Page last updated: 2024-08-18

thiophenes and chalcone

thiophenes has been researched along with chalcone in 14 studies

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19903 (21.43)18.7374
1990's0 (0.00)18.2507
2000's2 (14.29)29.6817
2010's5 (35.71)24.3611
2020's4 (28.57)2.80

Authors

AuthorsStudies
Soldati, G1
Hirose, K; Kayano, M; Ukai, S1
Hirose, K; Ukai, S1
Curti, C; Gellis, A; Vanelle, P1
Huang, TF; Lin, CN; Lo, HM; Peng, HC; Wu, WB1
Asiri, AM; Khan, SA1
Borges, F; Kachler, S; Klotz, KN; Matos, MJ; Santana, L; Uriarte, E; Vazquez-Rodriguez, S1
Dodda, RP; Haque, R; Jadiya, P; Kumar, M; Kumar, V; Modukuri, RK; Nazir, A; Sashidhara, KV; Siddiqi, MI; Sridhar, B1
Bilge, M; Chandraju, S; Fun, HK; Kumar, CS; Parlak, C; Quah, CK; Ramasami, P; Rhyman, L; Tursun, M1
Begnini, KR; Carapina, C; Collares, T; de Pereira, CM; Fogaça, TB; Martins, RM; Ritter, M; Seixas, FK1
Abdelhamid, IA; Hassaneen, HM; Helmy, MT; Mahmoud, K; Mahrous, KF; Mohamed Teleb, MA; Saleh, FM; Sroor, FM1
Alanazi, MM; Amran, SI; Biswas, S; Chander, S; Das, B; Hadda, TB; Hasan, AH; Jamalis, J; Murugesan, S; Pratama, MRF; Shakya, S1
Abreu, HR; Andricopulo, AD; Braga, AL; de Oliveira, AS; Ferreira, LL; Krogh, R; Llanes, LC; Meier, L; Nunes, RJ; Souza, JM; Valli, M; Voltolini, BG1
Kamra, N; Kumar, D; Rani, S; Sangwan, PL; Singh, A; Singh, SK; Singh, V; Thakral, S1

Other Studies

14 other study(ies) available for thiophenes and chalcone

ArticleYear
New compounds: addition products of heterocyclic chalcones.
    Journal of pharmaceutical sciences, 1975, Volume: 64, Issue:2

    Topics: Chalcone; Fungicides, Industrial; Furans; Propiophenones; Sulfides; Thiophenes

1975
[Synthesis and biological activity of sulfur containing derivatives of chalcone. IV. A novel method for the synthesis of thioaurones (author's transl)].
    Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan, 1975, Volume: 95, Issue:3

    Topics: Chalcone; Chemical Phenomena; Chemistry; Propiophenones; Thiophenes

1975
[Synthesis and biological activity of sulfur containing derivatives of chalcone. III. The diastereomeric form of an adduct in the reaction of trans-4-nitrochalcone oxide with thiophenol].
    Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan, 1974, Volume: 94, Issue:10

    Topics: Chalcone; Chemical Phenomena; Chemistry; Isomerism; Nitro Compounds; Oxides; Propiophenones; Thiophenes

1974
Synthesis of alpha,beta-unsaturated ketones as chalcone analogues via a S(RN)1 mechanism.
    Molecules (Basel, Switzerland), 2007, Apr-18, Volume: 12, Issue:4

    Topics: Anions; Chalcone; Chemistry; Electrons; Ketones; Magnetic Resonance Spectroscopy; Models, Chemical; Molecular Conformation; Molecular Structure; Propane; Quaternary Ammonium Compounds; Solvents; Temperature; Thiophenes

2007
2'-Ethoxy-5'-methoxy-2-(5-methylthienyl)chalcone inhibits collagen-induced protein tyrosine phosphorylation and thromboxane formation during platelet aggregation and adhesion.
    Pharmacology, 2009, Volume: 84, Issue:3

    Topics: Animals; Chalcone; Collagen; Crotalid Venoms; Focal Adhesion Protein-Tyrosine Kinases; Humans; Inhibitory Concentration 50; Lectins, C-Type; Phosphorylation; Platelet Adhesiveness; Platelet Aggregation; Prostaglandin-Endoperoxide Synthases; Thiophenes; Thromboxane B2; Thromboxane-A Synthase; Tyrosine

2009
Synthesis and anti-bacterial activities of a bis-chalcone derived from thiophene and its bis-cyclized products.
    Molecules (Basel, Switzerland), 2011, Jan-12, Volume: 16, Issue:1

    Topics: Anti-Bacterial Agents; Chalcone; Cyclization; Gas Chromatography-Mass Spectrometry; Gram-Negative Bacteria; Gram-Positive Bacteria; Magnetic Resonance Spectroscopy; Microbial Sensitivity Tests; Spectrophotometry, Infrared; Thiophenes

2011
Chalcone-based derivatives as new scaffolds for hA3 adenosine receptor antagonists.
    The Journal of pharmacy and pharmacology, 2013, Volume: 65, Issue:5

    Topics: Animals; Binding, Competitive; Chalcone; CHO Cells; Coumarins; Cricetinae; Cricetulus; Humans; Ligands; Purinergic P1 Receptor Antagonists; Radioligand Assay; Receptor, Adenosine A1; Receptor, Adenosine A2A; Receptor, Adenosine A2B; Receptor, Adenosine A3; Structure-Activity Relationship; Thiophenes

2013
Benzofuran-chalcone hybrids as potential multifunctional agents against Alzheimer's disease: synthesis and in vivo studies with transgenic Caenorhabditis elegans.
    ChemMedChem, 2014, Volume: 9, Issue:12

    Topics: Acetylcholine; Acetylcholinesterase; Alzheimer Disease; Amyloid beta-Peptides; Animals; Animals, Genetically Modified; Antioxidants; Benzofurans; Binding Sites; Caenorhabditis elegans; Chalcone; Chalcones; Crystallography, X-Ray; Disease Models, Animal; Humans; Microscopy, Fluorescence; Molecular Conformation; Molecular Docking Simulation; Oxidative Stress; Protein Structure, Tertiary; Structure-Activity Relationship; Thiophenes

2014
(2E)-1-(5-Chlorothiophen-2-yl)-3-{4-[(E)-2-phenylethenyl]phenyl}prop-2-en-1-one: Synthesis, XRD, FT-IR, Raman and DFT studies.
    Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy, 2015, Volume: 149

    Topics: Chalcone; Crystallography, X-Ray; Halogenation; Isomerism; Models, Molecular; Quantum Theory; Spectroscopy, Fourier Transform Infrared; Spectrum Analysis, Raman; Thiophenes

2015
Apoptotic effect of chalcone derivatives of 2-acetylthiophene in human breast cancer cells.
    Pharmacological reports : PR, 2017, Volume: 69, Issue:1

    Topics: Apoptosis; Breast Neoplasms; Cell Survival; Chalcone; Dose-Response Relationship, Drug; Female; Growth Inhibitors; Humans; MCF-7 Cells; Thiophenes

2017
Anticancer activity of novel 3-(furan-2-yl)pyrazolyl and 3-(thiophen-2-yl)pyrazolyl hybrid chalcones: Synthesis and in vitro studies.
    Archiv der Pharmazie, 2022, Volume: 355, Issue:3

    Topics: Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Cell Survival; Chalcone; Chalcones; Drug Screening Assays, Antitumor; Furans; Humans; Structure-Activity Relationship; Thiophenes

2022
Novel thiophene Chalcones-Coumarin as acetylcholinesterase inhibitors: Design, synthesis, biological evaluation, molecular docking, ADMET prediction and molecular dynamics simulation.
    Bioorganic chemistry, 2022, Volume: 119

    Topics: Acetylcholinesterase; Alzheimer Disease; Cells, Cultured; Chalcone; Cholinesterase Inhibitors; Coumarins; Dose-Response Relationship, Drug; Drug Design; Humans; Models, Molecular; Molecular Structure; Structure-Activity Relationship; Thiophenes

2022
Novel trypanocidal thiophen-chalcone cruzain inhibitors: structure- and ligand-based studies.
    Future medicinal chemistry, 2022, Volume: 14, Issue:11

    Topics: Chagas Disease; Chalcone; Chalcones; Cysteine Endopeptidases; Humans; Ligands; Molecular Docking Simulation; Protozoan Proteins; Structure-Activity Relationship; Thiophenes; Trypanocidal Agents; Trypanosoma cruzi

2022
Synthesis, Biological Activity and Molecular Docking Studies of Heterocyclic Chalcones.
    Chemistry & biodiversity, 2022, Volume: 19, Issue:9

    Topics: Aldehydes; Anti-Infective Agents; Antineoplastic Agents; Candida albicans; Chalcone; Chalcones; Imidazoles; Indoles; Molecular Docking Simulation; Molecular Structure; Pyrazoles; Staphylococcus aureus; Structure-Activity Relationship; Thiophenes; Triazoles

2022