Compounds > thiazoles
Page last updated: 2024-08-21

thiazoles and ssr 69071

thiazoles has been researched along with ssr 69071 in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (60.00)29.6817
2010's2 (40.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bidouard, JP; Duval, N; Herbert, JM; Janiak, P; Kapui, Z; O'Connor, SE1
Aranyi, P; Batori, S; Finance, O; Kapui, Z; Mikus, E; Szabo, T; Szeredi, J; Urban-Szabo, K; Varga, M1
Arányi, P; Bátori, S; Kapui, Z; Mikus, E; Nagy, LT; Urbán-Szabó, K; Varga, M; Vasvári-Debreczy, L1
Beel, S; De Muynck, L; Herdewyn, S; Robberecht, W; Scheveneels, W; Van Damme, P; Van Den Bosch, L1
Bali, KK; Kuner, R1

Other Studies

5 other study(ies) available for thiazoles and ssr 69071

ArticleYear
SSR69071, an elastase inhibitor, reduces myocardial infarct size following ischemia-reperfusion injury.
    European journal of pharmacology, 2003, Feb-07, Volume: 461, Issue:1

    Topics: Animals; Cyclic S-Oxides; Dose-Response Relationship, Drug; Leukocyte Elastase; Male; Myocardial Infarction; Myocardial Reperfusion Injury; Rabbits; Thiazoles

2003
Biochemical and pharmacological characterization of 2-(9-(2-piperidinoethoxy)-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yloxymethyl)-4-(1-methylethyl)-6-methoxy-1,2-benzisothiazol-3(2H)-one-1,1-dioxide (SSR69071), a novel, orally active elastase inhibitor.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 305, Issue:2

    Topics: Algorithms; Animals; Bronchoalveolar Lavage Fluid; Carrageenan; Cyclic S-Oxides; Dose-Response Relationship, Drug; Edema; Elastin; Enzyme Inhibitors; Hemorrhage; Humans; Hydrolysis; Kinetics; Leukocyte Elastase; Male; Mice; Oligopeptides; Rabbits; Rats; Thiazoles

2003
A novel orally active inhibitor of HLE.
    European journal of medicinal chemistry, 2003, Volume: 38, Issue:4

    Topics: Administration, Oral; Animals; Asthma; Cyclic S-Oxides; Cystic Fibrosis; Dose-Response Relationship, Drug; Enzyme Inhibitors; Hemorrhage; Humans; Inflammation; Leukocyte Elastase; Lung Diseases, Obstructive; Mice; Models, Chemical; Pulmonary Emphysema; Thiazoles

2003
The neurotrophic properties of progranulin depend on the granulin E domain but do not require sortilin binding.
    Neurobiology of aging, 2013, Volume: 34, Issue:11

    Topics: Adaptor Proteins, Vesicular Transport; Animals; Animals, Newborn; Antibodies; Binding Sites; Cell Survival; Cells, Cultured; Cerebral Cortex; Cyclic S-Oxides; Embryo, Nonmammalian; Embryonic Development; Endocytosis; Enzyme Inhibitors; Immunoprecipitation; Intercellular Signaling Peptides and Proteins; Morpholines; Motor Neurons; Nerve Growth Factors; Neurites; Progranulins; Protein Structure, Tertiary; Rats; Rats, Wistar; Thiazoles; Zebrafish

2013
Therapeutic potential for leukocyte elastase in chronic pain states harboring a neuropathic component.
    Pain, 2017, Volume: 158, Issue:11

    Topics: Analgesics; Animals; Cancer Pain; Chronic Pain; Cyclic S-Oxides; Disease Models, Animal; Female; Glycine; Hyperalgesia; Leukocyte Elastase; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Motor Activity; Neuralgia; Pain Measurement; Pain Threshold; Pregabalin; Serine Proteinase Inhibitors; Sulfonamides; Thiazoles

2017