Page last updated: 2024-08-21

thiazoles and ponatinib

thiazoles has been researched along with ponatinib in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's12 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Clackson, T; Deininger, MW; Druker, BJ; Eide, CA; O'Hare, T1
Quintás-Cardama, A; Santos, FP1
Pfirrmann, M; Saussele, S1
Kantarjian, H; Liu-Dumlao, T; O'Brien, S; Ravandi, F; Thomas, DA1
Azam, M1
Auberger, P; Cassuto, JP; Cassuto, O; Dubois, A; Dufies, M; Ginet, C; Hamouda, A; Jacquel, A; Karsenti, JM; Legros, L; Lenain, P; Luciano, F; Puissant, A; Robert, G1
Dolgin, E1
Tojo, A1
Bengió, RM; Bianchini, M; Ferri, CA; Gonzalez, MS; Larripa, IB; Moiraghi, EB; Noriega, MF1
Takahashi, N1
Eigendorff, E; Ernst, T; Hochhaus, A; La Rosée, P1
Kim, HH; Korade, Z; Porter, NA; Wages, PA1

Reviews

5 review(s) available for thiazoles and ponatinib

ArticleYear
New drugs for chronic myelogenous leukemia.
    Current hematologic malignancy reports, 2011, Volume: 6, Issue:2

    Topics: Benzamides; Dasatinib; Drug Resistance, Neoplasm; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Imidazoles; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Neoplastic Stem Cells; Piperazines; Protein Kinase Inhibitors; Pyridazines; Pyrimidines; Thiazoles

2011
Clinical trials in chronic myeloid leukemia.
    Current hematologic malignancy reports, 2012, Volume: 7, Issue:2

    Topics: Aniline Compounds; Benzamides; Dasatinib; Humans; Imatinib Mesylate; Imidazoles; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Nitriles; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyridazines; Pyrimidines; Quality of Life; Quinolines; Randomized Controlled Trials as Topic; Survival Analysis; Thiazoles

2012
Philadelphia-positive acute lymphoblastic leukemia: current treatment options.
    Current oncology reports, 2012, Volume: 14, Issue:5

    Topics: Aniline Compounds; Antineoplastic Agents; Benzamides; Dasatinib; Humans; Imatinib Mesylate; Imidazoles; Neoplasm, Residual; Nitriles; Piperazines; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Protein Kinase Inhibitors; Pyridazines; Pyrimidines; Quinolines; Stem Cell Transplantation; Thiazoles

2012
[Management of advanced stage chronic myeloid leukemia].
    [Rinsho ketsueki] The Japanese journal of clinical hematology, 2014, Volume: 55, Issue:10

    Topics: Allografts; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Dasatinib; Disease Progression; Drug Design; Fusion Proteins, bcr-abl; Hematopoietic Stem Cell Transplantation; Humans; Imatinib Mesylate; Imidazoles; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Molecular Targeted Therapy; Neoplasm Staging; Piperazines; Point Mutation; Protein Kinase Inhibitors; Pyridazines; Pyrimidines; Randomized Controlled Trials as Topic; Thiazoles

2014
Causes of resistance and treatment choices of second- and third-line treatment in chronic myelogenous leukemia patients.
    Annals of hematology, 2015, Volume: 94 Suppl 2

    Topics: Aniline Compounds; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Dasatinib; Disease Progression; Drug Monitoring; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Fusion Proteins, bcr-abl; Humans; Imidazoles; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Molecular Targeted Therapy; Mutation; Nitriles; Prognosis; Protein Kinase Inhibitors; Pyridazines; Pyrimidines; Quinolines; Thiazoles

2015

Other Studies

7 other study(ies) available for thiazoles and ponatinib

ArticleYear
Targeting the BCR-ABL signaling pathway in therapy-resistant Philadelphia chromosome-positive leukemia.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2011, Jan-15, Volume: 17, Issue:2

    Topics: Antineoplastic Agents; Dasatinib; Drug Resistance, Neoplasm; Drugs, Investigational; Fusion Proteins, bcr-abl; Humans; Imidazoles; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Molecular Targeted Therapy; Mutation; Pyridazines; Pyrimidines; Signal Transduction; Thiazoles

2011
An in vitro screening to identify drug-resistant mutations for target-directed chemotherapeutic agents.
    Methods in molecular biology (Clifton, N.J.), 2012, Volume: 928

    Topics: Benzamides; Cell Line; Dasatinib; Drug Discovery; Drug Evaluation, Preclinical; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Imidazoles; Mutation; Piperazines; Protein Kinase Inhibitors; Pyridazines; Pyrimidines; Thiazoles

2012
All tyrosine kinase inhibitor-resistant chronic myelogenous cells are highly sensitive to ponatinib.
    Oncotarget, 2012, Volume: 3, Issue:12

    Topics: Animals; Antineoplastic Agents; Apoptosis; Benzamides; Cell Survival; Dasatinib; Dose-Response Relationship, Drug; Drug Resistance, Neoplasm; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Imidazoles; Inhibitory Concentration 50; K562 Cells; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Mice; Mutation; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyridazines; Pyrimidines; Signal Transduction; Thiazoles; Tumor Cells, Cultured

2012
As leukemia options grow, drugs jockey to be first-line therapies.
    Nature medicine, 2013, Volume: 19, Issue:1

    Topics: Antineoplastic Agents; Benzamides; Dasatinib; Drug Resistance, Neoplasm; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Imidazoles; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Piperazines; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyridazines; Pyrimidines; Thiazoles

2013
[Chronic myeloid leukemia].
    Nihon rinsho. Japanese journal of clinical medicine, 2012, Volume: 70 Suppl 8

    Topics: Dasatinib; Humans; Imidazoles; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Molecular Targeted Therapy; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyridazines; Pyrimidines; Thiazoles

2012
Clinical activity of ponatinib in one patient with chronic myeloid leukemia in chronic phase with e19a2 transcript and T315I mutation.
    European journal of haematology, 2015, Volume: 94, Issue:3

    Topics: Antineoplastic Agents; Dasatinib; Drug Resistance, Neoplasm; Female; Fusion Proteins, bcr-abl; Gene Expression; Humans; Hydroxyurea; Imidazoles; Leukemia, Myeloid, Chronic-Phase; Middle Aged; Mutation; Pyridazines; Pyrimidines; RNA, Messenger; Thiazoles; Treatment Outcome

2015
Identification and characterization of prescription drugs that change levels of 7-dehydrocholesterol and desmosterol.
    Journal of lipid research, 2018, Volume: 59, Issue:10

    Topics: Benzamides; Cell Line, Tumor; Dehydrocholesterols; Desmosterol; Drug Evaluation, Preclinical; Gene Expression Regulation; High-Throughput Screening Assays; Humans; Imidazoles; Nerve Tissue Proteins; Oxidoreductases Acting on CH-CH Group Donors; Piperidines; Prescription Drugs; Pyridazines; Pyridines; Thiazoles; United States; United States Food and Drug Administration

2018