Page last updated: 2024-08-21

thiazoles and ro 41-1049

thiazoles has been researched along with ro 41-1049 in 44 studies

Research

Studies (44)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's32 (72.73)18.2507
2000's11 (25.00)29.6817
2010's1 (2.27)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fernandes, MH; Pestana, M; Soares-da-Silva, P1
Cesura, AM; Colzi, A; d'Agostini, F; Da Prada, M1
Da Prada, M; Richards, JG; Saura, J; Ulrich, J1
Da Prada, M; Kettler, R; Richards, JG; Saura, J1
Fernandes, MH; Soares-da-Silva, P2
Cesura, AM; Da Prada, M; Imhof, R; Lang, G; Muggli-Maniglio, D1
Da Prada, M; Kettler, R; Richards, JG; Saura Marti, J1
Borroni, E; Colzi, A; d'Agostini, F; Da Prada, M; Kettler, R1
Cesura, AM; Da Prada, M; Imhof, R; Keller, HH; Kettler, R; Kyburz, E; Muggli-Maniglio, D; Richards, JG; Saura Marti, J; Wyss, PC1
Bös, M; Cesura, AM; Da Prada, M; Galva, MD; Imhof, R1
Cesura, AM; Chan-Palay, V; Da Prada, M; Huber, G; Löffler, J; Luque, JM; Richards, JG; Saura, J1
Pestana, M; Soares-da-Silva, P1
Brannan, T; Prikhojan, A; Yahr, MD1
Fernandes, MH; Soares-da-Silva, P; Vieira-Coelho, MA1
García-Sevilla, JA; Miralles, A; Olmos, G; Ribas, C1
Bryan-Lluka, LJ; Westwood, NN1
Escriba, PV; Gabilondo, AM; García-Sevilla, JA; Miralles, A; Olmos, G1
García-Sevilla, JA; Sastre, M1
Abell, CW; Da Prada, M; Kwan, SW; Luque, JM; Richards, JG1
Bombi, JA; Mahy, N; Nadal, E; Saura, J; van den Berg, B; Vila, M1
Bleuel, Z; Chen, K; Da Prada, M; Malherbe, P; Mendelowitsch, A; Richards, JG; Saura, J; Shih, JC; Ulrich, J1
Boronat, MA; García-Sevilla, JA; Lizcano, JM; Olmos, G; Ozaita, A; Unzeta, M1
d'Agostini, F; Damsma, G; DaPrada, M; DeBoer, P; Heeringa, MJ1
Guimarães, JT; Soares-Da-Silva, P2
Cesura, AM; Da Prada, M; Gottowik, J; Lang, G; Malherbe, P1
Gundlach, AL; Hosseini, AR; Iakovidis, D; Jackman, GP; King, PR; Louis, WJ; Nero, TL; Suzuki, S1
Gundlach, AL; Hosseini, AR; Jackman, GP; King, PR; Louis, WJ1
Gundlach, AL; King, PR; Louis, WJ1
Balraj, EK; Dilley, GE; Farley, JT; Klimek, V; Meltzer, HY; Ordway, GA; Overholser, JC; Stockmeier, CA1
Mukherjee, J; Yang, ZY1
Alper, RH; Gilliland, SL; Levant, B1
Archer, T; Fredriksson, A; Palomo, T1
Ahlgren-Beckendorf, JA; Chen, K; Grandy, DK; Levant, B; Morgan, KA; Seif, I; Shih, JC1
Culver, KE; Szechtman, H1
Asensio, VJ; Esteban, S; García-Sevilla, JA; Miralles, A; Moranta, D; Sastre-Coll, A1
Anderson, NJ; Hudson, AL; Lupo, PA; Nutt, DJ; Robinson, ES1
Anderson, NJ; Hudson, AL; Husbands, SM; Nutt, DJ; Robinson, ES; Tyacke, RJ1
Anderson, NJ; Hudson, AL; Nutt, DJ; Robinson, ES; Seif, I1
Auge, N; Coatrieux, C; Hannun, Y; Itohara, S; Negre-Salvayre, A; Parini, A; Salvayre, R; Sanson, M1
Culver, KE; Levant, B; Szechtman, H1
Cao, X; Li, XM; Mousseau, DD1
García-Fuster, MJ; García-Sevilla, JA1

Reviews

1 review(s) available for thiazoles and ro 41-1049

ArticleYear
From moclobemide to Ro 19-6327 and Ro 41-1049: the development of a new class of reversible, selective MAO-A and MAO-B inhibitors.
    Journal of neural transmission. Supplementum, 1990, Volume: 29

    Topics: Animals; Benzamides; Brain; Enzyme Inhibitors; Moclobemide; Monoamine Oxidase; Picolinic Acids; Rats; Thiazoles

1990

Other Studies

43 other study(ies) available for thiazoles and ro 41-1049

ArticleYear
Deamination of newly-formed dopamine in rat renal tissues.
    British journal of pharmacology, 1991, Volume: 102, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Deamination; Dopamine; In Vitro Techniques; Kidney; Levodopa; Male; Pargyline; Picolinic Acids; Rats; Rats, Wistar; Thiazoles

1991
Brain microdialysis in rats: a technique to reveal competition in vivo between endogenous dopamine and moclobemide, a RIMA antidepressant.
    Psychopharmacology, 1992, Volume: 106 Suppl

    Topics: 2H-Benzo(a)quinolizin-2-ol, 2-Ethyl-1,3,4,6,7,11b-hexahydro-3-isobutyl-9,10-dimethoxy-; 3,4-Dihydroxyphenylacetic Acid; Animals; Benzamides; Binding, Competitive; Brain Chemistry; Dialysis; Dopamine; Male; Moclobemide; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Neurons; Rats; Rats, Inbred Strains; Thiazoles

1992
Molecular neuroanatomy of monoamine oxidases in human brainstem.
    Psychopharmacology, 1992, Volume: 106 Suppl

    Topics: Aged; Autoradiography; Brain Stem; Chromosome Mapping; Female; Humans; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Nucleic Acid Hybridization; Oligonucleotide Probes; Picolinic Acids; RNA, Messenger; Thiazoles

1992
Quantitative enzyme radioautography with 3H-Ro 41-1049 and 3H-Ro 19-6327 in vitro: localization and abundance of MAO-A and MAO-B in rat CNS, peripheral organs, and human brain.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1992, Volume: 12, Issue:5

    Topics: Animals; Autoradiography; Binding Sites; Brain; Central Nervous System; Humans; Isoenzymes; Kinetics; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Picolinic Acids; Rats; Thiazoles; Tissue Distribution; Tritium

1992
Role of monoamine oxidase A and B in the deamination of newly-formed dopamine in the rat kidney.
    Journal of neural transmission. Supplementum, 1990, Volume: 32

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Deamination; Dopamine; In Vitro Techniques; Kidney; Levodopa; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Picolinic Acids; Rats; Rats, Inbred Strains; Thiazoles

1990
Monoamine oxidase inhibition by moclobemide and 2-amino-ethyl carboxamide derivatives: mode of action and kinetic characteristics.
    Journal of neural transmission. Supplementum, 1990, Volume: 32

    Topics: Animals; Benzamides; Blood Platelets; Brain; Cell Membrane; Female; Humans; In Vitro Techniques; Kinetics; Moclobemide; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Picolinic Acids; Placenta; Pregnancy; Rats; Thiazoles

1990
Molecular neuroanatomy of MAO-A and MAO-B.
    Journal of neural transmission. Supplementum, 1990, Volume: 32

    Topics: Animals; Autoradiography; Brain; Histocytochemistry; Humans; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Nervous System; Nucleic Acid Hybridization; Picolinic Acids; Rats; Thiazoles

1990
Effect of selective and reversible MAO inhibitors on dopamine outflow in rat striatum: a microdialysis study.
    Journal of neural transmission. Supplementum, 1990, Volume: 32

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Benzamides; Corpus Striatum; Deamination; Dialysis; Dopamine; Homovanillic Acid; Male; Moclobemide; Monoamine Oxidase Inhibitors; Picolinic Acids; Rats; Rats, Inbred Strains; Thiazoles

1990
Effects of MAO-A and MAO-B selective inhibitors Ro 41-1049 and Ro 19-6327 on the deamination of newly formed dopamine in the rat kidney.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 255, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Dihydroxyphenylalanine; Dopamine; Isoenzymes; Kidney; Kinetics; Male; Monoamine Oxidase Inhibitors; Norepinephrine; Picolinic Acids; Rats; Rats, Inbred Strains; Thiazoles

1990
Characterization of the binding of [3H]Ro 41-1049 to the active site of human monoamine oxidase-A.
    Molecular pharmacology, 1990, Volume: 37, Issue:3

    Topics: Affinity Labels; Binding Sites; Binding, Competitive; Cerebral Cortex; Chromatography, High Pressure Liquid; Humans; In Vitro Techniques; Molecular Weight; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Placenta; Structure-Activity Relationship; Thiazoles; Trypsin

1990
Increased monoamine oxidase B activity in plaque-associated astrocytes of Alzheimer brains revealed by quantitative enzyme radioautography.
    Neuroscience, 1994, Volume: 62, Issue:1

    Topics: Aged; Aged, 80 and over; Alzheimer Disease; Astrocytes; Autoradiography; Brain; Female; Humans; Image Processing, Computer-Assisted; Immunohistochemistry; Isoquinolines; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Picolinic Acids; Thiazoles

1994
Effect of type A and B monoamine oxidase selective inhibition by Ro 41-1049 and Ro 19-6327 on dopamine outflow in rat kidney slices.
    British journal of pharmacology, 1994, Volume: 113, Issue:4

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Benserazide; Dopamine; In Vitro Techniques; Isoenzymes; Kidney Cortex; Levodopa; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Pargyline; Picolinic Acids; Rats; Rats, Wistar; Thiazoles

1994
Effect of a selective MAO-A inhibitor (Ro 41-1049) on striatal L-dopa and dopamine metabolism: an in vivo study.
    Journal of neural transmission. Parkinson's disease and dementia section, 1994, Volume: 8, Issue:1-2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Catechols; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Levodopa; Male; Monoamine Oxidase Inhibitors; Rats; Rats, Sprague-Dawley; Thiazoles

1994
In vivo effects of the monoamine oxidase inhibitors Ro 41-1049 and Ro 19-6327 on the production and fate of renal dopamine.
    Journal of neural transmission. Supplementum, 1994, Volume: 41

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Dopamine; Kidney; Levodopa; Male; Monoamine Oxidase Inhibitors; Picolinic Acids; Rats; Rats, Wistar; Thiazoles; Tissue Distribution

1994
Differential effects of the alkylating agent N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline on brain alpha 2-adrenoceptors and I2-imidazoline sites in vitro and in vivo.
    Journal of neurochemistry, 1993, Volume: 61, Issue:5

    Topics: Animals; Binding Sites; Brain; Cell Membrane; Dioxanes; Idazoxan; Imidazoles; Isoenzymes; Kinetics; Male; Monoamine Oxidase; Neurons; Picolinic Acids; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Thermodynamics; Thiazoles; Tritium

1993
Types A and B monoamine oxidase contribute to the metabolism of norepinephrine in perfused lungs of rats.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 267, Issue:2

    Topics: Animals; Deamination; Female; In Vitro Techniques; Isoenzymes; Kinetics; Lung; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Norepinephrine; Perfusion; Picolinic Acids; Rats; Rats, Wistar; Thiazoles; Vas Deferens

1993
Chronic treatment with the monoamine oxidase inhibitors clorgyline and pargyline down-regulates non-adrenoceptor [3H]-idazoxan binding sites in the rat brain.
    British journal of pharmacology, 1993, Volume: 108, Issue:3

    Topics: Animals; Binding, Competitive; Brain Chemistry; Cerebral Cortex; Clorgyline; Dioxanes; Down-Regulation; Idazoxan; In Vitro Techniques; Male; Monoamine Oxidase Inhibitors; Pargyline; Psychotropic Drugs; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Receptors, Drug; Thiazoles

1993
Opposite age-dependent changes of alpha 2A-adrenoceptors and nonadrenoceptor [3H]idazoxan binding sites (I2-imidazoline sites) in the human brain: strong correlation of I2 with monoamine oxidase-B sites.
    Journal of neurochemistry, 1993, Volume: 61, Issue:3

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Aging; Binding Sites; Brain; Child; Child, Preschool; Dioxanes; Female; Humans; Idazoxan; Imidazoline Receptors; Male; Middle Aged; Monoamine Oxidase; Picolinic Acids; Receptors, Adrenergic, alpha; Receptors, Drug; Thiazoles

1993
Cellular expression of mRNAs encoding monoamine oxidases A and B in the rat central nervous system.
    The Journal of comparative neurology, 1995, Dec-25, Volume: 363, Issue:4

    Topics: Animals; Autoradiography; Biomarkers; Central Nervous System; Histamine; Immunohistochemistry; In Situ Hybridization; Isoenzymes; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Oligonucleotide Probes; Picolinic Acids; Rats; RNA, Messenger; Sulfur Radioisotopes; Thiazoles

1995
Localization of monoamine oxidases in human peripheral tissues.
    Life sciences, 1996, Volume: 59, Issue:16

    Topics: Aged; Aged, 80 and over; Autoradiography; Duodenum; Humans; Isoenzymes; Kidney; Liver; Lung; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Myocardium; Picolinic Acids; Receptors, Adrenergic, beta; Spleen; Thiazoles

1996
Molecular neuroanatomy of human monoamine oxidases A and B revealed by quantitative enzyme radioautography and in situ hybridization histochemistry.
    Neuroscience, 1996, Volume: 70, Issue:3

    Topics: Aged; Aged, 80 and over; Autoradiography; Brain; Female; Histocytochemistry; Humans; In Situ Hybridization; Male; Middle Aged; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Picolinic Acids; Thiazoles

1996
Inhibition of monoamine oxidase A and B activities by imidazol(ine)/guanidine drugs, nature of the interaction and distinction from I2-imidazoline receptors in rat liver.
    British journal of pharmacology, 1997, Volume: 121, Issue:5

    Topics: Animals; Clonidine; Guanidines; Imidazoles; Imidazoline Receptors; Isoenzymes; Kinetics; Liver; Male; Mitochondria, Liver; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Picolinic Acids; Rats; Rats, Sprague-Dawley; Receptors, Drug; Thiazoles

1997
Effect of monoamine oxidase A and B and of catechol-O-methyltransferase inhibition on L-DOPA-induced circling behavior.
    Journal of neural transmission (Vienna, Austria : 1996), 1997, Volume: 104, Issue:6-7

    Topics: Animals; Antiparkinson Agents; Benzophenones; Catechol O-Methyltransferase Inhibitors; Enzyme Inhibitors; Levodopa; Male; Monoamine Oxidase Inhibitors; Motor Activity; Nitrophenols; Oxidopamine; Picolinic Acids; Rats; Rotation; Thiazoles; Tolcapone

1997
Unusual pattern of beta-phenylethylamine deamination in the rat heart.
    Biochemical Society transactions, 1997, Volume: 25, Issue:4

    Topics: Animals; Isoenzymes; Kidney Cortex; Kinetics; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Myocardium; Phenethylamines; Picolinic Acids; Psychotropic Drugs; Rats; Rats, Wistar; Serotonin; Substrate Specificity; Thiazoles

1997
The activity of MAO A and B in rat renal cells and tubules.
    Life sciences, 1998, Volume: 62, Issue:8

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Dopamine; Kidney; Kidney Tubules; Kinetics; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Picolinic Acids; Rats; Rats, Wistar; Thiazoles

1998
Structure-function relationships of mitochondrial monoamine oxidase A and B: chimaeric enzymes and site-directed mutagenesis studies.
    Journal of neural transmission. Supplementum, 1998, Volume: 52

    Topics: Amino Acid Substitution; Binding Sites; Cell Line; Cloning, Molecular; Histidine; Humans; Isoenzymes; Kidney; Kinetics; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Mutagenesis, Site-Directed; Polymerase Chain Reaction; Recombinant Fusion Proteins; Thiazoles; Threonine; Transfection

1998
[3H]Rilmenidine-labelled imidazoline-receptor binding sites co-localize with [3H]2-(benzofuranyl)-2-imidazoline-labelled imidazoline-receptor binding sites and monoamine oxidase-B in rabbit, but not rat, kidney.
    Journal of the autonomic nervous system, 1998, Oct-15, Volume: 72, Issue:2-3

    Topics: Adrenergic alpha-Agonists; Animals; Autoradiography; Benzofurans; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Isoenzymes; Kidney; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Oxazoles; Picolinic Acids; Rabbits; Rats; Rats, Inbred WKY; Receptors, Drug; Rilmenidine; Species Specificity; Thiazoles

1998
Pharmacology and subcellular distribution of [3H]rilmenidine binding sites in rat brain.
    Journal of the autonomic nervous system, 1998, Oct-15, Volume: 72, Issue:2-3

    Topics: Adrenergic alpha-Agonists; Animals; Binding Sites; Brain; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Male; Membranes; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Oxazoles; Picolinic Acids; Radioligand Assay; Rats; Rats, Inbred WKY; Receptors, Drug; Rilmenidine; Subcellular Fractions; Thiazoles

1998
Identification of imidazoline-receptor binding sites in cortex and medulla of the bovine adrenal gland. Colocalization with MAO-A and MAO-B.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Adrenal Cortex; Adrenal Medulla; Adrenergic beta-Agonists; Animals; Autoradiography; Benzofurans; Binding Sites; Cattle; Clonidine; Imidazoles; Imidazoline Receptors; Isoenzymes; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Oxazoles; Picolinic Acids; Rats; Receptors, Drug; Rilmenidine; Thiazoles; Tritium

1999
Quantitative distribution of monoamine oxidase A in brainstem monoamine nuclei is normal in major depression.
    Brain research, 1999, Nov-13, Volume: 847, Issue:1

    Topics: Adult; Aged; Biogenic Monoamines; Brain Stem; Depressive Disorder; Female; Humans; Locus Coeruleus; Male; Middle Aged; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Radioligand Assay; Raphe Nuclei; Thiazoles

1999
Development of N-[3-(2',4'-dichlorophenoxy)-2-18F-fluoropropyl]-N-methylpropargylamine (18F-fluoroclorgyline) as a potential PET radiotracer for monoamine oxidase-A.
    Nuclear medicine and biology, 1999, Volume: 26, Issue:6

    Topics: Animals; Brain; Clorgyline; Fluorine Radioisotopes; Kinetics; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Selegiline; Thiazoles; Tissue Distribution; Tomography, Emission-Computed

1999
Pharmacology of quinpirole-stimulated [35S]GTPgammaS binding: discrepancy with receptor binding profile.
    European journal of pharmacology, 2000, Mar-31, Volume: 392, Issue:3

    Topics: Animals; Benzazepines; Binding, Competitive; Clorgyline; Clozapine; Corpus Striatum; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Male; Membranes; Monoamine Oxidase Inhibitors; Quinpirole; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Selegiline; Spiperone; Sulfur Radioisotopes; Thiazoles

2000
Effects of MAO inhibitors upon MPTP mice chronically treated with suprathreshold doses of L-dopa.
    Behavioural pharmacology, 2000, Volume: 11, Issue:7-8

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Behavior, Animal; Clorgyline; Corpus Striatum; Dopamine; Dopamine Agents; Dose-Response Relationship, Drug; Levodopa; Locomotion; Male; Mice; Mice, Inbred C57BL; Monoamine Oxidase Inhibitors; Motor Activity; Phenelzine; Phenethylamines; Selegiline; Thiazoles; Tryptamines

2000
Modulation of [3H]quinpirole binding at striatal D2 dopamine receptors by a monoamine oxidaseA-like site: evidence from radioligand binding studies and D2 receptor- and MAO(A)-deficient mice.
    Life sciences, 2001, Nov-30, Volume: 70, Issue:2

    Topics: Animals; Binding Sites; Corpus Striatum; Dopamine Agonists; Female; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quinpirole; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Spiperone; Thiazoles; Tritium

2001
Clorgyline-induced switch from locomotion to mouthing in sensitization to the dopamine D2/D3 agonist quinpirole in rats: role of sigma and imidazoline I2 receptors.
    Psychopharmacology, 2003, Volume: 167, Issue:2

    Topics: Animals; Behavior, Animal; Benzofurans; Clorgyline; Dopamine; Dopamine Agonists; Drug Administration Schedule; Imidazoles; Imidazoline Receptors; Injections, Subcutaneous; Ligands; Male; Monoamine Oxidase Inhibitors; Motor Activity; Quinpirole; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Drug; Receptors, sigma; Thiazoles

2003
High-affinity binding of beta-carbolines to imidazoline I2B receptors and MAO-A in rat tissues: norharman blocks the effect of morphine withdrawal on DOPA/noradrenaline synthesis in the brain.
    European journal of pharmacology, 2005, Aug-22, Volume: 518, Issue:2-3

    Topics: Animals; Benzofurans; Binding, Competitive; Brain; Carbolines; Cerebral Cortex; Dihydroxyphenylalanine; Dose-Response Relationship, Drug; Harmine; Hippocampus; Imidazoles; Imidazoline Receptors; Liver; Male; Monoamine Oxidase; Morphine; Morphine Dependence; Naloxone; Norepinephrine; Picolinic Acids; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Drug; Substance Withdrawal Syndrome; Thiazoles; Tritium; Tyrosine 3-Monooxygenase

2005
Characterisation of imidazoline I2 binding sites in pig brain.
    European journal of pharmacology, 2005, Sep-05, Volume: 519, Issue:1-2

    Topics: Animals; Benzofurans; Binding Sites; Binding, Competitive; Brain; Carbolines; Clonidine; Dose-Response Relationship, Drug; Female; Idazoxan; Imidazoles; Imidazoline Receptors; Kinetics; Male; Monoamine Oxidase Inhibitors; Picolinic Acids; Radioligand Assay; Receptors, Drug; Swine; Thiazoles; Tritium

2005
In vitro and ex vivo distribution of [3H]harmane, an endogenous beta-carboline, in rat brain.
    Neuropharmacology, 2006, Volume: 50, Issue:3

    Topics: Animals; Autoradiography; Brain; Harmine; In Vitro Techniques; Male; Monoamine Oxidase Inhibitors; Neurotoxins; Protein Binding; Radionuclide Imaging; Rats; Rats, Wistar; Receptors, Drug; Thiazoles; Tissue Distribution; Tritium

2006
Autoradiographical distribution of imidazoline binding sites in monoamine oxidase A deficient mice.
    Journal of neurochemistry, 2006, Volume: 96, Issue:6

    Topics: Animals; Autoradiography; Benzofurans; Binding Sites; Binding, Competitive; Brain; Cell Membrane; Epithelial Cells; Harmine; Idazoxan; Imidazoles; Imidazoline Receptors; Imidazolines; Iodine Radioisotopes; Kidney; Mice; Mice, Inbred C3H; Mice, Knockout; Monoamine Oxidase; Neurons; Picolinic Acids; Radioligand Assay; Receptors, Drug; Thiazoles

2006
MAO-A-induced mitogenic signaling is mediated by reactive oxygen species, MMP-2, and the sphingolipid pathway.
    Free radical biology & medicine, 2007, Jul-01, Volume: 43, Issue:1

    Topics: Animals; Biogenic Amines; Blood Vessels; Butylated Hydroxytoluene; Cell Proliferation; Free Radical Scavengers; Hydrogen Peroxide; Matrix Metalloproteinase 2; Matrix Metalloproteinase Inhibitors; Mice; Mice, Mutant Strains; Mitogens; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Myocytes, Smooth Muscle; Oxidation-Reduction; Pargyline; Phenylalanine; Rabbits; Reactive Oxygen Species; RNA, Small Interfering; Serotonin; Signal Transduction; Sphingolipids; Thiazoles; Thiophenes; Tyramine

2007
Altered dopamine D2-like receptor binding in rats with behavioral sensitization to quinpirole: effects of pre-treatment with Ro 41-1049.
    European journal of pharmacology, 2008, Sep-11, Volume: 592, Issue:1-3

    Topics: Animals; Behavior, Animal; Dopamine Agonists; Dopamine Antagonists; Kinetics; Male; Monoamine Oxidase Inhibitors; Motor Activity; Neostriatum; Nucleus Accumbens; Quinpirole; Radioligand Assay; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Spiperone; Thiazoles

2008
Calcium alters monoamine oxidase-A parameters in human cerebellar and rat glial C6 cell extracts: possible influence by distinct signalling pathways.
    Life sciences, 2009, Jul-31, Volume: 85, Issue:5-6

    Topics: Aged; Animals; Binding Sites; Calcium; Calcium Signaling; Cell Line, Tumor; Cerebellum; Gene Expression; Glioblastoma; Humans; Male; Mice; Middle Aged; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Neuroglia; Neurons; p38 Mitogen-Activated Protein Kinases; Protein Binding; Rats; RNA, Messenger; Thiazoles

2009
Effects of anti-depressant treatments on FADD and p-FADD protein in rat brain cortex: enhanced anti-apoptotic p-FADD/FADD ratio after chronic desipramine and fluoxetine administration.
    Psychopharmacology, 2016, Volume: 233, Issue:15-16

    Topics: Adrenergic alpha-Antagonists; Animals; Antidepressive Agents; Apoptosis; Autoreceptors; Blotting, Western; Brain; CASP8 and FADD-Like Apoptosis Regulating Protein; Cerebral Cortex; Clorgyline; Desipramine; Electroshock; Excitatory Amino Acid Antagonists; Fas-Associated Death Domain Protein; Fluoxetine; Idazoxan; Indans; Ketamine; Male; Mianserin; Mirtazapine; Monoamine Oxidase Inhibitors; Norepinephrine Plasma Membrane Transport Proteins; Phenelzine; Phosphoproteins; Phosphorylation; Rats; RNA-Binding Proteins; Thiazoles

2016