Page last updated: 2024-08-21

thiazoles and saracatinib

thiazoles has been researched along with saracatinib in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (15.38)29.6817
2010's11 (84.62)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gautschi, O; Lee, D1
Saad, F1
Botta, M; Brullo, C; Musumeci, F; Schenone, S2
Dempke, W; Zippel, R1
Eadens, M; Messersmith, W; Puls, LN1
Bareford, MD; Cruickshanks, N; Dai, Y; Dent, P; Grant, S; Hamed, HA; Hubbard, N; Mitchell, C; Tang, Y; Tye, G; Yacoub, A1
Knecht, R; Kurzweg, T; Laban, S; Möckelmann, N1
de Wispelaere, M; LaCroix, AJ; Yang, PL1
Dai, B; Fang, B; Gao, W; Hofstetter, WL; Lu, H; Meng, J; Minna, J; Roth, JA; Swisher, SG; Wang, L; Wu, S1
Barth, C; Massard, C; Vignot, S1
Cho, H; Gray, NS; Liu, S; Vetter, ML; Wang, J; Yang, PL; Zhang, J; Zhang, W; Zhang, Z1
Abad, S; Auladell, C; Beas-Zarate, C; Camins, A; Ettcheto, M; Folch, J; García, ML; Olloquequi, J; Petrov, D; Sánchez-López, E1

Reviews

9 review(s) available for thiazoles and saracatinib

ArticleYear
Clinical development of SRC tyrosine kinase inhibitors in lung cancer.
    Clinical lung cancer, 2006, Volume: 7, Issue:6

    Topics: Benzodioxoles; Clinical Trials, Phase I as Topic; Dasatinib; Drug Evaluation, Preclinical; Humans; Lung Neoplasms; Protein Kinase Inhibitors; Pyrimidines; Quinazolines; Receptor Protein-Tyrosine Kinases; src-Family Kinases; Thiazoles

2006
Src as a therapeutic target in men with prostate cancer and bone metastases.
    BJU international, 2009, Volume: 103, Issue:4

    Topics: Antineoplastic Agents; Benzodioxoles; Bone Neoplasms; Dasatinib; Humans; Male; Prostatic Neoplasms; Protein Kinase Inhibitors; Proto-Oncogene Mas; Pyrimidines; Quinazolines; Receptors, Androgen; src-Family Kinases; Thiazoles

2009
Novel dual Src/Abl inhibitors for hematologic and solid malignancies.
    Expert opinion on investigational drugs, 2010, Volume: 19, Issue:8

    Topics: Aniline Compounds; Animals; Antineoplastic Agents; Benzodioxoles; Clinical Trials as Topic; CSK Tyrosine-Protein Kinase; Dasatinib; Dogs; Drug Evaluation, Preclinical; Fusion Proteins, bcr-abl; Hematologic Neoplasms; Humans; Mice; Mice, Knockout; Mice, Nude; Mice, SCID; Neoplasms; Nitriles; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines; Quinazolines; Quinolines; Rats; src-Family Kinases; Thiazoles; Triazines

2010
[SRC kinases in tumor therapy].
    Medizinische Klinik (Munich, Germany : 1983), 2010, Volume: 105, Issue:10

    Topics: Aniline Compounds; Benzodioxoles; Cell Physiological Phenomena; Cell Transformation, Neoplastic; Clinical Trials, Phase II as Topic; Dasatinib; Disease Progression; DNA Mutational Analysis; Drug Delivery Systems; Enzyme Activation; Humans; Neoplasms; Nitriles; Protein Kinase Inhibitors; Proto-Oncogene Mas; Pyrimidines; Quinazolines; Quinolines; src-Family Kinases; Thiazoles

2010
Current status of SRC inhibitors in solid tumor malignancies.
    The oncologist, 2011, Volume: 16, Issue:5

    Topics: Aniline Compounds; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Benzodioxoles; Clinical Trials as Topic; Dasatinib; Dose-Response Relationship, Drug; Humans; Neoplasms; Nitriles; Protein Kinase Inhibitors; Pyrimidines; Quinazolines; Quinolines; src-Family Kinases; Thiazoles

2011
Current treatment options for recurrent/metastatic head and neck cancer: a post-ASCO 2011 update and review of last year's literature.
    European archives of oto-rhino-laryngology : official journal of the European Federation of Oto-Rhino-Laryngological Societies (EUFOS) : affiliated with the German Society for Oto-Rhino-Laryngology - Head and Neck Surgery, 2012, Volume: 269, Issue:10

    Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzodioxoles; Carcinoma, Squamous Cell; Cetuximab; Combined Modality Therapy; Dasatinib; ErbB Receptors; Fluorouracil; Gefitinib; Head and Neck Neoplasms; Humans; Indoles; Neoplasm Recurrence, Local; Palliative Care; Pyrimidines; Pyrroles; Quinazolines; Quinazolinones; Salvage Therapy; Squamous Cell Carcinoma of Head and Neck; Sunitinib; Thiazoles

2012
An update on dual Src/Abl inhibitors.
    Future medicinal chemistry, 2012, Volume: 4, Issue:6

    Topics: Aniline Compounds; Animals; Antineoplastic Agents; Benzodioxoles; Dasatinib; Fusion Proteins, bcr-abl; Humans; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Models, Molecular; Nitriles; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-abl; Pyrimidines; Quinazolines; Quinolines; src-Family Kinases; Thiazoles

2012
[Bone targeted therapies: new agents].
    Bulletin du cancer, 2013, Volume: 100, Issue:11

    Topics: Aniline Compounds; Benzodioxoles; Bone Density Conservation Agents; Bone Resorption; Cathepsin K; Dasatinib; Diphosphonates; Humans; Molecular Targeted Therapy; Nitriles; Parathyroid Hormone-Related Protein; Pyrimidines; Quinazolines; Quinolines; RANK Ligand; Receptors, Chemokine; src-Family Kinases; Thiazoles; Transforming Growth Factor beta1

2013
Current Research Therapeutic Strategies for Alzheimer's Disease Treatment.
    Neural plasticity, 2016, Volume: 2016

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Animals; Benzamides; Benzodioxoles; Brain; Disease Models, Animal; Humans; Mice; Neurons; Piperidines; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-fyn; PrPC Proteins; Pyridines; Quinazolines; Receptor, Metabotropic Glutamate 5; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Synapses; Thiazoles

2016

Other Studies

4 other study(ies) available for thiazoles and saracatinib

ArticleYear
Simultaneous exposure of transformed cells to SRC family inhibitors and CHK1 inhibitors causes cell death.
    Cancer biology & therapy, 2011, Aug-01, Volume: 12, Issue:3

    Topics: Animals; bcl-2 Homologous Antagonist-Killer Protein; bcl-2-Associated X Protein; bcl-X Protein; Benzimidazoles; Benzodioxoles; Breast Neoplasms; Cell Death; Cell Line, Transformed; Cell Transformation, Neoplastic; Checkpoint Kinase 1; Dasatinib; Female; Fibroblasts; Humans; MAP Kinase Kinase 1; MAP Kinase Kinase 2; Mice; Protease Inhibitors; Protein Kinases; Proto-Oncogene Proteins c-fyn; Proto-Oncogene Proteins c-yes; Pyrimidines; Quinazolines; Radiation Tolerance; src-Family Kinases; Thiazoles

2011
The small molecules AZD0530 and dasatinib inhibit dengue virus RNA replication via Fyn kinase.
    Journal of virology, 2013, Volume: 87, Issue:13

    Topics: Antibodies, Monoclonal; Benzodioxoles; Blotting, Northern; Blotting, Western; Cell Survival; Dasatinib; Dengue Virus; Dimethyl Sulfoxide; DNA Primers; HEK293 Cells; Humans; Mycophenolic Acid; Polymerase Chain Reaction; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-fyn; Pyrimidines; Quinazolines; Replicon; RNA Interference; RNA, Viral; Thiazoles; Virus Replication

2013
IGFBP2/FAK pathway is causally associated with dasatinib resistance in non-small cell lung cancer cells.
    Molecular cancer therapeutics, 2013, Volume: 12, Issue:12

    Topics: Animals; Antineoplastic Agents; Benzodioxoles; Carcinoma, Non-Small-Cell Lung; Cell Line, Tumor; Dasatinib; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Resistance, Neoplasm; Enzyme Activation; Female; Focal Adhesion Protein-Tyrosine Kinases; Gene Expression; Humans; Inhibitory Concentration 50; Insulin-Like Growth Factor Binding Protein 2; Lung Neoplasms; Mice; Mutation; Phosphorylation; Protein Kinase Inhibitors; Pyrimidines; Quinazolines; Signal Transduction; Thiazoles; Xenograft Model Antitumor Assays

2013
Fluorescent visualization of Src by using dasatinib-BODIPY.
    Chembiochem : a European journal of chemical biology, 2014, Jun-16, Volume: 15, Issue:9

    Topics: Animals; Benzodioxoles; Boron Compounds; Cell Line; Cell Proliferation; Cell Survival; Dasatinib; Dose-Response Relationship, Drug; Fluorescence; Humans; Mice; Microscopy, Fluorescence; Molecular Probes; Molecular Structure; Protein Kinase Inhibitors; Pyrimidines; Quinazolines; src-Family Kinases; Structure-Activity Relationship; Thiazoles

2014