Page last updated: 2024-08-21

thiazoles and reserpine

thiazoles has been researched along with reserpine in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-199014 (63.64)18.7374
1990's3 (13.64)18.2507
2000's2 (9.09)29.6817
2010's3 (13.64)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Strosberg, AM1
Waldeck, B1
Bell, SC; Wei, PH1
Algeri, S; Cioce, V; Duvert, L; Garattini, S; Legeai, J; Manuel, C; Notelle, C; Ponzio, F; Rusconi, L; Sacchetti, G1
Gray, WD; Rauh, CE1
Götz, HG1
Inoki, R; Otori, K; Yamamoto, I1
Ashford, A; Brown, GR; Evans, DE; King, G; Palmer, PJ; Ross, JW; Shadbolt, RS; Sharpe, CJ; Trigg, RB; Ward, RJ1
Breese, GR; Cooper, BR; Grant, LD1
Brunaud, M; Laborit, H; Vallée, E1
Ashford, A; Ross, JW; Shadbolt, RS; Sharpe, CJ1
Glatt, MM1
Barbarino, F; Brilinschi, C; Togănel, E1
Felix, G; Otrzonsek, G; Schneider, B; Windsheimer, F1
Gujrati, VR; Palit, G; Shanker, K; Tripathi, M; Verma, M1
Adell, A; Artigas, F1
Lorenc-Koci, E; Wolfarth, S1
Farde, L; Gulyás, B; Halldin, C; Kiss, B; Laszlovszky, I; Schou, M; Schukin, E; Sóvágó, J1
Johansen, JL; Leist, M; Lotharius, J; Vergo, S1
Antonio, T; Dutta, AK; Ghosh, B; Kharkar, P; Reith, ME; Zhen, J1
Antonio, T; Dutta, AK; Johnson, M; Reith, ME1
Alfonso, M; Durán, R; Faro, LR; Oliveira, IM1

Reviews

1 review(s) available for thiazoles and reserpine

ArticleYear
[Antithyroid agents. 15].
    Pharmazeutische Praxis, 1967, Volume: 9

    Topics: Antithyroid Agents; Barbiturates; Carbimazole; Diiodotyrosine; Estrogens; Fluorides; Humans; Hyperthyroidism; Imidazoles; Iodine; Iodine Isotopes; Methylthiouracil; Perchlorates; Phenylacetates; Plant Extracts; Potassium; Propiophenones; Reserpine; Sodium; Sulfonamides; Thiazoles; Thiocyanates; Thiouracil; Tissue Extracts; Tyrosine; Vitamins

1967

Trials

2 trial(s) available for thiazoles and reserpine

ArticleYear
Controlled trials of non-barbiturate hypnotics and tranquillisers. With special reference to their use in alcoholics.
    Psychiatria et neurologia, 1966, Volume: 152, Issue:1

    Topics: Alcoholism; Amobarbital; Chlormethiazole; Chlorpromazine; Clinical Trials as Topic; Female; Glutethimide; Humans; Hypnotics and Sedatives; Male; Placebos; Promazine; Reserpine; Thiazoles; Tranquilizing Agents

1966
[Long-term antihypertensive therapy with Etozoline].
    Die Medizinische Welt, 1980, Apr-18, Volume: 31, Issue:16

    Topics: Adult; Drug Evaluation; Female; Humans; Hypertension; Inositol; Male; Mefruside; Middle Aged; Reserpine; Thiazoles

1980

Other Studies

19 other study(ies) available for thiazoles and reserpine

ArticleYear
The cardiovascular pharmacology and hemodynamic activity of tazolol, a selective myocardial beta-stimulant.
    Archives internationales de pharmacodynamie et de therapie, 1976, Volume: 222, Issue:2

    Topics: Adrenergic beta-Agonists; Amphetamine; Animals; Blood Pressure; Dogs; Drug Interactions; Female; Heart Rate; Hemodynamics; Isoproterenol; Male; Myocardial Contraction; Propanolamines; Propranolol; Reserpine; Thiazoles; Time Factors

1976
Analysis of the beta-receptor mediated effect on slow-contracting skeletal muscle in vitro.
    The Journal of pharmacy and pharmacology, 1977, Volume: 29, Issue:9

    Topics: Adrenergic beta-Antagonists; Animals; Dopamine; Electric Stimulation; Epinephrine; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Norepinephrine; Propanolamines; Receptors, Adrenergic; Receptors, Adrenergic, beta; Reserpine; Terbutaline; Thiazoles; Tyramine

1977
Syntheses of heterocylic fused thiazole acetic acids. 2.
    Journal of medicinal chemistry, 1976, Volume: 19, Issue:4

    Topics: Acetates; Animals; Antidepressive Agents; Antineoplastic Agents; Antitubercular Agents; Bridged-Ring Compounds; Humans; Mice; Neoplasms, Experimental; Reserpine; Thiazoles

1976
Behavioural and biochemical studies on 6-methylamino-4,5,6,7-tetrahydrobenzothiazole (14.839JL), a new potent dopaminergic agonist.
    Pharmacological research communications, 1987, Volume: 19, Issue:8

    Topics: Adenylyl Cyclases; Animals; Biogenic Amines; Brain Chemistry; Corpus Striatum; Female; Male; Mice; Motor Activity; Prolactin; Rats; Receptors, Dopamine; Reserpine; Stereotyped Behavior; Sulpiride; Thiazoles

1987
The anticonvulsant action of the carbonic anhydrase inhibitor methazolamide: possible involvement of a noradrenergic mechanism.
    European journal of pharmacology, 1974, Volume: 28, Issue:1

    Topics: Animals; Anticonvulsants; Benserazide; Body Temperature; Carbonic Anhydrase Inhibitors; Dihydroxyphenylalanine; Dopamine beta-Hydroxylase; Dose-Response Relationship, Drug; Electroshock; Ethanolamines; Isoproterenol; Levobunolol; Male; Methazolamide; Mice; Motor Activity; Norepinephrine; Phenoxybenzamine; Phentolamine; Phenytoin; Practolol; Propranolol; Rats; Reserpine; Serotonin; Thiazoles; Thiourea; Tolazoline

1974
Pharmacological studies on antagonists against nicotine-induced convulsions and death.
    Japanese journal of pharmacology, 1966, Volume: 16, Issue:4

    Topics: Animals; Anticonvulsants; Chlorpromazine; Drug Antagonism; Female; Ganglionic Blockers; Hexamethonium Compounds; Histamine H1 Antagonists; Male; Meprobamate; Mice; Nicotine; Parasympatholytics; Perphenazine; Phenobarbital; Phentolamine; Reserpine; Seizures; Sympatholytics; Thiazoles; Tolazoline; Tranquilizing Agents; Urea

1966
Basic ethers of 2-anilinobenzothiazoles and 2-anilinobenzoxazoles as potential antidepressants.
    Journal of medicinal chemistry, 1972, Volume: 15, Issue:5

    Topics: Abnormalities, Drug-Induced; Aniline Compounds; Animals; Antidepressive Agents; Behavior, Animal; Benzoxazoles; Body Weight; Cats; Dogs; Ethers; Female; Haplorhini; Mice; Motor Activity; Pregnancy; Rabbits; Rats; Reserpine; Stimulation, Chemical; Structure-Activity Relationship; Thiazoles

1972
Comparison of the behavioral depressant effects of biogenic amine depleting and neuroleptic agents following various 6-hydroxydopamine treatments.
    Psychopharmacologia, 1973, Jul-17, Volume: 31, Issue:2

    Topics: Animals; Behavior, Animal; Brain; Brain Chemistry; Chlorpromazine; Depression, Chemical; Dopamine; Dopamine beta-Hydroxylase; Haloperidol; Hydroxydopamines; Male; Methyltyrosines; Norepinephrine; Pimozide; Rats; Reinforcement, Psychology; Reserpine; Thiazoles; Thiourea; Time Factors; Tranquilizing Agents

1973
[The action of 2-amino-4-(isothioureyl methyl)-thiazol dihydrochloride (Agr 307) on the catecholamines of the central nervous system in the rat. Possible inhibition of dopamine beta-hydroxylase].
    Agressologie: revue internationale de physio-biologie et de pharmacologie appliquees aux effets de l'agression, 1971, Volume: 12, Issue:2

    Topics: Animals; Brain; Catecholamines; Dopamine; Hypertension; Male; Mixed Function Oxygenases; Monoamine Oxidase Inhibitors; Myocardial Infarction; Nialamide; Norepinephrine; Rats; Reserpine; Thiazoles

1971
Phenacylthioimidazolines and 3-aryl-5,6-dihydroimidazo(2,1-b)thiazoles with antidepressant activity.
    Journal of medicinal chemistry, 1971, Volume: 14, Issue:10

    Topics: Administration, Oral; Animals; Antidepressive Agents; Cats; Dihydroxyphenylalanine; Drug Synergism; Female; Fetus; Guinea Pigs; Hypothermia, Induced; Imidazoles; Male; Mice; Monoamine Oxidase Inhibitors; Motor Activity; Norepinephrine; Pregnancy; Rabbits; Rats; Reserpine; Stimulation, Chemical; Structure-Activity Relationship; Tetrabenazine; Thiazoles; Vas Deferens

1971
The effects of acetazolamide and of ethoxzolamide on gastric microcirculation in rats (histochemical study).
    Annals of the New York Academy of Sciences, 1984, Volume: 429

    Topics: Acetazolamide; Adenosine Triphosphatases; Animals; Ethoxzolamide; Female; Gastric Mucosa; Histocytochemistry; Microcirculation; Rats; Reserpine; Stomach Ulcer; Thiazoles

1984
Thiazolidinone congeners as central nervous system active agents.
    Arzneimittel-Forschung, 1993, Volume: 43, Issue:6

    Topics: Amphetamine; Animals; Brain; Central Nervous System Agents; Drug Synergism; Female; Helplessness, Learned; In Vitro Techniques; Male; Mice; Monoamine Oxidase Inhibitors; Pilocarpine; Rats; Reserpine; Salivation; Thiazoles

1993
A microdialysis study of the in vivo release of 5-HT in the median raphe nucleus of the rat.
    British journal of pharmacology, 1998, Volume: 125, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic Uptake Inhibitors; Animals; Benzopyrans; Male; Microdialysis; Piperazines; Pyridines; Quinolines; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Reserpine; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Thiazoles

1998
Efficacy of pramipexole, a new dopamine receptor agonist, to relieve the parkinsonian-like muscle rigidity in rats.
    European journal of pharmacology, 1999, Nov-26, Volume: 385, Issue:1

    Topics: alpha-Methyltyrosine; Animals; Benzothiazoles; Dopamine Agonists; Dose-Response Relationship, Drug; Electromyography; Haloperidol; Male; Muscle Rigidity; Muscle, Skeletal; Parkinson Disease, Secondary; Pramipexole; Rats; Rats, Wistar; Reserpine; Thiazoles; Treatment Outcome

1999
Lack of effect of reserpine-induced dopamine depletion on the binding of the dopamine-D3 selective radioligand, [11C]RGH-1756.
    Brain research bulletin, 2005, Oct-15, Volume: 67, Issue:3

    Topics: Adrenergic Uptake Inhibitors; Animals; Binding, Competitive; Brain; Carbon Isotopes; Dopamine; Female; Macaca fascicularis; Piperazines; Positron-Emission Tomography; Protein Binding; Reserpine; Thiazoles; Time Factors

2005
Vesicular monoamine transporter 2 regulates the sensitivity of rat dopaminergic neurons to disturbed cytosolic dopamine levels.
    Brain research, 2007, Dec-14, Volume: 1185

    Topics: Adrenergic Uptake Inhibitors; Analysis of Variance; Animals; Cell Proliferation; Cytosol; Dopamine; Drug Interactions; Green Fluorescent Proteins; L-Lactate Dehydrogenase; Methamphetamine; PC12 Cells; Potassium Chloride; Rats; Reserpine; Tetrazolium Salts; Thiazoles; Time Factors; Transfection; Tyrosine 3-Monooxygenase; Vesicular Monoamine Transport Proteins

2007
Development of (S)-N6-(2-(4-(isoquinolin-1-yl)piperazin-1-yl)ethyl)-N6-propyl-4,5,6,7-tetrahydrobenzo[d]-thiazole-2,6-diamine and its analogue as a D3 receptor preferring agonist: potent in vivo activity in Parkinson's disease animal models.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Animals; Antiparkinson Agents; Benzothiazoles; CHO Cells; Cricetinae; Cricetulus; Disease Models, Animal; Free Radical Scavengers; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Isoquinolines; Locomotion; Mice; Parkinson Disease; Radioligand Assay; Rats; Receptors, Dopamine D2; Receptors, Dopamine D3; Reserpine; Structure-Activity Relationship; Thiazoles

2010
Structure-activity relationship study of N⁶-(2-(4-(1H-Indol-5-yl)piperazin-1-yl)ethyl)-N⁶-propyl-4,5,6,7-tetrahydrobenzo[d]thiazole-2,6-diamine analogues: development of highly selective D3 dopamine receptor agonists along with a highly potent D2/D3 agoni
    Journal of medicinal chemistry, 2012, 06-28, Volume: 55, Issue:12

    Topics: Animals; CHO Cells; Cricetinae; Cricetulus; Drug Discovery; Female; Free Radical Scavengers; HEK293 Cells; Humans; Indoles; Locomotion; Male; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Reserpine; Structure-Activity Relationship; Substrate Specificity; Thiazoles

2012
In vivo neurochemical characterization of clothianidin induced striatal dopamine release.
    Toxicology, 2012, Dec-16, Volume: 302, Issue:2-3

    Topics: Animals; Calcium; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Exocytosis; Female; Guanidines; Insecticides; Microdialysis; Neonicotinoids; Nomifensine; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Reserpine; Tetrodotoxin; Thiazoles

2012