Page last updated: 2024-08-21

thiazoles and osimertinib

thiazoles has been researched along with osimertinib in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's4 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Liu, C; Liu, D; Song, Y; Tsui, ST; Wang, S1
Liu, D; Song, Y; Wang, S; Yan, F1
Jiang, Y; Li, Z; Wan, S; Wu, X; Yan, R; Zhang, J1
Cameron, MD; Chen, T; Dahlberg, SE; De Clercq, DJH; Eck, MJ; Gero, TW; Gray, NS; Heppner, DE; Jang, J; Jänne, PA; Mushajiang, M; Park, E; Shin, BH; To, C; Wang, S; Wong, KK; Xu, M; Yang, A1

Reviews

2 review(s) available for thiazoles and osimertinib

ArticleYear
EGFR C797S mutation mediates resistance to third-generation inhibitors in T790M-positive non-small cell lung cancer.
    Journal of hematology & oncology, 2016, 07-22, Volume: 9, Issue:1

    Topics: Acrylamides; Aniline Compounds; Benzeneacetamides; Carcinoma, Non-Small-Cell Lung; Drug Resistance, Neoplasm; ErbB Receptors; Humans; Lung Neoplasms; Mutation; Piperazines; Protein Kinase Inhibitors; Thiazoles

2016
Mechanisms of resistance to third-generation EGFR tyrosine kinase inhibitors.
    Frontiers of medicine, 2016, Volume: 10, Issue:4

    Topics: Acrylamides; Aniline Compounds; Antineoplastic Agents; Benzeneacetamides; Carcinoma, Non-Small-Cell Lung; Drug Resistance, Neoplasm; ErbB Receptors; Humans; Lung Neoplasms; Mutation; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-met; Receptor, ErbB-2; Thiazoles

2016

Other Studies

2 other study(ies) available for thiazoles and osimertinib

ArticleYear
Insight into binding mechanisms of EGFR allosteric inhibitors using molecular dynamics simulations and free energy calculations.
    Journal of biomolecular structure & dynamics, 2019, Volume: 37, Issue:16

    Topics: Acrylamides; Allosteric Regulation; Aniline Compounds; Benzeneacetamides; Carcinoma, Non-Small-Cell Lung; Drug Resistance, Neoplasm; ErbB Receptors; Erlotinib Hydrochloride; Gefitinib; Humans; Molecular Dynamics Simulation; Mutation; Protein Binding; Protein Kinase Inhibitors; Pyrimidines; Thiazoles

2019
Single and Dual Targeting of Mutant EGFR with an Allosteric Inhibitor.
    Cancer discovery, 2019, Volume: 9, Issue:7

    Topics: Acrylamides; Allosteric Regulation; Aniline Compounds; Animals; Antineoplastic Combined Chemotherapy Protocols; Benzeneacetamides; Cell Line, Tumor; Cell Survival; Drug Resistance, Neoplasm; ErbB Receptors; Humans; Lung Neoplasms; Mice; Mice, Transgenic; Mutation; NIH 3T3 Cells; Protein Kinase Inhibitors; Thiazoles; Xenograft Model Antitumor Assays

2019