thiazoles has been researched along with sr 27897 in 31 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 14 (45.16) | 18.2507 |
| 2000's | 14 (45.16) | 29.6817 |
| 2010's | 2 (6.45) | 24.3611 |
| 2020's | 1 (3.23) | 2.80 |
| Authors | Studies |
|---|---|
| Fréhel, D; Gully, D; Le Fur, G; Lespy, L; Maffrand, JP; Marcy, C; Neliat, G; Spinazzé, A | 1 |
| Bonouali-Pellissier, S | 1 |
| Gueudet, C; Gully, D; Le Fur, G; Santucci, V; Soubrie, P; Thurneyssen, O | 1 |
| Arnone, M; Gonalons, N; Gueudet, C; Gully, D; Heaulme, M; Keane, P; Le Fur, G; Poncelet, M; Santucci, V; Thurneyssen, O | 1 |
| Beart, PM; Krstew, E; Widdop, RE | 1 |
| Debonnel, G; Gronier, B | 1 |
| Allikmets, L; Harro, J; Matto, V | 1 |
| Beart, PM; Bunting, MW; Widdop, RE | 1 |
| Bischof Delaloye, A; Borovicka, J; Bouloux, C; Fried, M; Jansen, JB; Kreiss, C; Pignol, R; Schwizer, W | 1 |
| Bachy, A; Bignon, E; Boigegrain, R; Brodin, R; Cottineau, M; Gully, D; Herbert, JM; Keane, P; Labie, C; Le Fur, G; Maffrand, JP; Molimard, JC; Olliero, D; Oury-Donat, F; Pascal, M; Petereau, C; Prabonnaud, V; Rockstroh, MP; Schaeffer, P; Servant, O; Soubrié, P; Thurneyssen, O | 1 |
| Black, JW; Griffin, EP; Harper, EA; Shankley, NP | 1 |
| Bernard, C; Chayvialle, JA; Desbois, C; Dufresne, M; Fourmy, D; Gestin, M; Guilloteau, P; Gully, D; Le Dréan, G; Le Huërou-Luron, I; Moroder, L; Romé, V | 1 |
| Carillon, C; Delpech, B; Ferrara, P; Gouldson, P; Le Fur, G; Legoux, P; Shire, D | 2 |
| Bouisson, M; Escrieut, C; Fehrentz, JA; Fourmy, AD; Gigoux, V; Gully, D; Maigret, B; Martinez, J; Moroder, L; Silvente-Poirot, S; Vaysse, N | 1 |
| Felicio, LF; Ferreira, FS; Nasello, AG; Sassatani, AS; Tieppo, CA | 1 |
| Carillon, C; Dumont, X; Ferrara, P; Gouldson, P; Le Fur, G; Legoux, P; Shire, D | 1 |
| Fuentes, JA; Garrido, MM; Ruiz-Gayo, M | 1 |
| Bernard, C; Chayvialle, JA; Fourmy, D; Gestin, M; Guilloteau, P; Le Dréan, G; Le Huërou-Luron, I; Romé, V | 1 |
| Capellà, G; Clavé, P; Farré, R; González, AA; Monés, J | 1 |
| Agid, Y; Arnulf, I; Bonnet, AM; Brefel, C; Cattelin, F; Descombes, S; Jaillon, C; Pollak, P; Rascol, O; Vidailhet, M; Xie, J | 1 |
| Harper, EA; Morton, MF; Shankley, NP; Tavares, IA | 1 |
| Decker, M; Eckel, F; Frank, R; Helmberger, H; Lersch, C; Lippl, F; Neverve, J; Schulte-Frohlinde, E; Schusdziarra, V; Schwaiger, M; Weber, W | 1 |
| Cano, V; Ezquerra, L; Ramos, MP; Ruiz-Gayo, M | 2 |
| Chayvialle, JA; Guilloteau, P; Normand, V; Romé, V; Woliński, J; Zabielski, R | 1 |
| Archer-Lahlou, E; Dufresne, M; Escrieut, C; Fourmy, D; Maigret, B; Moroder, L; Pradayrol, L; Seva, C; Tikhonova, I | 1 |
| Cano, V; Ezquerra, L; Merino, B; Ruiz-Gayo, M; Somoza, B | 1 |
| Kim, BJ; Kim, SY; Kwon, YK; Lee, JH; So, I | 1 |
| Merino, B; Plaza, A; Rubio-Herrera, MA; Ruiz-Gayo, M; Sánchez-Pernaute, A; Torres-García, AJ | 1 |
| Chu, X; Dai, A; Feng, W; Han, S; He, C; Jiang, Y; Reedtz-Runge, S; Sensfuss, U; Tan, Q; Wang, J; Wang, M; Wang, MW; Wu, B; Xu, HE; Yang, D; Yang, Z; Zhang, H; Zhang, X; Zhao, Q; Zhao, S; Zhou, Q; Zhu, Y | 1 |
3 trial(s) available for thiazoles and sr 27897
| Article | Year |
|---|---|
Effect of lintitript, a new CCK-A receptor antagonist, on gastric emptying of a solid-liquid meal in humans.
Topics: Adult; Cholecystokinin; Cross-Over Studies; Double-Blind Method; Gastric Emptying; Humans; Indoleacetic Acids; Male; Pancreatic Polypeptide; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Thiazoles | 1998 |
Blockade of cholecystokinin-A receptors has no effect on dyskinesias in Parkinson's disease.
Topics: Administration, Oral; Disability Evaluation; Dyskinesia, Drug-Induced; Female; Humans; Indoleacetic Acids; Male; Middle Aged; Movement; Parkinson Disease; Random Allocation; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Thiazoles | 2001 |
Monitoring of tumour glucose metabolism by PET in a phase I study evaluating hormonal therapy in advanced pancreatic cancer.
Topics: Adenocarcinoma; Adult; Aged; Female; Fluorodeoxyglucose F18; Glucose; Hormone Antagonists; Humans; Indoleacetic Acids; Magnetic Resonance Imaging; Male; Middle Aged; Pancreatic Neoplasms; Radiopharmaceuticals; Receptors, Cholecystokinin; Thiazoles; Tomography, Emission-Computed | 2002 |
28 other study(ies) available for thiazoles and sr 27897
| Article | Year |
|---|---|
Peripheral biological activity of SR 27897: a new potent non-peptide antagonist of CCKA receptors.
Topics: Administration, Oral; Amylases; Animals; Benzodiazepinones; Binding, Competitive; Cholecystokinin; Devazepide; Dose-Response Relationship, Drug; Female; Gallbladder; Gastric Emptying; Gastrins; Guinea Pigs; In Vitro Techniques; Indoleacetic Acids; Injections, Intravenous; Male; Mice; Pancreas; Radioligand Assay; Rats; Rats, Wistar; Receptors, Cholecystokinin; Stomach; Thiazoles | 1993 |
Melatonin is involved in cholecystokinin-induced changes of ileal motility in rats.
Topics: Animals; Benzodiazepinones; Cholecystokinin; Devazepide; Electromyography; Gastrointestinal Motility; Ileum; Indoleacetic Acids; Male; Melatonin; Muscle, Smooth; Pineal Gland; Rats; Rats, Wistar; Receptors, Cholecystokinin; Thiazoles | 1994 |
The CCKA receptor antagonist SR 27897 differentially influences the activity of A9 and A10 dopaminergic neurons in the rat.
Topics: Animals; Apomorphine; Benzodiazepinones; Devazepide; Dopamine; Indoleacetic Acids; Male; Mesencephalon; Neurons; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Sincalide; Thiazoles | 1994 |
Neurobehavioural effects of SR 27897, a selective cholecystokinin type A (CCK-A) receptor antagonist.
Topics: Animals; Apomorphine; Brain; Cyclic GMP; Dose-Response Relationship, Drug; Female; Indoleacetic Acids; Male; Mice; Motor Activity; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Cholecystokinin; Thiazoles | 1993 |
Electrophysiological studies of the cholecystokininA receptor antagonists SR27897B and PD140548 in the rat isolated nodose ganglion.
Topics: Animals; Dose-Response Relationship, Drug; Electrophysiology; Hormone Antagonists; Indoleacetic Acids; Nodose Ganglion; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Thiazoles | 1996 |
Electrophysiological evidence for the implication of cholecystokinin in the modulation of the N-methyl-D-aspartate response by sigma ligands in the rat CA3 dorsal hippocampus.
Topics: Animals; Cholecystokinin; Cinnamates; Cyclopropanes; Drug Synergism; Electrophysiology; Hippocampus; Hormone Antagonists; Indoleacetic Acids; Male; N-Methylaspartate; Pentazocine; Rats; Rats, Sprague-Dawley; Receptors, sigma; Sincalide; Thiazoles | 1996 |
The effects of cholecystokinin A and B receptor antagonists on exploratory behaviour in the elevated zero-maze in rat.
Topics: Animals; Behavior, Animal; Benzodiazepinones; Devazepide; Dose-Response Relationship, Drug; Exploratory Behavior; Female; Hormone Antagonists; Indoleacetic Acids; Maze Learning; Rats; Rats, Wistar; Receptors, Cholecystokinin; Thiazoles | 1997 |
Effects of the CCK(A) receptor antagonists SR 27897B and PD140548 on baroreflex function in conscious rats.
Topics: Animals; Baroreflex; Blood Pressure; Heart Rate; Hormone Antagonists; Indoleacetic Acids; Indoles; Male; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Thiazoles | 1997 |
SR146131: a new potent, orally active, and selective nonpeptide cholecystokinin subtype 1 receptor agonist. I. In vitro studies.
Topics: 3T3 Cells; Animals; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; CHO Cells; Cricetinae; Devazepide; DNA-Binding Proteins; Early Growth Response Protein 1; Genes, Immediate-Early; Hormone Antagonists; Humans; Immediate-Early Proteins; Indoleacetic Acids; Indoles; Inosine Monophosphate; Mice; Neuroblastoma; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Recombinant Proteins; Sincalide; Thiazoles; Transcription Factors; Tumor Cells, Cultured | 1999 |
Analysis of the behaviour of selected CCKB/gastrin receptor antagonists in radioligand binding assays performed in mouse and rat cerebral cortex.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Binding Sites; Binding, Competitive; Bridged-Ring Compounds; Cerebral Cortex; Dipeptides; Guinea Pigs; Hormone Antagonists; Indoleacetic Acids; Indoles; Iodine Radioisotopes; Male; Meglumine; Mice; Pancreas; Phenylurea Compounds; Radioligand Assay; Rats; Rats, Wistar; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Sincalide; Succinimides; Thiazoles; Tritium | 1999 |
Exogenous CCK and gastrin stimulate pancreatic exocrine secretion via CCK-A but also via CCK-B/gastrin receptors in the calf.
Topics: Animals; Cattle; Cholecystokinin; Gastrins; In Vitro Techniques; Indoleacetic Acids; Indoles; Male; Meglumine; Pancreas; Pancreatic Juice; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Stimulation, Chemical; Thiazoles | 1999 |
Contrasting roles of leu(356) in the human CCK(1) receptor for antagonist SR 27897 and agonist SR 146131 binding.
Topics: Animals; Binding Sites; COS Cells; Hormone Antagonists; Humans; Indoleacetic Acids; Indoles; Leucine; Point Mutation; Receptors, Cholecystokinin; Sincalide; Thiazoles | 1999 |
Arginine 197 of the cholecystokinin-A receptor binding site interacts with the sulfate of the peptide agonist cholecystokinin.
Topics: Amino Acid Sequence; Amino Acid Substitution; Animals; Arginine; Binding Sites; Cholecystokinin; Computer Simulation; COS Cells; Humans; Indoleacetic Acids; Inositol Phosphates; Iodine Radioisotopes; Kinetics; Models, Molecular; Mutagenesis, Site-Directed; Protein Conformation; Radioligand Assay; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Recombinant Proteins; Thiazoles; Transfection; Tritium | 1999 |
Opposite modulation of apomorphine- or amphetamine-induced stereotypy by antagonists of CCK receptors.
Topics: Amphetamine; Animals; Apomorphine; Benzodiazepinones; Dopamine; Indoleacetic Acids; Male; Phenylurea Compounds; Rats; Rats, Wistar; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Stereotyped Behavior; Thiazoles | 2000 |
Essential role of extracellular charged residues of the human CCK(1) receptor for interactions with SR 146131, SR 27897 and CCK-8S.
Topics: Amino Acid Sequence; Animals; COS Cells; Dose-Response Relationship, Drug; Humans; Indoleacetic Acids; Indoles; Inositol Phosphates; Molecular Sequence Data; Mutation; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Sincalide; Structure-Activity Relationship; Thiazoles | 2000 |
Inhibition of the hypothalamic-pituitary-adrenal axis in food-deprived rats by a CCK-A receptor antagonist.
Topics: Adrenocorticotropic Hormone; Animals; Benzodiazepinones; Corticosterone; Eating; Food Deprivation; Hormone Antagonists; Hypothalamo-Hypophyseal System; Indoleacetic Acids; Male; Phenylurea Compounds; Pituitary-Adrenal System; Rats; Rats, Wistar; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Thiazoles | 2000 |
The agonist SR 146131 and the antagonist SR 27897 occupy different sites on the human CCK(1) receptor.
Topics: Amino Acid Sequence; Animals; Binding Sites; Binding, Competitive; COS Cells; Hormone Antagonists; Humans; Indoleacetic Acids; Indoles; Models, Molecular; Molecular Sequence Data; Mutagenesis, Site-Directed; Point Mutation; Protein Conformation; Protein Structure, Tertiary; Receptors, Cholecystokinin; Thiazoles | 2000 |
Pancreatic secretory response to feeding in the calf: CCK-A receptors, but not CCK-B/gastrin receptors are involved.
Topics: Animals; Cattle; Cholecystokinin; Eating; Gastrins; Hormone Antagonists; Indoleacetic Acids; Male; Pancreas; Pancreatic Juice; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Secretin; Thiazoles; Trypsin | 2000 |
Pharmacological and molecular characterization of muscular cholecystokinin receptors in the human lower oesophageal sphincter.
Topics: Adult; Aged; Benzodiazepines; Benzodiazepinones; Esophagogastric Junction; Female; Gastric Emptying; Gastrins; Gastrointestinal Agents; Gene Expression; Hormone Antagonists; Humans; In Vitro Techniques; Indoleacetic Acids; Male; Middle Aged; Phenylurea Compounds; Proglumide; Receptors, Cholecystokinin; Restriction Mapping; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sincalide; Thiazoles | 2000 |
Pharmacological evidence for putative CCK(1) receptor heterogeneity in human colon smooth muscle.
Topics: Aspartic Acid; Binding Sites; Binding, Competitive; Colon; Devazepide; Diazepam; Gallbladder; Humans; Indoleacetic Acids; Kinetics; Membranes; Models, Biological; Muscle, Smooth; Naphthalenesulfonates; Organ Culture Techniques; Organ Specificity; Protease Inhibitors; Radioligand Assay; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Thiazoles; Time Factors | 2002 |
Characterization of the role of endogenous cholecystokinin on the activity of the paraventricular nucleus of the hypothalamus in rats.
Topics: Animals; Cholecystokinin; Food Deprivation; Genes, fos; Indoleacetic Acids; Male; Paraventricular Hypothalamic Nucleus; Rats; Rats, Wistar; Receptors, Cholecystokinin; Thiazoles | 2003 |
Regulation of leptin distribution between plasma and cerebrospinal fluid by cholecystokinin receptors.
Topics: Animals; Benzodiazepinones; Blood Glucose; Cholecystokinin; Eating; Fasting; Indoleacetic Acids; Injections, Intraperitoneal; Injections, Subcutaneous; Insulin; Leptin; Male; Phenylurea Compounds; Rats; Rats, Wistar; Receptors, Cholecystokinin; Thiazoles; Tissue Distribution | 2003 |
The role of luminal gastrin in the regulation of pancreatic juice secretion in preruminant calves.
Topics: Animals; Anti-Anxiety Agents; Cattle; Cholecystokinin; Duodenum; Gastrins; Gastrointestinal Motility; Hormone Antagonists; Indoleacetic Acids; Indoles; Infusion Pumps; Infusions, Parenteral; Meglumine; Pancreas; Peptide Fragments; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Thiazoles | 2004 |
Modeled structure of a G-protein-coupled receptor: the cholecystokinin-1 receptor.
Topics: Amino Acid Motifs; Amino Acid Sequence; Animals; Benzodiazepinones; Binding Sites; Chlorocebus aethiops; Cholecystokinin; COS Cells; Devazepide; Humans; Indoleacetic Acids; Indoles; Ligands; Lipid Metabolism; Lipids; Magnetic Resonance Spectroscopy; Models, Molecular; Molecular Sequence Data; Mutagenesis, Site-Directed; Phenylurea Compounds; Protein Conformation; Receptor, Cholecystokinin A; Rhodopsin; Sequence Homology, Amino Acid; Thiazoles | 2005 |
A cholecystokinin-1 receptor agonist (CCK-8) mediates increased permeability of brain barriers to leptin.
Topics: Animals; Benzodiazepinones; Blood Glucose; Blood-Brain Barrier; Cell Membrane Permeability; Eating; Indoleacetic Acids; Injections, Intraperitoneal; Insulin; Kinetics; Leptin; Male; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Recombinant Proteins; Sincalide; Thiazoles | 2008 |
Characteristics of the cholecystokinin-induced depolarization of pacemaking activity in cultured interstitial cells of Cajal from murine small intestine.
Topics: Animals; Cells, Cultured; Chemokines, CC; Cholecystokinin; Cyclic AMP-Dependent Protein Kinases; Estrenes; Gastrins; Indoleacetic Acids; Interstitial Cells of Cajal; Intestine, Small; Membrane Potentials; Mice; Mice, Inbred BALB C; Patch-Clamp Techniques; Protein Kinase C; Pyrrolidinones; Quinazolinones; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Thiazoles; TRPC Cation Channels; Type C Phospholipases | 2013 |
Expression analysis of a cholecystokinin system in human and rat white adipose tissue.
Topics: Adipocytes; Adipose Tissue, White; Animals; Benzodiazepinones; Cholecystokinin; Gene Expression Regulation; Gene Silencing; Humans; Indoleacetic Acids; Male; Mesenchymal Stem Cells; Oncogene Protein v-akt; Phenylurea Compounds; Phosphorylation; Rats; Rats, Wistar; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Thiazoles | 2018 |
Structures of the human cholecystokinin receptors bound to agonists and antagonists.
Topics: Amino Acid Sequence; Cryoelectron Microscopy; Crystallization; Devazepide; Humans; Indoleacetic Acids; Ligands; Models, Molecular; Protein Binding; Protein Conformation; Receptors, Cholecystokinin; Structure-Activity Relationship; Thiazoles | 2021 |