Page last updated: 2024-08-18

thiophenes and pirenzepine

thiophenes has been researched along with pirenzepine in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19903 (25.00)18.7374
1990's8 (66.67)18.2507
2000's1 (8.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bartolini, A; Fantetti, L; Ghelardini, C; Giotti, A; Malcangio, M; Malmberg-Aiello, P1
Fisher, A; Segal, M1
Angeli, P; Brasili, L; Cantalamessa, F; Marucci, G; Wess, J1
Matsumoto, M; Morii, K; Saito, H; Togashi, H; Yoshioka, M1
Kato, T; Mizobe, F; Xu, M; Yamamoto, T1
Kawanishi, G; Mizobe, F; Ohgane, N; Ono, S; Saito, Y1
Althoff, PH; Hermann, GJ; Jungmann, E; Schöffling, K1
Ohno, M; Watanabe, S; Yamamoto, T1
Saito, Y1
Ikeda, T1
Bégos, A; Bizot, JC; Breton, P; Brochet, D; Tambuté, A; Trovero, F1
Mitchell, CA; Ward, MD; Yu, L1

Trials

1 trial(s) available for thiophenes and pirenzepine

ArticleYear
The effect of pizotifen, a serotonin antagonist, and of pirenzepine, a muscarinic antagonist, on hormonal responses to metoclopramide in healthy subjects.
    Arzneimittel-Forschung, 1984, Volume: 34, Issue:9

    Topics: Adult; Aldosterone; Benzodiazepinones; Hormones; Humans; Hydrocortisone; Male; Metoclopramide; Parasympatholytics; Pirenzepine; Pizotyline; Prolactin; Renin; Serotonin Antagonists; Thiophenes

1984

Other Studies

11 other study(ies) available for thiophenes and pirenzepine

ArticleYear
Role of muscarinic receptor subtypes in central antinociception.
    British journal of pharmacology, 1992, Volume: 105, Issue:1

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Analgesia; Animals; Male; Mice; Pain Measurement; Pirenzepine; Quinuclidines; Receptors, Muscarinic; Thiophenes

1992
AF102B, a muscarinic M1 receptor agonist, mimics some effects of acetylcholine on neurons of rat hippocampus slices.
    European journal of pharmacology, 1992, Sep-10, Volume: 220, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Electrophysiology; Hippocampus; In Vitro Techniques; Parasympathomimetics; Pirenzepine; Quinuclidines; Rats; Receptors, Muscarinic; Thiophenes

1992
Determination of muscarinic agonist potencies at M1 and M2 muscarinic receptors in a modified pithed rat preparation.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 342, Issue:6

    Topics: Animals; Bradycardia; Diamines; Dimethylamines; Dose-Response Relationship, Drug; Heart Rate; Heterocyclic Compounds; Male; Muscarine; Muscarinic Antagonists; Parasympatholytics; Pirenzepine; Rats; Receptors, Muscarinic; Stereoisomerism; Thiophenes

1990
Sympathoexcitatory action of a novel muscarinic receptor agonist, AF102B, and its blockade by pirenzepine.
    Pharmacology & toxicology, 1990, Volume: 67, Issue:1

    Topics: Anesthesia; Animals; Blood Pressure; Heart; Heart Rate; In Vitro Techniques; Male; Parasympathomimetics; Pirenzepine; Quinuclidines; Rats; Rats, Inbred Strains; Sympathomimetics; Thiophenes

1990
Differential effects of M1- and M2-muscarinic drugs on striatal dopamine release and metabolism in freely moving rats.
    Brain research, 1989, Aug-28, Volume: 495, Issue:2

    Topics: Animals; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Male; Oxotremorine; Pirenzepine; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Thiophenes

1989
Heterogeneity of muscarinic autoreceptors and heteroreceptors in the rat brain: effects of a novel M1 agonist, AF102B.
    European journal of pharmacology, 1988, Oct-11, Volume: 155, Issue:1-2

    Topics: Acetylcholine; Animals; Brain Chemistry; Corpus Striatum; Dopamine; Hippocampus; In Vitro Techniques; Male; Oxotremorine; Parasympathomimetics; Pirenzepine; Potassium; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Synaptosomes; Thiophenes

1988
Blockade of hippocampal M1 muscarinic receptors impairs working memory performance of rats.
    Brain research, 1994, Jul-11, Volume: 650, Issue:2

    Topics: Animals; Conditioning, Operant; Diamines; Dose-Response Relationship, Drug; Hippocampus; Injections; Male; Memory, Short-Term; Muscarinic Agonists; Muscarinic Antagonists; Parasympatholytics; Parasympathomimetics; Pirenzepine; Psychomotor Performance; Quinuclidines; Rats; Rats, Wistar; Thiophenes

1994
[Effect of a muscarinic (M1) receptor agonist on sympathetic nerve activity in rats].
    [Hokkaido igaku zasshi] The Hokkaido journal of medical science, 1993, Volume: 68, Issue:2

    Topics: Adrenal Medulla; Animals; Blood Pressure; Dose-Response Relationship, Drug; Electrophysiology; Heart; Heart Rate; Male; Parasympathomimetics; Pirenzepine; Quinuclidines; Rats; Rats, Wistar; Receptors, Muscarinic; Sympathetic Nervous System; Thiophenes

1993
[Functional role of muscarinic M1 receptor for the ganglionic transmission in the rat superior cervical ganglion].
    [Hokkaido igaku zasshi] The Hokkaido journal of medical science, 1997, Volume: 72, Issue:3

    Topics: Animals; Dimethylphenylpiperazinium Iodide; Ganglionic Stimulants; Hexamethonium; Laser-Doppler Flowmetry; Male; Muscarinic Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Parasympathomimetics; Pirenzepine; Quinuclidines; Rats; Rats, Wistar; Receptors, Muscarinic; Receptors, Nicotinic; Superior Cervical Ganglion; Synaptic Transmission; Thiophenes; Thyroid Gland

1997
Pharmacological profile of CEB-1957 and atropine toward brain muscarinic receptors and comparative study of their efficacy against sarin poisoning.
    Toxicology and applied pharmacology, 1998, Volume: 150, Issue:2

    Topics: Animals; Atropine; Autoradiography; Binding, Competitive; Brain; Cholinesterase Inhibitors; Male; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Poisoning; Rats; Rats, Wistar; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Sarin; Thiophenes

1998
Selective nucleation and discovery of organic polymorphs through epitaxy with single crystal substrates.
    Journal of the American Chemical Society, 2001, Nov-07, Volume: 123, Issue:44

    Topics: Benzodiazepines; Crystallization; Models, Chemical; Olanzapine; Pimelic Acids; Pirenzepine; Substrate Specificity; Succinic Acid; Thiophenes

2001