thiazoles has been researched along with urea in 173 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 22 (12.72) | 18.7374 |
| 1990's | 6 (3.47) | 18.2507 |
| 2000's | 48 (27.75) | 29.6817 |
| 2010's | 87 (50.29) | 24.3611 |
| 2020's | 10 (5.78) | 2.80 |
| Authors | Studies |
|---|---|
| Craig, JW; Reed, SE; Tyrrell, DA | 1 |
| Cheng, CC; Zee-Cheng, RK | 1 |
| Dienstbier, Z; Kozák, I; Kronrád, L | 1 |
| Castell, JV; Gómez-Lechón, MJ; Jover, R; Ponsoda, X | 1 |
| Dodgson, SJ; Forster, RE | 1 |
| Amacker, PA; Favet, J; Griffiths, W; Hunziker, N; Schorer, E | 1 |
| Kumar, A; Mishra, DN; Pandeya, SN; Singh, BN | 1 |
| Cantino, EC; Matsumae, A | 1 |
| Eisenbrand, G; Siebert, D | 1 |
| Heller, J; Tata, PS | 1 |
| Inoki, R; Otori, K; Yamamoto, I | 1 |
| Carone, FA; Krumlovsky, FA; Perlman, SG; Roberts, TH; Rowland, RG; Stolarczyk, J | 1 |
| Cooper, AJ; Meister, A | 1 |
| Suzuki, M; Taen, S | 1 |
| Bellare, RA; Deliwala, CV; Fernandez, BS; Kulkarni, BS; Patel, MR | 1 |
| Closier, MD; Islip, PJ | 1 |
| Capps, DB; Degnan, MB; Harger, GF; Werbel, LM | 1 |
| DeLong, DC; Kisner, K; Paget, CJ; Stone, RL | 1 |
| Moore, KE; Von Voigtlander, PF | 1 |
| Dekarz, B; Kozakiewicz, I; Lewicka, J; Polkowska-Krajewska, H; Rylski, L | 1 |
| Davies, P; Jackson, H | 1 |
| Pohloudek-Fabini, R; Schröpl, E | 1 |
| Cortese, I; Ermili, A | 1 |
| Andersen, KE; Frosch, PJ; Hannuksela, M; Lachapelle, JM; Lahti, A; Shaw, S; Wilkinson, JD | 1 |
| Biffi, M; Coppi, G; Mailland, F; Silingardi, S; Spotti, D | 1 |
| Brems, DN; Kaiser, RE; Roychoudhury, S; Yeh, WK | 1 |
| Cattel, L; Milla, P; Romeo, G; Russo, F; Salerno, L; Siracusa, M | 1 |
| Chang, JH; Cho, YB; Kim, CN; Lim, NG; Roh, J | 1 |
| Allen, SN; Bowling, JJ; Dayan, FE; Duke, MV; Duke, SO; Romagni, JG; Vincent, AC; Zjawiony, JK | 1 |
| Brange, J; Coats, A; Fink, AL; Frokjaer, S; Khurana, R; Nielsen, L; Uversky, VN; Vyas, S | 1 |
| Bucciantini, M; Capanni, C; Chiti, F; Dobson, CM; Stefani, M; Taddei, N | 1 |
| Andreassi, M; Anselmi, C; Centini, M; Di Stefano, A; Ettorre, A; Neri, P | 1 |
| Carpenter, JF; Kim, YS; Randolph, TW; Stevens, FJ | 1 |
| Bansal, A; De Lucca, I; King, RW; Priestley, ES; Scarnati, HT; Williams, JK | 1 |
| Barrish, JC; Das, J; DeFex, HF; Doweyko, AM; Fang, Q; Lin, J; Moquin, RV; Pang, S; Pitt, S; Schieven, GL; Shen, DR; Shen, Z; Spergel, SH; Wityak, J | 1 |
| Jones, S; Radford, SE; Serpell, LC; Smith, DP; Sunde, M | 1 |
| Avila, J; Berg, S; Bhat, R; Borgegård, T; Díaz-Nido, J; Giménez-Cassina, A; Hellberg, S; Hernández, F; Jerning, E; Lucas, JJ; Markgren, PO; Nilsson, Y; Nylöf, M; Ormö, M; Radesäter, AC; Xue, Y | 1 |
| Blystone, L; De Crescenzo, GA; Funkes-Shippy, CL; Getman, DP; Houseman, KA; Kishore, N; Kocan, GP; Lu, HF; McDonald, JJ; Mehta, PP; Nagarajan, SR; Sikorski, JA; Walker, JL | 1 |
| Atherton, J; Beebe, JS; Emerson, E; Finkelstein, M; Floyd, E; Foster, B; Gant, T; Goodwin, P; Harriman, S; Higdon, C; Hillerman, S; Jani, JP; Knauth, E; Kou, K; Marx, MA; Noe, MC; Rastinejad, F; Roberts, WG; Rossi, AM; Schaeffer, T; Soderstrom, C; Whalen, PM | 1 |
| Dusci, L; Guttner, Y; Marshall, BJ; Viiala, CH; Windsor, HM | 1 |
| Barsomian, G; Gourlie, BB; Hirth, BH; Kane, JL; Liang, B; Nahill, S | 1 |
| Brough, SJ; Herdon, HJ; Jerman, JC; Langmead, CJ; Porter, RA; Scott, C | 1 |
| Asuni, AA; Berg, S; Bhat, R; Drummond, JA; Jukes, JP; Lovestone, S; MacKay, D; Mears, A; Mildren, P; Mudher, A; Newman, TA; Shepherd, D; Squire, A | 1 |
| Bhat, R; Einat, H; Gould, TD; Manji, HK | 1 |
| Crandell, DE; Dyson, DH; Mathews, KA | 1 |
| Anborgh, PH; Okamura, S; Parmeggiani, A | 1 |
| Calloni, G; Chiti, F; Dobson, CM; Stefani, M; Zoffoli, S | 1 |
| Chimenti, R; Martino, G; Mazzulla, S; Sesti, S | 1 |
| Chao, BB; Peng, YP; Qiu, YH; Wang, JJ | 1 |
| He, Y; Luo, Y; Tang, H; Yi, Z; Zhou, H | 1 |
| Billadeau, DD; Fernandez-Zapico, ME; Ougolkov, AV; Savoy, DN; Urrutia, RA | 1 |
| Garcia, A; Houle, S; Meyer, JH; Stableford, WT; Vasdev, N; Wilson, AA; Young, AB | 1 |
| Laufer, S; Wagner, G | 1 |
| Caricasole, A; Gaviraghi, G; Terstappen, GC | 1 |
| Bilim, VN; Billadeau, DD; Chari, ST; Fernandez-Zapico, ME; Ougolkov, AV; Smyrk, TC | 1 |
| Cohen, RB; Cosgriff, TM; Eisenberg, PD; Hainsworth, JD; Healey, D; Langer, CJ; Liau, K; Madajewicz, S; Pierce, K; Simon, GR; Xu, H | 1 |
| Hwang, S; Kim, HY; Kim, SH; Kim, Y; Koh, SH; Lee, CH | 1 |
| Chen, R; Han, Y; Li, M; Li, W; Ruan, H; Wang, W; Wang, Y; Yang, Y; Ying, C; You, Y; Zhu, X | 1 |
| Abad, MA; Camins, A; Enguita, M; Folch, J; Pallàs, M; Trullàs, R; Yeste-Velasco, M | 1 |
| Iida, M; Kitagawa, H; Ozawa, T; Saito, J; Takahata, S; Yamada, M | 1 |
| Faghih, R; Gfesser, GA; Gopalakrishnan, M | 1 |
| Iida, M; Kitagawa, H; Ohsawa, F; Ozawa, T; Saito, J; Takahata, S; Takeuchi, Y; Watanabe, T; Yamada, M | 1 |
| Desfontis, JC; Fusellier, M; Gautier, F; Gogny, M; Le Roux, A; Madec, S; Thuleau, A | 1 |
| Chang, DI; Hwang, SJ; Kim, SH; Koh, SH; Yoo, AR | 1 |
| Binfaré, RW; García, AG; Kaster, MP; López, MG; Martín-Aparicio, E; Martinez, A; Medina, M; Morales, S; Navarro-Rico, ML; Rodrigues, AL; Rosa, AO | 1 |
| Allameh, A; Amirizadeh, N; Esmaeili, S; Gharehbaghian, A; Kazemnejad, S; Mohammadi, Y; Seoleimani, M | 1 |
| Baldwin, AS; Wilson, W | 1 |
| Bauchwitz, RP; Chen, S; Jope, RS; Min, WW; Sikorski, C; Yan, Q; Yuskaitis, CJ | 1 |
| Fujisawa, H; Hamada, J; Hayashi, Y; Kawakami, K; Mai, W; Minamoto, T; Miyashita, K; Nakada, M; Shakoori, A | 1 |
| Cavalli, A; Gervasio, FL; Masetti, M; Recanatini, M | 1 |
| de Lima, AF; de Souza Costa, CA; Gasparoto Mancini, MN; Hebling, J; Lessa, FC; Marchi, GM | 1 |
| Chen, YX; Filion, L; Hibbert, B; Holm, E; Ma, X; O'Brien, ER; Pourdjabbar, A; Rayner, K; Sun, J | 1 |
| Bhattacharya, R; Karmakar, R; Kulshrestha, G | 1 |
| Achim, CL; Chana, G; Everall, IP; Grant, I; Hult, BJ; Lucero, GR; Masliah, E; Nguyen, TB; Tatro, ET | 1 |
| Delgado-Martín, C; Escribano, C; Rodríguez-Fernández, JL | 1 |
| Aponte, AM; Murphy, E; Steenbergen, C; Wong, R | 1 |
| Bilim, V; Billadeau, D; Kawazoe, H; Motoyama, T; Muto, A; Naito, S; Ougolkov, A; Oya, M; Tomita, Y; Yuuki, K | 1 |
| Klein, RQ; Lok, W; Saif, MW | 1 |
| Dykstra, H; Fan, S; Mercer, AJ; Papugani, A; Persidsky, Y; Ramirez, SH; Reichenbach, N; Tuma, RF; Zhang, M | 1 |
| Costa, CA; Hebling, J; Lessa, FC; Lima, AF; Mancini, MN; Marchi, GM | 1 |
| Blood, JD; Pekary, AE; Sattin, A; Stevens, SA | 1 |
| Blumenthal, R; Drevets, W; Du, J; Hunsberger, JG; Khairova, R; Liu, L; Machado-Vieira, R; Manji, HK; Tragon, T; Wang, Y; Wang, YT; Wei, Y | 1 |
| Egea, J; Gadotti, VM; López, MG; Martins, DF; Mazzardo-Martins, L; Nascimento, FP; Rosa, AO; Santos, AR | 1 |
| Chang, WT; Chen, CL; Huang, WC; Kai, JI; Lin, CF; Tsai, CC | 1 |
| Christen, P; De los Rios, P; Goloubinoff, P; Lustig, A; Sharma, SK | 1 |
| Milligan, G; Pediani, JD; Ward, RJ | 1 |
| Dawson, LA; Kalinichev, M | 1 |
| Bécsi, B; Csortos, C; Czikora, I; Erdodi, F; Gergely, P; Kása, A; Kim, KM; Verin, AD | 1 |
| Krett, NL; Rosen, ST; Rovedo, MA | 1 |
| Ban, JO; Han, SB; Hong, JT; Kang, KW; Moon, DC; Oh, JH; Son, SM; Song, HS; Song, MJ; Won, D | 1 |
| Boländer, A; Dominguez, J; Eldar-Finkelman, H; Fuertes, A; Kramer, T; Monte, FL; Plotkin, B; Schmidt, B | 1 |
| Boey, L; Claes, L; Drieghe, J; Goossens, A; Travassos, AR | 1 |
| Ishigaki, Y; Kawakami, K; Kitano, A; Minamoto, T; Motoo, Y; Nakajima, H; Nakamura, Y; Nakaya, N; Sato, I; Shimasaki, T; Takata, T; Takegami, T; Tanaka, T; Tomosugi, N; Zhao, X | 1 |
| Aust, B; Getlik, M; Grütter, C; Nguyen, HD; Rauh, D; Robubi, A; Simard, JR; van Otterlo, WA | 1 |
| Hicks, JW; Houle, S; Rubie, EA; Vasdev, N; Wilson, AA; Woodgett, JR | 1 |
| Hu, Q; Lee, SY; O'Kusky, JR; Ye, P | 1 |
| Aarts, M; Ashworth, A; Garcia-Murillas, I; Gevensleben, H; Hurd, MS; Sharpe, R; Shumway, SD; Toniatti, C; Turner, NC | 1 |
| Fedoročko, P; Jendželovský, R; Koval, J; Mikeš, J; Papčová, Z; Plšíková, J | 1 |
| Ahn, SW; Choi, WJ; Hong, YH; Kim, JE; Kim, SH; Kim, SM; Lee, KW; Park, KS; Sung, JJ | 1 |
| Adelekun, AE; Hannaway, KE; Horiguchi, M; Jayathilake, K; Meltzer, HY | 1 |
| Azam, F; Mohan, G; Prasad, MV; Shrivastava, AK; Thangavel, N | 1 |
| Abraham, CJ; Aravantinou, M; Blanchard, J; Calenda, G; Derby, N; Fernández-Romero, JA; Gettie, A; Goldman, D; Kenney, J; Lifson, JD; Mawson, P; Menon, R; Piatak, M; Robbiani, M; Seidor, S; Singer, R; Teleshova, N; Villegas, G; Zydowsky, TM | 1 |
| Forinash, KD; Lawrence, NJ; Martin, MP; Patel, RA; Pireddu, R; Schönbrunn, E; Sebti, SM; Sun, N; Sun, Y | 1 |
| Cidral-Filho, FJ; Martins, DF; Mazzardo-Martins, L; Santos, AR; Stramosk, J | 1 |
| Andersen, KE; Brandão, FM; Bruynzeel, DP; Bruze, M; Diepgen, TL; Frosch, PJ; Giménez-Arnau, A; Gonçalo, M; Goossens, A; Johansen, JD; Lahti, A; Menné, T; Mowitz, M; Rustemeyer, T; Seidenari, S; Svedman, C; Tosti, A; Wahlberg, JE; White, IR; Wilkinson, JD | 1 |
| Dionyssiou, MG; Hashemi, S; Kerr, A; McDermott, JC; Nowacki, NB; Tsushima, RG; Zhao, J | 1 |
| Behnke, CA; Igaki, S; Kawamura, T; Kiyota, Y; Kono, M; Kori, M; Matsumoto, T; Miyazaki, J; Nishimura, A; Oki, H; Shimojo, M | 1 |
| Anderson, NJ; Guernsey, LS; Jolivalt, CG; King, MR | 1 |
| Roux, PP; Shin, S; Tcherkezian, J; Vallabhapurapu, S; Wolgamott, L; Yoon, SO; Yu, Y | 1 |
| Gowda, DC; Sharma, A; Suhas, R | 1 |
| Banu, SH; Chandana, KV; Channe Gowda, D; Sharma, A; Suhas, R | 1 |
| Chiappinelli, KB; Goodfellow, PJ; Kizer, NT; Ma, L; Thaker, PH; Trinkaus, KM; Yin, Y | 1 |
| Gowda, R; Madhunapantula, SV; Robertson, GP; Sharma, A | 1 |
| Dong, Y; Tu, X; Yu, J; Zhang, X | 1 |
| Carlson, TJ; Davis, J; Deprez, P; Fotsch, CH; Grillo, MP; Harrington, PE; Henley, C; Lively, SE; Lu, JY; Morony, S; Pattabiraman, K; Poon, SF; Reagan, JD; St Jean, DJ; Temal, T; Wang, M; Wehn, PM; Yang, Y | 1 |
| Gao, M; Maixner, DW; Weng, HR | 1 |
| Ahuja, V; Basavarajappa, H; Boriack-Sjodin, PA; de Sousa, SM; Ganguly, S; Gaonkar, S; Ghorpade, SR; Hameed, SP; Humnabadkar, V; Jena, LK; Kale, MG; Kale, RR; Kishore Reddy, BK; Koushik, K; Madhavapeddi, P; Mahesh Kumar, KN; Malolanarasimhan, K; Manjunatha, MR; Menasinakai, S; Nandishaiah, R; Naveen Kumar, CN; Ogg, D; Raichurkar, A; Sambandamurthy, VK; Sharma, S; Shinde, V; Waterson, D | 1 |
| Azim, K; Butt, A; Cantù, C; Draganova, K; Fischer, B; Hurtado-Chong, A; Raineteau, O; Sommer, L; Zemke, M | 1 |
| Adam, S; Krishna Reddy, RC; Raju, CN; Rasheed, S; Subba Rao, D; Venkata Rami Reddy, Y | 1 |
| Bostwick, JS; Chacko, SA; Chen, BC; Chen, XQ; Clark, CG; Hiebert, S; Hua, J; Huang, CS; Jeon, YT; Lam, PY; Levesque, PC; Li, D; Li, L; Liu, Y; Malley, M; Mathur, A; Price, LA; Qiao, JX; Rehfuss, R; Ruel, R; Schumacher, WA; Seiffert, DA; Shen, H; Stewart, AB; Sun, D; Thibeault, C; Wang, TC; Wang, Y; Wexler, RR; Wong, HS; Wu, DR; Yang, W; Zhu, J | 1 |
| Carter, YM; Chen, H; Gamblin, TC; Kunnimalaiyaan, M; Kunnimalaiyaan, S | 1 |
| Dent, P | 1 |
| Cho, YJ; Liu, J; MacDonald, TJ; Petersen, W; Schneiderjan, M; Yuan, L; Zhang, H | 1 |
| Banu, SH; Chandrashekar, S; Gowda, DC; Sharma, A; Suhas, R | 1 |
| Basak, S; Chattopadhyay, K; Prasad, GV; Varkey, J | 1 |
| Gazioglu, I; Kucukislamoglu, M; Kurt, BZ; Sonmez, F | 1 |
| Chang, MS; Cho, SJ; Choi, Y; Choi, YS; Kim, MA; Ko, YS; Lee, BL; Lee, JS; Park, J; Pyo, JS; Ye, SK; Yoon, J; Youn, HD | 1 |
| Cárcamo, HA; Herle, CE; Lupwayi, NZ | 1 |
| Ishioka, C; Suzuki, M; Takahashi, H; Yoshino, Y | 1 |
| Gui, Y; Li, L; Shi, Z; Singh, P; Walsh, MP; Yin, H; Yu, YN; Zheng, XL; Zhou, YX | 1 |
| Gamblin, TC; Kunnimalaiyaan, M; Kunnimalaiyaan, S | 1 |
| Arz, D; Caravatti, G; Fairhurst, RA; Fritsch, C; Furet, P; Gerspacher, M; Guthy, DA; Haasen, D; Imbach-Weese, P; Trappe, J; Wirth, J; Zoller, T | 1 |
| Basile, L; Gazioglu, I; Ginex, T; Guccione, S; Kucukislamoglu, M; Kurt, BZ; Sonmez, F | 1 |
| Ishioka, C; Yoshino, Y | 1 |
| Everett, M; Hardke, J; Lorenz, G; Slaton, N | 1 |
| Giordano, A; Morales, F | 1 |
| Bali, A; Jaggi, AS | 2 |
| Hirohama, M; Ito, A; Kumar, A; Yoshida, M; Zhang, KY | 1 |
| Andoh, T; Kuraishi, Y; Mizoguchi, S; Yakura, T | 1 |
| Brun, R; Patrick, DA; Tidwell, RR; Wang, MZ; Weiser, PT; Wenzler, T; Yang, S | 1 |
| Al-Onaizi, M; Barbash, S; Bekenstein, U; Fahnestock, M; Haberman, N; Hanin, G; Kish, MT; Kolisnyk, B; Prado, MAM; Prado, VF; Soreq, H; Soreq, L; Souza da Silva, J; Ule, J | 1 |
| Aichholz, R; Blanz, J; Blasco, F; Caravatti, G; Fairhurst, RA; Fritsch, C; Guagnano, V; Maira, SM; Schnell, C; Seiler, FH; Wipfli, P | 1 |
| Carvalho, AF; Dal-Pont, GC; de Souza, CT; Farias, HR; Jornada, LK; Machado, AG; Peterle, BR; Quevedo, J; Resende, WR; Valvassori, SS | 1 |
| Feng, Y; Hu, B; Rong, N; Yang, R; Zhang, J; Zhang, Q; Zhang, W | 1 |
| Agrawal, S; Kumari, N; Luthra, PM | 1 |
| Huang, CF; Liu, HS; Ramesh, C; Su, CL; Tseng, CL; Yao, CF | 1 |
| Ensom, MHH; Johnson, EG; Johnson, HE; Wilby, KJ | 1 |
| Kiran Kumar, E; Prakash Prabhu, N; Prasad, DK | 1 |
| Ail, D; Chesneau, A; Colozza, G; Hidalgo, M; Langhe, R; Locker, M; Perron, M | 1 |
| Abdel-Hakeem, MS; Houghton, M; Mason, AL; Sarhan, MA; Tyrrell, DL | 1 |
| Liu, Y; Zhang, M; Zhang, P; Zhou, Y | 1 |
| Aristizabal Prada, ET; Auernhammer, CJ; Grabowski, P; Grossman, A; Lauseker, M; Maurer, J; Nölting, S; Orth, M; Spöttl, G; Weis, C | 1 |
| Barančoková, M; Ilaš, J; Kikelj, D; Tammela, P; Tomašič, T; Zidar, N | 1 |
| Deng, H; Deng, Z; Liu, L; Liu, X; Liu, Y; Pang, W; Song, D; Zeng, Q; Zhang, N | 1 |
| Agrawal, S; Kumari, N; Kumari, R; Luthra, PM; Sharma, D | 1 |
| Ahmed, E; Ballabh, P; Cheng, B; Dohare, P; Kayton, R; Singla, P; Thomas, S; Ungvari, Z; Yadala, V | 1 |
| Dal-Pont, GC; Menegas, S; Peterle, BR; Quevedo, J; Resende, WR; Trajano, KS; Valvassori, SS; Varela, RB | 1 |
| Chung, YH; Hsu, PH; Lin, KJ; Lin, YT; Liu, HL; Yang, LY; Yen, TC | 1 |
| Ballabh, P; Dohare, P; Hevner, R; Kaur, J; Kidwai, A; Klebe, D; Krishna, S; Singla, P; Zhang, X | 1 |
| Dang, Y; Loewen, NA; Loewen, RT; Shah, P; Wang, C; Waxman, S | 1 |
| Deng, YH; Liu, JP; Liu, Y; Sun, LP; Xue, WJ; Yan, ZH | 1 |
| Chai, HH; Chen, GZ; Chen, WX; Chen, YS; Fu, XC; Guo, YW; Li, SP; Ma, L; Song, MY; Sun, HT; Tan, MX | 1 |
| Chang, H; Chen, H; Chen, Q; Huang, Y; Li, L; Li, P; Lu, M; Yu, Y | 1 |
| Abe, K; Aiba, H; Aoki, Y; Araki, Y; Bolidong, D; Domoto, T; Hayashi, K; Higuchi, T; Igarashi, K; Inatani, H; Minamoto, T; Miwa, S; Takeuchi, A; Taniguchi, Y; Tsuchiya, H; Yamamoto, N; Yonezawa, H | 1 |
| Jiang, W; Wang, J | 1 |
| Cogdill, AG; Guevara, B | 1 |
| Blackmore, TR; Jacobson, J; Jarman, KE; Lewin, SR; Nguyen, W; Purcell, DF; Sabroux, HJ; Sleebs, BE | 1 |
| Chang, LS; Chiou, JT; Huang, CH; Lee, YC; Shi, YJ; Wang, LJ | 1 |
| Besen, MH; Dalsenter, YO; Kaufmann, FN; Moretti, M; Neis, VB; Platt, N; Rodrigues, ALS; Rosa, PB; Rosado, AF; Werle, I | 1 |
| Aasen, T; Abdul Moin, NI; Abdul Wafi, S; Aboukameel, A; Abu-Bakar, N; Acharya, A; Ackermans, L; Adaramoye, O; Adarsh, KV; Adeosun, WA; Ahmad, NH; Ahmadi, F; Akanni, O; Akbar, M; Akbulak, RO; Akev, N; Akkaya, Ö; Al-Rashed, S; AlAbbad, S; Alabi, O; Alappat, BJ; Alcalá, S; Alcoutlabi, M; Aleppo, G; Alexander Ross, JB; Alexander, JH; Alexander, R; Alias, A; Alimba, C; Alken, FA; Allan, R; Alpers, M; Alsbou, EM; Amarasiri, SS; An, T; Anastasiadis, F; Anastassiadou, M; Anderson, KC; Andronikos, P; Anheyer, D; Annapurna, K; Anorlu, RI; Anten, MM; Anthopoulos, TD; Araujo-Castillo, RV; Aravamudhan, S; Arawwawala, LDAM; Arulsamy, N; Arunamata, A; Asghar, A; Asiri, AM; Aslanidou, T; Astrakhantseva, IV; Astutik, E; Attanayake, AP; Atwater, BD; Audureau, E; Augusto, S; Bakare, A; Banach, M; Bandelier, P; Banerjee, S; Barral, M; Bascuñán, J; Bates, FS; Bauer, NJC; Bayrak, BB; Beck, RW; Beckervordersantforth, J; Beeri, R; Begum, R; Beldi-Ferchiou, A; Bellingham, G; Ben-Tal, N; Bendib, I; Bergenstal, RM; Berger, MF; Bernasconi, G; Berry, S; Beuvon, F; Bi, WJ; Bi, Z; Bianconi, V; Bibi, I; Blank, BR; Bliemeister, E; Bobkowski, W; Bode, AM; Booth, CM; Bose, U; Boyd, K; Brancato, A; Brenmoehl, J; Brogi, E; Bronzo, P; Brooks, T; Brown, D; Brown, DN; Bruce, D; Buan, MEM; Bueno-Hernández, F; Bugielski, B; Bulavaitė, A; Buscagan, TM; Buxton, R; Caffaro, MM; Cai, Q; Cai, X; Cai, Y; Calhoun, P; Callander, N; Cambier, S; Camparo, P; Canales-Vargas, EJ; Canham, K; Cantu, J; Cao, J; Cao, JW; Cao, P; Cao, T; Cao, X; Caravella, BA; Carcadea, E; Carè, J; Carmichael, P; Carrasco Cabrera, L; Carteaux, G; Carvalho, PDS; Casarez, E; Cazorla, M; Celestrin, CP; Chakraborty, NK; Chan, B; Chandarlapaty, S; Chandgude, AL; Chang, CC; Chang, JH; Chang, X; Chang, Y; Chankhanittha, T; Chantanis, S; Chapovetsky, A; Chavan, S; Chen, B; Chen, D; Chen, F; Chen, G; Chen, H; Chen, J; Chen, K; Chen, KJ; Chen, KP; Chen, L; Chen, MA; Chen, Q; Chen, S; Chen, W; Chen, WF; Chen, X; Chen, Y; Cheng, D; Cheng, J; Cheng, Q; Cheon, GJ; 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Yang, S; Yang, T; Yang, X; Yang, Y; Yao, H; Yao, Y; Yari, D; Yassin, MT; Ye, C; Ye, J; Ye, Q; Yildiz, EA; Ying, S; Yoon, H; Yu, D; Yu, K; Yu, N; Yu, PL; Yuan, C; Yuan, D; Yuan, LJ; Yuan, Z; Yuen, N; Zagatto, AM; Zakaria, Y; Zalewski, AM; Zamora, S; Zavorotinskaya, T; Zeid, JL; Zeinoun, T; Zeng, C; Zerby, HN; Zhan, X; Zhang, A; Zhang, D; Zhang, E; Zhang, F; Zhang, H; Zhang, J; Zhang, L; Zhang, M; Zhang, P; Zhang, Q; Zhang, QY; Zhang, RG; Zhang, S; Zhang, T; Zhang, X; Zhang, Y; Zhang, YY; Zhao, CK; Zhao, H; Zhao, J; Zhao, K; Zhao, Q; Zhao, S; Zhao, T; Zhao, XQ; Zhao, Y; Zhao, Z; Zheng, J; Zheng, L; Zheng, Y; Zhou, B; Zhou, G; Zhou, L; Zhou, T; Zhou, X; Zhu, C; Zhu, J; Zhu, Y; Zhu, ZQ; Zhuang, T; Zimmermannova, O; Zin, NNINM; Zisimos, K; Zoghebi, KA; Zonder, JA; Zou, C; Zwirner, J | 1 |
| Abadi, AH; Abdel-Halim, M; AlNajjar, YT; Becker, W; ElHady, AK; Engel, M; Gabr, M; Salah, M; Wilms, G | 1 |
| Gao, L; Li, X; Ning, L; Wang, T; Zhang, F | 1 |
8 review(s) available for thiazoles and urea
| Article | Year |
|---|---|
[Pharmacotherapy of epilepsy].
Topics: Amino Acids; Anticonvulsants; Butyrophenones; Chemical Phenomena; Chemistry; Chlordiazepoxide; Epilepsy; Humans; Oxyphenbutazone; Succinates; Sulfonamides; Thiazoles; Urea | 1968 |
Small molecular anti-cytokine agents.
Topics: ADAM Proteins; ADAM17 Protein; Animals; Caspase Inhibitors; Cytochrome P-450 Enzyme Inhibitors; Cytokines; Humans; Hydroxamic Acids; Imidazoles; Matrix Metalloproteinase Inhibitors; Oligopeptides; p38 Mitogen-Activated Protein Kinases; Protein Kinase Inhibitors; Pyridazines; Pyridines; Pyrimidines; Quinazolines; Structure-Activity Relationship; Succinates; Thiazoles; Tumor Necrosis Factor-alpha; Urea | 2006 |
Advances in the discovery of novel positive allosteric modulators of the alpha7 nicotinic acetylcholine receptor.
Topics: Allosteric Regulation; alpha7 Nicotinic Acetylcholine Receptor; Animals; Bridged Bicyclo Compounds, Heterocyclic; Cognition Disorders; Drug Design; Humans; Nicotinic Agonists; Quinolines; Receptors, Nicotinic; Thiazoles; Urea | 2007 |
Aurora kinase inhibitors as anti-cancer therapy.
Topics: Antineoplastic Agents; Aurora Kinase B; Aurora Kinase C; Aurora Kinases; Benzamides; Benzimidazoles; Cyclohexanecarboxylic Acids; Drug Screening Assays, Antitumor; Enzyme Activation; Humans; Neoplasms; Organophosphates; Phenylurea Compounds; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Pyrazoles; Quinazolines; Thiazoles; Urea | 2010 |
Overview of CDK9 as a target in cancer research.
Topics: Bridged Bicyclo Compounds, Heterocyclic; Cell Cycle; Cyclic N-Oxides; Cyclin-Dependent Kinase 9; Flavonoids; Humans; Indolizines; Molecular Targeted Therapy; Neoplasms; Oxazoles; Piperidines; Protein Kinase Inhibitors; Purines; Pyrazoles; Pyridinium Compounds; Roscovitine; Thiazoles; Urea | 2016 |
Evidence-Based Review of Pharmacotherapy Used for Parkinson's Disease Psychosis.
Topics: Antipsychotic Agents; Benzodiazepines; Clozapine; Evidence-Based Medicine; Humans; Olanzapine; Parkinson Disease; Piperazines; Piperidines; Practice Guidelines as Topic; Psychotic Disorders; Quetiapine Fumarate; Randomized Controlled Trials as Topic; Risperidone; Thiazoles; Urea | 2017 |
Helicobacter pylori: A Review of Current Diagnostic and Management Strategies.
Topics: Amoxicillin; Anti-Bacterial Agents; Anti-Ulcer Agents; Antigens, Bacterial; Biopsy; Bismuth; Breath Tests; Clarithromycin; Culture Techniques; Doxycycline; Drug Resistance, Bacterial; Drug Therapy, Combination; Dyspepsia; Feces; Gastroscopy; Helicobacter Infections; Helicobacter pylori; Humans; Levofloxacin; Lymphoma, B-Cell, Marginal Zone; Metronidazole; Nitro Compounds; Organometallic Compounds; Peptic Ulcer; Polymerase Chain Reaction; Proton Pump Inhibitors; Rifabutin; Salicylates; Salvage Therapy; Serologic Tests; Stomach Neoplasms; Tetracycline; Thiazoles; Treatment Outcome; Urea | 2020 |
Psychological distress among health care professionals of the three COVID-19 most affected Regions in Cameroon: Prevalence and associated factors.
Topics: 3' Untranslated Regions; 5'-Nucleotidase; A549 Cells; Accidental Falls; Acetylcholinesterase; Acrylic Resins; Actinobacillus; Acute Disease; Acute Kidney Injury; Adaptor Proteins, Signal Transducing; Adenosine; Adenosine Triphosphate; Administration, Inhalation; Administration, Oral; Adolescent; Adult; Advance Care Planning; Africa, Northern; Age Factors; Aged; Aged, 80 and over; Air Pollutants; Air Pollution; Air Pollution, Indoor; Albendazole; Aluminum Oxide; Anastomosis, Surgical; Ancylostoma; Ancylostomiasis; Androstadienes; Angiogenesis Inhibitors; Angiotensin II; Animals; Anti-Bacterial Agents; Anti-Infective Agents; Antibodies, Bispecific; Antibodies, Viral; Anticoagulants; Antihypertensive Agents; Antinematodal Agents; Antineoplastic Agents; Antineoplastic Agents, Immunological; Antineoplastic Combined Chemotherapy Protocols; Antioxidants; Antiporters; Antiviral Agents; Apoptosis; Aptamers, Nucleotide; Aromatase Inhibitors; Asian People; Astrocytes; Atrial Fibrillation; Auditory Threshold; Aurora Kinase B; Australia; Autophagy; Autophagy-Related Protein 5; Autotrophic Processes; Bacillus cereus; Bacillus thuringiensis; Bacterial Proteins; Beclin-1; Belgium; Benzene; Benzene Derivatives; Benzhydryl Compounds; beta Catenin; beta-Arrestin 2; Biliary Tract Diseases; Biofilms; Biofuels; Biomarkers; Biomarkers, Tumor; Biomass; Biomechanical Phenomena; Bioreactors; Biosensing Techniques; Biosynthetic Pathways; Bismuth; Blood Platelets; Bone and Bones; Bone Regeneration; Bortezomib; Botulinum Toxins, Type A; Brain; Brain Injuries; Brain Ischemia; Brain Neoplasms; Breast Neoplasms; Breath Tests; Bronchodilator Agents; Calcium Phosphates; Cannabis; Carbon Dioxide; Carbon Isotopes; Carcinogenesis; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Cardiac Resynchronization Therapy; Cardiac Resynchronization Therapy Devices; Cardiomyopathies; Cardiovascular Diseases; Cariostatic Agents; Case Managers; Case-Control Studies; Catalysis; Cation Transport Proteins; CD8-Positive T-Lymphocytes; Cecropia Plant; Cell Adhesion; Cell Count; Cell Differentiation; Cell Division; Cell Line; Cell Line, Tumor; Cell Membrane; Cell Movement; Cell Proliferation; Cell Self Renewal; Cell Survival; Cells, Cultured; Cellular Reprogramming; Cellulose; Charcoal; Chemical and Drug Induced Liver Injury; Chemical Phenomena; Chemokines; Chemoradiotherapy; Chemoreceptor Cells; Child; Child Abuse; Child, Preschool; China; Chlorogenic Acid; Chloroquine; Chromatography, Gas; Chronic Disease; Clinical Competence; Coated Materials, Biocompatible; Cochlea; Cohort Studies; Color; Comorbidity; Computer Simulation; Computer-Aided Design; Contraception; Contraceptive Agents, Female; Contrast Media; COP-Coated Vesicles; Coronavirus Infections; Cost of Illness; Coturnix; COVID-19; Creatinine; Cross-Over Studies; Cross-Sectional Studies; Culex; Curriculum; Cyclic N-Oxides; Cytokines; Cytoplasm; Cytotoxicity, Immunologic; Cytotoxins; Databases, Factual; Deep Learning; Delivery, Obstetric; Denitrification; Dental Caries; Denture, Complete; Dexamethasone; Diabetes Complications; Diabetes Mellitus; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 2; Dielectric Spectroscopy; Diet, High-Fat; Dietary Fiber; Disease Models, Animal; Disease Progression; DNA; DNA Copy Number Variations; DNA, Mitochondrial; Dog Diseases; Dogs; Dopaminergic Neurons; Double-Blind Method; Down-Regulation; Doxorubicin; Drug Carriers; Drug Design; Drug Interactions; Drug Resistance, Bacterial; Drug Resistance, Neoplasm; Drug-Related Side Effects and Adverse Reactions; Drugs, Chinese Herbal; Dry Powder Inhalers; Dust; E2F1 Transcription Factor; Ecosystem; Education, Nursing; Education, Nursing, Baccalaureate; Electric Impedance; Electricity; Electrocardiography; Electrochemical Techniques; Electrochemistry; Electrodes; Electrophoresis, Polyacrylamide Gel; Endoplasmic Reticulum; Endothelial Cells; Environmental Monitoring; Enzyme Inhibitors; Epithelial Cells; Epithelial-Mesenchymal Transition; Esophageal Neoplasms; Esophageal Squamous Cell Carcinoma; Estrogen Receptor Modulators; Europe; Evoked Potentials, Auditory, Brain Stem; Exosomes; Feasibility Studies; Female; Ferricyanides; Ferrocyanides; Fibrinogen; Finite Element Analysis; Fistula; Fluorescent Dyes; Fluorides, Topical; Fluorodeoxyglucose F18; Fluticasone; Follow-Up Studies; Food Contamination; Food Microbiology; Foods, Specialized; Forensic Medicine; Frail Elderly; France; Free Radicals; Fresh Water; Fungi; Fungicides, Industrial; Galactosamine; Gastrointestinal Neoplasms; Gene Expression Profiling; Gene Expression Regulation, Neoplastic; Gene Frequency; Genetic Predisposition to Disease; Genotype; Gingival Hemorrhage; Glioblastoma; Glioma; Glomerular Filtration Rate; Glomerulosclerosis, Focal Segmental; Glucose; Glucose Transport Proteins, Facilitative; Glucosides; Glutamine; Glycolysis; Gold; GPI-Linked Proteins; Gram-Negative Bacteria; Gram-Positive Bacteria; Graphite; Haplotypes; HCT116 Cells; Healthy Volunteers; Hearing Loss; Heart Failure; Hedgehog Proteins; HEK293 Cells; HeLa Cells; Hemodynamics; Hemorrhage; Hepatocytes; Hippo Signaling Pathway; Histone Deacetylases; Homeostasis; Hospital Mortality; Hospitalization; Humans; Hydantoins; Hydrazines; Hydrogen Peroxide; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Hydroxylamines; Hypoglycemic Agents; Immunity, Innate; Immunoglobulin G; Immunohistochemistry; Immunologic Factors; Immunomodulation; Immunophenotyping; Immunotherapy; Incidence; Indazoles; Indonesia; Infant; Infant, Newborn; Infarction, Middle Cerebral Artery; Inflammation; Injections, Intramuscular; Insecticides; Insulin-Like Growth Factor I; Insurance, Health; Intention to Treat Analysis; Interleukin-1 Receptor-Associated Kinases; Interleukin-6; Intrauterine Devices; Intrauterine Devices, Copper; Iron; Ischemia; Jordan; Keratinocytes; Kidney; Kidney Diseases; Kir5.1 Channel; Klebsiella Infections; Klebsiella pneumoniae; Lab-On-A-Chip Devices; Laparoscopy; Lasers; Lasers, Semiconductor; Lenalidomide; Leptin; Lethal Dose 50; Levonorgestrel; Limit of Detection; Lipid Metabolism; Lipid Metabolism Disorders; Lipogenesis; Lipopolysaccharides; Liquid Biopsy; Liver; Liver Abscess, Pyogenic; Liver Cirrhosis; Liver Diseases; Liver Neoplasms; Longevity; Lung Neoplasms; Luteolin; Lymph Nodes; Lymphocyte Activation; Macaca fascicularis; Macrophages; Mad2 Proteins; Magnetic Resonance Imaging; Male; Mammary Glands, Human; Manganese; Manganese Compounds; MAP Kinase Signaling System; Materials Testing; Maternal Health Services; MCF-7 Cells; Medicaid; Medicine, Chinese Traditional; Melanoma; Membrane Proteins; Mental Health; Mercury; Metal Nanoparticles; Metals, Heavy; Metformin; Methionine Adenosyltransferase; Mice; Mice, Inbred BALB C; Mice, Inbred C3H; Mice, Inbred C57BL; Mice, Inbred CBA; Mice, Knockout; Mice, Nude; Microalgae; Microbial Sensitivity Tests; Microglia; MicroRNAs; Microscopy, Atomic Force; Microscopy, Electron, Scanning; Middle Aged; Mitochondria; Mitochondrial Proteins; Mitral Valve; Mitral Valve Insufficiency; Models, Anatomic; Molecular Structure; Molybdenum; Monocarboxylic Acid Transporters; Moths; MPTP Poisoning; Multigene Family; Multiparametric Magnetic Resonance Imaging; Multiple Myeloma; Muscle, Skeletal; Mutagens; Mutation; Myeloid Cells; Nanocomposites; Nanofibers; Nanomedicine; Nanoparticles; Nanowires; Neoadjuvant Therapy; Neomycin; Neoplasm Grading; Neoplasm Recurrence, Local; Neoplasms; Neoplastic Stem Cells; Neostriatum; Neovascularization, Pathologic; Netherlands; Neuromuscular Agents; Neurons; NF-E2-Related Factor 2; NF-kappa B; Nickel; Nitrogen Oxides; Non-alcoholic Fatty Liver Disease; Nucleosides; Nucleotidyltransferases; Nutritional Status; Obesity, Morbid; Ofloxacin; Oils, Volatile; Oligopeptides; Oncogene Protein v-akt; Optical Imaging; Organic Cation Transport Proteins; Organophosphonates; Osteoarthritis; Osteoarthritis, Hip; Osteoarthritis, Knee; Osteoblasts; Osteogenesis; Oxidation-Reduction; Oxidative Stress; Oxides; Oxygen Isotopes; Pancreas; Pancreaticoduodenectomy; Pandemics; Particle Size; Particulate Matter; Patient Acceptance of Health Care; Patient Compliance; PC-3 Cells; Peptide Fragments; Peptides; Periodontal Attachment Loss; Periodontal Index; Periodontal Pocket; Periodontitis; Peroxides; Peru; Pest Control, Biological; Phosphatidylinositol 3-Kinase; Phosphatidylinositol 3-Kinases; Phylogeny; Pilot Projects; Piperidines; Plant Bark; Plant Extracts; Plant Leaves; Plasmids; Platelet Function Tests; Pneumonia, Viral; Podocytes; Poly (ADP-Ribose) Polymerase-1; Poly(ADP-ribose) Polymerase Inhibitors; Polyethylene Terephthalates; Polymers; Polymorphism, Single Nucleotide; Porosity; Portugal; Positron-Emission Tomography; Postoperative Complications; Postural Balance; Potassium Channels, Inwardly Rectifying; Povidone; Powders; Precancerous Conditions; Precision Medicine; Predictive Value of Tests; Pregnancy; Prenatal Care; Prognosis; Promoter Regions, Genetic; Prospective Studies; Prostatectomy; Prostatic Neoplasms; Proteasome Inhibitors; Protective Agents; Protein Binding; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Protein Transport; Proto-Oncogene Proteins B-raf; Proto-Oncogene Proteins c-akt; Psychiatric Nursing; PTEN Phosphohydrolase; Pulmonary Embolism; Pyrimethamine; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Rats, Wistar; Reactive Oxygen Species; Receptor, ErbB-2; Receptor, IGF Type 1; Receptors, Estrogen; Receptors, G-Protein-Coupled; Recombinational DNA Repair; Recovery of Function; Regional Blood Flow; Renal Dialysis; Renin; Renin-Angiotensin System; Reperfusion Injury; Reproducibility of Results; Republic of Korea; Respiratory Distress Syndrome; Retrospective Studies; Rhodamines; Risk Assessment; Risk Factors; RNA, Long Noncoding; RNA, Messenger; Running; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Salinity; Salmeterol Xinafoate; Sarcoma; Seasons; Shoulder Injuries; Signal Transduction; Silicon Dioxide; Silver; Sirtuin 1; Sirtuins; Skull Fractures; Social Determinants of Health; Sodium; Sodium Fluoride; Sodium Potassium Chloride Symporter Inhibitors; Sodium-Glucose Transporter 2 Inhibitors; Soil; Soil Pollutants; Spain; Spectrophotometry; Spectroscopy, Fourier Transform Infrared; Staphylococcal Protein A; Staphylococcus aureus; Stem Cells; Stereoisomerism; Stomach Neoplasms; Streptomyces; Strontium; Structure-Activity Relationship; Students, Nursing; Substance-Related Disorders; Succinic Acid; Sulfur; Surface Properties; Survival Rate; Survivin; Symporters; T-Lymphocytes; Temozolomide; Tensile Strength; Thiazoles; Thiobacillus; Thiohydantoins; Thiourea; Thrombectomy; Time Factors; Titanium; Tobacco Mosaic Virus; Tobacco Use Disorder; Toll-Like Receptor 4; Toluene; Tomography, X-Ray Computed; TOR Serine-Threonine Kinases; Toxicity Tests, Acute; Toxicity Tests, Subacute; Transcriptional Activation; Treatment Outcome; Troponin I; Tumor Cells, Cultured; Tumor Escape; Tumor Hypoxia; Tumor Microenvironment; Tumor Necrosis Factor Inhibitors; Tumor Necrosis Factor-alpha; Tyrosine; Ubiquitin-Protein Ligases; Ubiquitination; Ultrasonic Waves; United Kingdom; United States; United States Department of Veterans Affairs; Up-Regulation; Urea; Uric Acid; Urinary Bladder Neoplasms; Urinary Bladder, Neurogenic; Urine; Urodynamics; User-Computer Interface; Vemurafenib; Verbenaceae; Veterans; Veterans Health; Viral Load; Virtual Reality; Vitiligo; Water Pollutants, Chemical; Wildfires; Wnt Signaling Pathway; Wound Healing; X-Ray Diffraction; Xenograft Model Antitumor Assays; Xylenes; Young Adult; Zinc; Zinc Oxide; Zinc Sulfate; Zoonoses | 2021 |
7 trial(s) available for thiazoles and urea
| Article | Year |
|---|---|
Four compounds active against rhinovirus: comparison in vitro and in volunteers.
Topics: Adolescent; Adult; Antiviral Agents; Cell Line; Clinical Trials as Topic; Female; HeLa Cells; Humans; In Vitro Techniques; Male; Middle Aged; Oxadiazoles; Respiratory Tract Infections; Rhinovirus; Thiazoles; Urea; Virus Diseases | 1976 |
Chloromethylisothiazolone/methylisothiazolone (CMI/MI) use test with a shampoo on patch-test-positive subjects. Results of a multicentre double-blind crossover trial.
Topics: Cross-Over Studies; Dermatitis, Allergic Contact; Double-Blind Method; Hair Preparations; Humans; Patch Tests; Preservatives, Pharmaceutical; Thiazoles; Urea | 1995 |
Pharmacokinetics of pidotimod in elderly volunteers and in renal failure patients.
Topics: Administration, Oral; Adult; Aged; Aged, 80 and over; Female; Half-Life; Humans; Immunologic Factors; Injections, Intravenous; Intestinal Absorption; Male; Middle Aged; Pyrrolidonecarboxylic Acid; Renal Insufficiency; Thiazoles; Thiazolidines; Urea | 1994 |
Nitazoxanide in treatment of Helicobacter pylori: a clinical and in vitro study.
Topics: Adult; Aged; Anti-Infective Agents; Biotransformation; Breath Tests; Drug Therapy, Combination; Enzyme Inhibitors; Female; Helicobacter Infections; Helicobacter pylori; Humans; Male; Microbial Sensitivity Tests; Middle Aged; Nitro Compounds; Proton Pump Inhibitors; Thiazoles; Urea | 2003 |
A phase I/randomized phase II, non-comparative, multicenter, open label trial of CP-547,632 in combination with paclitaxel and carboplatin or paclitaxel and carboplatin alone as first-line treatment for advanced non-small cell lung cancer (NSCLC).
Topics: Administration, Oral; Adult; Aged; Antineoplastic Combined Chemotherapy Protocols; Area Under Curve; Carboplatin; Carcinoma, Non-Small-Cell Lung; Diarrhea; Dose-Response Relationship, Drug; Drug Administration Schedule; Exanthema; Female; Gastrointestinal Diseases; Half-Life; Hematologic Diseases; Humans; Lung Neoplasms; Male; Middle Aged; Neoplasm Staging; Paclitaxel; Prognosis; Thiazoles; Treatment Outcome; Urea | 2007 |
Effect of short-term treatment with meloxicam and pimobendan on the renal function in healthy beagle dogs.
Topics: Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Creatinine; Cross-Over Studies; Dogs; Female; Glomerular Filtration Rate; Kidney; Meloxicam; Pyridazines; Radionuclide Imaging; Technetium Tc 99m Pentetate; Thiazines; Thiazoles; Urea | 2008 |
Psychological distress among health care professionals of the three COVID-19 most affected Regions in Cameroon: Prevalence and associated factors.
Topics: 3' Untranslated Regions; 5'-Nucleotidase; A549 Cells; Accidental Falls; Acetylcholinesterase; Acrylic Resins; Actinobacillus; Acute Disease; Acute Kidney Injury; Adaptor Proteins, Signal Transducing; Adenosine; Adenosine Triphosphate; Administration, Inhalation; Administration, Oral; Adolescent; Adult; Advance Care Planning; Africa, Northern; Age Factors; Aged; Aged, 80 and over; Air Pollutants; Air Pollution; Air Pollution, Indoor; Albendazole; Aluminum Oxide; Anastomosis, Surgical; Ancylostoma; Ancylostomiasis; Androstadienes; Angiogenesis Inhibitors; Angiotensin II; Animals; Anti-Bacterial Agents; Anti-Infective Agents; Antibodies, Bispecific; Antibodies, Viral; Anticoagulants; Antihypertensive Agents; Antinematodal Agents; Antineoplastic Agents; Antineoplastic Agents, Immunological; Antineoplastic Combined Chemotherapy Protocols; Antioxidants; Antiporters; Antiviral Agents; Apoptosis; Aptamers, Nucleotide; Aromatase Inhibitors; Asian People; Astrocytes; Atrial Fibrillation; Auditory Threshold; Aurora Kinase B; Australia; Autophagy; Autophagy-Related Protein 5; Autotrophic Processes; Bacillus cereus; Bacillus thuringiensis; Bacterial Proteins; Beclin-1; Belgium; Benzene; Benzene Derivatives; Benzhydryl Compounds; beta Catenin; beta-Arrestin 2; Biliary Tract Diseases; Biofilms; Biofuels; Biomarkers; Biomarkers, Tumor; Biomass; Biomechanical Phenomena; Bioreactors; Biosensing Techniques; Biosynthetic Pathways; Bismuth; Blood Platelets; Bone and Bones; Bone Regeneration; Bortezomib; Botulinum Toxins, Type A; Brain; Brain Injuries; Brain Ischemia; Brain Neoplasms; Breast Neoplasms; Breath Tests; Bronchodilator Agents; Calcium Phosphates; Cannabis; Carbon Dioxide; Carbon Isotopes; Carcinogenesis; Carcinoma, Hepatocellular; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Cardiac Resynchronization Therapy; Cardiac Resynchronization Therapy Devices; Cardiomyopathies; Cardiovascular Diseases; Cariostatic Agents; Case Managers; Case-Control Studies; Catalysis; Cation Transport Proteins; CD8-Positive T-Lymphocytes; Cecropia Plant; Cell Adhesion; Cell Count; Cell Differentiation; Cell Division; Cell Line; Cell Line, Tumor; Cell Membrane; Cell Movement; Cell Proliferation; Cell Self Renewal; Cell Survival; Cells, Cultured; Cellular Reprogramming; Cellulose; Charcoal; Chemical and Drug Induced Liver Injury; Chemical Phenomena; Chemokines; Chemoradiotherapy; Chemoreceptor Cells; Child; Child Abuse; Child, Preschool; China; Chlorogenic Acid; Chloroquine; Chromatography, Gas; Chronic Disease; Clinical Competence; Coated Materials, Biocompatible; Cochlea; Cohort Studies; Color; Comorbidity; Computer Simulation; Computer-Aided Design; Contraception; Contraceptive Agents, Female; Contrast Media; COP-Coated Vesicles; Coronavirus Infections; Cost of Illness; Coturnix; COVID-19; Creatinine; Cross-Over Studies; Cross-Sectional Studies; Culex; Curriculum; Cyclic N-Oxides; Cytokines; Cytoplasm; Cytotoxicity, Immunologic; Cytotoxins; Databases, Factual; Deep Learning; Delivery, Obstetric; Denitrification; Dental Caries; Denture, Complete; Dexamethasone; Diabetes Complications; Diabetes Mellitus; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 2; Dielectric Spectroscopy; Diet, High-Fat; Dietary Fiber; Disease Models, Animal; Disease Progression; DNA; DNA Copy Number Variations; DNA, Mitochondrial; Dog Diseases; Dogs; Dopaminergic Neurons; Double-Blind Method; Down-Regulation; Doxorubicin; Drug Carriers; Drug Design; Drug Interactions; Drug Resistance, Bacterial; Drug Resistance, Neoplasm; Drug-Related Side Effects and Adverse Reactions; Drugs, Chinese Herbal; Dry Powder Inhalers; Dust; E2F1 Transcription Factor; Ecosystem; Education, Nursing; Education, Nursing, Baccalaureate; Electric Impedance; Electricity; Electrocardiography; Electrochemical Techniques; Electrochemistry; Electrodes; Electrophoresis, Polyacrylamide Gel; Endoplasmic Reticulum; Endothelial Cells; Environmental Monitoring; Enzyme Inhibitors; Epithelial Cells; Epithelial-Mesenchymal Transition; Esophageal Neoplasms; Esophageal Squamous Cell Carcinoma; Estrogen Receptor Modulators; Europe; Evoked Potentials, Auditory, Brain Stem; Exosomes; Feasibility Studies; Female; Ferricyanides; Ferrocyanides; Fibrinogen; Finite Element Analysis; Fistula; Fluorescent Dyes; Fluorides, Topical; Fluorodeoxyglucose F18; Fluticasone; Follow-Up Studies; Food Contamination; Food Microbiology; Foods, Specialized; Forensic Medicine; Frail Elderly; France; Free Radicals; Fresh Water; Fungi; Fungicides, Industrial; Galactosamine; Gastrointestinal Neoplasms; Gene Expression Profiling; Gene Expression Regulation, Neoplastic; Gene Frequency; Genetic Predisposition to Disease; Genotype; Gingival Hemorrhage; Glioblastoma; Glioma; Glomerular Filtration Rate; Glomerulosclerosis, Focal Segmental; Glucose; Glucose Transport Proteins, Facilitative; Glucosides; Glutamine; Glycolysis; Gold; GPI-Linked Proteins; Gram-Negative Bacteria; Gram-Positive Bacteria; Graphite; Haplotypes; HCT116 Cells; Healthy Volunteers; Hearing Loss; Heart Failure; Hedgehog Proteins; HEK293 Cells; HeLa Cells; Hemodynamics; Hemorrhage; Hepatocytes; Hippo Signaling Pathway; Histone Deacetylases; Homeostasis; Hospital Mortality; Hospitalization; Humans; Hydantoins; Hydrazines; Hydrogen Peroxide; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Hydroxylamines; Hypoglycemic Agents; Immunity, Innate; Immunoglobulin G; Immunohistochemistry; Immunologic Factors; Immunomodulation; Immunophenotyping; Immunotherapy; Incidence; Indazoles; Indonesia; Infant; Infant, Newborn; Infarction, Middle Cerebral Artery; Inflammation; Injections, Intramuscular; Insecticides; Insulin-Like Growth Factor I; Insurance, Health; Intention to Treat Analysis; Interleukin-1 Receptor-Associated Kinases; Interleukin-6; Intrauterine Devices; Intrauterine Devices, Copper; Iron; Ischemia; Jordan; Keratinocytes; Kidney; Kidney Diseases; Kir5.1 Channel; Klebsiella Infections; Klebsiella pneumoniae; Lab-On-A-Chip Devices; Laparoscopy; Lasers; Lasers, Semiconductor; Lenalidomide; Leptin; Lethal Dose 50; Levonorgestrel; Limit of Detection; Lipid Metabolism; Lipid Metabolism Disorders; Lipogenesis; Lipopolysaccharides; Liquid Biopsy; Liver; Liver Abscess, Pyogenic; Liver Cirrhosis; Liver Diseases; Liver Neoplasms; Longevity; Lung Neoplasms; Luteolin; Lymph Nodes; Lymphocyte Activation; Macaca fascicularis; Macrophages; Mad2 Proteins; Magnetic Resonance Imaging; Male; Mammary Glands, Human; Manganese; Manganese Compounds; MAP Kinase Signaling System; Materials Testing; Maternal Health Services; MCF-7 Cells; Medicaid; Medicine, Chinese Traditional; Melanoma; Membrane Proteins; Mental Health; Mercury; Metal Nanoparticles; Metals, Heavy; Metformin; Methionine Adenosyltransferase; Mice; Mice, Inbred BALB C; Mice, Inbred C3H; Mice, Inbred C57BL; Mice, Inbred CBA; Mice, Knockout; Mice, Nude; Microalgae; Microbial Sensitivity Tests; Microglia; MicroRNAs; Microscopy, Atomic Force; Microscopy, Electron, Scanning; Middle Aged; Mitochondria; Mitochondrial Proteins; Mitral Valve; Mitral Valve Insufficiency; Models, Anatomic; Molecular Structure; Molybdenum; Monocarboxylic Acid Transporters; Moths; MPTP Poisoning; Multigene Family; Multiparametric Magnetic Resonance Imaging; Multiple Myeloma; Muscle, Skeletal; Mutagens; Mutation; Myeloid Cells; Nanocomposites; Nanofibers; Nanomedicine; Nanoparticles; Nanowires; Neoadjuvant Therapy; Neomycin; Neoplasm Grading; Neoplasm Recurrence, Local; Neoplasms; Neoplastic Stem Cells; Neostriatum; Neovascularization, Pathologic; Netherlands; Neuromuscular Agents; Neurons; NF-E2-Related Factor 2; NF-kappa B; Nickel; Nitrogen Oxides; Non-alcoholic Fatty Liver Disease; Nucleosides; Nucleotidyltransferases; Nutritional Status; Obesity, Morbid; Ofloxacin; Oils, Volatile; Oligopeptides; Oncogene Protein v-akt; Optical Imaging; Organic Cation Transport Proteins; Organophosphonates; Osteoarthritis; Osteoarthritis, Hip; Osteoarthritis, Knee; Osteoblasts; Osteogenesis; Oxidation-Reduction; Oxidative Stress; Oxides; Oxygen Isotopes; Pancreas; Pancreaticoduodenectomy; Pandemics; Particle Size; Particulate Matter; Patient Acceptance of Health Care; Patient Compliance; PC-3 Cells; Peptide Fragments; Peptides; Periodontal Attachment Loss; Periodontal Index; Periodontal Pocket; Periodontitis; Peroxides; Peru; Pest Control, Biological; Phosphatidylinositol 3-Kinase; Phosphatidylinositol 3-Kinases; Phylogeny; Pilot Projects; Piperidines; Plant Bark; Plant Extracts; Plant Leaves; Plasmids; Platelet Function Tests; Pneumonia, Viral; Podocytes; Poly (ADP-Ribose) Polymerase-1; Poly(ADP-ribose) Polymerase Inhibitors; Polyethylene Terephthalates; Polymers; Polymorphism, Single Nucleotide; Porosity; Portugal; Positron-Emission Tomography; Postoperative Complications; Postural Balance; Potassium Channels, Inwardly Rectifying; Povidone; Powders; Precancerous Conditions; Precision Medicine; Predictive Value of Tests; Pregnancy; Prenatal Care; Prognosis; Promoter Regions, Genetic; Prospective Studies; Prostatectomy; Prostatic Neoplasms; Proteasome Inhibitors; Protective Agents; Protein Binding; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Protein Transport; Proto-Oncogene Proteins B-raf; Proto-Oncogene Proteins c-akt; Psychiatric Nursing; PTEN Phosphohydrolase; Pulmonary Embolism; Pyrimethamine; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Rats, Wistar; Reactive Oxygen Species; Receptor, ErbB-2; Receptor, IGF Type 1; Receptors, Estrogen; Receptors, G-Protein-Coupled; Recombinational DNA Repair; Recovery of Function; Regional Blood Flow; Renal Dialysis; Renin; Renin-Angiotensin System; Reperfusion Injury; Reproducibility of Results; Republic of Korea; Respiratory Distress Syndrome; Retrospective Studies; Rhodamines; Risk Assessment; Risk Factors; RNA, Long Noncoding; RNA, Messenger; Running; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Salinity; Salmeterol Xinafoate; Sarcoma; Seasons; Shoulder Injuries; Signal Transduction; Silicon Dioxide; Silver; Sirtuin 1; Sirtuins; Skull Fractures; Social Determinants of Health; Sodium; Sodium Fluoride; Sodium Potassium Chloride Symporter Inhibitors; Sodium-Glucose Transporter 2 Inhibitors; Soil; Soil Pollutants; Spain; Spectrophotometry; Spectroscopy, Fourier Transform Infrared; Staphylococcal Protein A; Staphylococcus aureus; Stem Cells; Stereoisomerism; Stomach Neoplasms; Streptomyces; Strontium; Structure-Activity Relationship; Students, Nursing; Substance-Related Disorders; Succinic Acid; Sulfur; Surface Properties; Survival Rate; Survivin; Symporters; T-Lymphocytes; Temozolomide; Tensile Strength; Thiazoles; Thiobacillus; Thiohydantoins; Thiourea; Thrombectomy; Time Factors; Titanium; Tobacco Mosaic Virus; Tobacco Use Disorder; Toll-Like Receptor 4; Toluene; Tomography, X-Ray Computed; TOR Serine-Threonine Kinases; Toxicity Tests, Acute; Toxicity Tests, Subacute; Transcriptional Activation; Treatment Outcome; Troponin I; Tumor Cells, Cultured; Tumor Escape; Tumor Hypoxia; Tumor Microenvironment; Tumor Necrosis Factor Inhibitors; Tumor Necrosis Factor-alpha; Tyrosine; Ubiquitin-Protein Ligases; Ubiquitination; Ultrasonic Waves; United Kingdom; United States; United States Department of Veterans Affairs; Up-Regulation; Urea; Uric Acid; Urinary Bladder Neoplasms; Urinary Bladder, Neurogenic; Urine; Urodynamics; User-Computer Interface; Vemurafenib; Verbenaceae; Veterans; Veterans Health; Viral Load; Virtual Reality; Vitiligo; Water Pollutants, Chemical; Wildfires; Wnt Signaling Pathway; Wound Healing; X-Ray Diffraction; Xenograft Model Antitumor Assays; Xylenes; Young Adult; Zinc; Zinc Oxide; Zinc Sulfate; Zoonoses | 2021 |
159 other study(ies) available for thiazoles and urea
| Article | Year |
|---|---|
Antileukemic activity of substituted ureidothiazoles, ureidothiadiazoles, and related compounds.
Topics: Animals; Antineoplastic Agents; Leukemia, Experimental; Mice; Structure-Activity Relationship; Thiadiazoles; Thiazoles; Urea | 1979 |
Distribution and behaviour of isoselenium salts in organism. III. Radioprotective effect of selenium derivatives.
Topics: Animals; Cobalt Radioisotopes; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Guanidines; Isothiuronium; Mice; Radiation Injuries, Experimental; Radiation-Protective Agents; Selenium; Structure-Activity Relationship; Thiazoles; Urea | 1975 |
Potentiation of heroin and methadone hepatotoxicity by ethanol: an in vitro study using cultured human hepatocytes.
Topics: Biopsy; Cells, Cultured; Drug Interactions; Ethanol; Female; Glutathione; Glycogen; Heroin; Humans; L-Lactate Dehydrogenase; Liver; Male; Methadone; Oxidation-Reduction; Prospective Studies; Tetrazolium Salts; Thiazoles; Urea | 1992 |
Carbonic anhydrase: inhibition results in decreased urea production by hepatocytes.
Topics: Animals; Carbon Dioxide; Carbonic Anhydrases; Cytosol; Ethoxzolamide; Guinea Pigs; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Liver; Male; Mitochondria, Liver; Thiazoles; Urea | 1986 |
[Skin tests for hypersensitivity to Kathon CG and Germall II].
Topics: Adolescent; Adult; Aged; Drug Hypersensitivity; Female; Humans; Male; Middle Aged; Pharmaceutic Aids; Preservatives, Pharmaceutical; Skin Tests; Thiazoles; Urea | 1987 |
Synthesis and biological activity of isodithiobiurets, dithiobiurets, and dithiazoles.
Topics: Analgesics; Animals; Anticonvulsants; Antifungal Agents; Biuret; Drug Synergism; Female; Fusarium; Hypnotics and Sedatives; Insecticides; Male; Mice; Periplaneta; Rats; Thiazoles; Urea | 1987 |
Sensitivity of the spores of Blastocladiella emersonii and related fungi to antibiotics and some other drugs.
Topics: Acridines; Aniline Compounds; Anti-Bacterial Agents; Antifungal Agents; Antimycin A; Carbamates; Chloramphenicol; Chlortetracycline; Coloring Agents; Cycloheximide; Dactinomycin; Fungi; Mercury; Microbial Sensitivity Tests; Mitomycins; Nitrobenzenes; Nystatin; Phenols; Spores; Staphylococcus; Sulfonic Acids; Tetracycline; Thiazoles; Triazines; Urea | 1971 |
Induction of mitotic gene conversion in Saccharomyces cerevisiae by N-nitrosated pesticides.
Topics: Alleles; Carbaryl; Cells, Cultured; Chromosome Mapping; Herbicides; Insecticides; Mitosis; Mutagens; Mutation; Nitroso Compounds; Propoxur; Recombination, Genetic; Saccharomyces cerevisiae; Thiazoles; Urea | 1974 |
The influence of chlorthalidone, etozoline and triamterene on electrolyte and urea concentration gradients in the rat kidney.
Topics: Acetates; Animals; Carbonic Anhydrase Inhibitors; Chlorthalidone; Diuretics; Electrolytes; Female; Kidney; Natriuresis; Osmolar Concentration; Potassium; Rats; Sodium; Thiazoles; Triamterene; Urea | 1968 |
Pharmacological studies on antagonists against nicotine-induced convulsions and death.
Topics: Animals; Anticonvulsants; Chlorpromazine; Drug Antagonism; Female; Ganglionic Blockers; Hexamethonium Compounds; Histamine H1 Antagonists; Male; Meprobamate; Mice; Nicotine; Parasympatholytics; Perphenazine; Phenobarbital; Phentolamine; Reserpine; Seizures; Sympatholytics; Thiazoles; Tolazoline; Tranquilizing Agents; Urea | 1966 |
The nature of a drug-induced renal concentrating defect in rats.
Topics: Amines; Animals; Biological Transport; Carbon Radioisotopes; Dehydration; Disease Models, Animal; Glomerular Filtration Rate; Inulin; Kidney; Kidney Concentrating Ability; Kidney Cortex; Kidney Diseases; Kidney Medulla; Kidney Tubules; Male; Microscopy, Electron; Osmolar Concentration; Photometry; Potassium; Punctures; Quaternary Ammonium Compounds; Rats; Sodium; Thiazoles; Urea; Vasopressins; Water | 1974 |
Action of liver glutamine transaminase and L-amino acid oxidase on several glutamine analogs. Preparation and properties of the 4-S, O, and NH analogs of alpha-ketoglutaramic acid.
Topics: Amidohydrolases; Amino Acid Oxidoreductases; Amino Acids, Diamino; Animals; Carbamates; Carboxylic Acids; Chemical Phenomena; Chemistry; Chromatography, Paper; Cysteine; Glutamine; Glyoxylates; Hydrogen Peroxide; Imidazoles; Lactams; Liver; Propionates; Rats; Semicarbazides; Serine; Snakes; Spectrophotometry, Infrared; Spectrophotometry, Ultraviolet; Thiazoles; Transaminases; Urea; Venoms | 1973 |
Chemotherapy of tuberculosis. IX. Synthesis and screening of new thiazolyl thiocarbanilides.
Topics: Animals; Antitubercular Agents; Chemical Phenomena; Chemistry; Guinea Pigs; Isoniazid; Mycobacterium tuberculosis; Thiazoles; Urea | 1969 |
Nitrofuryl heterocyclics. 2.
Topics: Amides; Animals; Enterococcus faecalis; Mice; Nitrofurans; Shigella sonnei; Staphylococcal Infections; Staphylococcus; Streptococcal Infections; Thiazoles; Urea | 1971 |
1-Alkyl-3-(3-alkyl-5-nitro-4-thiazolin-2-ylidene)ureas and related compounds as schistosomicides.
Topics: Alkylation; Animals; Anthelmintics; Mice; Schistosomiasis; Structure-Activity Relationship; Thiazoles; Urea | 1972 |
Heterocyclic substituted ureas. II. Immunosuppressive and antiviral activity of benzothiazole- and benzoxazoleureas.
Topics: Animals; Antibody Formation; Antigen-Antibody Reactions; Antiviral Agents; Benzoxazoles; Chemical Phenomena; Chemistry; Coxsackievirus Infections; Erythrocytes; Immunosuppressive Agents; Mice; Sheep; Thiazoles; Urea | 1969 |
Behavioral and brain catecholamine depleting actions of U-14,624, an inhibitor of dopamine beta-hydroxylase.
Topics: Animals; Brain; Depression, Chemical; Dopamine; Male; Mice; Mixed Function Oxygenases; Motor Activity; Norepinephrine; Thiazoles; Urea | 1970 |
[Synthesis of some acyl derivatives of sulfonamides].
Topics: Chemistry, Pharmaceutical; Pyrazoles; Pyrimidines; Sulfanilamides; Sulfonamides; Thiazoles; Urea | 1970 |
Experimental studies on the chemosterilization of Schistosoma mansoni.
Topics: Amides; Animals; Azirines; Chemosterilants; Esters; Female; Imidazoles; Male; Mice; Nitrogen Mustard Compounds; Ovary; Phosphoric Acids; Propylene Glycols; Schistosoma; Snails; Sulfonic Acids; Testis; Thiazoles; Urea | 1970 |
[Attempts of halogen exchange against rhodan group in chain halogenized carbonyl compounds. 2. 35. On the organic rhodan compounds].
Topics: Chemistry, Pharmaceutical; Halogens; Phenylthiourea; Potassium; Thiazines; Thiazoles; Thiocyanates; Urea | 1969 |
[Chemical and pharmacological studies of ureas with hypoglycemic action. 3. Synthesis of asymmetrical 1,3-bis-(5-alkyl-1,3,4-thiadiazol-2-yl) ureas].
Topics: Animals; Hypoglycemic Agents; Rats; Thiazoles; Urea | 1967 |
Specific interaction between beta-lactams and soluble penicillin-binding protein 2a from methicillin-resistant Staphylococcus aureus: development of a chromogenic assay.
Topics: Acylation; Anti-Bacterial Agents; Bacterial Proteins; beta-Lactams; Carrier Proteins; Cephalosporins; Chromogenic Compounds; Hexosyltransferases; Kinetics; Lactams; Mass Spectrometry; Methicillin Resistance; Muramoylpentapeptide Carboxypeptidase; Penicillin V; Penicillin-Binding Proteins; Penicillins; Peptidyl Transferases; Protein Binding; Staphylococcus aureus; Thiazoles; Urea | 1996 |
Synthesis of novel 4,5-diphenylthiazole derivatives as potential acyl-CoA:cholesterol O-acyltransferase inhibitors.
Topics: Animals; Enzyme Inhibitors; In Vitro Techniques; Male; Microsomes, Liver; Phenylurea Compounds; Rats; Rats, Wistar; Sterol O-Acyltransferase; Structure-Activity Relationship; Thiazoles; Urea | 1999 |
Simultaneous analysis of urinary 2-thiothiazolidine-4-carboxylic acid and thiocarbamide as a biological exposure index for carbon disulfide exposure.
Topics: Animals; Carbon Disulfide; Environmental Exposure; Rats; Rats, Sprague-Dawley; Thiazoles; Thiazolidines; Thiourea; Urea | 1999 |
Amino- and urea-substituted thiazoles inhibit photosynthetic electron transfer.
Topics: Amines; Electron Transport; Herbicides; Magnoliopsida; Molecular Structure; Photosynthesis; Thiazoles; Urea | 2000 |
Effect of environmental factors on the kinetics of insulin fibril formation: elucidation of the molecular mechanism.
Topics: Anilino Naphthalenesulfonates; Animals; Anions; Benzothiazoles; Cattle; Chemistry, Physical; Excipients; Fluorescent Dyes; Hydrogen-Ion Concentration; Insulin; Kinetics; Methylamines; Models, Chemical; Osmolar Concentration; Protein Denaturation; Salts; Sonication; Sucrose; Surface Properties; Thiazoles; Urea | 2001 |
Solution conditions can promote formation of either amyloid protofilaments or mature fibrils from the HypF N-terminal domain.
Topics: Amyloid; Amyloid beta-Peptides; Bacterial Proteins; Benzothiazoles; Circular Dichroism; Cloning, Molecular; Coloring Agents; Congo Red; Escherichia coli; Fluorescent Dyes; Hot Temperature; Hydrogen-Ion Concentration; Microscopy, Electron; Protein Structure, Tertiary; Thiazoles; Time Factors; Trifluoroethanol; Urea | 2001 |
In vitro induction of apoptosis vs. necrosis by widely used preservatives: 2-phenoxyethanol, a mixture of isothiazolinones, imidazolidinyl urea and 1,2-pentanediol.
Topics: Apoptosis; DNA; DNA Fragmentation; Ethylene Glycols; Food Preservatives; Glycols; HL-60 Cells; Humans; Necrosis; Pentanes; Pentanols; Thiazoles; Urea | 2002 |
Kinetics and energetics of assembly, nucleation, and growth of aggregates and fibrils for an amyloidogenic protein. Insights into transition states from pressure, temperature, and co-solute studies.
Topics: Amyloid; Benzothiazoles; Chromatography, High Pressure Liquid; Coloring Agents; Congo Red; Humans; Immunoglobulin Light Chains; Kinetics; Microscopy, Electron; Microscopy, Fluorescence; Pressure; Protein Binding; Protein Folding; Protein Structure, Tertiary; Spectroscopy, Fourier Transform Infrared; Temperature; Thermodynamics; Thiazoles; Time Factors; Ultraviolet Rays; Urea | 2002 |
Selection of a thiazole urea-resistant variant of bovine viral diarrhoea virus that maps to the RNA-dependent RNA polymerase.
Topics: Animals; Antiviral Agents; Cell Line; Diarrhea Viruses, Bovine Viral; Drug Resistance, Viral; Inhibitory Concentration 50; Molecular Structure; RNA-Dependent RNA Polymerase; RNA, Viral; Selection, Genetic; Thiazoles; Urea; Virus Replication | 2002 |
Molecular design, synthesis, and structure-Activity relationships leading to the potent and selective p56(lck) inhibitor BMS-243117.
Topics: Adenosine Triphosphate; Binding Sites; Cell Division; Drug Design; Enzyme Inhibitors; Humans; Lymphocyte Specific Protein Tyrosine Kinase p56(lck); Models, Molecular; Molecular Conformation; Structure-Activity Relationship; Substrate Specificity; T-Lymphocytes; Thiazoles; Urea | 2003 |
A systematic investigation into the effect of protein destabilisation on beta 2-microglobulin amyloid formation.
Topics: Amyloid; Benzothiazoles; beta 2-Microglobulin; Circular Dichroism; Coloring Agents; Congo Red; Dose-Response Relationship, Drug; Escherichia coli; Humans; Hydrogen-Ion Concentration; Microscopy, Electron; Models, Molecular; Mutagenesis, Site-Directed; Point Mutation; Protein Denaturation; Sodium Chloride; Thiazoles; Time Factors; Ultraviolet Rays; Urea; X-Ray Diffraction | 2003 |
Structural insights and biological effects of glycogen synthase kinase 3-specific inhibitor AR-A014418.
Topics: Adenosine Triphosphate; Animals; CDC2-CDC28 Kinases; Cell Death; Cell Line, Tumor; Cell Survival; Crystallography, X-Ray; Cyclin-Dependent Kinase 2; Cyclin-Dependent Kinase 5; Cyclin-Dependent Kinases; Dose-Response Relationship, Drug; Electrons; Enzyme Inhibitors; Glycogen Synthase Kinase 3; Humans; Inhibitory Concentration 50; Kinetics; Mice; Models, Chemical; Models, Molecular; Neurons; NIH 3T3 Cells; Peptides; Protein Binding; Signal Transduction; tau Proteins; Thiazoles; Urea | 2003 |
Discovery of novel benzothiazolesulfonamides as potent inhibitors of HIV-1 protease.
Topics: Administration, Oral; Animals; Biological Availability; HIV Protease; HIV Protease Inhibitors; Humans; Inhibitory Concentration 50; Rats; Structure-Activity Relationship; Sulfonamides; Thiazoles; Urea | 2003 |
Pharmacological characterization of CP-547,632, a novel vascular endothelial growth factor receptor-2 tyrosine kinase inhibitor for cancer therapy.
Topics: Animals; Endothelium, Vascular; Enzyme Inhibitors; Female; Humans; Kinetics; Male; Mice; Mice, Inbred C3H; Mice, Nude; Neoplasms, Experimental; Neovascularization, Pathologic; NIH 3T3 Cells; Phosphorylation; Rats; Rats, Sprague-Dawley; Thiazoles; Urea; Vascular Endothelial Growth Factor Receptor-2; Xenograft Model Antitumor Assays | 2003 |
Ureas of 5-aminopyrazole and 2-aminothiazole inhibit growth of gram-positive bacteria.
Topics: Anti-Bacterial Agents; Gram-Positive Bacteria; Methicillin Resistance; Microbial Sensitivity Tests; Molecular Conformation; Molecular Structure; Pyrazoles; Staphylococcus aureus; Structure-Activity Relationship; Thiazoles; Urea | 2003 |
Characterisation of the binding of [3H]-SB-674042, a novel nonpeptide antagonist, to the human orexin-1 receptor.
Topics: Animals; Benzoxazoles; CHO Cells; Cricetinae; Humans; Naphthyridines; Orexin Receptors; Protein Binding; Pyrrolidines; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Thiazoles; Tritium; Urea | 2004 |
GSK-3beta inhibition reverses axonal transport defects and behavioural phenotypes in Drosophila.
Topics: Animals; Axonal Transport; Axons; Drosophila melanogaster; Drosophila Proteins; Enzyme Inhibitors; Glycogen Synthase Kinase 3; Humans; Larva; Lithium Chloride; Locomotion; Phosphorylation; Protein Processing, Post-Translational; Recombinant Fusion Proteins; tau Proteins; Tauopathies; Thiazoles; Urea | 2004 |
AR-A014418, a selective GSK-3 inhibitor, produces antidepressant-like effects in the forced swim test.
Topics: Amphetamine; Animals; Antidepressive Agents; Central Nervous System Stimulants; Enzyme Inhibitors; Glycogen Synthase Kinase 3; Male; Motor Activity; Rats; Rats, Sprague-Dawley; Swimming; Thiazoles; Urea | 2004 |
Effect of meloxicam and carprofen on renal function when administered to healthy dogs prior to anesthesia and painful stimulation.
Topics: Anesthesia; Animals; Anti-Inflammatory Agents, Non-Steroidal; Area Under Curve; Blood Pressure; Carbazoles; Creatine; Cross-Over Studies; Dogs; Electric Stimulation; Female; Glomerular Filtration Rate; Heart Rate; Kidney; Male; Meloxicam; Respiration; Thiazines; Thiazoles; Urea | 2004 |
Effects of the antibiotic pulvomycin on the elongation factor Tu-dependent reactions. Comparison with other antibiotics.
Topics: Aminoglycosides; Anti-Bacterial Agents; Binding Sites; Enzyme Inhibitors; Enzyme Stability; GTP Phosphohydrolases; Guanosine Diphosphate; Guanosine Triphosphate; Hydrolysis; Peptide Elongation Factor Tu; Peptide Elongation Factors; Peptides, Cyclic; Protein Denaturation; Pyridones; Thiazoles; Trypsin; Urea | 2004 |
Investigating the effects of mutations on protein aggregation in the cell.
Topics: Animals; Benzothiazoles; Biotechnology; Blotting, Western; Chickens; Cloning, Molecular; Cytosol; DNA Mutational Analysis; Dose-Response Relationship, Drug; Electrophoresis, Polyacrylamide Gel; Escherichia coli; Macromolecular Substances; Muramidase; Mutation; Peptides; Point Mutation; Protein Binding; Protein Conformation; Protein Denaturation; Protein Engineering; Protein Folding; Protein Structure, Tertiary; Solubility; Thiazoles; Urea | 2005 |
Effect of bradykinin on nitric oxide production, urea synthesis and viability of rat hepatocyte cultures.
Topics: Animals; Bradykinin; Cell Survival; Cells, Cultured; Coloring Agents; Enzyme Inhibitors; Fluorescein; Hepatocytes; Indicators and Reagents; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Rats; Rats, Wistar; Tetrazolium Salts; Thiazoles; Time Factors; Urea | 2005 |
Effect of lesions of cerebellar fastigial nuclei on lymphocyte functions of rats.
Topics: Animals; Biogenic Monoamines; Brain Chemistry; Brain Diseases; Cell Death; Cell Proliferation; Cerebellar Nuclei; Chromatography, High Pressure Liquid; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Flow Cytometry; Glutamic Acid; Hypothalamus; Kainic Acid; Killer Cells, Natural; Lymphocyte Activation; Lymphocytes; Macrolides; Quinolines; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Staining and Labeling; Tetrazolium Salts; Thiazoles; Time Factors; Urea | 2005 |
Fibrillogenesis of apomyoglobin facilitated by aggregation sequence of yeast Sup35 in various regions.
Topics: Amino Acid Sequence; Animals; Apoproteins; Benzothiazoles; Hydrogen-Ion Concentration; Male; Microscopy, Electron; Models, Molecular; Molecular Sequence Data; Mutation; Myoglobin; Peptide Termination Factors; Prions; Protein Denaturation; Protein Structure, Tertiary; Recombinant Fusion Proteins; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Thiazoles; Urea; Whales | 2005 |
Glycogen synthase kinase-3beta participates in nuclear factor kappaB-mediated gene transcription and cell survival in pancreatic cancer cells.
Topics: Apoptosis; Cell Growth Processes; Cell Line, Tumor; Cell Survival; Gene Expression Regulation, Neoplastic; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; NF-kappa B; Pancreatic Neoplasms; Thiazoles; Transcription, Genetic; Urea | 2005 |
Synthesis and ex vivo evaluation of carbon-11 labelled N-(4-methoxybenzyl)-N'-(5-nitro-1,3-thiazol-2-yl)urea ([11C]AR-A014418): a radiolabelled glycogen synthase kinase-3beta specific inhibitor for PET studies.
Topics: Animals; Carbon Radioisotopes; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Isotope Labeling; Positron-Emission Tomography; Rats; Rats, Sprague-Dawley; Thiazoles; Tissue Distribution; Urea | 2005 |
The Wnt signaling pathway as a target for the treatment of neurodegenerative disorders.
Topics: Animals; Enzyme Inhibitors; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Homeostasis; Humans; Indoles; Lithium Chloride; Maleimides; Models, Biological; Nervous System; Neurodegenerative Diseases; Pyridines; Pyrimidines; Signal Transduction; Thiazoles; Urea; Wnt Proteins | 2006 |
Aberrant nuclear accumulation of glycogen synthase kinase-3beta in human pancreatic cancer: association with kinase activity and tumor dedifferentiation.
Topics: Adenocarcinoma; Animals; Apoptosis; Cell Differentiation; Cell Line, Tumor; Cell Nucleus; Cell Proliferation; Female; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Male; Mice; Mice, Nude; Middle Aged; NF-kappa B; Pancreatic Neoplasms; Structure-Activity Relationship; Survival Rate; Thiazoles; Transplantation, Heterologous; Urea; Xenograft Model Antitumor Assays | 2006 |
Inhibition of glycogen synthase kinase-3 suppresses the onset of symptoms and disease progression of G93A-SOD1 mouse model of ALS.
Topics: Amyotrophic Lateral Sclerosis; Animals; Blotting, Western; Caspase 3; Cell Death; Cyclooxygenase 2; Cytochromes c; Cytosol; Disease Progression; Enzyme Inhibitors; Glycogen Synthase Kinase 3; Humans; In Situ Nick-End Labeling; Intercellular Adhesion Molecule-1; Mice; Mice, Transgenic; Motor Neurons; Poly(ADP-ribose) Polymerases; Postural Balance; Spinal Cord; Superoxide Dismutase; Superoxide Dismutase-1; Thiazoles; Urea | 2007 |
Inhibition of glycogen synthase kinase-3beta protects dopaminergic neurons from MPTP toxicity.
Topics: Analysis of Variance; Animals; Apoptosis; Corpus Striatum; Disease Models, Animal; Dopamine; Dose-Response Relationship, Drug; Enzyme Inhibitors; Freezing Reaction, Cataleptic; Glycogen Synthase Kinase 3; Indoles; Male; Mice; Mice, Inbred C57BL; MPTP Poisoning; Neurons; Oximes; tau Proteins; Thiazoles; Tyrosine 3-Monooxygenase; Urea | 2007 |
Glycogen synthase kinase-3 is involved in the regulation of the cell cycle in cerebellar granule cells.
Topics: Analysis of Variance; Animals; Animals, Newborn; Apoptosis; Cell Cycle; Cells, Cultured; Cerebellum; Cyclin E; Enzyme Activation; Enzyme Inhibitors; Flow Cytometry; Glycogen Synthase Kinase 3; Immunoprecipitation; Lithium; Neurons; Potassium Deficiency; Rats; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serum; Thiazoles; Time Factors; Urea | 2007 |
Phenylimidazole derivatives of 4-pyridone as dual inhibitors of bacterial enoyl-acyl carrier protein reductases FabI and FabK.
Topics: Anti-Bacterial Agents; Bacterial Proteins; Benzothiazoles; Binding Sites; Cell Line, Tumor; Crystallography, X-Ray; Enoyl-(Acyl-Carrier-Protein) Reductase (NADH); Escherichia coli Proteins; Fatty Acid Synthase, Type II; Fatty Acids; Humans; Imidazoles; Microbial Sensitivity Tests; Models, Molecular; Molecular Structure; Mutation; Pyridones; Staphylococcus aureus; Streptococcus pneumoniae; Thiazoles; Urea | 2007 |
Crystal structure of enoyl-acyl carrier protein reductase (FabK) from Streptococcus pneumoniae reveals the binding mode of an inhibitor.
Topics: Binding, Competitive; Crystallography, X-Ray; Enoyl-(Acyl-Carrier-Protein) Reductase (NADH); Kinetics; Models, Molecular; NAD; Streptococcus pneumoniae; Thiazoles; Urea | 2008 |
Inhibition of GSK-3 reduces infarct volume and improves neurobehavioral functions.
Topics: Animals; Behavior, Animal; Blood Glucose; Brain Edema; Calcium-Binding Proteins; Caspase 3; Cerebral Infarction; Cyclooxygenase 2; Disease Models, Animal; Glial Fibrillary Acidic Protein; Glycogen Synthase Kinase 3; Microfilament Proteins; Oxadiazoles; Poly(ADP-ribose) Polymerases; Protein Kinase Inhibitors; Pyridines; Rats; Rats, Sprague-Dawley; Thiazoles; Urea | 2008 |
Antidepressant-like effect of the novel thiadiazolidinone NP031115 in mice.
Topics: Animals; Antidepressive Agents; Cyclic AMP-Dependent Protein Kinases; Cyclin-Dependent Kinase 5; Enzyme Inhibitors; Female; Glycogen Synthase Kinase 3; Male; Mice; Mitogen-Activated Protein Kinases; Motor Activity; PPAR gamma; Rosiglitazone; Swimming; Thiazoles; Thiazolidinediones; Urea | 2008 |
Functional hepatocyte-like cells derived from human bone marrow mesenchymal stem cells on a novel 3-dimensional biocompatible nanofibrous scaffold.
Topics: Alanine Transaminase; Albumins; Biocompatible Materials; Biomarkers; Cell Differentiation; Cells, Cultured; Flow Cytometry; Hepatocytes; Humans; Mesenchymal Stem Cells; Microscopy, Electron, Scanning; Nanotechnology; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetrazolium Salts; Thiazoles; Tissue Engineering; Tissue Scaffolds; Transferrin; Urea | 2008 |
Maintenance of constitutive IkappaB kinase activity by glycogen synthase kinase-3alpha/beta in pancreatic cancer.
Topics: Cell Proliferation; Cell Survival; Enzyme Activation; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; I-kappa B Kinase; Isoenzymes; NF-kappa B; Pancreatic Neoplasms; Protein Binding; Thiazoles; Tumor Cells, Cultured; Urea | 2008 |
Elevated glycogen synthase kinase-3 activity in Fragile X mice: key metabolic regulator with evidence for treatment potential.
Topics: Acoustic Stimulation; Analysis of Variance; Animals; Antimanic Agents; Brain; Citrates; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Routes; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Exploratory Behavior; Fragile X Mental Retardation Protein; Gene Expression Regulation; Glycogen Synthase Kinase 3; Indoles; Lithium Chloride; Male; Maleimides; Mice; Mice, Knockout; Pyridines; Seizures; Serine; Thiazoles; Urea | 2009 |
Potential therapeutic effect of glycogen synthase kinase 3beta inhibition against human glioblastoma.
Topics: Apoptosis; Brain Neoplasms; Cell Line, Tumor; Cell Proliferation; Cell Survival; Drug Evaluation, Preclinical; Glioblastoma; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Radiation-Sensitizing Agents; RNA Interference; Thiazoles; Urea | 2009 |
Exploring complex protein-ligand recognition mechanisms with coarse metadynamics.
Topics: Binding Sites; Computer Simulation; Crystallography, X-Ray; Enoyl-(Acyl-Carrier-Protein) Reductase (NADH); Escherichia coli; Estrogen Receptor alpha; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Ligands; Models, Chemical; Models, Molecular; Molecular Structure; Tamoxifen; Thermodynamics; Thiazoles; Triclosan; Urea | 2009 |
Cytotoxic effects of different concentrations of a carbamide peroxide bleaching gel on odontoblast-like cells MDPC-23.
Topics: Carbamide Peroxide; Cell Line; Dental Enamel; Dose-Response Relationship, Drug; Drug Combinations; Gels; Humans; Hydrogen Peroxide; Microscopy, Electron, Scanning; Odontoblasts; Peroxides; Tetrazolium Salts; Thiazoles; Time Factors; Tooth Bleaching; Tooth Discoloration; Urea | 2009 |
Inhibition of endothelial progenitor cell glycogen synthase kinase-3beta results in attenuated neointima formation and enhanced re-endothelialization after arterial injury.
Topics: Animals; Apoptosis; Arteries; Cell Adhesion; Cell Survival; Cells, Cultured; Endothelium, Vascular; Enzyme Inhibitors; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Homeostasis; Humans; Integrin alpha4; Mesenchymal Stem Cells; Mice; Models, Animal; Neovascularization, Pathologic; Thiazoles; Tunica Intima; Urea; Vascular Endothelial Growth Factor A | 2009 |
Comparative metabolite profiling of the insecticide thiamethoxam in plant and cell suspension culture of tomato.
Topics: Cells, Cultured; Fruit; Guanidines; Insecticides; Neonicotinoids; Nitro Compounds; Nitroso Compounds; Oxazines; Solanum lycopersicum; Thiamethoxam; Thiazoles; Urea | 2009 |
Glycogen synthase kinase-3beta (GSK-3beta) inhibitors AR-A014418 and B6B3O prevent human immunodeficiency virus-mediated neurotoxicity in primary human neurons.
Topics: AIDS Dementia Complex; Caspase 3; Caspase 7; Cells, Cultured; Enzyme Inhibitors; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Indoles; L-Lactate Dehydrogenase; Macrophages; Necrosis; Nerve Degeneration; Neurons; Oximes; Thiazoles; Urea | 2009 |
CCR7-dependent stimulation of survival in dendritic cells involves inhibition of GSK3beta.
Topics: Adjuvants, Immunologic; Animals; Apoptosis; Cell Survival; Chemokine CCL19; Chemokine CCL21; Dendritic Cells; Extracellular Signal-Regulated MAP Kinases; Forkhead Box Protein O1; Forkhead Transcription Factors; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; I-kappa B Kinase; Lithium Chloride; Mice; Mice, Inbred C57BL; NF-kappa B; Phosphorylation; Proto-Oncogene Proteins c-akt; Receptors, CCR7; Signal Transduction; Thiazoles; Urea | 2009 |
Cardioprotection leads to novel changes in the mitochondrial proteome.
Topics: Animals; Blotting, Western; Cardiotonic Agents; Cytochromes c; Electron Transport; Electrophoresis, Polyacrylamide Gel; Energy Metabolism; Enzyme Inhibitors; Glycogen Synthase Kinase 3; Hemodynamics; Ischemic Preconditioning, Myocardial; Mice; Mice, Inbred C57BL; Mitochondria, Heart; Myocardium; Necrosis; Proteome; Thiazoles; Urea | 2010 |
Glycogen synthase kinase-3: a new therapeutic target in renal cell carcinoma.
Topics: Adult; Aged; Carcinoma, Renal Cell; Cell Proliferation; Cell Survival; Docetaxel; Female; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Kidney Neoplasms; Male; Middle Aged; NF-kappa B; Proto-Oncogene Proteins c-bcl-2; Taxoids; Thiazoles; Urea; X-Linked Inhibitor of Apoptosis Protein | 2009 |
Inhibition of glycogen synthase kinase 3beta (GSK3beta) decreases inflammatory responses in brain endothelial cells.
Topics: AIDS Dementia Complex; Animals; Blood-Brain Barrier; Brain; Case-Control Studies; Cell Adhesion; Cells, Cultured; Drug Evaluation, Preclinical; Encephalitis; Endothelial Cells; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Inflammation Mediators; Male; Mice; Mice, Inbred C57BL; Monocytes; Protein Kinase Inhibitors; Thiadiazoles; Thiazoles; Urea | 2010 |
Transdentinal protective role of sodium ascorbate against the cytopathic effects of H2O2 released from bleaching agents.
Topics: Antioxidants; Ascorbic Acid; Carbamide Peroxide; Cell Adhesion; Cell Culture Techniques; Cell Line; Cell Survival; Coloring Agents; Dentin; Dentin Permeability; Diffusion; Humans; Hydrogen Peroxide; Materials Testing; Microscopy, Electron, Scanning; Odontoblasts; Oxidants; Peroxides; Protective Agents; Spectrophotometry, Ultraviolet; Tetrazolium Salts; Thiazoles; Time Factors; Tooth Bleaching; Urea | 2010 |
Rapid modulation of TRH and TRH-like peptide release in rat brain, pancreas, and testis by a GSK-3beta inhibitor.
Topics: Animals; Brain; Cerebellum; Corticosterone; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Male; Oligopeptides; Pancreas; Rats; Rats, Sprague-Dawley; Testis; Thiazoles; Thyrotropin-Releasing Hormone; Time Factors; Urea | 2010 |
A kinesin signaling complex mediates the ability of GSK-3beta to affect mood-associated behaviors.
Topics: Affect; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antidepressive Agents; Bipolar Disorder; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Hippocampus; Kinesins; Lithium; Male; Mice; Microtubule-Associated Proteins; Models, Biological; Neuronal Plasticity; Receptors, AMPA; Synapses; Thiazoles; Urea | 2010 |
The antinociceptive effects of AR-A014418, a selective inhibitor of glycogen synthase kinase-3 beta, in mice.
Topics: Abdominal Pain; Aggression; Analgesics; Analysis of Variance; Animals; Anti-Inflammatory Agents, Non-Steroidal; Azides; Cytokines; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Routes; Formaldehyde; Glutamic Acid; Glycogen Synthase Kinase 3; Inflammation; Male; Mice; N-Methylaspartate; Pain Measurement; Sugar Acids; Thiazoles; Urea; Xylose | 2011 |
Glycogen synthase kinase-3β indirectly facilitates interferon-γ-induced nuclear factor-κB activation and nitric oxide biosynthesis.
Topics: Animals; Blotting, Western; Cell Line; Electrophoretic Mobility Shift Assay; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Indoles; Interferon-gamma; Mice; NF-kappa B; Nitric Oxide; Oximes; RNA Interference; Signal Transduction; Thiazoles; Urea | 2010 |
The kinetic parameters and energy cost of the Hsp70 chaperone as a polypeptide unfoldase.
Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Benzothiazoles; Energy Metabolism; Escherichia coli; Fluorescent Dyes; Freezing; Genes, Reporter; HSP70 Heat-Shock Proteins; Kinetics; Luciferases; Molecular Chaperones; Polynucleotide 5'-Hydroxyl-Kinase; Protein Folding; Substrate Specificity; Thiazoles; Urea | 2010 |
Ligand-induced internalization of the orexin OX(1) and cannabinoid CB(1) receptors assessed via N-terminal SNAP and CLIP-tagging.
Topics: Alkyl and Aryl Transferases; Benzoxazoles; Cell Line; Cell Membrane; Cloning, Molecular; Cyclohexanols; Extracellular Signal-Regulated MAP Kinases; Humans; Intracellular Signaling Peptides and Proteins; Ligands; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Phenylurea Compounds; Phosphorylation; Piperidines; Plasmids; Pyrazoles; Pyrrolidines; Receptor, Cannabinoid, CB1; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Rimonabant; Thiazoles; Urea | 2011 |
Evidence for antimanic efficacy of glycogen synthase kinase-3 (GSK3) inhibitors in a strain-specific model of acute mania.
Topics: Amphetamine; Animals; Antimanic Agents; Antipsychotic Agents; Bipolar Disorder; Blood-Brain Barrier; Central Nervous System Stimulants; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Therapy, Combination; Glycogen Synthase Kinase 3; Humans; Indoles; Male; Maleimides; Mice; Mice, Mutant Strains; Molecular Targeted Therapy; Motor Activity; Reproducibility of Results; Thiadiazoles; Thiazoles; Urea | 2011 |
Characterization of the effect of TIMAP phosphorylation on its interaction with protein phosphatase 1.
Topics: Animals; Blotting, Western; Cell Line; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cytoskeletal Proteins; Endothelial Cells; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Kinetics; Membrane Proteins; Microfilament Proteins; Microscopy, Fluorescence; Phosphorylation; Protein Binding; Protein Phosphatase 1; Surface Plasmon Resonance; Thiazoles; Urea | 2011 |
Inhibition of glycogen synthase kinase-3 increases the cytotoxicity of enzastaurin.
Topics: Antineoplastic Agents; beta Catenin; Cells, Cultured; Glycogen Synthase Kinase 3; Humans; Hyaluronan Receptors; Indoles; Lymphoma, T-Cell, Cutaneous; Protein Kinase C; Protein Kinase Inhibitors; Skin Neoplasms; TCF Transcription Factors; Thiazoles; Urea | 2011 |
Troglitazone, a PPAR agonist, inhibits human prostate cancer cell growth through inactivation of NFκB via suppression of GSK-3β expression.
Topics: Apoptosis; Cell Cycle; Cell Line, Tumor; Cell Nucleus; Cell Proliferation; Chromans; Dose-Response Relationship, Drug; G1 Phase; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Immunoblotting; Male; Microscopy, Fluorescence; NF-kappa B; PPAR gamma; Prostatic Neoplasms; Resting Phase, Cell Cycle; RNA Interference; Thiazoles; Thiazolidinediones; Troglitazone; Urea | 2011 |
Synthesis and biological evaluation of glycogen synthase kinase 3 (GSK-3) inhibitors: an fast and atom efficient access to 1-aryl-3-benzylureas.
Topics: Animals; Chemistry Techniques, Synthetic; Dose-Response Relationship, Drug; Glycogen Synthase Kinase 3; Microwaves; Models, Molecular; Molecular Structure; Phenotype; Protein Kinase Inhibitors; Small Molecule Libraries; Stereoisomerism; Structure-Activity Relationship; Thiazoles; Urea; Zebrafish | 2011 |
Non-fragrance allergens in specific cosmetic products.
Topics: Acrylates; Allergens; Antioxidants; Cosmetics; Cross-Sectional Studies; Databases, Factual; Dermatitis, Allergic Contact; Emulsifying Agents; Ethylene Glycols; Formaldehyde; Humans; Hydantoins; Methacrylates; Methenamine; Nickel; Parabens; Plant Extracts; Preservatives, Pharmaceutical; Propylene Glycols; Sunscreening Agents; Thiazoles; Urea | 2011 |
Glycogen synthase kinase 3β inhibition sensitizes pancreatic cancer cells to gemcitabine.
Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Blotting, Western; Cell Line, Tumor; Deoxycytidine; DNA Repair; Drug Resistance, Neoplasm; Female; Gemcitabine; Gene Expression Regulation; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; HEK293 Cells; Humans; Mice; Mice, Inbred BALB C; Mice, Nude; Oligonucleotide Array Sequence Analysis; Pancreatic Neoplasms; Phosphorylation; Reverse Transcriptase Polymerase Chain Reaction; Thiazoles; Urea; Xenograft Model Antitumor Assays | 2012 |
Structure-based design, synthesis and biological evaluation of N-pyrazole, N'-thiazole urea inhibitors of MAP kinase p38α.
Topics: Humans; Inhibitory Concentration 50; Magnetic Resonance Spectroscopy; Mitogen-Activated Protein Kinase 14; Models, Molecular; Protein Kinase Inhibitors; Pyrazoles; Spectrometry, Mass, Electrospray Ionization; Structure-Activity Relationship; Thiazoles; Urea; X-Ray Diffraction | 2012 |
Towards the preparation of radiolabeled 1-aryl-3-benzyl ureas: Radiosynthesis of [(11)C-carbonyl] AR-A014418 by [(11)C]CO(2) fixation.
Topics: Carbon Dioxide; Carbon Radioisotopes; Glycogen Synthase Kinase 3; Humans; Positron-Emission Tomography; Radiopharmaceuticals; Thiazoles; Urea | 2012 |
Signalling through the type 1 insulin-like growth factor receptor (IGF1R) interacts with canonical Wnt signalling to promote neural proliferation in developing brain.
Topics: Adjuvants, Immunologic; Animals; beta Catenin; beta-Galactosidase; Brain; Cell Proliferation; Cells, Cultured; Embryo, Mammalian; Enzyme Inhibitors; Frontal Lobe; Gene Expression Regulation, Developmental; Lithium Chloride; Mice; Mice, Transgenic; Neurons; Receptor, IGF Type 1; RNA, Messenger; Signal Transduction; Thiazoles; Urea; Wnt Proteins | 2012 |
Forced mitotic entry of S-phase cells as a therapeutic strategy induced by inhibition of WEE1.
Topics: Animals; Antineoplastic Agents; Apoptosis; Breast Neoplasms; Cell Cycle Proteins; Cell Line; Cell Line, Tumor; Checkpoint Kinase 1; Cyclins; Deoxycytidine; DNA-Binding Proteins; Enhancer of Zeste Homolog 2 Protein; Female; Gemcitabine; Gene Expression Regulation, Neoplastic; Humans; Mice; Mice, SCID; Mitosis; Nuclear Proteins; Polycomb Repressive Complex 2; Protein Kinase Inhibitors; Protein Kinases; Protein-Tyrosine Kinases; Pyrazoles; Pyrimidines; Pyrimidinones; Quinolines; S Phase; Thiazoles; Thiophenes; Transcription Factors; Tumor Burden; Tumor Suppressor Protein p53; Urea; Xenograft Model Antitumor Assays | 2012 |
Inhibition of GSK-3β reverses the pro-apoptotic effect of proadifen (SKF-525A) in HT-29 colon adenocarcinoma cells.
Topics: Adenocarcinoma; Antineoplastic Agents; Apoptosis; Caspase 3; Cell Cycle; Cell Proliferation; Colonic Neoplasms; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; HT29 Cells; Humans; Proadifen; Protein Kinase Inhibitors; Thiazoles; Urea | 2012 |
The neuroprotective effect of the GSK-3β inhibitor and influence on the extrinsic apoptosis in the ALS transgenic mice.
Topics: Amyotrophic Lateral Sclerosis; Animals; Apoptosis; Caspase 8; Cell Count; Disease Models, Animal; fas Receptor; Fas-Associated Death Domain Protein; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Mice; Mice, Transgenic; Motor Neurons; Neuroprotective Agents; Phosphorylation; Rotarod Performance Test; Signal Transduction; Spinal Cord; Superoxide Dismutase; Superoxide Dismutase-1; Thiazoles; Urea | 2012 |
Prevention of the phencyclidine-induced impairment in novel object recognition in female rats by co-administration of lurasidone or tandospirone, a 5-HT(1A) partial agonist.
Topics: Animals; Cognition Disorders; Disease Models, Animal; Dopamine D2 Receptor Antagonists; Female; Haloperidol; Isoindoles; Lurasidone Hydrochloride; Phencyclidine; Piperazines; Piperidines; Pyridines; Pyrimidines; Rats; Rats, Long-Evans; Receptors, N-Methyl-D-Aspartate; Schizophrenia; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Agonists; Thiazoles; Urea | 2012 |
Structure-based design, synthesis and molecular modeling studies of thiazolyl urea derivatives as novel anti-parkinsonian agents.
Topics: Animals; Antiparkinson Agents; Catalepsy; Chemistry Techniques, Synthetic; Drug Design; Haloperidol; Humans; Male; Mice; Molecular Docking Simulation; Oxidative Stress; Protein Conformation; Receptors, Adenosine A2; Thiazoles; Urea | 2012 |
The nonnucleoside reverse transcription inhibitor MIV-160 delivered from an intravaginal ring, but not from a carrageenan gel, protects against simian/human immunodeficiency virus-RT Infection.
Topics: Administration, Intravaginal; Administration, Rectal; Animals; Carrageenan; Enzyme Inhibitors; Female; HIV Reverse Transcriptase; Humans; Macaca mulatta; Pyridines; Rectum; Simian Acquired Immunodeficiency Syndrome; Simian Immunodeficiency Virus; Thiazoles; Thiourea; Treatment Outcome; Urea; Vagina | 2012 |
RKI-1447 is a potent inhibitor of the Rho-associated ROCK kinases with anti-invasive and antitumor activities in breast cancer.
Topics: Animals; Antineoplastic Agents; Binding Sites; Blotting, Western; Breast Neoplasms; Cell Line, Tumor; Cell Movement; Crystallography, X-Ray; Cytoskeleton; Humans; Mammary Neoplasms, Experimental; Mice; Mice, Transgenic; Models, Molecular; Molecular Structure; Neoplasm Invasiveness; NIH 3T3 Cells; Protein Binding; Protein Kinase Inhibitors; Protein Structure, Tertiary; rho-Associated Kinases; Substrate Specificity; Thiazoles; Tumor Burden; Urea | 2012 |
Glycogen synthase kinase 3-specific inhibitor AR-A014418 decreases neuropathic pain in mice: evidence for the mechanisms of action.
Topics: Analgesics; Animals; Arginine; Cytokines; Enzyme Inhibitors; Glycogen Synthase Kinase 3; Hyperalgesia; Ligation; Male; Mice; Motor Activity; Neuralgia; Nitric Oxide; Pain Measurement; Parasympathetic Nervous System; Sciatic Neuropathy; Serotonin; Spinal Cord; Thiazoles; Urea | 2012 |
Follow-up of the monitored levels of preservative sensitivity in Europe: overview of the years 2001-2008.
Topics: Dermatitis, Allergic Contact; Disinfectants; Europe; Female; Follow-Up Studies; Formaldehyde; Humans; Male; Methenamine; Nitriles; Parabens; Patch Tests; Preservatives, Pharmaceutical; Thiazoles; Urea | 2012 |
Cross-talk between glycogen synthase kinase 3β (GSK3β) and p38MAPK regulates myocyte enhancer factor 2 (MEF2) activity in skeletal and cardiac muscle.
Topics: Animals; Cell Line; Enhancer Elements, Genetic; Female; Gene Expression Regulation; Genes, Reporter; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Imidazoles; Luciferases; Male; MEF2 Transcription Factors; Mice; Mice, Inbred C57BL; Mice, Transgenic; Muscle, Skeletal; Myoblasts; Myoblasts, Skeletal; Myocardium; Myocytes, Cardiac; Myogenic Regulatory Factors; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Primary Cell Culture; Protein Processing, Post-Translational; Pyridines; Signal Transduction; Thiazoles; Transcriptional Activation; Urea | 2013 |
Synthesis, SAR study, and biological evaluation of a series of piperazine ureas as fatty acid amide hydrolase (FAAH) inhibitors.
Topics: Amidohydrolases; Analgesics; Animals; Humans; Mice; Molecular Docking Simulation; Pain; Piperazine; Piperazines; Rats; Structure-Activity Relationship; Thiazoles; Urea | 2013 |
Glycogen synthase kinase-3 inhibition prevents learning deficits in diabetic mice.
Topics: Animals; Cerebral Cortex; Cognition Disorders; Diabetes Mellitus, Experimental; Female; Glycogen Synthase Kinase 3; Hippocampus; Maze Learning; Mice; Motor Skills; Nerve Growth Factors; Recognition, Psychology; Rotarod Performance Test; Thiazoles; Urea | 2013 |
Glycogen synthase kinase-3β positively regulates protein synthesis and cell proliferation through the regulation of translation initiation factor 4E-binding protein 1.
Topics: Adaptor Proteins, Signal Transducing; Animals; Cell Cycle Proteins; Cell Growth Processes; Enzyme Inhibitors; Female; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Mice; Mice, Nude; Peptide Initiation Factors; Phosphoproteins; Phosphorylation; Protein Binding; Protein Biosynthesis; Random Allocation; Thiazoles; Triple Negative Breast Neoplasms; Urea; Xenograft Model Antitumor Assays | 2014 |
Ureas/thioureas of benzo[d]isothiazole analog conjugated glutamic acid: synthesis and biological evaluation.
Topics: Enzyme Inhibitors; Glutamic Acid; Glycation End Products, Advanced; Structure-Activity Relationship; Thiazoles; Thiourea; Urea; Urease | 2013 |
tert-Butyl 1,5-bis(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)-1,5-dioxopentan-2-ylcarbamate urea/thiourea derivatives as potent H+/K(+)-ATPase inhibitors.
Topics: Animals; Anti-Ulcer Agents; Carbamates; Gastric Mucosa; Glutamic Acid; H(+)-K(+)-Exchanging ATPase; Proton Pump Inhibitors; Sheep; Thiazoles; Thiourea; Urea | 2013 |
Glycogen synthase kinase 3β inhibition as a therapeutic approach in the treatment of endometrial cancer.
Topics: Adjuvants, Immunologic; Animals; Carcinogenesis; Cell Line, Tumor; Cell Proliferation; Drug Synergism; Endometrial Neoplasms; Female; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Lithium Chloride; M Phase Cell Cycle Checkpoints; Mice; Neoplasm Transplantation; Paclitaxel; Signal Transduction; Thiazoles; Urea; Xenograft Model Antitumor Assays | 2013 |
Identification of glycogen synthase kinase 3α as a therapeutic target in melanoma.
Topics: Apoptosis; Cell Line, Tumor; Cell Proliferation; Down-Regulation; G1 Phase; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Melanocytes; Melanoma; Molecular Targeted Therapy; Neoplasm Staging; Resting Phase, Cell Cycle; RNA, Small Interfering; Skin Neoplasms; Thiazoles; Urea; Xenograft Model Antitumor Assays | 2013 |
Effects of environmental factors on MSP21-25 aggregation indicate the roles of hydrophobic and electrostatic interactions in the aggregation process.
Topics: Anilino Naphthalenesulfonates; Antigens, Protozoan; Benzothiazoles; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Methylamines; Peptide Fragments; Protein Multimerization; Protozoan Proteins; Sodium Dodecyl Sulfate; Static Electricity; Thiazoles; Urea | 2014 |
Metabolism-guided discovery of a potent and orally bioavailable urea-based calcimimetic for the treatment of secondary hyperparathyroidism.
Topics: Administration, Oral; Animals; Biological Availability; Half-Life; Hyperparathyroidism, Secondary; Male; Parathyroid Hormone; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Calcium-Sensing; Thiazoles; Urea | 2013 |
Glycogen synthase kinase 3 beta regulates glial glutamate transporter protein expression in the spinal dorsal horn in rats with neuropathic pain.
Topics: Amino Acid Transport System X-AG; Animals; Astrocytes; Disease Models, Animal; Drug Administration Routes; Enzyme Inhibitors; Excitatory Amino Acid Transporter 2; Gene Expression Regulation; Glial Fibrillary Acidic Protein; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Hyperalgesia; Interleukin-1beta; Male; Neurons; Oncogene Protein v-akt; Pain Measurement; Pain Threshold; Rats; Rats, Sprague-Dawley; Sciatica; Serine; Spinal Cord; Thiazoles; Time Factors; Urea | 2014 |
Thiazolopyridone ureas as DNA gyrase B inhibitors: optimization of antitubercular activity and efficacy.
Topics: Administration, Oral; Animals; Antitubercular Agents; Disease Models, Animal; Inhibitory Concentration 50; Mice; Microbial Sensitivity Tests; Molecular Structure; Mycobacterium tuberculosis; Pyridones; Thiazoles; Topoisomerase II Inhibitors; Urea | 2014 |
Persistent Wnt/β-catenin signaling determines dorsalization of the postnatal subventricular zone and neural stem cell specification into oligodendrocytes and glutamatergic neurons.
Topics: Animals; beta Catenin; Blotting, Western; Cell Proliferation; Glutamic Acid; Glycogen Synthase Kinase 3; Green Fluorescent Proteins; Lateral Ventricles; Mice, Transgenic; Microscopy, Confocal; Neural Stem Cells; Neurons; Oligodendroglia; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Thiazoles; Urea; Wnt3 Protein | 2014 |
New urea and thiourea derivatives of piperazine doped with febuxostat: synthesis and evaluation of anti-TMV and antimicrobial activities.
Topics: Anti-Infective Agents; Antiviral Agents; Bacterial Physiological Phenomena; Febuxostat; Piperazine; Piperazines; Thiazoles; Thiourea; Tobacco Mosaic Virus; Urea | 2013 |
Identification of 1-{2-[4-chloro-1'-(2,2-dimethylpropyl)-7-hydroxy-1,2-dihydrospiro[indole-3,4'-piperidine]-1-yl]phenyl}-3-{5-chloro-[1,3]thiazolo[5,4-b]pyridin-2-yl}urea, a potent, efficacious and orally bioavailable P2Y(1) antagonist as an antiplatelet
Topics: Administration, Oral; Animals; Dogs; Half-Life; Macaca fascicularis; Phenylurea Compounds; Platelet Aggregation; Platelet Aggregation Inhibitors; Purinergic P2Y Receptor Antagonists; Rats; Receptors, Purinergic P2Y1; Structure-Activity Relationship; Thiazoles; Thrombosis; Urea | 2014 |
Specific glycogen synthase kinase-3 inhibition reduces neuroendocrine markers and suppresses neuroblastoma cell growth.
Topics: Antineoplastic Agents; Apoptosis; Basic Helix-Loop-Helix Transcription Factors; Biomarkers, Tumor; Bone Marrow Neoplasms; Cell Line, Tumor; Cell Proliferation; Chromogranin A; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Neuroblastoma; Phosphorylation; Thiazoles; Tyrosine; Urea | 2014 |
New methods to control neuroblastoma growth.
Topics: Antineoplastic Agents; Biomarkers, Tumor; Bone Marrow Neoplasms; Cell Proliferation; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Neuroblastoma; Thiazoles; Urea | 2014 |
Dasatinib suppression of medulloblastoma survival and migration is markedly enhanced by combining treatment with the aurora kinase inhibitor AT9283.
Topics: Animals; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Aurora Kinase A; Autophagy; Benzimidazoles; Cell Line, Tumor; Cell Movement; Cell Proliferation; Cell Survival; Dasatinib; Enzyme Inhibitors; G2 Phase; Humans; Medulloblastoma; Mice; Mice, Inbred C57BL; Neoplasm Transplantation; Protein Kinase Inhibitors; Pyrimidines; Thiazoles; Tumor Suppressor Protein p53; Urea | 2014 |
Implications of N-capped urea/thiourea and C-capped 3-(1-piperazinyl)-1,2-benzisothiazole with bridging Gly-Val/Phe-Gly-Val-Pro as therapeutic targets.
Topics: Oligopeptides; Piperazines; Thiazoles; Thiourea; Urea | 2014 |
Early sodium dodecyl sulfate induced collapse of α-synuclein correlates with its amyloid formation.
Topics: alpha-Synuclein; Amyloid; Benzothiazoles; Circular Dichroism; Entropy; Escherichia coli; Fluorescence Resonance Energy Transfer; Glycerol; Microscopy, Electron, Transmission; Mutation; Protein Structure, Secondary; Recombinant Proteins; Sodium Dodecyl Sulfate; Solutions; Solvents; Spectrometry, Fluorescence; Thiazoles; Urea | 2015 |
Synthesis, antioxidant and anticholinesterase activities of novel coumarylthiazole derivatives.
Topics: Acetylcholinesterase; Animals; Antioxidants; Butyrylcholinesterase; Cholinesterase Inhibitors; Coumarins; Electrophorus; Horses; Structure-Activity Relationship; Thiazoles; Urea | 2015 |
Signal transducers and activators of transcription 3-induced metastatic potential in gastric cancer cells is enhanced by glycogen synthase kinase-3β.
Topics: Amino Acid Substitution; Biomarkers, Tumor; Cell Line, Tumor; Cell Movement; Epithelial-Mesenchymal Transition; Gene Knockdown Techniques; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Immunohistochemistry; Mutant Proteins; Neoplasm Invasiveness; RNA, Small Interfering; Signal Transduction; STAT3 Transcription Factor; Stomach Neoplasms; Thiazoles; Tyrphostins; Urea | 2015 |
Sitona lineatus (Coleoptera: Curculionidae) Larval Feeding on Pisum sativum L. Affects Soil and Plant Nitrogen.
Topics: Animals; Female; Fertilizers; Herbivory; Insecticides; Larva; Male; Neonicotinoids; Nitro Compounds; Nitrogen; Oxazines; Pisum sativum; Plant Roots; Soil; Thiamethoxam; Thiazoles; Urea; Weevils | 2015 |
Inhibition of invasion by glycogen synthase kinase-3 beta inhibitors through dysregulation of actin re-organisation via down-regulation of WAVE2.
Topics: Actin Cytoskeleton; Actins; Cell Adhesion; Cell Line, Tumor; Cell Movement; Collagen; Drug Combinations; Focal Adhesions; Gene Expression; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Laminin; Protein Kinase Inhibitors; Proteoglycans; Thiazoles; Urea; Wiskott-Aldrich Syndrome Protein Family | 2015 |
Potential Role of Glycogen Synthase Kinase-3β in Regulation of Myocardin Activity in Human Vascular Smooth Muscle Cells.
Topics: Actins; Calcium-Binding Proteins; Calponins; Cell Differentiation; Cell Line; Gene Expression Regulation; Gene Knockout Techniques; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Membrane Proteins; Microfilament Proteins; Muscle Proteins; Myocytes, Smooth Muscle; Nuclear Proteins; Phosphoproteins; Promoter Regions, Genetic; Protein Kinase Inhibitors; Pyrimidines; Pyrroles; Recombinant Proteins; RNA, Small Interfering; Serine; Thiazoles; Threonine; Trans-Activators; Urea | 2016 |
Glycogen synthase kinase-3 inhibitor AR-A014418 suppresses pancreatic cancer cell growth via inhibition of GSK-3-mediated Notch1 expression.
Topics: Apoptosis; Blotting, Western; Cell Line, Tumor; Cell Proliferation; Cell Survival; Glycogen Synthase Kinase 3; Humans; Immunoprecipitation; Pancreas; Pancreatic Neoplasms; Receptor, Notch1; Thiazoles; Urea | 2015 |
Identification and optimisation of a 4',5-bisthiazole series of selective phosphatidylinositol-3 kinase alpha inhibitors.
Topics: Animals; Class I Phosphatidylinositol 3-Kinases; Humans; Models, Molecular; Molecular Dynamics Simulation; Phosphatidylinositol 3-Kinases; Phosphatidylinositols; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase Inhibitors; Thiazoles; Urea | 2015 |
Potential of aryl-urea-benzofuranylthiazoles hybrids as multitasking agents in Alzheimer's disease.
Topics: Acetylcholinesterase; Alzheimer Disease; Animals; Antioxidants; Benzofurans; Butyrylcholinesterase; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Humans; Molecular Dynamics Simulation; Molecular Structure; Structure-Activity Relationship; Thiazoles; Torpedo; Urea | 2015 |
Inhibition of glycogen synthase kinase-3 beta induces apoptosis and mitotic catastrophe by disrupting centrosome regulation in cancer cells.
Topics: Apoptosis; Cell Cycle; Cell Line, Tumor; Cell Proliferation; Cell Survival; Centrosome; Chromosomal Instability; Down-Regulation; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Mitosis; Neoplasms; NF-kappa B; Phosphatidylinositol 3-Kinases; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Signal Transduction; Spindle Apparatus; Thiazoles; Urea | 2015 |
Efficacy of Rice Insecticide Seed Treatments at Selected Nitrogen Rates for Control of the Rice Water Weevil (Coleoptera: Curculionidae).
Topics: Animals; Fertilizers; Guanidines; Insect Control; Insecticides; Larva; Neonicotinoids; Nitro Compounds; Nitrogen; Oryza; Oxazines; Seeds; Thiamethoxam; Thiazoles; Urea; Weevils | 2015 |
Investigations on GSK-3β/NF-kB signaling in stress and stress adaptive behavior in electric foot shock subjected mice.
Topics: Adaptation, Psychological; Adjuvants, Immunologic; Animals; Brain; Corticosterone; Disease Models, Animal; Ditiocarb; Dose-Response Relationship, Drug; Electroshock; Enzyme Inhibitors; Exploratory Behavior; Gene Expression Regulation; Glycogen Synthase Kinase 3 beta; Interpersonal Relations; Locomotion; Mice; NF-kappa B; Signal Transduction; Stress, Psychological; Thiazoles; Urea | 2016 |
Identification of new SUMO activating enzyme 1 inhibitors using virtual screening and scaffold hopping.
Topics: Binding Sites; Humans; Inhibitory Concentration 50; Molecular Conformation; Molecular Docking Simulation; Protein Structure, Tertiary; Pyrazoles; Small Ubiquitin-Related Modifier Proteins; Structure-Activity Relationship; Thiazoles; Urea | 2016 |
Involvement of c-Myc-mediated transient receptor potential melastatin 8 expression in oxaliplatin-induced cold allodynia in mice.
Topics: Animals; Benzyl Compounds; Ganglia, Spinal; Hyperalgesia; Male; Mice; Organoplatinum Compounds; Oxaliplatin; Proto-Oncogene Proteins c-myc; Skin; Thiazoles; Transient Receptor Potential Channels; TRPA1 Cation Channel; TRPM Cation Channels; Urea | 2016 |
Synthesis of novel amide and urea derivatives of thiazol-2-ethylamines and their activity against Trypanosoma brucei rhodesiense.
Topics: Amides; Amines; Animals; Antiprotozoal Agents; Cell Survival; Dose-Response Relationship, Drug; Humans; Mice; Microsomes, Liver; Molecular Structure; Myoblasts; Parasitic Sensitivity Tests; Rats; Structure-Activity Relationship; Thiazoles; Trypanosoma brucei rhodesiense; Urea | 2016 |
Cholinergic Surveillance over Hippocampal RNA Metabolism and Alzheimer's-Like Pathology.
Topics: Acetylcholine; Alzheimer Disease; Amyloid beta-Peptides; Amyloid Precursor Protein Secretases; Animals; Aspartic Acid Endopeptidases; Cells, Cultured; Disease Models, Animal; Embryo, Mammalian; Enzyme Inhibitors; Gene Expression Regulation; Glycogen Synthase Kinase 3; Hippocampus; Humans; Learning Disabilities; Mice; Mice, Inbred C57BL; Mice, Transgenic; RNA; Thiazoles; Thyroid Nuclear Factor 1; Urea; Vesicular Acetylcholine Transport Proteins | 2017 |
Increasing metabolic stability via the deuterium kinetic isotope effect: An example from a proline-amide-urea aminothiazole series of phosphatidylinositol-3 kinase alpha inhibitors.
Topics: Amides; Animals; Biological Availability; Class I Phosphatidylinositol 3-Kinases; Deuterium; Enzyme Inhibitors; Kinetics; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Proline; Rats; Thiazoles; Urea | 2016 |
Lithium and valproate act on the GSK-3β signaling pathway to reverse manic-like behavior in an animal model of mania induced by ouabain.
Topics: Animals; Antimanic Agents; Bipolar Disorder; Disease Models, Animal; Frontal Lobe; Glycogen Synthase Kinase 3 beta; Hippocampus; Lithium Compounds; Locomotion; Male; Ouabain; Phosphatidylinositol 3-Kinases; Phosphorylation; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Rats, Wistar; Signal Transduction; Thiazoles; Urea; Valproic Acid | 2017 |
Angiotensin II degrades myeloid cell leukemia 1 in human umbilical vein endothelial cells.
Topics: Angiotensin II; Cell Survival; Dose-Response Relationship, Drug; Glycogen Synthase Kinase 3; Human Umbilical Vein Endothelial Cells; Humans; Myeloid Cell Leukemia Sequence 1 Protein; Phosphorylation; Thiazoles; Urea | 2017 |
Pharmacological assessments of potent A
Topics: Adenosine A2 Receptor Antagonists; Adenosine-5'-(N-ethylcarboxamide); Animals; Antiparkinson Agents; Catalepsy; Female; Haloperidol; Male; Mice; Motor Activity; Parkinson Disease; Rats, Wistar; Receptor, Adenosine A2A; Thiazoles; Toxicity Tests, Acute; Toxicity Tests, Subacute; Urea | 2017 |
Using gene expression database to uncover biology functions of 1,4-disubstituted 1,2,3-triazole analogues synthesized via a copper (I)-catalyzed reaction.
Topics: Antineoplastic Agents; Apoptosis; Autophagy; Carcinoma, Hepatocellular; Cell Line, Tumor; Copper; Curcumin; Databases, Genetic; Glycogen Synthase Kinase 3; Humans; Liver Neoplasms; Structure-Activity Relationship; Thiazoles; Triazoles; Urea | 2017 |
Concentration dependent switch in the kinetic pathway of lysozyme fibrillation: Spectroscopic and microscopic analysis.
Topics: Amyloid; Benzothiazoles; Hydrogen-Ion Concentration; Kinetics; Microscopy; Muramidase; Polymerization; Protein Conformation; Spectrometry, Fluorescence; Thiazoles; Urea | 2017 |
Müller glial cell reactivation in Xenopus models of retinal degeneration.
Topics: Age Factors; Animals; Animals, Genetically Modified; Animals, Newborn; Bromodeoxyuridine; Cell Proliferation; Diamines; Disease Models, Animal; Ependymoglial Cells; Gene Expression Regulation; Green Fluorescent Proteins; Metronidazole; Proliferating Cell Nuclear Antigen; Radiation-Sensitizing Agents; Regeneration; Retinal Degeneration; Rhodopsin; SOX9 Transcription Factor; Thiazoles; Urea; Xenopus laevis | 2017 |
Glycogen synthase kinase 3β inhibitors prevent hepatitis C virus release/assembly through perturbation of lipid metabolism.
Topics: Apolipoproteins B; Apolipoproteins E; Cell Line; Glycogen Synthase Kinase 3 beta; Hepacivirus; Hepatitis C; Humans; Lipid Metabolism; Lithium Chloride; Thiazoles; Urea; Virion; Virus Replication | 2017 |
Anti-stress effects of a GSK-3β inhibitor, AR-A014418, in immobilization stress of variable duration in mice.
Topics: Animals; Behavior, Animal; Brain; Corticosterone; Disease Models, Animal; Glycogen Synthase Kinase 3 beta; Mice; Motor Activity; Stress, Psychological; Thiazoles; Urea | 2017 |
GSK3 inhibitor AR-A014418 promotes osteogenic differentiation of human adipose-derived stem cells via ERK and mTORC2/Akt signaling pathway.
Topics: Adipose Tissue; Butadienes; Cell Differentiation; Cell Proliferation; Cells, Cultured; Dose-Response Relationship, Drug; Extracellular Signal-Regulated MAP Kinases; Humans; Mechanistic Target of Rapamycin Complex 2; Multiprotein Complexes; Nitriles; Osteogenesis; Proto-Oncogene Proteins c-akt; Signal Transduction; Stem Cells; Structure-Activity Relationship; Thiazoles; TOR Serine-Threonine Kinases; Urea | 2017 |
GSK3α/β: A Novel Therapeutic Target for Neuroendocrine Tumors.
Topics: Apoptosis; Cell Line, Tumor; Cell Movement; Cell Proliferation; Cell Survival; Glycogen Synthase Kinase 3 beta; Humans; Neuroendocrine Tumors; Thiazoles; Urea | 2018 |
Design, synthesis, and biological evaluation of 1-ethyl-3-(thiazol-2-yl)urea derivatives as Escherichia coli DNA gyrase inhibitors.
Topics: Anti-Bacterial Agents; Dose-Response Relationship, Drug; Drug Design; Enterococcus faecalis; Escherichia coli; Microbial Sensitivity Tests; Molecular Structure; Pseudomonas aeruginosa; Staphylococcus aureus; Structure-Activity Relationship; Thiazoles; Topoisomerase II Inhibitors; Urea | 2018 |
Glycogen synthase kinase-3β inhibition promotes lysosome-dependent degradation of c-FLIP
Topics: Amino Acid Sequence; AMP-Activated Protein Kinases; Apoptosis; CASP8 and FADD-Like Apoptosis Regulating Protein; Caspase 3; Cell Line, Tumor; Cell Nucleus; Cytoskeletal Proteins; Cytosol; Gene Expression Regulation; Hep G2 Cells; Humans; Lysosomes; Nuclear Proteins; Protein Stability; Proteolysis; RNA, Small Interfering; Signal Transduction; Thiazoles; TOR Serine-Threonine Kinases; Urea | 2018 |
Neuroprotective effect of IDPU (1-(7-imino-3-propyl-2,3-dihydrothiazolo [4,5-d]pyrimidin-6(7H)-yl)urea) in 6-OHDA induced rodent model of hemiparkinson's disease.
Topics: Animals; Antiparkinson Agents; Behavior, Animal; Depression; Disease Models, Animal; Male; Neuroprotective Agents; Oxidopamine; Parkinson Disease; Parkinsonian Disorders; Rats, Wistar; Reactive Oxygen Species; Rotarod Performance Test; Thiazoles; Tyrosine 3-Monooxygenase; Urea | 2018 |
Glycogen synthase kinase-3β inhibition enhances myelination in preterm newborns with intraventricular hemorrhage, but not recombinant Wnt3A.
Topics: Animals; Brain; Female; Glycogen Synthase Kinase 3 beta; Humans; Infant, Newborn; Infant, Premature; Male; Nerve Fibers, Myelinated; Rabbits; Recombinant Proteins; Thiazoles; Urea; Wnt3A Protein | 2018 |
Inhibition of GSK-3β on Behavioral Changes and Oxidative Stress in an Animal Model of Mania.
Topics: Aldehydes; Animals; Antioxidants; Behavior, Animal; Bipolar Disorder; Catalase; Dinoprost; Disease Models, Animal; Glutathione Peroxidase; Glycogen Synthase Kinase 3 beta; Lipid Peroxidation; Male; Motor Activity; Oxidative Stress; Protein Carbonylation; Rats, Wistar; Submitochondrial Particles; Superoxide Dismutase; Superoxides; Thiazoles; Tyrosine; Urea | 2019 |
Focused Ultrasound-Induced Blood-Brain Barrier Opening Enhances GSK-3 Inhibitor Delivery for Amyloid-Beta Plaque Reduction.
Topics: Amyloid beta-Peptides; Animals; Biomarkers; Blood-Brain Barrier; Brain; Enzyme Inhibitors; Glycogen Synthase Kinase 3; Immunohistochemistry; Male; Mice; Mice, Transgenic; Plaque, Amyloid; Protein Aggregates; Protein Aggregation, Pathological; Protein Binding; Thiazoles; Ultrasonic Waves; Urea | 2018 |
GSK3β Inhibition Restores Impaired Neurogenesis in Preterm Neonates With Intraventricular Hemorrhage.
Topics: Animals; Apoptosis; Blotting, Western; Case-Control Studies; Cell Count; Cell Proliferation; Cerebral Cortex; Cerebral Intraventricular Hemorrhage; Disease Models, Animal; Ependymoglial Cells; Glycogen Synthase Kinase 3 beta; Humans; Immunohistochemistry; Infant, Extremely Premature; Infant, Newborn; Ki-67 Antigen; Lateral Ventricles; Neural Stem Cells; Neurogenesis; PAX6 Transcription Factor; Phosphorylation; Pyramidal Cells; Rabbits; Real-Time Polymerase Chain Reaction; Retinoblastoma Protein; SOXB1 Transcription Factors; T-Box Domain Proteins; Thiazoles; Urea; White Matter | 2019 |
RKI-1447, a Rho kinase inhibitor, causes ocular hypotension, actin stress fiber disruption, and increased phagocytosis.
Topics: Animals; Cells, Cultured; Disease Models, Animal; Glaucoma, Open-Angle; Intraocular Pressure; Ocular Hypotension; Phagocytosis; rho-Associated Kinases; Stress Fibers; Swine; Thiazoles; Trabecular Meshwork; Urea | 2019 |
Phenyl and Diaryl Ureas with Thiazolo[5,4-d]pyrimidine Scaffold as Angiogenesis Inhibitors: Design, Synthesis and Biological Evaluation.
Topics: Angiogenesis Inhibitors; Cell Movement; Cell Proliferation; Dose-Response Relationship, Drug; Drug Design; Human Umbilical Vein Endothelial Cells; Humans; Molecular Structure; Neovascularization, Pathologic; Structure-Activity Relationship; Thiazoles; Urea; Wound Healing | 2019 |
The chemokine CXCL1 and its receptor CXCR2 contribute to chronic stress-induced depression in mice.
Topics: Animals; Antidepressive Agents, Second-Generation; Apoptosis; Brain-Derived Neurotrophic Factor; Chemokine CXCL1; Depression; Fluoxetine; Glycogen Synthase Kinase 3 beta; Hippocampus; Male; Mice; Mice, Inbred C57BL; Neuronal Plasticity; Phenylurea Compounds; Receptors, Interleukin-8B; Stress, Psychological; Thiazoles; Triazoles; Urea | 2019 |
RKI-1447 suppresses colorectal carcinoma cell growth via disrupting cellular bioenergetics and mitochondrial dynamics.
Topics: Animals; Antineoplastic Agents; Apoptosis; Cell Line, Tumor; Cell Proliferation; Colorectal Neoplasms; Endoplasmic Reticulum Stress; Energy Metabolism; Glycolysis; HCT116 Cells; Humans; Male; Mice; Mice, Inbred BALB C; Mitochondria; Mitochondrial Dynamics; Neoplasm Invasiveness; Reactive Oxygen Species; rho-Associated Kinases; Signal Transduction; Thiazoles; Transcription Factor CHOP; Urea; Xenograft Model Antitumor Assays | 2020 |
Glycogen synthase kinase 3β as a potential therapeutic target in synovial sarcoma and fibrosarcoma.
Topics: Animals; Cell Cycle Checkpoints; Cell Line, Tumor; Cell Proliferation; Cell Survival; Cyclin D1; Cyclin-Dependent Kinase 4; Fibrosarcoma; Gene Expression Regulation, Neoplastic; Glycogen Synthase Kinase 3 beta; Humans; Indoles; Injections, Intraperitoneal; Maleimides; Mice; Phosphorylation; RNA Interference; Sarcoma, Synovial; Thiazoles; Up-Regulation; Urea; Xenograft Model Antitumor Assays | 2020 |
The Effects of RKI-1447 in a Mouse Model of Nonalcoholic Fatty Liver Disease Induced by a High-Fat Diet and in HepG2 Human Hepatocellular Carcinoma Cells Treated with Oleic Acid.
Topics: Alanine Transaminase; Animals; Aspartate Aminotransferases; Carcinoma, Hepatocellular; Cholesterol; Diet, High-Fat; Disease Models, Animal; Glucose Tolerance Test; Hep G2 Cells; Humans; Insulin Resistance; Interleukin-6; Liver; Liver Neoplasms; Male; Malondialdehyde; Mice, Inbred ICR; Models, Biological; Non-alcoholic Fatty Liver Disease; Oleic Acid; Oxidative Stress; rhoA GTP-Binding Protein; Signal Transduction; Superoxide Dismutase; Thiazoles; Triglycerides; Tumor Necrosis Factor-alpha; Urea | 2020 |
Optimization of 5-substituted thiazolyl ureas and 6-substituted imidazopyridines as potential HIV-1 latency reversing agents.
Topics: Anti-HIV Agents; Drug Design; HEK293 Cells; HIV-1; Humans; Imidazoles; Pyridines; Thiazoles; Urea; Virus Latency | 2020 |
GSK3β suppression inhibits MCL1 protein synthesis in human acute myeloid leukemia cells.
Topics: Aniline Compounds; Antineoplastic Agents; Apoptosis; Autophagy; Cell Line, Tumor; Cell Proliferation; Down-Regulation; Glycogen Synthase Kinase 3 beta; HL-60 Cells; Humans; Leukemia, Myeloid, Acute; MAP Kinase Signaling System; Myeloid Cell Leukemia Sequence 1 Protein; RNA, Messenger; Sulfonamides; Thiazoles; U937 Cells; Urea | 2021 |
The involvement of PI3K/Akt/mTOR/GSK3β signaling pathways in the antidepressant-like effect of AZD6765.
Topics: Animals; Antidepressive Agents; Behavior, Animal; Depression; Drug Combinations; Female; Glycogen Synthase Kinase 3 beta; Hindlimb Suspension; Hippocampus; Ketamine; Lithium Chloride; Mice; Open Field Test; Phenethylamines; Phosphatidylinositol 3-Kinases; Phosphorylation; Proto-Oncogene Proteins c-akt; Pyridines; Ribosomal Protein S6 Kinases, 70-kDa; Signal Transduction; Sirolimus; Stress, Physiological; Thiazoles; TOR Serine-Threonine Kinases; Urea | 2020 |
Discovery of novel 6-hydroxybenzothiazole urea derivatives as dual Dyrk1A/α-synuclein aggregation inhibitors with neuroprotective effects.
Topics: alpha-Synuclein; Cell Survival; Dose-Response Relationship, Drug; Drug Discovery; Dyrk Kinases; HEK293 Cells; Humans; Molecular Structure; Neuroprotective Agents; Protein Aggregates; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Structure-Activity Relationship; Thiazoles; Urea | 2022 |
Mechanical Stretch Induces Annulus Fibrosus Cell Senescence through Activation of the RhoA/ROCK Pathway.
Topics: Animals; Annulus Fibrosus; Cell Proliferation; Cells, Cultured; Cellular Senescence; G1 Phase Cell Cycle Checkpoints; Intervertebral Disc Degeneration; Protein Kinase Inhibitors; Rats; Rats, Sprague-Dawley; rho GTP-Binding Proteins; rho-Associated Kinases; Signal Transduction; Stress, Mechanical; Telomerase; Thiazoles; Urea | 2021 |