thiazoles has been researched along with rhodanine in 61 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 46 (75.41) | 18.7374 |
| 1990's | 3 (4.92) | 18.2507 |
| 2000's | 4 (6.56) | 29.6817 |
| 2010's | 8 (13.11) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Eggers, HJ | 1 |
| Irons, RD; Lee, JC; Schenk, EA | 1 |
| Eggers, HJ; Rosenwirth, B | 2 |
| Salama, KhM; Vladzimirs'ka, OV | 1 |
| Reichardt, LF; Ross, WN | 1 |
| Buchanan, LL; Douch, PG | 1 |
| Strumwasser, F; Woolum, JC | 1 |
| Jenssen, HL; Jülich, WD; Köhler, H; Weuffen, W | 1 |
| Foye, WO; Tovivich, P | 1 |
| Olech, A | 1 |
| Kajikawa, N; Mukai, T; Nagahara, M; Ohishi, Y; Yajima, M | 1 |
| Hashimoto, H; Nakashima, M; Satoh, N; Takiguchi, Y | 1 |
| Iagodin, SV; Pushkarev, IuP; Romanov, NN; Slutskiĭ, VM; Sukhanov, VL | 1 |
| Dai, S | 1 |
| Hatanaka, I; Huitian, Z; Shigeta, Y; Sonobe, M; Terada, M; Yamashita, M; Yasuda, H | 1 |
| Consigli, RA; Guikema, JA; Ludlow, JW | 1 |
| Kondo, M; Nakano, K; Nishioka, H; Terashima, H; Yoshida, T; Yoshioka, K | 1 |
| Akiguchi, I; Kuriya, N; Miyake, S; Mori, T; Nakanishi, T; Takahashi, A; Toyama, K; Ueda, Y; Yamaguchi, Y; Yokota, A | 1 |
| Furukawa, A; Ikeda, K; Kurono, Y; Li, FL; Takesue, Y | 1 |
| Harada, T; Hotta, N; Kakuta, H; Kojima, K; Matsubara, H; Mizuno, K; Sakamoto, N; Suzuki, M | 2 |
| Hagerman, AE; Inoue, KH | 1 |
| Konnerth, A; Orkand, RK | 1 |
| Fukasawa, H; Hotta, N; Iida, M; Kakuta, H; Kimura, M; Koh, N; Morimura, T; Sakamoto, N; Terashima, H | 1 |
| Khromov, VE; Mavrina, EA | 1 |
| Bohnenstengel, C; Jülich, WD; Wagner, R; Weber, P; Weuffen, W | 1 |
| An, SH; Foye, WO | 1 |
| Warashina, A | 1 |
| Fujii, S; Hirano, Y; Hirota, A; Sawanobori, T | 1 |
| Heiny, JA; Vergara, J | 1 |
| Hatanaka, I; Kikkawa, R; Kobayashi, N; Morimura, T; Shigeta, Y; Terashima, H; Tsuboshima, M; Yasuda, H | 1 |
| Hatanaka, I; Kikkawa, R; Kobayashi, N; Shigeta, Y; Yasuda, H | 1 |
| Hama, K; Hatanaka, I; Kikkawa, R; Shigeta, Y; Terashima, H; Tsuboshima, M; Yamamoto, R | 1 |
| Fujii, S; Hirota, A; Kamino, K; Sawanobori, T | 1 |
| Fujii, S; Hirota, A; Kamino, K | 1 |
| Barth, P; Biellmann, JF; Potier, N; Tritsch, D; Van Dorsselaer, A | 1 |
| El-Bindary, AA; El-Dissouky, A; El-Gogary, TM; El-Sonbati, AZ; Hilali, AS | 1 |
| Bekhit, AA; Fahmy, HT | 1 |
| LAPIERE, CL; STAINIER, C | 1 |
| MUSTAFA, A; TAWAB, SA | 1 |
| ALLAN, FJ; ALLAN, GG; M'NEIL, CM | 1 |
| KURNITSKII, II | 1 |
| ZAPADNIUK, VI | 1 |
| MYNKA, AF | 1 |
| KURNYTSKYI, II | 1 |
| IRVIN, JL; PIANTADOSI, C; SKULASON, VG; ZAMBRANA, BF | 1 |
| MYNKA, AF; TURKEVICH, MN | 1 |
| MAZZANTI, L | 1 |
| DEMKIV, LP; DYBAN, AP | 1 |
| MORITA, M | 1 |
| Chen, Z; Demuth, TP; Frère, JM; Lu, WP; White, RE; Zervosen, A | 1 |
| Nakamura, J | 1 |
| Arora, P; Chudayeu, M; Kaushik-Basu, N; Kulkarni, SS; Patel, MR; Singh, S; Talele, TT | 1 |
| Chiruvella, KK; Hemlal, H; Joy, O; Moorthy, BT; Raghavan, SC; Ravi, S; Srivastava, M | 1 |
| Hayashi, S; Ihara, M; Kimura, H; Matsumura, K; Mori, H; Okamoto, Y; Ono, M; Saji, H; Takahashi, R | 1 |
| Cascioferro, S; Daidone, G; Maggio, B; Raffa, D; Raimondi, MV; Schillaci, D | 1 |
| Dun, Y; Fang, H; Fu, H; Hou, X; Wang, L; Yang, X | 1 |
| Kado, S; Kojima, H; Kumagai, K; Kunii, N; Liu, K; Mizuno, S; Nagano, T; Okabe, T; Sakai, H; Sakane, F; Sakuma, M; Sato, M; Shirai, Y; Yamaki, A | 1 |
| Botta, M; De Logu, A; Deodato, D; Ferraris, DM; Kasula, M; Mori, M; Rizzi, M; Sanna, A | 1 |
| Botta, M; Brai, A; Cagno, V; Canducci, F; Ceresola, ER; Dreassi, E; Ferrarese, R; Iovenitti, G; Lembo, D; Poli, G; Tintori, C; Zamperini, C | 1 |
1 review(s) available for thiazoles and rhodanine
| Article | Year |
|---|---|
[Development of therapeutic agents for diabetic neuropathies].
Topics: Aldehyde Reductase; Antioxidants; C-Peptide; Diabetic Neuropathies; Drug Design; Enzyme Inhibitors; Genetic Therapy; Glycation End Products, Advanced; Hedgehog Proteins; Humans; Indoles; Maleimides; Nerve Growth Factor; Oxidative Stress; Polymers; Protein Kinase C; Rhodanine; Thiadiazoles; Thiamine; Thiazoles; Thiazolidines; Trans-Activators; Vascular Endothelial Growth Factor A | 2005 |
60 other study(ies) available for thiazoles and rhodanine
| Article | Year |
|---|---|
Selective inhibiton of uncoating of echovirus 12 by rhodanine. A study on early virus-cell interactions.
Topics: Benzimidazoles; Cell Line; Drug Resistance; Enterovirus B, Human; Guanidines; Hydrogen-Ion Concentration; Light; Poliovirus; Protein Biosynthesis; Rhodanine; RNA, Viral; Thiazoles | 1977 |
Cytochemical methods for copper. Semiquantitative screening procedure for identification of abnormal copper levels in liver.
Topics: Copper; Evaluation Studies as Topic; Humans; Liver; Methods; Rhodanine; Spectrophotometry, Atomic; Staining and Labeling; Thiazoles | 1977 |
Early processes of echovirus 12-infection: elution, penetration, and uncoating under the influence of rhodanine.
Topics: Animals; Cell Line; Cell Membrane; Centrifugation, Density Gradient; Cytoplasm; Enterovirus B, Human; Haplorhini; Rhodanine; Temperature; Thiazoles | 1979 |
Echovirus 12-induced host cell shutoff is prevented by rhodanine.
Topics: Cell Line; Echovirus Infections; Enterovirus B, Human; Poliovirus; Protein Biosynthesis; Rhodanine; Thiazoles; Virus Replication | 1977 |
[Synthesis and properties of bis-(thiazolidone-2-thion-4-yl-3)-butane and its derivatives].
Topics: Chemistry, Pharmaceutical; Isomerism; Rhodanine; Thiazoles; Thiones | 1979 |
Species-specific effects on the optical signals of voltage-sensitive dyes.
Topics: Action Potentials; Animals; Coloring Agents; Electric Stimulation; Electrophysiology; Membrane Potentials; Neurons; Optics and Photonics; Oxazoles; Oxazolone; Rhodanine; Species Specificity; Thiazoles | 1979 |
The metabolism of nitrophenolic and 5-arylazorhodanine anthelmintics by Ascaris suum, Moniezia expansa and by mouse- and sheep-liver enzymes.
Topics: Animals; Anthelmintics; Ascaris; Cestoda; In Vitro Techniques; Liver; Male; Mice; Monieziasis; Nitrophenols; Nitroxinil; Rhodanine; Sheep; Species Specificity; Thiazoles | 1979 |
Membrane-potential-sensitive dyes for optical monitoring of activity in Aplysia neurons.
Topics: Action Potentials; Animals; Aplysia; Circadian Rhythm; Coloring Agents; Membrane Potentials; Neurons; Optic Nerve; Oxazoles; Rhodanine; Thiazoles | 1978 |
[Relations between the macrophage electrophoretic mobility test and the rhodanide level in patients with malignant tumors, autoaggression diseases and after transplantation].
Topics: Animals; Antibody Formation; Autoimmune Diseases; Guinea Pigs; Humans; Kidney Transplantation; Lymphocyte Activation; Macrophages; Neoplasms; Postoperative Complications; Rhodanine; Thiazoles; Transplantation, Homologous | 1975 |
N-Glucopyranosyl-5-aralkylidenerhodanines: synthesis and antibacterial and antiviral activities.
Topics: Animals; Anti-Bacterial Agents; Antiviral Agents; Bacteria; Blood Glucose; Cells, Cultured; Cricetinae; Rhodanine; RNA; RNA, Viral; Thiazoles | 1977 |
[Complex rhodanate salts as precipitating reagents for assaying organic bases. III. Use of potassium hexarhodanochromate for the determination of imipramine and some other dibenzoazepine derivatives].
Topics: Chemical Phenomena; Chemical Precipitation; Chemistry; Chromium; Dibenzazepines; Imipramine; Indicators and Reagents; Rhodanine; Thiazoles | 1975 |
Preparation of 5-alkyl-3-carboxymethylrhodanines and their aldose reductase inhibitory activity.
Topics: Aldehyde Reductase; Animals; Rats; Rhodanine; Thiazoles | 1992 |
Effects of an aldose reductase inhibitor, ONO-2235, insulin and their combination on the altered responsiveness to the nerve stimulation and agonists of the isolated atria of diabetic rats.
Topics: Aldehyde Reductase; Animals; Blood Glucose; Diabetes Mellitus, Experimental; Electric Stimulation; Heart Atria; In Vitro Techniques; Insulin; Male; Muscle, Smooth; Myocardial Contraction; Norepinephrine; Rats; Rats, Inbred Strains; Rhodanine; Sugar Alcohol Dehydrogenases; Synaptic Transmission; Thiazoles; Thiazolidines | 1990 |
[Optical signals from the nerve fibers of fresh-water mollusks stained with the potential-sensitive dye WW375].
Topics: Action Potentials; Animals; In Vitro Techniques; Lymnaea; Nerve Fibers; Optics and Photonics; Rhodanine; Staining and Labeling; Thiazoles | 1986 |
Ventricular histamine concentrations and arrhythmias during acute myocardial ischaemia in rats.
Topics: Acute Disease; Animals; Arrhythmias, Cardiac; Blood Pressure; Coronary Disease; Guanidines; Heart Rate; Heart Ventricles; Histamine; Histamine Release; Male; Myocardium; Rats; Rats, Inbred Strains; Rhodanine; Thiazoles | 1987 |
Effect of prostaglandin E1 analogue TFC 612 on diabetic neuropathy in streptozocin-induced diabetic rats. Comparison with aldose reductase inhibitor ONO 2235.
Topics: Adenosine Triphosphate; Aldehyde Reductase; Alprostadil; Animals; Diabetes Mellitus, Experimental; Diabetic Neuropathies; Electrophysiology; Inositol; Lactates; Male; Myelin Sheath; Nerve Fibers; Phosphocreatine; Rats; Rats, Inbred Strains; Rhodanine; Sciatic Nerve; Sorbitol; Streptozocin; Sugar Alcohol Dehydrogenases; Thiazoles; Thiazolidines | 1989 |
Use of 5-(4-dimethylaminobenzylidene)rhodanine in quantitating silver grains eluted from autoradiograms of biological material.
Topics: Autoradiography; Colorimetry; Coloring Agents; Densitometry; Molecular Weight; Polyomavirus; Rhodanine; Silver; Thiazoles; Viral Proteins; Viral Structural Proteins | 1986 |
Effect of aldose reductase inhibitor ONO 2235 on reduced sympathetic nervous system activity and peripheral nerve disorders in STZ-induced diabetic rats.
Topics: Aldehyde Reductase; alpha-Methyltyrosine; Animals; Autonomic Nervous System Diseases; Diabetes Mellitus, Experimental; Diabetic Neuropathies; Erythrocytes; Female; Methyltyrosines; Neural Conduction; Norepinephrine; Peripheral Nervous System Diseases; Rats; Rats, Inbred Strains; Rhodanine; Sciatic Nerve; Sorbitol; Streptozocin; Sugar Alcohol Dehydrogenases; Sympathetic Nervous System; Thiazoles; Thiazolidines; Triiodothyronine | 1987 |
Effects of aldose reductase inhibitor on the peripheral nerve function during ischemia in diabetics.
Topics: Action Potentials; Adolescent; Adult; Aldehyde Reductase; Arm; Child; Diabetic Neuropathies; Female; Humans; Ischemia; Male; Middle Aged; Peripheral Nerves; Rhodanine; Sugar Alcohol Dehydrogenases; Thiazoles; Thiazolidines | 1987 |
Photo-stabilization and solubilization of an aldose reductase inhibitor, (E)-3-carboxymethyl-5-[(2E)-methyl-3-phenylpropenylidene]rhodani ne (ONO-2235), by human serum albumin.
Topics: Aldehyde Reductase; Drug Stability; Humans; Photochemistry; Rhodanine; Serum Albumin; Sugar Alcohol Dehydrogenases; Thiazoles; Thiazolidines | 1987 |
Effects of aldose reductase inhibitor on retinal microangiopathy in streptozotocin-diabetic rats.
Topics: Aldehyde Reductase; Animals; Basement Membrane; Blood Glucose; Body Weight; Capillaries; Diabetes Mellitus, Experimental; Diabetic Angiopathies; Male; Microscopy, Electron; Rats; Rats, Inbred Strains; Retinal Vessels; Rhodanine; Streptozocin; Sugar Alcohol Dehydrogenases; Thiazoles; Thiazolidines | 1985 |
Determination of gallotannin with rhodanine.
Topics: Colorimetry; Esters; Gallic Acid; Hydrogen-Ion Concentration; Hydrolysis; Plants; Rhodanine; Tannins; Thiazoles | 1988 |
Voltage-sensitive dyes measure potential changes in axons and glia of the frog optic nerve.
Topics: Animals; Axons; Benzoxazoles; Electric Stimulation; Electrophysiology; Microelectrodes; Neuroglia; Optic Nerve; Oxazoles; Oxazolone; Rana pipiens; Rhodanine; Thiazoles; Thiazolidines | 1986 |
Effects of a fructose-rich diet and the aldose reductase inhibitor, ONO-2235, on the development of diabetic neuropathy in streptozotocin-treated rats.
Topics: Aldehyde Reductase; Animals; Diabetes Mellitus, Experimental; Diabetic Neuropathies; Dietary Carbohydrates; Erythrocytes; Fructose; Male; Motor Neurons; Neural Conduction; Rats; Retina; Rhodanine; Sciatic Nerve; Sorbitol; Sugar Alcohol Dehydrogenases; Thiazoles; Thiazolidines | 1985 |
[Experimentally induced diabetic retinal microangiopathy and polyol pathway. II. Effect of aldose reductase inhibitors on microangiopathy].
Topics: Aldehyde Reductase; Animals; Diabetic Retinopathy; Male; Rats; Rats, Inbred Strains; Rhodanine; Sugar Alcohol Dehydrogenases; Thiazoles; Thiazolidines | 1985 |
[Functional changes in the body of workers engaged in production of nitron fibers].
Topics: Acrylates; Chemical Industry; Dermatitis, Contact; Dermatitis, Occupational; Female; Humans; Male; Neurasthenia; Occupational Diseases; Rhodanine; Russia; Thiazoles | 1974 |
[Studies on the influence of electrolytes upon immunization processes. I. Immunological reactivity as a function of the rhodanide level in guinea pigs sensitized with horse serum].
Topics: Animals; Antibodies; Antibody Formation; Binding Sites, Antibody; Body Weight; Cell Membrane Permeability; Cell Migration Inhibition; DNA; Guinea Pigs; Hemagglutination Tests; Horses; Immune Sera; Rhodanine; RNA; Thiazoles | 1974 |
Synthesis of N-glycosylthioureas, N-glycosylrhodanines, and N-glycosyl-2-aminothiazoles and their antimicrobial activity.
Topics: Anti-Infective Agents; Glycosylation; Microbial Sensitivity Tests; Rhodanine; Thiazoles; Thiourea | 1981 |
Further studies on absorption changes arising in dye-stained nerves during excitation.
Topics: Animals; Benzoxazoles; Brachyura; Electric Stimulation; Ganglia, Sympathetic; Light; Nerve Fibers; Rabbits; Rats; Rhodanine; Spectrophotometry; Staining and Labeling; Thiazoles; Thiazolidines; Vagus Nerve | 1980 |
Circus-movement tachycardia in frog atrium monitored by voltage-sensitive dyes.
Topics: Acetylcholine; Action Potentials; Animals; Benzoxazoles; Fluorescent Dyes; Heart; Heart Atria; Microelectrodes; Rana catesbeiana; Rhodanine; Tachycardia; Thiazoles; Thiazolidines | 1984 |
Dichroic behavior of the absorbance signals from dyes NK2367 and WW375 in skeletal muscle fibers.
Topics: Absorption; Animals; Membranes; Models, Biological; Muscles; Oxazoles; Oxazolone; Potentiometry; Rana catesbeiana; Rhodanine; Spectrum Analysis; Thiazoles | 1984 |
Effect of a new aldose reductase inhibitor, (E)-3-carboxymethyl-5-[(2E)-methyl-3-phenylpropenylidene]rhodanine (ONO-2235) on peripheral nerve disorders in streptozotocin-diabetic rats.
Topics: Aldehyde Reductase; Animals; Diabetes Mellitus, Experimental; Diabetic Neuropathies; Erythrocytes; Insulin; Male; Neural Conduction; Rats; Rats, Inbred Strains; Rhodanine; Sciatic Nerve; Sorbitol; Sugar Alcohol Dehydrogenases; Thiazoles; Thiazolidines | 1983 |
Prevention of peripheral nerve dysfunction by an aldose reductase inhibitor in streptozotocin-diabetic rats.
Topics: Aldehyde Reductase; Animals; Diabetes Mellitus, Experimental; Diabetic Neuropathies; Male; Motor Neurons; Neural Conduction; Rats; Rats, Inbred Strains; Rhodanine; Sciatic Nerve; Sorbitol; Sugar Alcohol Dehydrogenases; Thiazoles; Thiazolidines | 1984 |
Effects of a new aldose reductase inhibitor on various tissues in vitro.
Topics: Aldehyde Reductase; Animals; Erythrocytes; Kinetics; Lens, Crystalline; Male; Rats; Rats, Inbred Strains; Rhodanine; Sciatic Nerve; Sorbitol; Sugar Alcohol Dehydrogenases; Thiazoles; Thiazolidines | 1984 |
Optical recording of conducted action potential in heart muscle using a voltage-sensitive dye.
Topics: Action Potentials; Animals; Benzoxazoles; Coloring Agents; Heart; In Vitro Techniques; Methods; Optics and Photonics; Rana catesbeiana; Rhodanine; Thiazoles; Thiazolidines | 1981 |
Localization of pacemaking activity in early embryonic heart monitored using voltage-sensitive dye.
Topics: Action Potentials; Animals; Chick Embryo; Fluorescent Dyes; Heart; Heart Atria; Heart Rate; Myocardial Contraction; Pyrimidines; Rhodanine; Thiazoles; Thiazolidines | 1981 |
Study of non-covalent enzyme-inhibitor complexes of aldose reductase by electrospray mass spectrometry.
Topics: Acetates; Aldehyde Reductase; Animals; Apoenzymes; Enzyme Inhibitors; Furans; Imidazoles; Imidazolidines; Lens, Crystalline; Mass Spectrometry; NADP; Naphthalenes; Rhodanine; Swine; Thiazoles; Thiazolidines | 1997 |
Substituents effect on the spectral studies on rutheninum(III) complexes of 5(-4'-derivatives phenyldiazo)-3-phenyl-2-thioxo-4-thiazolidinone.
Topics: Chemical Phenomena; Chemistry, Physical; Electrochemistry; Hydrogen Bonding; Ligands; Magnetics; Organometallic Compounds; Rhodanine; Ruthenium; Spectrophotometry, Infrared; Thiazoles | 2002 |
Synthesis of some new bis-thiazoles as possible anticancer agents.
Topics: Antineoplastic Agents; Chemical Phenomena; Chemistry, Physical; Drug Screening Assays, Antitumor; Humans; Indicators and Reagents; Magnetic Resonance Spectroscopy; Rhodanine; Spectrophotometry, Infrared; Thiazoles; Tumor Cells, Cultured | 2002 |
[Some derivatives of rhodanine with in-vitro tuberculostatic action].
Topics: Humans; Mycobacterium tuberculosis; Rhodanine; Thiazoles | 1958 |
A comparative study of pharmacological and toxicological action of 2,4-thiazolidinedione and rhodanine and its derivatives.
Topics: Rhodanine; Thiazoles; Thiazolidinediones | 1960 |
Mothicidal rhodanine derivatives.
Topics: Insecticides; Rhodanine; Thiazoles | 1959 |
[Studies on the properties of the complex of copper and 4-(3-rhodanine)-benzoic acid].
Topics: Benzoates; Benzoic Acid; Copper; Rhodanine; Thiazoles | 1962 |
[Relation of anti-spastic properties and toxicity to the chemical structure of thiohydantoin and rhodanine derivatives].
Topics: Hydantoins; Muscle Spasticity; Rhodanine; Thiazoles; Thiohydantoins | 1962 |
[SYNTHESIS AND STUDIES ON 5-ALKYL DERIVATIVES OF RHODANINE].
Topics: Ammonium Compounds; Chemistry, Pharmaceutical; Pharmacy; Quaternary Ammonium Compounds; Research; Rhodanine; Thiazoles | 1963 |
[ON THE COMBINATION OF COPPER WITH RHODANINE-3-BENZOIC ACID AND ON ITS CONSTANT INSTABILITY].
Topics: Benzoates; Benzoic Acid; Chemistry, Pharmaceutical; Copper; Pharmacy; Research; Rhodanine; Thiazoles | 1963 |
SYNTHESIS OF SOME PYRIMIDINE AMINO ACIDS BY THE RHODANINE METHOD AND TESTS VS. THE EHRLICH ASCITES CARCINOMA.
Topics: Amino Acids; Animals; Ascites; Carbon Isotopes; Carcinoma; Carcinoma, Ehrlich Tumor; Chemistry, Pharmaceutical; Mice; Pharmacology; Proteins; Pyrimidines; Research; Rhodanine; Thiazoles | 1965 |
[ON THE EFFECT OF ALKYL SUBSTITUTES IN THE 5TH POSITION ON THE ULTRAVIOLET SPECTRUM OF RHODANINE ABSORPTION].
Topics: Chemistry, Pharmaceutical; Pharmacy; Research; Rhodanine; Spectrum Analysis; Thiazoles; Ultraviolet Rays | 1964 |
[Different reactions of the endocrine pancreas to intramine and rhodanine in animal species].
Topics: Animals; Benzidines; Islets of Langerhans; Pancreas; Rhodanine; Thiazoles | 1954 |
[Goitrogenic effect of rhodanine].
Topics: Antithyroid Agents; Humans; Rhodanine; Thiazoles | 1954 |
[Synthesis and antibacterial activity of antipyrine derivative. I. 4-Thiazoline-2-thiones, dithiocarbamic acid esters and rhodanines].
Topics: Anti-Bacterial Agents; Antipyrine; Esters; Rhodanine; Thiazoles; Thiazolidines | 1962 |
Interactions between penicillin-binding proteins (PBPs) and two novel classes of PBP inhibitors, arylalkylidene rhodanines and arylalkylidene iminothiazolidin-4-ones.
Topics: Algorithms; Alkenes; Bacillus megaterium; Bacteria; Bacterial Proteins; Carrier Proteins; Cell Wall; Dipeptidyl-Peptidases and Tripeptidyl-Peptidases; Escherichia coli; Hexosyltransferases; Kinetics; Muramoylpentapeptide Carboxypeptidase; Penicillin-Binding Proteins; Peptidoglycan; Peptidyl Transferases; Protease Inhibitors; Rhodanine; Streptococcus pneumoniae; Structure-Activity Relationship; Thiazoles | 2004 |
Structure-based virtual screening, synthesis and SAR of novel inhibitors of hepatitis C virus NS5B polymerase.
Topics: Allosteric Regulation; Antiviral Agents; Benzylidene Compounds; Binding Sites; Computer Simulation; Databases, Factual; Enzyme Inhibitors; Hepacivirus; Rhodanine; Structure-Activity Relationship; Thiazoles; Viral Nonstructural Proteins | 2010 |
Novel rhodanine derivatives induce growth inhibition followed by apoptosis.
Topics: Antineoplastic Agents; Apoptosis; Cell Line, Tumor; Cell Membrane; Cell Proliferation; Cell Survival; Coloring Agents; DNA Fragmentation; Dose-Response Relationship, Drug; Humans; L-Lactate Dehydrogenase; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Reactive Oxygen Species; Rhodanine; Tetrazolium Salts; Thiazoles; Trypan Blue | 2010 |
Rhodanine and thiohydantoin derivatives for detecting tau pathology in Alzheimer's brains.
Topics: Alzheimer Disease; Animals; Autoradiography; Benzothiazoles; Brain; Humans; Iodine Radioisotopes; Mice; Neurofibrillary Tangles; Positron-Emission Tomography; Radiopharmaceuticals; Recombinant Proteins; Rhodanine; Tauopathies; Thiazoles; Thiohydantoins; Tissue Distribution | 2011 |
Sortase A Inhibitors: Recent Advances and Future Perspectives.
Topics: Adamantane; Aminoacyltransferases; Animals; Anti-Bacterial Agents; Bacterial Adhesion; Bacterial Proteins; Benzoates; Carbolines; Cysteine Endopeptidases; Enzyme Inhibitors; Humans; Models, Molecular; Nitriles; Protein Conformation; Rhodanine; Small Molecule Libraries; Staphylococcal Infections; Staphylococcus aureus; Thiazoles; Thiones | 2015 |
Design, synthesis and biological evaluation of 3-aryl-rhodanine benzoic acids as anti-apoptotic protein Bcl-2 inhibitors.
Topics: Antineoplastic Agents; bcl-X Protein; Benzoates; Cell Line, Tumor; Humans; Molecular Docking Simulation; Myeloid Cell Leukemia Sequence 1 Protein; Proto-Oncogene Proteins c-bcl-2; Rhodanine; Sulfonamides; Thiazoles | 2015 |
A novel diacylglycerol kinase α-selective inhibitor, CU-3, induces cancer cell apoptosis and enhances immune response.
Topics: Animals; Antineoplastic Agents; Apoptosis; Cell Line, Tumor; Cell Proliferation; Chlorocebus aethiops; COS Cells; Diacylglycerol Kinase; Drug Screening Assays, Antitumor; Enzyme Inhibitors; HeLa Cells; Humans; Inhibitory Concentration 50; Interleukin-2; Isoenzymes; Lymphocyte Activation; Rhodanine; Substrate Specificity; Sulfonamides; T-Lymphocytes; Thiazoles | 2016 |
Design, synthesis, SAR and biological investigation of 3-(carboxymethyl)rhodanine and aminothiazole inhibitors of Mycobacterium tuberculosis Zmp1.
Topics: Antitubercular Agents; Bacterial Proteins; Enzyme Inhibitors; Humans; Metalloproteases; Microbial Sensitivity Tests; Molecular Docking Simulation; Molecular Structure; Mycobacterium tuberculosis; Rhodanine; Structure-Activity Relationship; Thiazoles; THP-1 Cells | 2018 |
Rhodanine derivatives as potent anti-HIV and anti-HSV microbicides.
Topics: Animals; Antiviral Agents; Chlorocebus aethiops; Drug Resistance, Viral; Female; HeLa Cells; Herpes Simplex; Herpesvirus 1, Human; Herpesvirus 2, Human; HIV Infections; HIV-1; Humans; Molecular Structure; Pre-Exposure Prophylaxis; Rhodanine; Simplexvirus; Thiazoles; Vaginal Creams, Foams, and Jellies; Vero Cells; Virus Replication | 2018 |