Page last updated: 2024-08-18

thiophenes and agn 194310

thiophenes has been researched along with agn 194310 in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (12.50)18.2507
2000's6 (75.00)29.6817
2010's1 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chandraratna, RA; Escobar, M; Johnson, AT; Standeven, AM; Wang, L1
Brown, G; Burnett, RD; Chandraratna, RA; Durham, J; Hammond, LA; Jones, EL; Tomkins, SE; Van Krinks, CH1
Chandraratna, RA; Torchia, J; Underhill, TM; Weston, AD1
Chandraratna, RA; McArthur, GA; Walkley, CR; Yuan, YD1
Alexander, G; Austenaa, LM; Blomhoff, HK; Blomhoff, R; Carlsen, H; Ertesvag, A1
Atangan, LI; Bird, R; Brown, G; Chandraratna, RA; Hammond, LA; Keedwell, RG; Qin, S; Reitmair, A; Shurland, DL; Wallace, DM; Wen, K; Zhao, Y1
Chandraratna, RA; Fibach, E; Prus, E1
Andersson, G; Hu, L; Jacobson, A; Lind, T; Melhus, H; Pejler, G; Sundqvist, A1

Other Studies

8 other study(ies) available for thiophenes and agn 194310

ArticleYear
Synthesis and biological activity of high-affinity retinoic acid receptor antagonists.
    Bioorganic & medicinal chemistry, 1999, Volume: 7, Issue:7

    Topics: Animals; Benzoates; Heterocyclic Compounds; Inhibitory Concentration 50; Naphthalenes; Receptors, Retinoic Acid; Recombinant Proteins; Retinoid X Receptors; Retinoids; Structure-Activity Relationship; Thiophenes; Transcription Factors; Transcription, Genetic

1999
Antagonists of retinoic acid receptors (RARs) are potent growth inhibitors of prostate carcinoma cells.
    British journal of cancer, 2001, Aug-03, Volume: 85, Issue:3

    Topics: Antineoplastic Agents; Apoptosis; Benzoates; Cell Cycle; Humans; Male; Prostatic Neoplasms; Receptors, Retinoic Acid; Retinoids; Thiophenes; Tretinoin; Tumor Cells, Cultured

2001
Requirement for RAR-mediated gene repression in skeletal progenitor differentiation.
    The Journal of cell biology, 2002, Jul-08, Volume: 158, Issue:1

    Topics: Activating Transcription Factor 2; Animals; Benzoates; Blotting, Northern; Blotting, Western; Bone and Bones; Cell Differentiation; Chondrocytes; COS Cells; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Genes, Dominant; Genes, Reporter; High Mobility Group Proteins; Histone Deacetylase Inhibitors; Hydroxamic Acids; Imidazoles; Luciferases; Mesoderm; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Phenotype; Plasmids; Pyridines; Receptors, Retinoic Acid; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; SOX9 Transcription Factor; Stem Cells; Thiophenes; Transcription Factors; Transcription, Genetic; Transcriptional Activation; Transfection

2002
Retinoic acid receptor antagonism in vivo expands the numbers of precursor cells during granulopoiesis.
    Leukemia, 2002, Volume: 16, Issue:9

    Topics: Animals; Benzoates; Bone Marrow Cells; Cell Death; Cell Line; Colony-Forming Units Assay; Female; Flow Cytometry; Granulocytes; Hematopoiesis; Mice; Mice, Inbred C57BL; Receptors, Retinoic Acid; Stem Cells; Thiophenes

2002
Vitamin A status significantly alters nuclear factor-kappaB activity assessed by in vivo imaging.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2004, Volume: 18, Issue:11

    Topics: Animals; Benzoates; Genes, Reporter; Immunoglobulin kappa-Chains; Luciferases; Lymphoid Tissue; Mice; Mice, Transgenic; NF-kappa B; Skin; T-Lymphocytes; Thiophenes; Transcriptional Activation; Tretinoin; Ultraviolet Rays; Vitamin A Deficiency

2004
An antagonist of retinoic acid receptors more effectively inhibits growth of human prostate cancer cells than normal prostate epithelium.
    British journal of cancer, 2004, Aug-02, Volume: 91, Issue:3

    Topics: Apoptosis; Benzoates; Carcinoma; Caspases; DNA Damage; Epithelial Cells; Humans; Male; Prostate; Prostatic Neoplasms; Receptors, Retinoic Acid; Thiophenes; Tumor Cells, Cultured

2004
Retinoic acid receptor antagonist inhibits CD38 antigen expression on human hematopoietic cells in vitro.
    Leukemia & lymphoma, 2004, Volume: 45, Issue:5

    Topics: ADP-ribosyl Cyclase; ADP-ribosyl Cyclase 1; Antigens, CD; Antigens, CD34; Benzoates; Cell Culture Techniques; Cell Differentiation; Cell Line; Cell Proliferation; Drug Interactions; Fetal Blood; Hematopoietic Stem Cells; Humans; Membrane Glycoproteins; Receptors, Retinoic Acid; Thiophenes

2004
Vitamin a is a negative regulator of osteoblast mineralization.
    PloS one, 2013, Volume: 8, Issue:12

    Topics: Animals; Benzoates; Benzothiazoles; Calcification, Physiologic; Cell Line; Core Binding Factor Alpha 1 Subunit; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Femur; Humans; Male; Osteoblasts; Rats; Rats, Sprague-Dawley; Receptors, Retinoic Acid; Retinoic Acid 4-Hydroxylase; Signal Transduction; Sp7 Transcription Factor; Thiophenes; Transcription Factors; Triazoles; Vitamin A; Vitamins

2013