Page last updated: 2024-08-21

thiazoles and tacrolimus

thiazoles has been researched along with tacrolimus in 23 studies

Research

Studies (23)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's9 (39.13)18.2507
2000's10 (43.48)29.6817
2010's4 (17.39)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bergstrand, H; Lundquist, B1
Bergstrand, H; Eriksson, T; Hallberg, A; Johansson, B; Karabelas, K; Michelsen, P; Nybom, A1
Cooper, MH; Gregory, SH; Starzl, TE; Wing, EJ1
Leduc, D; Pretolani, M; Vargaftig, BB; Zuany-Amorim, C1
Cai, W; Foulkes, JG; Hu, L1
Claude, JR; Duc, HT; Dutertre-Catella, H; Ellouk-Achard, S; Martin, C; Pham-Huy, C; Thevenin, M; Warnet, JM1
Claude, JR; Dutertre-Catella, H; Ellouk-Achard, S; Martin, C; Massicot, F; Pham-Huy, C; Rucay, P; Thevenin, M; Warnet, JM1
Finney, NS1
Morin, C; Simon, N; Thiault, L; Tillement, JP; Zini, R1
Heuser, J; McGraw, TE; Moskowitz, HS; Ryan, TA1
Araki, N; Fukuuchi, Y; Gotoh, J; Hamada, J; Sasaki, T; Shibata, M1
Gotham, S1
Castilho, RF; Kowaltowski, AJ; Maciel, EN; Rodrigues, JM; Schwalm, FD; Souza, DO; Vercesi, AE; Wajner, M1
Gabryel, B; Małecki, A; Toborek, T1
Arakawa, K; Hirano, T; Saito, K; Saito, N; Satoh, H; Sugiyama, K; Takahashi, K1
Kaminska, B; Szydlowska, K; Zawadzka, M1
Cárcamo, JG; Claude, AA; Garrido, WX; González-Oyarzún, MA; Quezada, CA; Rauch, MC; Salas, MR; San Martín, RE; Slebe, JC; Yañez, AJ1
Dannaoui, E; Lortholary, O; Schwarz, P1
Bandin, F; Baudouin, V; Carol, A; Cassaing, S; Decramer, S; Garnier, A; Guigonis, V; Kwon, T; Linas, MD; Valentin, A1
de Ruiter, P; Janssen, HL; Kwekkeboom, J; Metselaar, HJ; Pan, Q; Tilanus, HW; van der Laan, LJ1
Hirano, T; Isogai, K; Nakagawa, Y; Saito, K; Satoh, H; Sugiyama, K; Takahashi, K; Tasaki, M; Toyama, A1
Aikawa, Y; Akashi, K; Cleary, ML; Katsumoto, T; Kitabayashi, I; Shima, Y; Shino, M; Stanley, ER; Tenen, DG; Yamagata, K1
Huang, F; Rowland, L; Sabo, JP; Schultz, A; Trampisch, M; Voelk, C1

Reviews

2 review(s) available for thiazoles and tacrolimus

ArticleYear
Transcription-modulating drugs: mechanism and selectivity.
    Current opinion in biotechnology, 1996, Volume: 7, Issue:6

    Topics: Animals; Anti-Inflammatory Agents; Aspirin; Cyclosporine; Drug Design; Estrogen Antagonists; Humans; Hypoglycemic Agents; Immunosuppressive Agents; Polyenes; Sirolimus; Tacrolimus; Thiazoles; Transcription, Genetic

1996
Enantioselective epoxide hydrolysis: catalysis involving microbes, mammals and metals.
    Chemistry & biology, 1998, Volume: 5, Issue:4

    Topics: Antibodies, Catalytic; Antihypertensive Agents; Antineoplastic Agents; Catalysis; Diltiazem; Epothilones; Epoxy Compounds; Hydrolysis; Immunosuppressive Agents; Tacrolimus; Thiazoles

1998

Trials

1 trial(s) available for thiazoles and tacrolimus

ArticleYear
Pharmacokinetic Interaction between Faldaprevir and Cyclosporine or Tacrolimus in Healthy Volunteers: A Prospective, Open-Label, Fixed-Sequence, Crossover Study.
    Basic & clinical pharmacology & toxicology, 2018, Volume: 123, Issue:1

    Topics: Adolescent; Adult; Aminoisobutyric Acids; Antiviral Agents; Area Under Curve; Cross-Over Studies; Cyclosporine; Drug Interactions; Female; Graft Rejection; Healthy Volunteers; Hepatitis C; Humans; Immunosuppressive Agents; Leucine; Liver Transplantation; Male; Middle Aged; Oligopeptides; Proline; Prospective Studies; Quinolines; Secondary Prevention; Tacrolimus; Thiazoles; Young Adult

2018

Other Studies

20 other study(ies) available for thiazoles and tacrolimus

ArticleYear
Human basophil histamine release is differently affected by inhibitors of calmodulin, diacylglycerol kinase and peptidyl prolyl cis-trans isomerase in a secretagogue specific manner.
    Allergy, 1992, Volume: 47, Issue:4 Pt 2

    Topics: Amino Acid Isomerases; Basophils; Benzimidazoles; Calmodulin; Carrier Proteins; Diacylglycerol Kinase; Felodipine; Histamine Release; Humans; Imidazoles; Isoquinolines; Peptidylprolyl Isomerase; Phenothiazines; Phosphotransferases; Pyrimidinones; Tacrolimus; Thiazoles

1992
Modulation of neutrophil superoxide generation by inhibitors of protein kinase C, calmodulin, diacylglycerol and myosin light chain kinases, and peptidyl prolyl cis-trans isomerase.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 263, Issue:3

    Topics: Amino Acid Isomerases; Basophils; Calmodulin; Carbazoles; Carrier Proteins; Diacylglycerol Kinase; Histamine Release; Humans; Indole Alkaloids; Myosin-Light-Chain Kinase; Neutrophils; Peptidylprolyl Isomerase; Phosphotransferases; Protein Kinase C; Pyrimidinones; Superoxides; Tacrolimus; Tetradecanoylphorbol Acetate; Thiazoles

1992
Rapamycin but not FK506 inhibits the proliferation of mononuclear phagocytes induced by colony-stimulating factors.
    Transplantation, 1994, Volume: 57, Issue:3

    Topics: Animals; Bone Marrow Cells; Cell Count; Cell Division; Colony-Stimulating Factors; Concanavalin A; Culture Media, Conditioned; Cyclosporine; Female; Lymphocyte Activation; Mice; Mice, Inbred C57BL; Phagocytes; Polyenes; Sirolimus; Spleen; T-Lymphocytes; Tacrolimus; Tetrazolium Salts; Thiazoles; Thymidine; Tritium

1994
Characterization and pharmacological modulation of antigen-induced peritonitis in actively sensitized mice.
    British journal of pharmacology, 1993, Volume: 110, Issue:2

    Topics: Animals; Benzeneacetamides; Cetirizine; Cycloheximide; Dexamethasone; Eosinophils; Histamine Release; Hydroxamic Acids; Indomethacin; Kinetics; Leukocyte Count; Leukotriene B4; Leukotriene C4; Lipoxygenase Inhibitors; Male; Mice; Mice, Inbred BALB C; Ovalbumin; Peritoneal Cavity; Peritonitis; Platelet Activating Factor; T-Lymphocytes; Tacrolimus; Terfenadine; Thiazoles; Zymosan

1993
Implication of CYP 3A in the toxicity of cyclosporin G (CsG), cyclosporin A (CsA) and FK506 on rat hepatocytes in primary culture.
    Archives of toxicology, 1997, Volume: 71, Issue:7

    Topics: Animals; Aryl Hydrocarbon Hydroxylases; Calcium; Cell Survival; Cells, Cultured; Coloring Agents; Cyclosporine; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Flow Cytometry; Immunosuppressive Agents; Intracellular Fluid; Liver; Male; Oxidoreductases, N-Demethylating; Rats; Rats, Wistar; Tacrolimus; Tetrazolium Salts; Thiazoles

1997
Modulation of energy status and cytotoxicity induced by FK506 and cyclosporin A in a renal epithelial cell line.
    Archives of toxicology, 1997, Volume: 71, Issue:8

    Topics: Adenosine Triphosphate; Animals; Cell Survival; Cyclosporine; Energy Metabolism; Immunosuppressive Agents; Kidney; LLC-PK1 Cells; Nucleotides; Swine; Tacrolimus; Tetrazolium Salts; Thiazoles; Time Factors

1997
Tacrolimus decreases in vitro oxidative phosphorylation of mitochondria from rat forebrain.
    Life sciences, 1998, Volume: 63, Issue:5

    Topics: Adenosine Triphosphate; Animals; Antimycin A; Cerebral Cortex; Dose-Response Relationship, Drug; Enzyme Inhibitors; Immunosuppressive Agents; In Vitro Techniques; Male; Methacrylates; Mitochondria; Multienzyme Complexes; Oxidative Phosphorylation; Oxygen Consumption; Proton-Translocating ATPases; Rats; Rats, Wistar; Tacrolimus; Thiazoles

1998
Targeted chemical disruption of clathrin function in living cells.
    Molecular biology of the cell, 2003, Volume: 14, Issue:11

    Topics: Animals; Bridged Bicyclo Compounds, Heterocyclic; CHO Cells; Clathrin; Cloning, Molecular; Coated Pits, Cell-Membrane; Cricetinae; Cricetulus; Fluorescence Recovery After Photobleaching; Microscopy; Microscopy, Electron; Protein Binding; Tacrolimus; Tacrolimus Binding Proteins; Thiazoles; Thiazolidines

2003
FK506 abrogates delayed neuronal death via suppression of nitric oxide production in rats.
    Brain research, 2004, May-29, Volume: 1009, Issue:1-2

    Topics: Analysis of Variance; Animals; Brain Ischemia; Cell Count; Cell Death; Cell Line; Cell Survival; Dose-Response Relationship, Drug; Hippocampus; Humans; L-Lactate Dehydrogenase; Male; Microdialysis; Neuroblastoma; Neurons; Neuroprotective Agents; Nitric Oxide; Nitric Oxide Donors; Nitroso Compounds; Rats; Rats, Sprague-Dawley; Reperfusion; Staining and Labeling; Tacrolimus; Tetrazolium Salts; Thiazoles

2004
Digestive Disease Week 2004. Bowel inflammation.
    IDrugs : the investigational drugs journal, 2004, Volume: 7, Issue:6

    Topics: Azepines; Cholinergic Agents; Colitis, Ulcerative; Crohn Disease; Humans; Immunosuppressive Agents; Inflammatory Bowel Diseases; Isoquinolines; Pyridazines; Tacrolimus; Thiazoles

2004
Mitochondrial permeability transition in neuronal damage promoted by Ca2+ and respiratory chain complex II inhibition.
    Journal of neurochemistry, 2004, Volume: 90, Issue:5

    Topics: Animals; Antimycin A; Bongkrekic Acid; Brain; Calcimycin; Calcium; Catalase; Cell Survival; Cyclosporins; Dose-Response Relationship, Drug; Drug Interactions; Electron Transport Complex II; Enzyme Inhibitors; Female; In Vitro Techniques; Ionophores; Malonates; Membrane Potentials; Methylmalonic Acid; Mitochondria; NADP; Neurons; Nitro Compounds; Oxygen Consumption; PC12 Cells; Permeability; Propionates; Rats; Rotenone; Tacrolimus; Tetrazolium Salts; Thiazoles; Uncoupling Agents

2004
Immunosuppressive immunophilin ligands attenuate damage in cultured rat astrocytes depleted of glutathione and exposed to simulated ischemia in vitro. Comparison with N-acetylcysteine.
    Neurotoxicology, 2005, Volume: 26, Issue:3

    Topics: Acetylcysteine; Animals; Apoptosis; Astrocytes; Benzimidazoles; Brain Ischemia; Cell Separation; Cells, Cultured; Cyclosporine; Fluorescent Dyes; Free Radical Scavengers; Glutathione; Immunophilins; Immunosuppressive Agents; Ligands; Mitochondria; Oxidative Stress; Rats; Rats, Wistar; Reactive Oxygen Species; Tacrolimus; Tetrazolium Salts; Thiazoles

2005
Correlation between pharmacological efficacy of cyclosporine A and tacrolimus, evaluated by lymphocyte immunosuppressant-sensitivity test (LIST) with MTT assay procedure in renal transplant recipients.
    Journal of immunoassay & immunochemistry, 2006, Volume: 27, Issue:2

    Topics: Adult; Calcineurin Inhibitors; Cyclosporine; Female; Graft Rejection; Humans; Immunoassay; Immunosuppressive Agents; Kidney Transplantation; Lymphocyte Activation; Lymphocytes; Male; Middle Aged; Tacrolimus; Tetrazolium Salts; Thiazoles

2006
Neuroprotectant FK506 inhibits glutamate-induced apoptosis of astrocytes in vitro and in vivo.
    Journal of neurochemistry, 2006, Volume: 99, Issue:3

    Topics: Animals; Apoptosis; Astrocytes; Blotting, Western; Caspases; Cell Size; Cell Survival; Cells, Cultured; Cerebral Cortex; DNA Fragmentation; Enzyme Activation; Excitatory Amino Acid Antagonists; Fluorescent Dyes; Glial Fibrillary Acidic Protein; Glutamic Acid; In Situ Nick-End Labeling; Indoles; Infarction, Middle Cerebral Artery; Male; Membrane Potentials; Mitochondria; Neuroprotective Agents; Rats; Reperfusion Injury; Tacrolimus; Tetrazolium Salts; Thiazoles

2006
Effect of tacrolimus on activity and expression of P-glycoprotein and ATP-binding cassette transporter A5 (ABCA5) proteins in hematoencephalic barrier cells.
    Biological & pharmaceutical bulletin, 2008, Volume: 31, Issue:10

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Blood-Brain Barrier; Blotting, Western; Caspase 3; Cells, Cultured; Endothelial Cells; Fluoresceins; Humans; Immunosuppressive Agents; Reverse Transcriptase Polymerase Chain Reaction; Tacrolimus; Tetrazolium Salts; Thiazoles

2008
In vitro interactions between antifungals and immunosuppressive drugs against zygomycetes.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:8

    Topics: Amphotericin B; Antifungal Agents; Azoles; Cyclosporine; Drug Interactions; Immunosuppressive Agents; Itraconazole; Microbial Sensitivity Tests; Mucorales; Rhizopus; Sirolimus; Tacrolimus; Thiazoles; Triazoles

2009
Cryptosporidiosis in paediatric renal transplantation.
    Pediatric nephrology (Berlin, Germany), 2009, Volume: 24, Issue:11

    Topics: Adolescent; Antiparasitic Agents; Biopsy; Child; Cohort Studies; Cryptosporidiosis; Diarrhea; Drug Administration Schedule; Female; Follow-Up Studies; Humans; Immunosuppressive Agents; Kidney; Kidney Transplantation; Male; Mycophenolic Acid; Nitro Compounds; Prednisone; Sirolimus; Tacrolimus; Thiazoles; Time Factors; Transplantation, Homologous; Treatment Outcome

2009
Calcineurin inhibitor tacrolimus does not interfere with the suppression of hepatitis C virus infection by interferon-alpha.
    Liver transplantation : official publication of the American Association for the Study of Liver Diseases and the International Liver Transplantation Society, 2010, Volume: 16, Issue:4

    Topics: Antiviral Agents; Calcineurin Inhibitors; Cell Proliferation; Cell Survival; Gene Expression Regulation; Hepacivirus; Hepatitis C; Humans; Immunosuppressive Agents; Interferon-alpha; T-Lymphocytes; Tacrolimus; Tetrazolium Salts; Thiazoles

2010
Correlation between the pharmacological efficacy of cyclosporine and tacrolimus as evaluated by the lymphocyte immunosuppressant sensitivity test (LIST) and the MTT assay procedure in patients before and after renal transplantation.
    International journal of clinical pharmacology and therapeutics, 2011, Volume: 49, Issue:2

    Topics: Cyclosporine; Humans; Immunosuppressive Agents; Kidney Transplantation; Lymphocytes; Tacrolimus; Tetrazolium Salts; Thiazoles

2011
Essential role of PU.1 in maintenance of mixed lineage leukemia-associated leukemic stem cells.
    Cancer science, 2015, Volume: 106, Issue:3

    Topics: Animals; Carcinogenesis; Gene Expression Regulation, Leukemic; Genes, Homeobox; Histone-Lysine N-Methyltransferase; Leukemia, Myeloid, Acute; Mice; Mice, Inbred C57BL; Mice, Transgenic; Myeloid-Lymphoid Leukemia Protein; Neoplastic Stem Cells; Phenylurea Compounds; Prognosis; Proto-Oncogene Proteins; Receptor, Macrophage Colony-Stimulating Factor; Recombinant Fusion Proteins; Signal Transduction; Tacrolimus; Thiazoles; Trans-Activators; Transcription, Genetic; Transcriptional Activation; Up-Regulation

2015