Page last updated: 2024-08-21

thiazoles and nifedipine

thiazoles has been researched along with nifedipine in 37 studies

Research

Studies (37)

TimeframeStudies, this research(%)All Research%
pre-199010 (27.03)18.7374
1990's15 (40.54)18.2507
2000's8 (21.62)29.6817
2010's3 (8.11)24.3611
2020's1 (2.70)2.80

Authors

AuthorsStudies
Nebel, U; Wermelskirchen, D; Wilffert, B; Wirth, A1
Iso, T; Miyawaki, N; Nishimura, K; Yamauchi, H1
Bazill, GW; Dexter, TM1
Koch, P; Peters, T; Wilffert, B; Wilhelm, D1
Halabi, A; Kirch, W; Linde, M; Ohnhaus, EE; Santos, SR1
Ferry, DR; Glossmann, H; Goll, A; Linn, T1
Halabi, H; Kirch, W; Ohnhaus, EE1
Halabi, A; Kirch, W; Linde, M; Ohnhaus, EE1
Koch, P; Nebel, U; Peters, T; Wermelskirchen, D; Wilffert, B; Wilhelm, D1
Knee, CD; Krell, RD; Kusner, EJ1
Fischli, W; Hengartner, U; Holck, M1
Ito, K; Kanazawa, T; Morita, T; Nose, T2
Hashimoto, H; Kanda, A1
Chiba, K; Fukuzawa, A; Ishigai, Y; Mori, T; Shibano, T1
Decrinis, M; Kasper, K; Miyawaki, N; Stark, G; Stark, U; Tritthart, HA1
Mori, M; Ohtani, K; Sato, N; Shimizu, H; Tanaka, Y1
Balkan, A; Ertan, M; Ertekin, N; Sara, Y; Tozkoparan, B1
Aivasian, A; Akopov, S; Gabrielian, E; Grigorian, G; Markarian, E; Panossian, A; Vartanian, S1
Nakagawa, M; Sasaki, S1
Mori, M; Ohtani, KI; Sato, N; Shimizu, H1
Hisatome, I; Ikeda, T; Ogino, K; Shimoyama, M; Tanaka, Y1
Asano, M; Hazama, H; Imuta, H; Iwasawa, K; Kawakami, Y; Morita, T; Nakajima, T; Nakamura, F; Okuda, Y; Omata, M; Oonuma, H; Suzuki, J; Suzuki, S1
Beschke, K; Ebner, T; Ludwig, E; Schmid, J1
Finnerty, D; Freed, MI; Harris, RZ; Inglis, AM; Jorkasky, DK; Miller, AK; Patterson, S; Thompson, KA1
Kuwahara, M; Miyaji, T; Tsubone, H1
Harbour, C; Koutalistras, N; Li, L; Mears, D; Sheil, AG; Sun, J; Wang, L1
Adachi, Y; Karaki, H; Satake, N; Sato, K; Shibata, S1
Gokina, NI; Osol, G1
Abe, K; Inoue, R; Ito, Y; Morita, H1
Kritz, H; Oguogho, A; Sinzinger, H; Wolfram, RM1
Beaman-Hall, CM; Bui, CJ; Middleton, FA; Vallano, ML1
Bay, BH; Cheung, NS; Li, Y; Qi, RZ; Sheu, FS; Tan, CH; Whiteman, M; Yap, YW1
Ayon, RJ; Davis, AJ; Duan, DD; Forrest, AS; Freitas, N; Greenwood, IA; Huebner, ML; Joyce, J; Joyce, TC; Leblanc, N; Singer, CA; Valencik, ML; Wiwchar, M; Ye, L1
Di, CP; Ding, C; Fan, Y; Li, L; Sun, Y; Xu, Y; Zhao, L1
Chen, W; Cheng, X; Cui, H; He, K; Li, S; Wang, L; Zhang, B; Zhong, W1
Ahmed, B; Keshari, M; Khalilullah, H; Khan, RA; Yusuf, M1

Reviews

1 review(s) available for thiazoles and nifedipine

ArticleYear
[Calcium channel blocker for therapy of patients with hypertension].
    Nihon rinsho. Japanese journal of clinical medicine, 1997, Volume: 55, Issue:8

    Topics: Benzimidazoles; Calcium Channel Blockers; Dihydropyridines; Drug Interactions; Humans; Hypertension; Mibefradil; Nifedipine; Tetrahydronaphthalenes; Thiazoles

1997

Trials

4 trial(s) available for thiazoles and nifedipine

ArticleYear
Negative effects of famotidine on cardiac performance assessed by noninvasive hemodynamic measurements.
    Gastroenterology, 1989, Volume: 96, Issue:6

    Topics: Adult; Double-Blind Method; Drug Interactions; Famotidine; Half-Life; Hemodynamics; Histamine H2 Antagonists; Humans; Nifedipine; Random Allocation; Reference Values; Thiazoles

1989
Negative inotropic effects of famotidine.
    Lancet (London, England), 1987, Sep-19, Volume: 2, Issue:8560

    Topics: Adult; Depression, Chemical; Drug Interactions; Famotidine; Histamine H2 Antagonists; Humans; Myocardial Contraction; Nifedipine; Random Allocation; Thiazoles

1987
[Negative inotropic action of famotidine].
    Schweizerische medizinische Wochenschrift, 1988, Dec-17, Volume: 118, Issue:50

    Topics: Adult; Cardiac Output; Depression, Chemical; Drug Combinations; Famotidine; Histamine H2 Antagonists; Humans; Myocardial Contraction; Nifedipine; Stroke Volume; Thiazoles

1988
Rosiglitazone has no clinically significant effect on nifedipine pharmacokinetics.
    Journal of clinical pharmacology, 1999, Volume: 39, Issue:11

    Topics: Adolescent; Adult; Calcium Channel Blockers; Cross-Over Studies; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Humans; Hypoglycemic Agents; Male; Nifedipine; Rosiglitazone; Thiazoles; Thiazolidinediones; Time Factors

1999

Other Studies

32 other study(ies) available for thiazoles and nifedipine

ArticleYear
45Ca2+ movements induced by Ca2+ chloride in isolated rat aorta under K(+)-free conditions.
    European journal of pharmacology, 1991, Jan-17, Volume: 192, Issue:3

    Topics: Amiloride; Animals; Aorta, Thoracic; Benzothiazoles; Calcium; Calcium Chloride; Calcium Radioisotopes; Flunarizine; In Vitro Techniques; Indomethacin; Lanthanum; Lidocaine; Nifedipine; omega-Conotoxins; Peptides, Cyclic; Piperidines; Potassium; Rats; Thiazoles; Vasoconstriction

1991
Tissue selectivity of the novel calcium antagonist sesamodil fumarate in isolated smooth muscles and cardiac muscles.
    Arzneimittel-Forschung, 1990, Volume: 40, Issue:3

    Topics: Animals; Calcimycin; Calcium Channel Blockers; Diltiazem; Guinea Pigs; Heart; Male; Muscle Contraction; Muscle, Smooth, Vascular; Myocardial Contraction; Nicardipine; Nifedipine; Rabbits; Swine; Thiazoles; Verapamil

1990
Role of endocytosis in the action of ether lipids on WEHI-3B, HL60, and FDCP-mix A4 cells.
    Cancer research, 1990, Dec-01, Volume: 50, Issue:23

    Topics: Animals; Antineoplastic Agents; Azepines; Cell Survival; Chloroquine; Diltiazem; Drug Synergism; Endocytosis; Furans; Humans; Hydroxyzine; In Vitro Techniques; Leukemia, Myeloid; Mice; Nifedipine; Phospholipid Ethers; Platelet Activating Factor; Pyridines; Quinidine; Quinine; Sodium Fluoride; Thiazoles; Triazoles; Verapamil

1990
R 56865 differentiates between contractile agents with respect to the nifedipine-sensitive component in the isolated rat aorta.
    Pharmacology, 1989, Volume: 39, Issue:1

    Topics: Angiotensin II; Animals; Aorta, Thoracic; Arginine Vasopressin; Benzothiazoles; Calcium; Calcium Channels; Cytosol; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Thiazoles

1989
Molecular approach to the calcium channel.
    Advances in myocardiology, 1985, Volume: 5

    Topics: Animals; Benzothiazoles; Binding Sites; Brain; Calcium; Cattle; Chemical Phenomena; Chemistry; Diltiazem; Guinea Pigs; In Vitro Techniques; Ion Channels; Isradipine; Muscles; Myocardium; Nicotinic Acids; Nifedipine; Nimodipine; Nitrendipine; Oxadiazoles; Thiazoles; Verapamil

1985
Different effects of R 56865 and calcium entry blockers on K+- and noradrenaline-induced contractions and 45Ca uptake in rat aorta.
    European journal of pharmacology, 1988, Dec-13, Volume: 158, Issue:3

    Topics: Animals; Aorta; Benzothiazoles; Calcium; Calcium Channel Blockers; Diltiazem; Dose-Response Relationship, Drug; Flunarizine; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Norepinephrine; Piperidines; Potassium; Rats; Rats, Inbred Strains; Thiazoles; Verapamil

1988
Pharmacologic analysis of 1-0-alkyl-2-acetyl-sn-glycero-3-phosphocholine-induced increases in cutaneous vascular permeability in the rat.
    Agents and actions, 1987, Volume: 20, Issue:1-2

    Topics: Animals; Capillary Permeability; Chromones; Dose-Response Relationship, Drug; Indomethacin; Masoprocol; Methysergide; Nifedipine; Phenoxybenzamine; Phospholipid Ethers; Platelet Activating Factor; Pyrilamine; Rats; Theophylline; Thiazoles

1987
Effects of temperature and allosteric modulators on [3H] nitrendipine binding: methods for detecting potential Ca2+ channel blockers.
    Journal of receptor research, 1984, Volume: 4, Issue:1-6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Allosteric Regulation; Animals; Benzothiazoles; Binding Sites; Calcium Channel Blockers; Diltiazem; Guinea Pigs; Heart; In Vitro Techniques; Kinetics; Microsomes; Myocardium; Nifedipine; Nitrendipine; Propylamines; Temperature; Thiazoles; Tiapamil Hydrochloride; Verapamil

1984
Vasodilator mechanism of KB-944, a new calcium antagonist.
    Arzneimittel-Forschung, 1982, Volume: 32, Issue:9

    Topics: Adenosine; Animals; Benzothiazoles; Calcium Channel Blockers; Calcium Chloride; Coronary Vessels; Diltiazem; Dogs; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Nifedipine; Potassium; Rabbits; Thiazoles; Vasodilator Agents; Verapamil

1982
Antihypertensive effect of KB-944, a new calcium antagonist, in conscious normotensive and hypertensive rats.
    Arzneimittel-Forschung, 1982, Volume: 32, Issue:9

    Topics: Animals; Antihypertensive Agents; Benzothiazoles; Blood Pressure; Calcium Channel Blockers; Desoxycorticosterone; Diltiazem; Heart Rate; Hypertension; Hypertension, Renal; Nifedipine; Rats; Thiazoles

1982
Effects of semotiadil fumarate, a novel calcium antagonist, on blood pressure and heart rate in conscious spontaneously hypertensive rats.
    Japanese journal of pharmacology, 1993, Volume: 63, Issue:1

    Topics: Animals; Blood Pressure; Calcium Channel Blockers; Diltiazem; Dose-Response Relationship, Drug; Heart Rate; Hypertension; Male; Nifedipine; Rats; Rats, Inbred SHR; Thiazoles

1993
Pharmacological profile of semotiadil fumarate, a novel calcium antagonist, in rat experimental angina model.
    British journal of pharmacology, 1995, Volume: 116, Issue:1

    Topics: Acetylcholine; Angina Pectoris; Animals; Arginine Vasopressin; Calcium Channel Blockers; Coronary Vessels; Diltiazem; Disease Models, Animal; Electrocardiography; Male; Nifedipine; Nisoldipine; Rats; Rats, Inbred Strains; Rats, Sprague-Dawley; Thiazoles; Vasoconstrictor Agents

1995
Effects of semotiadil, a novel Ca2+ channel antagonist, on the electrical activity of Langendorff-perfused guinea pig hearts in comparison with diltiazem, amlodipine and nifedipine.
    European journal of pharmacology, 1995, Nov-03, Volume: 286, Issue:1

    Topics: Amlodipine; Animals; Calcium Channel Blockers; Depression, Chemical; Diltiazem; Electrocardiography; Female; Guinea Pigs; Heart Conduction System; Heart Rate; In Vitro Techniques; Male; Nifedipine; Thiazoles

1995
Pioglitazone hydrochloride stimulates insulin secretion in HIT-T 15 cells by inducing Ca2+ influx.
    The Journal of endocrinology, 1996, Volume: 150, Issue:1

    Topics: Animals; Calcium; Calcium Channel Blockers; Cell Line; Cricetinae; Glucose; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Nifedipine; Pioglitazone; Stimulation, Chemical; Thiazoles; Thiazolidinediones

1996
New thiazolo[3,2-a] pyrimidine derivatives, synthesis and calcium antagonistic activities.
    Bollettino chimico farmaceutico, 1996, Volume: 135, Issue:11

    Topics: Animals; Calcium Channel Blockers; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Nifedipine; Pyrimidines; Thiazoles

1996
Beditine, a new benzodioxane derivative, as a suppressor of human polymorphonuclear leukocyte and platelet activation.
    Biochemical pharmacology, 1997, Jun-01, Volume: 53, Issue:11

    Topics: Adenosine Triphosphate; Aspirin; Calcimycin; Dioxanes; Eicosanoids; Humans; Lipoxygenase Inhibitors; Neutrophils; Nifedipine; Platelet Aggregation Inhibitors; Superoxides; Thiazoles

1997
Troglitazone (CS-045) inhibits beta-cell proliferation rate following stimulation of insulin secretion in HIT-T 15 cells.
    Endocrinology, 1998, Volume: 139, Issue:1

    Topics: Animals; Calcium; Cell Division; Cells, Cultured; Chromans; Cricetinae; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Mesocricetus; Nifedipine; Thiazoles; Thiazolidinediones; Troglitazone

1998
Hemodynamic basis for the acute cardiac effects of troglitazone in isolated perfused rat hearts.
    Diabetes, 1999, Volume: 48, Issue:3

    Topics: Animals; Blood Pressure; Calcium Channels; Chromans; Coronary Circulation; Heart Rate; Hemodynamics; Humans; Hypoglycemic Agents; In Vitro Techniques; Male; Nifedipine; Nitroprusside; Prazosin; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Thiazoles; Thiazolidinediones; Troglitazone; Ventricular Function, Left

1999
Troglitazone inhibits voltage-dependent calcium currents in guinea pig cardiac myocytes.
    Circulation, 1999, Jun-08, Volume: 99, Issue:22

    Topics: Animals; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Calcium Channels, T-Type; Cardiotonic Agents; Chromans; Cyclic AMP; Electric Conductivity; Guinea Pigs; Hypoglycemic Agents; Isoproterenol; Kinetics; Myocardium; Nifedipine; Thiazoles; Thiazolidinediones; Troglitazone; Verapamil

1999
Activation of human cytochrome P-450 3A4-catalyzed meloxicam 5'-methylhydroxylation by quinidine and hydroquinidine in vitro.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:1

    Topics: 3-Oxo-5-alpha-Steroid 4-Dehydrogenase; Calcium Channel Blockers; Chromatography, High Pressure Liquid; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Enzyme Activation; Humans; Hydroxylation; In Vitro Techniques; Meloxicam; Microsomes, Liver; Mixed Function Oxygenases; Nifedipine; Oxidation-Reduction; Quinidine; Thiazines; Thiazoles

1999
Angiotensin II type 1 receptor-mediated increase in cytosolic Ca(2+) and proliferation in mesothelial cells.
    European journal of pharmacology, 2000, Jan-24, Volume: 388, Issue:1

    Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Angiotensin II; Angiotensin Receptor Antagonists; Angiotensin-Converting Enzyme Inhibitors; Animals; Buffers; Calcium; Calcium Channel Blockers; Calcium Signaling; Cell Division; Coloring Agents; Culture Media; Cytosol; Fluorescent Dyes; Fura-2; Indicators and Reagents; Nifedipine; Pertussis Toxin; Pleura; Rats; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; Tetrazolium Salts; Thiazoles; Virulence Factors, Bordetella

2000
Factors affecting hepatocyte viability and CYPIA1 activity during encapsulation.
    Artificial cells, blood substitutes, and immobilization biotechnology, 2000, Volume: 28, Issue:3

    Topics: Alginates; Animals; Apoptosis; Biocompatible Materials; Calcium; Calcium Chloride; Calcium Compounds; Cell Culture Techniques; Cell Survival; Coloring Agents; Cytochrome P-450 CYP1A1; Drug Compounding; Glutathione; Lactates; Liver; Necrosis; Nifedipine; Polylysine; Rats; Rats, Inbred Lew; Rats, Sprague-Dawley; Reproducibility of Results; Swine; Taurine; Temperature; Tetrazolium Salts; Thiazoles

2000
Mechanisms of vasoinhibitory effect of cardioprotective agent, CP-060S, in rat aorta.
    European journal of pharmacology, 2000, Jul-21, Volume: 400, Issue:2-3

    Topics: Angiotensin II; Animals; Anti-Arrhythmia Agents; Aorta, Thoracic; Arginine Vasopressin; Calcium; Calcium Channel Blockers; Cytosol; Dinoprost; Drug Interactions; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Phenylephrine; Rats; Rats, Wistar; Thiazoles; Thiazolidines; Vasoconstrictor Agents; Vasodilator Agents

2000
Actin cytoskeletal modulation of pressure-induced depolarization and Ca(2+) influx in cerebral arteries.
    American journal of physiology. Heart and circulatory physiology, 2002, Volume: 282, Issue:4

    Topics: Actins; Androstadienes; Animals; Blood Pressure; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Cerebral Arteries; Cytochalasin D; Cytoskeleton; Egtazic Acid; Endothelium, Vascular; In Vitro Techniques; Ionomycin; Male; Marine Toxins; Membrane Potentials; Muscle, Smooth, Vascular; Nifedipine; Nigericin; Rats; Rats, Inbred WKY; Thiazoles; Thiazolidines; Vasoconstriction; Wortmannin

2002
Possible involvement of M5 muscarinic receptor in the enhancing actions of the novel gastroprokinetic agent Z-338 on nifedipine-sensitive voltage-dependent Ca2+ currents in guinea pig stomach.
    Japanese journal of pharmacology, 2002, Volume: 89, Issue:4

    Topics: Animals; Benzamides; Calcium Channel Blockers; Calcium Channels, L-Type; Dose-Response Relationship, Drug; Drug Synergism; Female; Gastrointestinal Agents; Guinea Pigs; Male; Membrane Potentials; Nifedipine; Receptor, Muscarinic M5; Receptors, Muscarinic; Stomach; Thiazoles

2002
Antiplatelet activity of semotiadil fumarate.
    Thrombosis research, 2002, May-15, Volume: 106, Issue:4-5

    Topics: Adenosine Diphosphate; Adult; Amlodipine; Calcium Channel Blockers; Case-Control Studies; Collagen; Diltiazem; Humans; Hypertension; Middle Aged; Nifedipine; Platelet Aggregation; Platelet Aggregation Inhibitors; Thiazoles

2002
Depolarization and Ca(2+) down regulate CB1 receptors and CB1-mediated signaling in cerebellar granule neurons.
    Neuropharmacology, 2006, Volume: 50, Issue:6

    Topics: Age Factors; Analysis of Variance; Animals; Animals, Newborn; Blotting, Northern; Calcium; Calcium Channel Blockers; Cell Survival; Cells, Cultured; Cerebellum; Cyclohexanols; Dose-Response Relationship, Drug; Drug Interactions; Fluorescent Antibody Technique; Gene Expression Regulation, Developmental; In Situ Hybridization; Models, Biological; Neurons; Nifedipine; Potassium Chloride; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Signal Transduction; Tetrazolium Salts; Tetrodotoxin; Thiazoles; Time Factors

2006
Hypochlorous acid induces apoptosis of cultured cortical neurons through activation of calpains and rupture of lysosomes.
    Journal of neurochemistry, 2006, Volume: 98, Issue:5

    Topics: Adenosine Triphosphate; Animals; Apoptosis; Calcium; Calcium Channels; Calpain; Caspase 3; Caspases; Cell Survival; Cells, Cultured; Dipeptides; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Hypochlorous Acid; Lysosomes; Mice; Microscopy, Electron, Transmission; Neocortex; Neurons; Nifedipine; Oxidants; Tetrazolium Salts; Thiazoles; Time Factors

2006
Increased TMEM16A-encoded calcium-activated chloride channel activity is associated with pulmonary hypertension.
    American journal of physiology. Cell physiology, 2012, Dec-15, Volume: 303, Issue:12

    Topics: Animals; Anoctamin-1; Calcium Channel Blockers; Chloride Channel Agonists; Chloride Channels; Cyclooxygenase Inhibitors; Hypertension, Pulmonary; Hypertrophy, Right Ventricular; Indomethacin; Male; Monocrotaline; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Nifedipine; Niflumic Acid; Patch-Clamp Techniques; Pulmonary Artery; Pyrimidines; Rats; Rats, Wistar; Serotonin; Thiazoles

2012
Effect of nifedipine on the expression of keratinocyte growth factor and its receptor in cocultured/monocultured fibroblasts and keratinocytes.
    Journal of periodontal research, 2013, Volume: 48, Issue:6

    Topics: Calcium Channel Blockers; Cell Communication; Cell Culture Techniques; Cell Membrane; Cell Proliferation; Coculture Techniques; Coloring Agents; Fibroblast Growth Factor 7; Fibroblasts; Gene Expression Regulation; Gingiva; Humans; Keratinocytes; Nifedipine; Receptor, Fibroblast Growth Factor, Type 2; Tetrazolium Salts; Thiazoles

2013
Alagebrium (ALT-711) improves the anti-hypertensive efficacy of nifedipine in diabetic-hypertensive rats.
    Hypertension research : official journal of the Japanese Society of Hypertension, 2014, Volume: 37, Issue:10

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Diabetes Mellitus, Experimental; Drug Therapy, Combination; Endothelin-1; Epoprostenol; Heart Rate; Hypertension; Male; Nifedipine; Nitric Oxide; Rats; Rats, Wistar; Thiazoles

2014
Pharmacophore modeling, design, and synthesis of potent antihypertensives, oxazolo/thiazolo-[3,2-a]-pyrimidin-3(2H)-one, and 1,5-dihydroimidazo-[1,2-a]-pyrimidin-3(2H)-one derivatives: A pilot trial.
    Bioorganic & medicinal chemistry letters, 2020, 12-01, Volume: 30, Issue:23

    Topics: Animals; Antihypertensive Agents; Arterial Pressure; Drug Design; Female; Imidazoles; Male; Molecular Structure; Nifedipine; Oxazoles; Pilot Projects; Pyrimidines; Rats, Wistar; Structure-Activity Relationship; Thiazoles

2020