Page last updated: 2024-08-21

thiazoles and rifampin

thiazoles has been researched along with rifampin in 42 studies

Research

Studies (42)

TimeframeStudies, this research(%)All Research%
pre-19903 (7.14)18.7374
1990's4 (9.52)18.2507
2000's17 (40.48)29.6817
2010's18 (42.86)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ashtekar, DR; Fernandes, F; Khadse, BG; Shirodkar, MV1
Hermes, K; Ritzerfeld, W1
Hatano, M; Ishihara, M; Miura, K; Miyata, K; Okusawa, S; Shimizu, S; Yamada, T; Yoshida, A1
Furusawa, S; Nakano, S; Sasaki, K; Takayanagi, M; Takayanagi, Y; Wu, J1
Abate, G; Miörner, H; Mshana, RN; Tadesse, G1
Abate, G; Miörner, H; Mshana, RN1
Dorko, K; Esplen, JE; Komoroski, BJ; Kostrubsky, VE; Ramachandran, V; Strom, SC; Venkataramanan, R; Zhang, S1
Barros, S; Hamilton, G; Huang, SM; LeCluyse, EL; Lesko, LJ; Sahi, J; Sinz, M1
Boeddrich, A; Heiser, V; Lehrach, H; Lurz, R; Nordhoff, E; Scherzinger, E; Schugardt, N; Wanker, EE1
Lemus, D; Martin, A; Montoro, E; Palomino, JC; Portaels, F1
Boffo, MM; da Silva, PA; de Mattos, IG; Martin, A; Palomino, JC; Silva, AB; Takiff, HE1
Hirohata, M; Ono, K; Yamada, M1
Huang, JD; Lai, ML; Lu, WJ; Nezu, J; Tamai, I1
Faucette, SR; Lecluyse, EL; Negishi, M; Smith, CM; Sueyoshi, T; Wang, H1
Butler, PC; Glabe, CG; Gurlo, T; Haataja, L; Jayasinghe, S; Kayed, R; Langen, R; Lin, CY; Meier, JJ1
Anzenbacher, P; Anzenbacherova, E; Cerveny, L; Dvorak, Z; Pavek, P; Staud, F; Svecova, L; Ulrichova, J; Vrzal, R1
Antimisiaris, SG; Fadda, AM; Klepetsanis, P; Mourtas, S; Zaru, M1
Fu, M; Qu, X; Ren, J; Wang, X1
Balagopal, A; Sears, CL1
Antimisiaris, SG; Dracopoulos, V; Fadda, AM; Manca, ML; Mourtas, S1
Marek, P; Meng, F; Potter, KJ; Raleigh, DP; Verchere, CB1
Cheng, X; Li, D; Meng, Q; Shen, C1
Alvarenga, MA; Da Silva, EC; Durán, N; Marcato, PD; Melo, PS1
Boursier-Neyret, C; Cloarec, O; Croixmarie, V; Moreau, A; Pascussi, JM; Umbdenstock, T; Walther, B1
Jeong, H; Koh, KH; Yang, K1
Boursier-Neyret, C; Cloarec, O; Croixmarie, V; Moreau, A; Parmentier, Y; Pascussi, JM; Umbdenstock, T; Walther, B1
Chen, CC; Cheng, KC; Chiang, SR; Chuang, YC; Ko, WC; Su, BA; Tang, HJ; Toh, HS1
Leggio, M; Podos, SD; Pucci, MJ; Thanassi, JA1
Hirota, K; Kawamoto, T; Makino, K; Nakajima, T; Terada, H1
Hu, HH; Xu, C; Xu, SY; Yu, LS; Zeng, S1
Keirns, J; Kerbusch, V; Kowalski, D; Krauwinkel, W; Lee, J; Marion, A; Meijer, J; Moy, S; Roy, M; Sawamoto, T; Takusagawa, S; van Gelderen, M1
Chen, XY; Gao, ZW; Meng, J; Zhong, DF; Zhou, X1
Chiu, YY; Ereshefsky, L; Loebel, A; Poola, N; Preskorn, SH1
Benjaminsen, J; Fenaroli, F; Griffiths, G; Hildahl, J; Kolstad, T; Meijer, AH; Nyström, B; Roos, N; Skjeldal, FM; Ulanova, L; van der Vaart, M; Westmoreland, D1
Chen, S; Desai, M; He, L; Mendell, J; Parasramupria, DA1
Cushman, M; Hammac, GK; Mayhoub, AS; Mohammad, H; Monteleone, D; Reddy, PV; Seleem, MN1
Burk, O; Damm, G; Kandel, BA; Schwab, M; Seehofer, D; Thomas, M; Winter, S; Zanger, UM1
Inaba, M; Inouye, Y; Kanno, Y; Nakamura, S; Nemoto, K; Tanuma, N; Yazawa, S; Zhao, S1
Fattorini, L; Giannoni, F; Iacobino, A; Mustazzolu, A; Piccaro, G1
Kreiswirth, BN; Kurepina, N; Meinke, PT; Olsen, DB; Singh, SB; Xu, L; Young, K1
Aluri, J; Boyd, P; Chang, MK; Ferry, J; Lai, WG; Nomoto, M; Rege, B; Schuck, E; Siu, YA; Yasuda, S; Zamora, CA1
Goosen, TC; Lin, J; Malhotra, B; Tse, S; Yamagami, H1

Reviews

2 review(s) available for thiazoles and rifampin

ArticleYear
Clostridium difficile: new therapeutic options.
    Current opinion in pharmacology, 2007, Volume: 7, Issue:5

    Topics: Animals; Anti-Bacterial Agents; Clostridioides difficile; Clostridium Infections; Community-Acquired Infections; Depsipeptides; Diarrhea; Humans; Nitro Compounds; Polymers; Rifampin; Sulfonic Acids; Thiazoles

2007
Lurasidone drug-drug interaction studies: a comprehensive review.
    Drug metabolism and drug interactions, 2014, Volume: 29, Issue:3

    Topics: Antipsychotic Agents; Area Under Curve; Clinical Trials, Phase I as Topic; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inducers; Cytochrome P-450 CYP3A Inhibitors; Diltiazem; Drug Interactions; Drug Therapy, Combination; Humans; Isoindoles; Ketoconazole; Lithium Compounds; Lurasidone Hydrochloride; Rifampin; Thiazoles

2014

Trials

3 trial(s) available for thiazoles and rifampin

ArticleYear
Role of cytochrome p450 isoenzymes 3A and 2D6 in the in vivo metabolism of mirabegron, a β3-adrenoceptor agonist.
    Clinical drug investigation, 2013, Volume: 33, Issue:6

    Topics: Acetanilides; Adolescent; Adrenergic beta-3 Receptor Agonists; Adult; Area Under Curve; Cross-Over Studies; Cytochrome P-450 CYP2D6; Cytochrome P-450 CYP3A; Drug Interactions; Female; Half-Life; Humans; Ketoconazole; Male; Middle Aged; Rifampin; Thiazoles; Young Adult

2013
The effect of rifampin on the pharmacokinetics of edoxaban in healthy adults.
    Clinical drug investigation, 2015, Volume: 35, Issue:7

    Topics: Adult; Drug Interactions; Factor Xa Inhibitors; Female; Humans; Male; Prothrombin Time; Pyridines; Rifampin; Thiazoles

2015
Pharmacokinetic/pharmacodynamic drug-drug interactions of avatrombopag when coadministered with dual or selective CYP2C9 and CYP3A interacting drugs.
    British journal of clinical pharmacology, 2018, Volume: 84, Issue:5

    Topics: Adolescent; Adult; Cytochrome P-450 CYP2C9 Inducers; Cytochrome P-450 CYP2C9 Inhibitors; Cytochrome P-450 CYP3A Inducers; Cytochrome P-450 CYP3A Inhibitors; Drug Interactions; Female; Fluconazole; Healthy Volunteers; Humans; Itraconazole; Male; Middle Aged; Platelet Count; Receptors, Thrombopoietin; Rifampin; Thiazoles; Thiophenes; Young Adult

2018

Other Studies

37 other study(ies) available for thiazoles and rifampin

ArticleYear
A rapid method for the evaluation of new antituberculous agents.
    Chemotherapy, 1987, Volume: 33, Issue:1

    Topics: Antitubercular Agents; Carbon Dioxide; Ethambutol; Guanidines; Isoniazid; Mycobacterium tuberculosis; Pyrazinamide; Rifampin; Scintillation Counting; Streptomycin; Succinimides; Thiazoles; Time Factors

1987
[Antibiotic effect of Ciclacillin-Rifampicin combination].
    Arzneimittel-Forschung, 1971, Volume: 21, Issue:9

    Topics: Cyclohexanecarboxylic Acids; Cyclohexanes; Drug Synergism; Escherichia coli; Oxygen Consumption; Penicillanic Acid; Penicillins; Proteus; Rifampin; Staphylococcus; Thiazoles

1971
[Studies on isolated rat hepatocytes (5). Effects on platonin].
    Josai Shika Daigaku kiyo. The Bulletin of the Josai Dental University, 1983, Volume: 12, Issue:3

    Topics: Animals; Liver; Male; Rats; Rats, Inbred Strains; Rifampin; Thiazoles; Trapidil; Uncoupling Agents

1983
Potentiation of pirarubicin activity in multidrug resistant cells by rifampicin.
    Biological & pharmaceutical bulletin, 1997, Volume: 20, Issue:12

    Topics: Animals; Antibiotics, Antineoplastic; Antibiotics, Antitubercular; Apoptosis; Cell Cycle; Doxorubicin; Drug Resistance, Multiple; Drug Synergism; Gene Expression Regulation, Neoplastic; Genes, MDR; Leukemia P388; Mice; Rifampin; Tetrazolium Salts; Thiazoles

1997
Use of 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyl tetrazolium bromide for rapid detection of rifampin-resistant Mycobacterium tuberculosis.
    Journal of clinical microbiology, 1998, Volume: 36, Issue:5

    Topics: Antibiotics, Antitubercular; Colony Count, Microbial; Coloring Agents; Dose-Response Relationship, Drug; Drug Resistance, Microbial; Mycobacterium bovis; Mycobacterium tuberculosis; Rifampin; Tetrazolium Salts; Thiazoles; Tuberculosis, Multidrug-Resistant

1998
Evaluation of a colorimetric assay based on 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyl tetrazolium bromide (MTT) for rapid detection of rifampicin resistance in Mycobacterium tuberculosis.
    The international journal of tuberculosis and lung disease : the official journal of the International Union against Tuberculosis and Lung Disease, 1998, Volume: 2, Issue:12

    Topics: Antibiotics, Antitubercular; Colony Count, Microbial; Colorimetry; Drug Resistance, Microbial; Evaluation Studies as Topic; Humans; Mycobacterium tuberculosis; Rifampin; Tetrazolium Salts; Thiazoles; Tuberculosis, Multidrug-Resistant

1998
Troglitazone increases cytochrome P-450 3A protein and activity in primary cultures of human hepatocytes.
    Drug metabolism and disposition: the biological fate of chemicals, 1999, Volume: 27, Issue:10

    Topics: Aryl Hydrocarbon Hydroxylases; Cells, Cultured; Chromans; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Dose-Response Relationship, Drug; Enzyme Induction; Humans; Hypoglycemic Agents; Liver; Oxidoreductases, N-Demethylating; Rifampin; Thiazoles; Thiazolidinediones; Troglitazone

1999
Effect of troglitazone on cytochrome P450 enzymes in primary cultures of human and rat hepatocytes.
    Xenobiotica; the fate of foreign compounds in biological systems, 2000, Volume: 30, Issue:3

    Topics: Animals; Aryl Hydrocarbon Hydroxylases; Blotting, Western; Cells, Cultured; Chromans; Cytochrome P-450 CYP1A1; Cytochrome P-450 CYP1A2; Cytochrome P-450 CYP2B6; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Dexamethasone; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Activation; Enzyme Inhibitors; Glucocorticoids; Humans; Hypoglycemic Agents; Liver; Male; Microsomes, Liver; Mixed Function Oxygenases; Oxidoreductases, N-Demethylating; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; Rifampin; RNA, Messenger; Steroid Hydroxylases; Substrate Specificity; Thiazoles; Thiazolidinediones; Troglitazone

2000
Inhibition of huntingtin fibrillogenesis by specific antibodies and small molecules: implications for Huntington's disease therapy.
    Proceedings of the National Academy of Sciences of the United States of America, 2000, Jun-06, Volume: 97, Issue:12

    Topics: Animals; Antibodies, Monoclonal; Benzoates; Benzothiazoles; Biphenyl Compounds; Congo Red; COS Cells; Gossypol; Humans; Huntingtin Protein; Huntington Disease; Melatonin; Nerve Tissue Proteins; Nuclear Proteins; Peptides; Rifampin; Thiazoles

2000
Rapid alternative methods for detection of rifampicin resistance in Mycobacterium tuberculosis.
    The Journal of antimicrobial chemotherapy, 2004, Volume: 54, Issue:1

    Topics: Antibiotics, Antitubercular; Colorimetry; Culture Media; DNA-Directed RNA Polymerases; Drug Resistance, Bacterial; Humans; Indicators and Reagents; Microbial Sensitivity Tests; Mycobacterium tuberculosis; Nitrate Reductase; Nitrate Reductases; Oxazines; Oxidation-Reduction; Peru; Reagent Kits, Diagnostic; Rifampin; Tetrazolium Salts; Thiazoles; Tuberculosis; Xanthenes

2004
Comparison of redox and D29 phage methods for detection of isoniazid and rifampicin resistance in Mycobacterium tuberculosis.
    Clinical microbiology and infection : the official publication of the European Society of Clinical Microbiology and Infectious Diseases, 2006, Volume: 12, Issue:3

    Topics: Antitubercular Agents; Costs and Cost Analysis; Drug Resistance, Bacterial; Isoniazid; Microbial Sensitivity Tests; Mycobacteriophages; Mycobacterium tuberculosis; Oxazines; Oxidation-Reduction; Rifampin; Sensitivity and Specificity; Tetrazolium Salts; Thiazoles; Xanthenes

2006
Alpha-lipoic acid exhibits anti-amyloidogenicity for beta-amyloid fibrils in vitro.
    Biochemical and biophysical research communications, 2006, Mar-24, Volume: 341, Issue:4

    Topics: Amyloid; Amyloid beta-Peptides; Benzothiazoles; Masoprocol; Microscopy, Electron; Rifampin; Spectrometry, Fluorescence; Tetracycline; Thiazoles; Thioctic Acid

2006
Organic anion transporting polypeptide-C mediates arsenic uptake in HEK-293 cells.
    Journal of biomedical science, 2006, Volume: 13, Issue:4

    Topics: Arsenates; Arsenic; Arsenites; Biological Transport, Active; Cacodylic Acid; Cell Line; DNA Primers; DNA, Complementary; Estradiol; Humans; Immunoblotting; Lethal Dose 50; Liver-Specific Organic Anion Transporter 1; Reverse Transcriptase Polymerase Chain Reaction; Rifampin; Taurocholic Acid; Tetrazolium Salts; Thiazoles; Toxicity Tests; Transfection

2006
Differential regulation of hepatic CYP2B6 and CYP3A4 genes by constitutive androstane receptor but not pregnane X receptor.
    The Journal of pharmacology and experimental therapeutics, 2006, Volume: 317, Issue:3

    Topics: Aryl Hydrocarbon Hydroxylases; Base Sequence; Cell Line, Tumor; Constitutive Androstane Receptor; Cytochrome P-450 CYP2B6; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Electrophoretic Mobility Shift Assay; Gene Expression Regulation, Enzymologic; Genes, Reporter; Hepatocytes; Humans; Liver; Molecular Sequence Data; Oxidoreductases, N-Demethylating; Oximes; Pregnane X Receptor; Protein Binding; Receptor Cross-Talk; Receptors, Cytoplasmic and Nuclear; Receptors, Steroid; Reverse Transcriptase Polymerase Chain Reaction; Rifampin; Thiazoles; Transcription Factors

2006
Inhibition of human IAPP fibril formation does not prevent beta-cell death: evidence for distinct actions of oligomers and fibrils of human IAPP.
    American journal of physiology. Endocrinology and metabolism, 2006, Volume: 291, Issue:6

    Topics: Adenoviridae; Amyloid beta-Protein Precursor; Animals; Apoptosis; Benzothiazoles; Blotting, Western; Cell Death; Coloring Agents; DNA, Complementary; Fluorescent Dyes; Humans; In Situ Nick-End Labeling; Insulin-Secreting Cells; Islets of Langerhans; Propidium; Rats; Rats, Sprague-Dawley; Rifampin; Tetrazolium Salts; Thiazoles

2006
Valproic acid induces CYP3A4 and MDR1 gene expression by activation of constitutive androstane receptor and pregnane X receptor pathways.
    Drug metabolism and disposition: the biological fate of chemicals, 2007, Volume: 35, Issue:7

    Topics: Anticonvulsants; Aryl Hydrocarbon Hydroxylases; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line, Tumor; Constitutive Androstane Receptor; Cytochrome P-450 CYP2B6; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Drug Synergism; Electrophoretic Mobility Shift Assay; Enzyme Induction; Genes, Reporter; Hepatocytes; Humans; Hydroxylation; Luciferases; Oxidoreductases, N-Demethylating; Oximes; Pregnane X Receptor; Promoter Regions, Genetic; Receptors, Cytoplasmic and Nuclear; Receptors, Steroid; Retinoid X Receptor alpha; Reverse Transcriptase Polymerase Chain Reaction; Rifampin; RNA, Messenger; Testosterone; Thiazoles; Transcription Factors; Transcription, Genetic; Transcriptional Activation; Transfection; Up-Regulation; Valproic Acid

2007
Liposomes for drug delivery to the lungs by nebulization.
    European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V, 2007, Volume: 67, Issue:3

    Topics: Adhesives; Adsorption; Aerosols; Antibiotics, Antitubercular; Calorimetry, Differential Scanning; Cell Survival; Cells, Cultured; Chemistry, Pharmaceutical; Cholesterol; Drug Compounding; Drug Delivery Systems; Excipients; Freeze Drying; Humans; Liposomes; Lung; Mucous Membrane; Nebulizers and Vaporizers; Particle Size; Pulmonary Alveoli; Rifampin; Surface Properties; Tetrazolium Salts; Thermodynamics; Thiazoles

2007
Evaluation of different culture conditions for high-level soluble expression of human cyclin A2 with pET vector in BL21 (DE3) and spectroscopic characterization of its inclusion body structure.
    Protein expression and purification, 2007, Volume: 56, Issue:1

    Topics: Benzothiazoles; Chromatography, Affinity; Culture Media; Cyclin A; Cyclin A2; Escherichia coli; Genetic Vectors; Humans; Inclusion Bodies; Rifampin; Spectroscopy, Fourier Transform Infrared; Thiazoles

2007
PLGA, chitosan or chitosan-coated PLGA microparticles for alveolar delivery? A comparative study of particle stability during nebulization.
    Colloids and surfaces. B, Biointerfaces, 2008, Apr-01, Volume: 62, Issue:2

    Topics: Adhesiveness; Administration, Inhalation; Antibiotics, Antitubercular; Cell Line; Chemical Phenomena; Chemistry, Physical; Chitosan; Diffusion; Drug Compounding; Drug Delivery Systems; Drug Stability; Electrochemistry; Emulsions; Humans; Lactic Acid; Microscopy, Electron, Scanning; Microspheres; Molecular Weight; Mucins; Mucous Membrane; Nebulizers and Vaporizers; Particle Size; Polyglycolic Acid; Polylactic Acid-Polyglycolic Acid Copolymer; Polymers; Pulmonary Alveoli; Rifampin; Solvents; Tetrazolium Salts; Thiazoles

2008
Rifampicin does not prevent amyloid fibril formation by human islet amyloid polypeptide but does inhibit fibril thioflavin-T interactions: implications for mechanistic studies of beta-cell death.
    Biochemistry, 2008, Jun-03, Volume: 47, Issue:22

    Topics: Amyloid; Antioxidants; Benzothiazoles; Cell Death; Humans; Islet Amyloid Polypeptide; Islets of Langerhans; Microscopy, Electron, Transmission; Rifampin; Thiazoles

2008
Investigation of rifampicin-induced hepatotoxicity in rat hepatocytes maintained in gel entrapment culture.
    Cell biology and toxicology, 2009, Volume: 25, Issue:3

    Topics: Acetylcysteine; Albumins; Animals; Antitubercular Agents; Cell Culture Techniques; Cell Survival; Cells, Cultured; Chemical and Drug Induced Liver Injury; Cytochrome P-450 Enzyme Inhibitors; Drug Antagonism; Enzyme Inhibitors; Glutathione; Glycyrrhizic Acid; Hepatocytes; Lipid Metabolism; Male; Malondialdehyde; Oxidative Stress; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Rifampin; Tetrazolium Salts; Thiazoles

2009
Microencapsulation of antibiotic rifampicin in poly(3-hydroxybutyrate-co-3-hydroxyvalerate).
    Archives of pharmacal research, 2008, Volume: 31, Issue:11

    Topics: Animals; Antibiotics, Antitubercular; Cell Line; Cricetinae; Drug Compounding; Excipients; Microbial Sensitivity Tests; Microscopy, Electron, Scanning; Nanoparticles; Neutral Red; Nucleic Acid Synthesis Inhibitors; Particle Size; Polyesters; Rifampin; Staphylococcus aureus; Tetrazolium Salts; Thiazoles

2008
Integrated comparison of drug-related and drug-induced ultra performance liquid chromatography/mass spectrometry metabonomic profiles using human hepatocyte cultures.
    Analytical chemistry, 2009, Aug-01, Volume: 81, Issue:15

    Topics: Biomarkers; Chromatography, Liquid; Constitutive Androstane Receptor; Excitatory Amino Acid Antagonists; Hepatocytes; Humans; Mass Spectrometry; Metabolomics; Nucleic Acid Synthesis Inhibitors; Oximes; Phenobarbital; Rifampin; Thiazoles

2009
Induction of CYP2B6 and CYP3A4 expression by 1-aminobenzotriazole (ABT) in human hepatocytes.
    Drug metabolism letters, 2010, Volume: 4, Issue:3

    Topics: Aryl Hydrocarbon Hydroxylases; Constitutive Androstane Receptor; Cytochrome P-450 CYP2B6; Cytochrome P-450 CYP3A; Dose-Response Relationship, Drug; Enzyme Induction; Gene Expression Regulation, Enzymologic; Hep G2 Cells; Hepatocytes; Humans; Oxidoreductases, N-Demethylating; Oximes; Promoter Regions, Genetic; Receptors, Cytoplasmic and Nuclear; Rifampin; RNA, Messenger; Thiazoles; Transcriptional Activation; Transfection; Triazoles

2010
Metabonomic studies on human hepatocyte in primary culture.
    Methods in molecular biology (Clifton, N.J.), 2010, Volume: 640

    Topics: Cells, Cultured; Constitutive Androstane Receptor; Hepatocytes; Humans; Mass Spectrometry; Metabolomics; Models, Biological; Oximes; Phenobarbital; Pregnane X Receptor; Receptors, Cytoplasmic and Nuclear; Receptors, Steroid; Rifampin; Thiazoles

2010
In vitro efficacy of fosfomycin-containing regimens against methicillin-resistant Staphylococcus aureus in biofilms.
    The Journal of antimicrobial chemotherapy, 2012, Volume: 67, Issue:4

    Topics: Anti-Bacterial Agents; Biofilms; Drug Interactions; Fosfomycin; Humans; Methicillin-Resistant Staphylococcus aureus; Microbial Sensitivity Tests; Microbial Viability; Rifampin; Staining and Labeling; Tetrazolium Salts; Thiazoles

2012
Bactericidal activity of ACH-702 against nondividing and biofilm Staphylococci.
    Antimicrobial agents and chemotherapy, 2012, Volume: 56, Issue:7

    Topics: Acetamides; Anti-Bacterial Agents; Aza Compounds; Biofilms; Fluoroquinolones; Linezolid; Microbial Sensitivity Tests; Molecular Structure; Moxifloxacin; Oxazolidinones; Quinolines; Quinolones; Rifampin; Staphylococcus; Thiazoles; Vancomycin

2012
Distribution and deposition of respirable PLGA microspheres in lung alveoli.
    Colloids and surfaces. B, Biointerfaces, 2013, May-01, Volume: 105

    Topics: Administration, Inhalation; Animals; Antibiotics, Antitubercular; Antigens, CD; Antigens, Differentiation, Myelomonocytic; Coumarins; Fluorescence; Immunoenzyme Techniques; Lactic Acid; Lung; Macrophages, Alveolar; Male; Microspheres; Phagocytosis; Polyglycolic Acid; Polylactic Acid-Polyglycolic Acid Copolymer; Rats; Rats, Wistar; Rifampin; Thiazoles; Tissue Distribution; Trachea

2013
[Establishment of in vitro evaluation model for CYP2B6 induction and its application to screen inducers among TCMs].
    Yao xue xue bao = Acta pharmaceutica Sinica, 2013, Volume: 48, Issue:1

    Topics: Aryl Hydrocarbon Hydroxylases; Constitutive Androstane Receptor; Cytochrome P-450 CYP2B6; Drugs, Chinese Herbal; Genes, Reporter; Genetic Vectors; Hep G2 Cells; High-Throughput Screening Assays; Humans; Luciferases; Oximes; Plants, Medicinal; Plasmids; Pregnane X Receptor; Receptors, Cytoplasmic and Nuclear; Receptors, Steroid; Rifampin; Thiazoles; Transfection

2013
Effects of ketoconazole and rifampicin on the pharmacokinetics of GLS4, a novel anti-hepatitis B virus compound, in dogs.
    Acta pharmacologica Sinica, 2013, Volume: 34, Issue:11

    Topics: Administration, Oral; Animals; Antiviral Agents; Area Under Curve; Chromatography, High Pressure Liquid; Cytochrome P-450 CYP3A; Dogs; Drug Interactions; Enzyme Induction; Enzyme Inhibitors; Humans; Ketoconazole; Male; Microsomes, Liver; Pyrimidines; Rifampin; Species Specificity; Tandem Mass Spectrometry; Thiazoles

2013
Nanoparticles as drug delivery system against tuberculosis in zebrafish embryos: direct visualization and treatment.
    ACS nano, 2014, Jul-22, Volume: 8, Issue:7

    Topics: Animals; Anti-Bacterial Agents; Biological Transport; Coumarins; Drug Carriers; Embryo, Nonmammalian; Granuloma; Lactic Acid; Macrophages; Mycobacterium Infections, Nontuberculous; Mycobacterium marinum; Nanoparticles; Optical Imaging; Polyglycolic Acid; Polylactic Acid-Polyglycolic Acid Copolymer; Rhodamines; Rifampin; Thiazoles; Tuberculosis; Zebrafish

2014
Antibacterial Characterization of Novel Synthetic Thiazole Compounds against Methicillin-Resistant Staphylococcus pseudintermedius.
    PloS one, 2015, Volume: 10, Issue:6

    Topics: Animals; Anti-Bacterial Agents; Cell Line; Cell Survival; Dog Diseases; Dogs; Lysostaphin; Methicillin; Methicillin Resistance; Mice; Microbial Sensitivity Tests; Oxacillin; Rifampin; Staphylococcal Infections; Staphylococcus; Thiazoles; Vancomycin

2015
Genomewide comparison of the inducible transcriptomes of nuclear receptors CAR, PXR and PPARα in primary human hepatocytes.
    Biochimica et biophysica acta, 2016, Volume: 1859, Issue:9

    Topics: Adult; Constitutive Androstane Receptor; Cytochrome P-450 Enzyme System; Female; Gene Expression Profiling; Gene Expression Regulation; Gene Ontology; Genome-Wide Association Study; Hepatocytes; Humans; Inactivation, Metabolic; Ligands; Male; Metabolic Networks and Pathways; Middle Aged; Molecular Sequence Annotation; Oximes; PPAR alpha; Pregnane X Receptor; Primary Cell Culture; Pyrimidines; Receptors, Cytoplasmic and Nuclear; Receptors, Steroid; Rifampin; Signal Transduction; Thiazoles; Transcriptome

2016
Differences in Gene Regulation by Dual Ligands of Nuclear Receptors Constitutive Androstane Receptor (CAR) and Pregnane X Receptor (PXR) in HepG2 Cells Stably Expressing CAR/PXR.
    Drug metabolism and disposition: the biological fate of chemicals, 2016, Volume: 44, Issue:8

    Topics: Constitutive Androstane Receptor; Cytochrome P-450 CYP2B6; Cytochrome P-450 CYP2C9; Cytochrome P-450 CYP3A; Drug Partial Agonism; Gene Expression Regulation, Enzymologic; Glucuronosyltransferase; Hep G2 Cells; Humans; Isoquinolines; Ligands; Oximes; Pregnane X Receptor; Receptor Cross-Talk; Receptors, Cytoplasmic and Nuclear; Receptors, Steroid; Rifampin; RNA, Messenger; Thiazoles; Transfection

2016
Mycobacterium tuberculosis Is Selectively Killed by Rifampin and Rifapentine in Hypoxia at Neutral pH.
    Antimicrobial agents and chemotherapy, 2017, Volume: 61, Issue:3

    Topics: Anaerobiosis; Antitubercular Agents; Hydrogen-Ion Concentration; Isonicotinic Acids; Microbial Sensitivity Tests; Mycobacterium tuberculosis; Nitroimidazoles; Phenazines; Quinolines; Rifampin; Thiazoles

2017
Thiazomycin, nocathiacin and analogs show strong activity against clinical strains of drug-resistant Mycobacterium tuberculosis.
    The Journal of antibiotics, 2017, Volume: 70, Issue:5

    Topics: Antitubercular Agents; Drug Resistance, Multiple, Bacterial; Fluoroquinolones; Intercellular Signaling Peptides and Proteins; Isoniazid; Microbial Sensitivity Tests; Moxifloxacin; Mycobacterium tuberculosis; Peptides; Peptides, Cyclic; Rifampin; Solubility; Thiazoles

2017
Physiologically Based Pharmacokinetic Modeling Suggests Limited Drug-Drug Interaction for Fesoterodine When Coadministered With Mirabegron.
    Journal of clinical pharmacology, 2019, Volume: 59, Issue:11

    Topics: Acetanilides; Adult; Benzhydryl Compounds; Cresols; Cytochrome P-450 CYP2D6; Cytochrome P-450 CYP2D6 Inhibitors; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Drug Interactions; Female; Humans; Ketoconazole; Male; Middle Aged; Rifampin; Thiazoles; Urinary Bladder, Overactive

2019