Compounds > thiazoles

Page last updated: 2024-08-21

thiazoles and miltefosine

thiazoles has been researched along with miltefosine in 16 studies

Research

Studies (16)

Timeframe	Studies, this research(%)	All Research%
pre-1990	0 (0.00)	18.7374
1990's	1 (6.25)	18.2507
2000's	11 (68.75)	29.6817
2010's	4 (25.00)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Berger, MR; Sobottka, SB	1
Lobovská, A; Nohýnková, E	1
Bories, C; Bréard, J; Loiseau, PM; Paris, C	1
Dey, CS; Verma, NK	1
Bandyopadhyay, S; Chatterjee, M; Dutta, A; Mandal, C	1
Bandyopadhyay, S; Chatterjee, M; Ganguly, S; Sarkar, A	1
Bouchaud, O; Izri, A	1
Ben Brahim, M; Bories, C; Le Moyec, L; Loiseau, PM; Rakotomanga, M; Saint-Pierre-Chazalet, M	1
Mesquita, JT; Reimão, JQ; Tempone, AG	1
Chong, LS; Epp, JB; Fu, Q; Groutas, WC; He, S; Kuang, R; Li, YH; Ruan, S; Truong, TM; Tu, J; Venkataraman, R; Vu, NT; Yu, H	1
Chan, HK; Groutas, WC; He, S; Kuang, R; Ruan, S; Tu, J	1
Alliston, KR; Gan, X; Groutas, WC; Lai, Z; Li, YH; Wei, L; Yu, H	1
Alliston, KR; Dou, D; Groutas, WC; Hanzlik, RP; Huang, W; Li, Y; Williams, TD; Yamamoto, Y	1
Dou, D; Fu, Q; Groutas, WC; He, G; Kuang, R; Venkataraman, R	1
Caram, JA; Castro, EA; Duchowicz, PR; Fernández, FM; García, J; Mirífico, MV; Rozas, MF	1
Cummings, AH; Gates, KS; Hillebrand, R; Laciak, AR; Lewis, SM; Punthasee, P; Ruddraraju, KV; Singh, H; Tanner, JJ	1

Reviews

1 review(s) available for thiazoles and miltefosine

Article	Year
[New drugs for treatment of parasitic infections]. Casopis lekaru ceskych, 2003, Volume: 142, Issue:3 Topics: Antiparasitic Agents; Humans; Intestinal Diseases, Parasitic; Leishmaniasis; Nitro Compounds; Phosphorylcholine; Thiazoles	2003

Other Studies

15 other study(ies) available for thiazoles and miltefosine

Article	Year
Assessment of antineoplastic agents by MTT assay: partial underestimation of antiproliferative properties. Cancer chemotherapy and pharmacology, 1992, Volume: 30, Issue:5 Topics: Animals; Antineoplastic Agents; Cell Count; Cell Division; Coloring Agents; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Humans; Nitrosourea Compounds; Phosphorylcholine; Rats; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured; Vinblastine	1992
Miltefosine induces apoptosis-like death in Leishmania donovani promastigotes. Antimicrobial agents and chemotherapy, 2004, Volume: 48, Issue:3 Topics: Animals; Antiprotozoal Agents; Apoptosis; Cell Cycle; Chromatography, Agarose; Colorimetry; DNA Fragmentation; Flow Cytometry; Leishmania donovani; Phosphatidylserines; Phosphorylcholine; Protease Inhibitors; Tetrazolium Salts; Thiazoles	2004
Possible mechanism of miltefosine-mediated death of Leishmania donovani. Antimicrobial agents and chemotherapy, 2004, Volume: 48, Issue:8 Topics: Animals; Antiprotozoal Agents; Apoptosis; Cell Division; Coloring Agents; Cricetinae; Cricetulus; DNA Fragmentation; DNA, Protozoan; In Situ Nick-End Labeling; Indicators and Reagents; Leishmania donovani; Leishmaniasis, Visceral; Macrophages; Nucleosomes; Phosphorylcholine; Poly(ADP-ribose) Polymerases; Propidium; Tetrazolium Salts; Thiazoles	2004
Development of a modified MTT assay for screening antimonial resistant field isolates of Indian visceral leishmaniasis. Parasitology international, 2005, Volume: 54, Issue:2 Topics: Amphotericin B; Animals; Antimony Sodium Gluconate; Antiprotozoal Agents; Drug Resistance; Humans; Leishmania donovani; Leishmaniasis, Visceral; Parasitic Sensitivity Tests; Phosphorylcholine; Tetrazolium Salts; Thiazoles	2005
Development of a semi-automated colorimetric assay for screening anti-leishmanial agents. Journal of microbiological methods, 2006, Volume: 66, Issue:1 Topics: Amphotericin B; Animals; Antiprotozoal Agents; Colorimetry; Drug Evaluation, Preclinical; Humans; Indicators and Reagents; Inhibitory Concentration 50; Kinetics; Leishmania; Leishmania donovani; Leishmaniasis, Visceral; Pentamidine; Phosphorylcholine; Tetrazolium Salts; Thiazoles	2006
[New antiparasitic drugs]. La Revue de medecine interne, 2008, Volume: 29 Suppl 1 Topics: Albendazole; Antimalarials; Antiparasitic Agents; Benzimidazoles; Cyclohexanes; Fatty Acids, Unsaturated; Humans; Ivermectin; Nitro Compounds; Phosphorylcholine; Praziquantel; Sesquiterpenes; Thiazoles; Triclabendazole	2008
Membrane sterol depletion impairs miltefosine action in wild-type and miltefosine-resistant Leishmania donovani promastigotes. The Journal of antimicrobial chemotherapy, 2009, Volume: 64, Issue:5 Topics: Animals; Antiprotozoal Agents; Cell Membrane; Drug Resistance; Leishmania donovani; Lipid Metabolism; Microbial Viability; Mitochondria; Models, Molecular; Molecular Structure; Parasitic Sensitivity Tests; Phosphorylcholine; Sterols; Tetrazolium Salts; Thiazoles	2009
Combination therapy with nitazoxanide and amphotericin B, Glucantime®, miltefosine and sitamaquine against Leishmania (Leishmania) infantum intracellular amastigotes. Acta tropica, 2014, Volume: 130 Topics: Aminoquinolines; Amphotericin B; Animals; Antiprotozoal Agents; Drug Combinations; Leishmania infantum; Leishmaniasis, Visceral; Macrophages, Peritoneal; Meglumine; Meglumine Antimoniate; Mice; Nitro Compounds; Organometallic Compounds; Parasitic Sensitivity Tests; Phosphorylcholine; Thiazoles	2014
1,2,5-Thiadiazolidin-3-one 1,1 dioxide: a powerful scaffold for probing the S' subsites of (chymo)trypsin-like serine proteases. Archives of biochemistry and biophysics, 2001, Jan-01, Volume: 385, Issue:1 Topics: Cathepsin G; Cathepsins; Chymotrypsin; Cyclic S-Oxides; Humans; Kinetics; Leukocyte Elastase; Models, Chemical; Molecular Probes; Myeloblastin; Protein Binding; Serine Endopeptidases; Temperature; Thiazoles; Time Factors	2001
Inhibition of serine proteases by functionalized sulfonamides coupled to the 1,2,5-thiadiazolidin-3-one 1,1 dioxide scaffold. Bioorganic & medicinal chemistry, 2001, Volume: 9, Issue:6 Topics: Cathepsin G; Cathepsins; Cyclic S-Oxides; Drug Design; Leukocyte Elastase; Models, Molecular; Myeloblastin; Serine Endopeptidases; Serine Proteinase Inhibitors; Structure-Activity Relationship; Sulfonamides; Thiazoles	2001
Potent inhibition of human leukocyte elastase by 1,2,5-thiadiazolidin-3-one 1,1 dioxide-based sulfonamide derivatives. Archives of biochemistry and biophysics, 2004, Sep-15, Volume: 429, Issue:2 Topics: Cyclic S-Oxides; Enzyme Inhibitors; Humans; Leukocyte Elastase; Magnetic Resonance Spectroscopy; Sulfonamides; Thiazoles	2004
X-ray snapshot of the mechanism of inactivation of human neutrophil elastase by 1,2,5-thiadiazolidin-3-one 1,1-dioxide derivatives. Journal of medicinal chemistry, 2008, Apr-10, Volume: 51, Issue:7 Topics: Binding Sites; Crystallography, X-Ray; Cyclic S-Oxides; Enzyme Activation; Humans; Leukocyte Elastase; Models, Molecular; Molecular Structure; Protein Structure, Tertiary; Serine Proteinase Inhibitors; Structure-Activity Relationship; Thiazoles	2008
Effects of structure on inhibitory activity in a series of mechanism-based inhibitors of human neutrophil elastase. Bioorganic & medicinal chemistry, 2010, Sep-15, Volume: 18, Issue:18 Topics: Cyclic S-Oxides; Humans; Kinetics; Leukocyte Elastase; Myeloblastin; Protease Inhibitors; Thiazoles	2010
A comparative QSAR on 1,2,5-thiadiazolidin-3-one 1,1-dioxide compounds as selective inhibitors of human serine proteinases. Journal of molecular graphics & modelling, 2011, Volume: 31 Topics: Cyclic S-Oxides; Drug Design; Humans; Linear Models; Molecular Conformation; Molecular Dynamics Simulation; Quantitative Structure-Activity Relationship; Serine Proteases; Serine Proteinase Inhibitors; Thiazoles	2011
Covalent Allosteric Inactivation of Protein Tyrosine Phosphatase 1B (PTP1B) by an Inhibitor-Electrophile Conjugate. Biochemistry, 2017, 04-11, Volume: 56, Issue:14 Topics: Allosteric Regulation; Allosteric Site; Binding Sites; Crystallography, X-Ray; Cyclic S-Oxides; Enzyme Inhibitors; Escherichia coli; Gene Expression; Humans; Kinetics; Mutation; Protein Binding; Protein Tyrosine Phosphatase, Non-Receptor Type 1; Recombinant Proteins; Structure-Activity Relationship; Thermodynamics; Thiazoles	2017