Page last updated: 2024-08-18

thiophenes and 8-hydroxy-2-(di-n-propylamino)tetralin

thiophenes has been researched along with 8-hydroxy-2-(di-n-propylamino)tetralin in 23 studies

Research

Studies (23)

TimeframeStudies, this research(%)All Research%
pre-19902 (8.70)18.7374
1990's17 (73.91)18.2507
2000's3 (13.04)29.6817
2010's1 (4.35)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bervoets, K; Brocco, M; Canton, H; Gobert, A; Le Marouille-Girardon, S; Lefebvre de Ladonchamps, B; Lejeune, F; Millan, MJ; Rivet, JM; Verriele, L1
Bizot-Espiard, J; Costentin, J; Guardiola, B; Schiavi, P; Simon, P1
Laubie, M; Mennecier, P; Verbeuren, TJ1
Canton, H; Laubie, M; Lavielle, G; Lejeune, F; Millan, MJ; Rivet, JM1
De Vry, J; Glaser, T; Glennon, RA; Spencer, DG1
Barber, DJ; Cooper, SJ; Rusk, IN1
Hiner, BC; Peroutka, SJ; Roth, HL1
Adrien, J; Fattaccini, CM; Gozlan, H; Guardiola-Lemaitre, B; Haj-Dahmane, S; Hamon, M; Jolas, T; Kidd, EJ; Lanfumey, L1
Andrews, N; File, SE; Gonzalez, LE; Hogg, S1
Emerit, MB; Hamon, M; Riad, M1
Artigas, F; Celada, P; Romero, L1
Ishimoto, Y; Kamata, T; Katoh, S; Kawakubo, H; Mochizuki, D; Nagatani, T; Sasaki, Y; Takagi, S; Yamaura, Y1
Cagnotto, A; De Blasi, A; Esposito, E; Mennini, T; Prisco, S; Talone, D1
Bietti, G; Borsini, F; Ceci, A; Donetti, A1
File, SE; Gonzalez, LE1
Assie, MB; Koek, W1
Andrews, N; File, SE; Gonzalez, LE1
Dekeyne, A; Girardon, S; Millan, MJ1
Fornal, CA; Jacobs, BL; Martin, FJ; Metzler, CW1
Akunne, HC; Cooke, LW; Davis, MD; Georgic, LM; Heffner, TG; MacKenzie, RG; Meltzer, LT; Pugsley, TA; Shih, YH; Whetzel, SZ; Wise, LD; Wustrow, DJ; Zoski, KT1
Dijkstra, D; Rodenhuis, N; Timmerman, W; Wikström, HV1
Grandoso, L; Pineda, J; Torrecilla, M; Ugedo, L1
Banas, SM; Belmer, A; Diaz, SL; Doly, S; Fernandez, SP; Guiard, BP; Mameli, M; Maroteaux, L; Moutkine, I; Muzerelle, A; Pitychoutis, PM; Quentin, E; Roumier, A; Tchenio, A1

Other Studies

23 other study(ies) available for thiophenes and 8-hydroxy-2-(di-n-propylamino)tetralin

ArticleYear
S 14671: a naphtylpiperazine 5-hydroxytryptamine1A agonist of exceptional potency and high efficacy possessing antagonist activity at 5-hydroxytryptamine1C/2 receptors.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 262, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analgesia; Animals; Body Temperature; Corticosterone; In Vitro Techniques; Male; Mice; Phosphatidylinositols; Piperazines; Posture; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes; Thiophenes

1992
5-HT1A receptor agonists prevent in rats the yawning and penile erections induced by direct dopamine agonists.
    Psychopharmacology, 1992, Volume: 108, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Aminoquinolines; Animals; Body Temperature; Buspirone; Chromans; Dopamine Agents; Male; Mice; Penile Erection; Propanolamines; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Serotonin; Spiro Compounds; Thiophenes; Yawning

1992
5-Hydroxytryptamine-induced vasodilatation in the isolated perfused rat kidney: are endothelial 5-HT1A receptors involved?
    European journal of pharmacology, 1991, Aug-16, Volume: 201, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Angiotensin II; Animals; Atrial Natriuretic Factor; Endothelium, Vascular; Kidney; Male; Nitroglycerin; Papaverine; Piperazines; Propanolamines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes; Thiophenes; Vasodilation

1991
S 14671: a novel naphthylpiperazine 5-HT1A agonist of high efficacy and exceptional in vivo potency.
    European journal of pharmacology, 1991, Oct-15, Volume: 203, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Alprenolol; Animals; Behavior, Animal; Binding, Competitive; Dose-Response Relationship, Drug; Male; Piperazines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes; Thiophenes

1991
Stimulus properties of tiflucarbine: a novel antidepressant agent.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 37, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antidepressive Agents; Discrimination, Psychological; DOM 2,5-Dimethoxy-4-Methylamphetamine; Indoles; Male; Methoxydimethyltryptamines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes; Thiophenes

1990
Yawning induced by the selective dopamine D2 agonist N-0437 is blocked by the selective dopamine autoreceptor antagonist (+)-UH 232.
    Physiology & behavior, 1989, Volume: 45, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dopamine Agents; Dopamine Antagonists; Drug Interactions; Male; Naphthalenes; Raclopride; Rats; Salicylamides; Tetrahydronaphthalenes; Thiophenes; Time Factors; Yawning

1989
Antimigraine drug interactions with 5-hydroxytryptamine1A receptors.
    Annals of neurology, 1986, Volume: 19, Issue:5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain; Cyproheptadine; Dihydroalprenolol; Drug Interactions; Methysergide; Pizotyline; Propranolol; Rats; Receptors, Serotonin; Tetrahydronaphthalenes; Thiophenes

1986
(-)Tertatolol is a potent antagonist at pre- and postsynaptic serotonin 5-HT1A receptors in the rat brain.
    Naunyn-Schmiedeberg's archives of pharmacology, 1993, Volume: 347, Issue:5

    Topics: 5-Hydroxytryptophan; 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Brain; Electrophysiology; Hydroxyindoleacetic Acid; Isomerism; Male; Neurons; Propanolamines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Thiophenes

1993
5-HT1A receptors in the median raphe nucleus and dorsal hippocampus may mediate anxiolytic and anxiogenic behaviours respectively.
    European journal of pharmacology, 1994, Nov-03, Volume: 264, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Anxiety; Autoreceptors; Dendrites; Grooming; Hippocampus; Male; Motor Activity; Propanolamines; Raphe Nuclei; Rats; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Social Behavior; Thiophenes

1994
Neurotrophic effects of ipsapirone and other 5-HT1A receptor agonists on septal cholinergic neurons in culture.
    Brain research. Developmental brain research, 1994, Oct-14, Volume: 82, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Autoradiography; Brain; Cell Division; Cells, Cultured; Choline O-Acetyltransferase; Dose-Response Relationship, Drug; Female; Fetus; Immunohistochemistry; Nerve Growth Factors; Neurons; Piperazines; Pregnancy; Propanolamines; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiophenes; Tritium

1994
Reduction of in vivo striatal 5-hydroxytryptamine release by 8-OH-DPAT after inactivation of Gi/G(o) proteins in dorsal raphe nucleus.
    European journal of pharmacology, 1994, Nov-14, Volume: 265, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Autoreceptors; Citalopram; Corpus Striatum; GTP-Binding Proteins; Male; Pertussis Toxin; Potassium Channels; Propanolamines; Raphe Nuclei; Rats; Rats, Wistar; Serotonin; Thiophenes; Virulence Factors, Bordetella

1994
(R)-1,2,3,4-tetrahydro[1]benzothieno[2,3-c]pyridines: novel optically active compounds with strong 5-HT1A receptor binding ability exhibiting anticonflict activity and lessening of memory impairment.
    Journal of medicinal chemistry, 1993, Nov-12, Volume: 36, Issue:23

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amnesia; Animals; Anti-Anxiety Agents; Avoidance Learning; Conflict, Psychological; Male; Mice; Molecular Structure; Pyridines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Serotonin; Scopolamine; Stereoisomerism; Structure-Activity Relationship; Thienopyridines; Thiophenes

1993
Tertatolol, a new beta-blocker, is a serotonin (5-hydroxytryptamine1A) receptor antagonist in rat brain.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain; Electrophysiology; Male; Membranes; Neurons; Propanolamines; Radioligand Assay; Raphe Nuclei; Rats; Serotonin Antagonists; Thiophenes

1993
BIMT 17, a 5-HT1A receptor agonist/5-HT2A receptor antagonist, directly activates postsynaptic 5-HT inhibitory responses in the rat cerebral cortex.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Analysis of Variance; Animals; Antidepressive Agents; Benzimidazoles; Binding, Competitive; Buspirone; Cerebral Cortex; Dose-Response Relationship, Drug; In Vitro Techniques; Iontophoresis; Male; Microelectrodes; Neurons; Piperazines; Prazosin; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiophenes

1995
Anxiolytic effects in the plus-maze of 5-HT1A-receptor ligands in dorsal raphé and ventral hippocampus.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 54, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Anti-Anxiety Agents; Anxiety; Hippocampus; Ligands; Male; Propanolamines; Raphe Nuclei; Rats; Receptors, Serotonin; Serotonin Receptor Agonists; Stereotaxic Techniques; Thiophenes

1996
(-)-pindolol and (+/-)-tertatolol affect rat hippocampal 5-HT levels through mechanisms involving not only 5-HT1A, but also 5-HT1B receptors.
    Neuropharmacology, 1996, Volume: 35, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Betaxolol; Hippocampus; Male; Microdialysis; Pindolol; Propanolamines; Rats; Receptors, Serotonin; Serotonin; Thiophenes

1996
5-HT1A and benzodiazepine receptors in the basolateral amygdala modulate anxiety in the social interaction test, but not in the elevated plus-maze.
    Brain research, 1996, Sep-02, Volume: 732, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholinesterase; Adrenergic beta-Antagonists; Amygdala; Analysis of Variance; Animals; Anxiety; GABA Modulators; Infusions, Parenteral; Male; Maze Learning; Midazolam; Motor Activity; Neurons; Propanolamines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists; Social Behavior; Thiophenes

1996
Discriminative stimulus properties of the novel serotonin (5-HT)2C receptor agonist, RO 60-0175: a pharmacological analysis.
    Neuropharmacology, 1999, Volume: 38, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aminopyridines; Animals; Conditioning, Operant; Ethylamines; Fluorobenzenes; Indoles; Male; Mianserin; Piperazines; Piperidines; Pyrazines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Reinforcement, Psychology; Serotonin Antagonists; Serotonin Receptor Agonists; Thiophenes

1999
Pindolol suppresses serotonergic neuronal activity and does not block the inhibition of serotonergic neurons produced by 8-hydroxy-2-(di-n-propylamino)tetralin in awake cats.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 291, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Cats; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Neurons; Pindolol; Propanolamines; Raphe Nuclei; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Thiophenes

1999
PD 158771, a potential antipsychotic agent with D(2)/D(3) partial agonist and 5-HT(1A) agonist actions. I. Neurochemical effects.
    Neuropharmacology, 2000, Apr-27, Volume: 39, Issue:7

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Benzazepines; Biogenic Amines; Brain Chemistry; Cells, Cultured; CHO Cells; Cricetinae; Dopamine Agonists; Dopamine Antagonists; Electrophysiology; Humans; Male; Membranes; Neostriatum; Piperazines; Pyrimidines; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists; Spiperone; Tetrahydronaphthalenes; Thiophenes

2000
Thiophene analogs of naphthoxazines and 2-aminotetralins: bioisosteres with improved relative oral bioavailability, as compared to 5-OH-DPAT.
    European journal of pharmacology, 2000, Apr-14, Volume: 394, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Administration, Oral; Animals; Binding, Competitive; Biological Availability; Injections, Subcutaneous; Male; Microdialysis; Motor Activity; Naphthalenes; Neostriatum; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Serotonin; Reserpine; Sympatholytics; Tetrahydronaphthalenes; Thiophenes

2000
alpha(2)-Adrenoceptor involvement in the in vitro inhibitory effect of citalopram on a subpopulation of rat locus coeruleus neurons.
    European journal of pharmacology, 2005, Jul-04, Volume: 517, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Amphetamines; Animals; Bridged Bicyclo Compounds, Heterocyclic; Brimonidine Tartrate; Citalopram; Dose-Response Relationship, Drug; Duloxetine Hydrochloride; Idazoxan; In Vitro Techniques; Locus Coeruleus; Male; Methiothepin; Naloxone; Narcotic Antagonists; Neurons; Norepinephrine; Oxazines; Piperazines; Piperidines; Pyridines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Opioid, mu; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiophenes

2005
Positive regulation of raphe serotonin neurons by serotonin 2B receptors.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2018, Volume: 43, Issue:7

    Topics: 3,4-Methylenedioxyamphetamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Amphetamines; Animals; Body Temperature; Central Nervous System Sensitization; Female; Fluoxetine; Indoles; Male; Mice; Mice, Knockout; Mice, Transgenic; Neurogenesis; Prepulse Inhibition; Raphe Nuclei; Receptor, Serotonin, 5-HT2B; Serotonergic Neurons; Serotonin 5-HT2 Receptor Agonists; Thiophenes; Transcription Factors

2018