Compounds > thiazoles
Page last updated: 2024-08-21

thiazoles and sr141716

thiazoles has been researched along with sr141716 in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's6 (50.00)29.6817
2010's5 (41.67)24.3611
2020's1 (8.33)2.80

Authors

AuthorsStudies
Adolfs, TJ; Borst, AJ; Coolen, HK; de Looff, W; Keizer, HG; Kruse, CG; Lange, JH; McCreary, AC; van Stuivenberg, HH; Veerman, W; Verveer, PC; Wals, HC1
Cadet, JL; Chen, J; Deng, X; Errico, S; Freed, WJ; Lee, CT1
Schweitzer, P; Slanina, KA1
Finn, P1
Kruse, CG; Lange, JH1
Chu, KL; Dart, MJ; McGaraughty, S; Meyer, MD; Yao, BB1
Milligan, G; Pediani, JD; Ward, RJ1
Cox, BF; Dart, M; Diaz, G; Gintant, GA; Green, J; Limberis, JT; Liu, X; Martin, RL; Meyer, M; Polakowski, J; Preusser, L; Su, Z; Yao, B1
Gyertyán, I; Kassai, F; Varga, B1
Beggiato, S; Borelli, AC; Bradberry, CW; Ferraro, L; Ferré, S; Goldberg, SR; Justinova, Z; Mascia, P; Melis, M; Panlilio, LV; Pistis, M; Sagheddu, C; Schindler, CW; Schwarcz, R; Secci, ME; Tanda, G; Tomasini, MC1
Eiler, WJA; Gleason, SD; Smith, JL; Witkin, JM1
Bales, KL; Dreyer, BK; Freeman, SM; Lackey, NS; Manoli, DS; Simmons, TC1

Other Studies

12 other study(ies) available for thiazoles and sr141716

ArticleYear
Bioisosteric replacements of the pyrazole moiety of rimonabant: synthesis, biological properties, and molecular modeling investigations of thiazoles, triazoles, and imidazoles as potent and selective CB1 cannabinoid receptor antagonists.
    Journal of medicinal chemistry, 2005, Mar-24, Volume: 48, Issue:6

    Topics: Administration, Oral; Animals; CHO Cells; Cricetinae; Cricetulus; Cyclohexanols; Hypotension; Hypothermia; Imidazoles; Mice; Models, Molecular; Molecular Conformation; Piperidines; Pyrazoles; Radioligand Assay; Rats; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Stereoisomerism; Structure-Activity Relationship; Thiazoles; Triazoles

2005
Protective effects of Delta(9)-tetrahydrocannabinol against N-methyl-d-aspartate-induced AF5 cell death.
    Brain research. Molecular brain research, 2005, Apr-04, Volume: 134, Issue:2

    Topics: alpha-Tocopherol; Animals; Benzimidazoles; Benzoxazines; Blotting, Northern; Blotting, Western; Calcium Channel Blockers; Calcium Channels; Capsaicin; Cell Count; Cell Death; Cell Lineage; Dizocilpine Maleate; DNA, Single-Stranded; Dose-Response Relationship, Drug; Dronabinol; Drug Interactions; Excitatory Amino Acid Agonists; Immunohistochemistry; In Situ Nick-End Labeling; Morpholines; N-Methylaspartate; Naphthalenes; Neurons; Neuroprotective Agents; Piperidines; Pyrazoles; Rats; Receptor, Cannabinoid, CB1; Receptors, N-Methyl-D-Aspartate; Reverse Transcriptase Polymerase Chain Reaction; Rimonabant; RNA, Messenger; Ruthenium; Tetrazolium Salts; Thiazoles; TRPC Cation Channels

2005
Inhibition of cyclooxygenase-2 elicits a CB1-mediated decrease of excitatory transmission in rat CA1 hippocampus.
    Neuropharmacology, 2005, Volume: 49, Issue:5

    Topics: Animals; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Electrophysiology; Excitatory Postsynaptic Potentials; GABA Antagonists; Hippocampus; In Vitro Techniques; Male; Meloxicam; Membrane Potentials; Patch-Clamp Techniques; Piperidines; Prostaglandin-Endoperoxide Synthases; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, GABA-A; Rimonabant; Synaptic Transmission; Thiazines; Thiazoles

2005
American Heart Association--scientific sessions 2005. Potential new drugs for various indications. 13-16 November 2005, Dallas, TX, USA.
    IDrugs : the investigational drugs journal, 2006, Volume: 9, Issue:1

    Topics: American Heart Association; Animals; Cardiotonic Agents; Heart Diseases; Humans; Piperidines; Potassium Channel Blockers; PPAR delta; Pyrazoles; Rimonabant; Thiazoles

2006
Cannabinoid CB1 receptor antagonists in therapeutic and structural perspectives.
    Chemical record (New York, N.Y.), 2008, Volume: 8, Issue:3

    Topics: Animals; Anti-Obesity Agents; CHO Cells; Cricetinae; Cricetulus; Humans; Imidazoles; Isomerism; Models, Chemical; Obesity; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Solubility; Structure-Activity Relationship; Thiazoles; Triazoles; Water

2008
A CB(2) receptor agonist, A-836339, modulates wide dynamic range neuronal activity in neuropathic rats: contributions of spinal and peripheral CB(2) receptors.
    Neuroscience, 2009, Feb-18, Volume: 158, Issue:4

    Topics: Action Potentials; Animals; Camphanes; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Routes; Ganglia, Spinal; Male; Neurons; Peripheral Nervous System Diseases; Physical Stimulation; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB2; Rimonabant; Spinal Cord; Thiazoles

2009
Ligand-induced internalization of the orexin OX(1) and cannabinoid CB(1) receptors assessed via N-terminal SNAP and CLIP-tagging.
    British journal of pharmacology, 2011, Volume: 162, Issue:6

    Topics: Alkyl and Aryl Transferases; Benzoxazoles; Cell Line; Cell Membrane; Cloning, Molecular; Cyclohexanols; Extracellular Signal-Regulated MAP Kinases; Humans; Intracellular Signaling Peptides and Proteins; Ligands; Naphthyridines; Neuropeptides; Orexin Receptors; Orexins; Phenylurea Compounds; Phosphorylation; Piperidines; Plasmids; Pyrazoles; Pyrrolidines; Receptor, Cannabinoid, CB1; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Rimonabant; Thiazoles; Urea

2011
Negative inotropic effect of a CB2 agonist A-955840 in isolated rabbit ventricular myocytes is independent of CB1 and CB2 receptors.
    Current drug safety, 2011, Nov-01, Volume: 6, Issue:5

    Topics: Animals; Benzamides; Calcium Channels, L-Type; Dogs; Heart Ventricles; Inhibitory Concentration 50; Male; Myocardial Contraction; Myocytes, Cardiac; Patch-Clamp Techniques; Piperidines; Pyrazoles; Rabbits; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Sarcomeres; Thiazoles

2011
Interactions of CB1 and mGlu5 receptor antagonists in food intake, anxiety and memory models in rats.
    Pharmacology, biochemistry, and behavior, 2012, Volume: 103, Issue:2

    Topics: Animals; Anxiety; Disease Models, Animal; Fear; Feeding Behavior; Male; Memory; Piperidines; Pyrazoles; Pyridines; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Rimonabant; Thiazoles

2012
Astrocytic Mechanisms Involving Kynurenic Acid Control Δ
    Molecular neurobiology, 2019, Volume: 56, Issue:5

    Topics: Action Potentials; alpha7 Nicotinic Acetylcholine Receptor; Animals; Astrocytes; Brain; Cells, Cultured; Dronabinol; Glutamic Acid; Kynurenic Acid; Male; Nucleus Accumbens; Prefrontal Cortex; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Reward; Rimonabant; RNA, Messenger; Sulfonamides; Thiazoles; Ventral Tegmental Area

2019
A medium throughput rodent model of relapse from addiction with behavioral and pharmacological specificity.
    Pharmacology, biochemistry, and behavior, 2019, Volume: 183

    Topics: Amino Acids; Animals; Behavior, Addictive; Behavior, Animal; Bridged Bicyclo Compounds, Heterocyclic; Cannabinoid Receptor Antagonists; Conditioning, Operant; Drug Discovery; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Extinction, Psychological; Feeding Behavior; Male; Models, Animal; Pyridines; Rats; Rats, Sprague-Dawley; Recurrence; Rimonabant; Self Administration; Substance-Related Disorders; Thiazoles

2019
Cannabinoid receptor Type 1 densities reflect social organization in Microtus.
    The Journal of comparative neurology, 2021, 04-01, Volume: 529, Issue:5

    Topics: Animals; Arvicolinae; Brain Chemistry; Cannabinoid Receptor Antagonists; Female; Ligands; Male; Nerve Net; Organ Specificity; Pair Bond; Radioligand Assay; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Rimonabant; Sex Characteristics; Sexual Behavior, Animal; Species Specificity; Spleen; Thiazoles

2021