 on the Immune Response and Cell Metabolism of Microglia.
    Frontiers in immunology, 2020, Volume: 11

    Topics: Animals; CLOCK Proteins; Cytokines; Energy Metabolism; Gene Expression Regulation; Immunity; Immunity, Innate; Male; Microglia; Mitochondria; Nuclear Receptor Subfamily 1, Group D, Member 1; Phagocytosis; Pyrrolidines; Rats; Thiophenes

2020
A quantitative method for the simultaneous detection of SR9009 and SR9011 in equine plasma using liquid chromatography-electrospray ionization-tandem mass spectrometry.
    Drug testing and analysis, 2022, Volume: 14, Issue:8

    Topics: Animals; Chromatography, High Pressure Liquid; Chromatography, Liquid; Horses; Pyrrolidines; Reproducibility of Results; Spectrometry, Mass, Electrospray Ionization; Tandem Mass Spectrometry; Thiophenes

2022