Page last updated: 2024-08-21

thiazoles and melphalan

thiazoles has been researched along with melphalan in 14 studies

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19903 (21.43)18.7374
1990's3 (21.43)18.2507
2000's4 (28.57)29.6817
2010's4 (28.57)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fujimaru, J; Ogura, M; Takeda, Y; Tomiyoshi, Y; Wada, Y; Yoshida, S1
DeGraff, W; Friedman, N; Mitchell, JB; Russo, A1
Carmichael, J; DeGraff, WG; Gazdar, AF; Minna, JD; Mitchell, JB1
Addicks, HW; Norpoth, K; Witting, U1
Alaoui-Jamali, M; Aubin, R; Batist, G; Bramson, J; Christodoulopoulos, G; McQuillan, A; Panasci, LC1
Batist, G; Chen, X1
Beauséjour, CM; Cournoyer, D; Delisle, JS; Létourneau, S; Momparler, RL; Palerme, JS1
Adams, J; Altamirano, C; Berenson, JR; Borad, MJ; Frantzen, M; Friedman, JM; Ma, MH; Manyak, S; Mikail, A; Neeser, J; Parker, K; Roussos, E; Sjak-Shie, N; Vescio, RA; Wu, ZQ; Yang, HH1
Kutschy, P; McDonald, JF; Mezencev, R; Salayova, A; Updegrove, T1
Forman, SJ; Kogut, NM; O'Donnell, MR; Palmer, JM; Senitzer, D; Slovak, ML; Snyder, DS; Spielberger, RT; Stein, AS; Thomas, SH; Tsai, NC1
Baumann, P; Leban, J; Mandl-Weber, S; Meinel, FG; Schmidmaier, R1
Fujiwara, D; Imano, M; Itoh, T; Komai, M; Mashimo, K; Mukai, J; Nishida, S; Ogawa, N; Sakaguchi, K; Sakamoto, K; Satou, T; Shimaoka, H; Takeda, T; Tsubaki, M1
Augustine, CK; Beasley, GM; Lidsky, ME; Sharma, K; Tokuhisa, Y; Toshimitsu, H; Turley, RS; Tyler, DS; Ueno, T1
Mahmoud, MY; Ramasubramanian, A; Sims, LB; Steinbach-Rankins, JM; Stocke, S; Tyo, KM1

Other Studies

14 other study(ies) available for thiazoles and melphalan

ArticleYear
[Sensitivity test of anti-tumor agents. 2. Application of MTT assay].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1991, Volume: 18, Issue:10

    Topics: Antineoplastic Agents; Cisplatin; Doxorubicin; Drug Screening Assays, Antitumor; Melphalan; Mitomycin; Mitomycins; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1991
Selective modulation of glutathione levels in human normal versus tumor cells and subsequent differential response to chemotherapy drugs.
    Cancer research, 1986, Volume: 46, Issue:6

    Topics: Antineoplastic Agents; Bleomycin; Buthionine Sulfoximine; Cell Survival; Cells, Cultured; Cisplatin; Glutathione; Humans; Lung; Lung Neoplasms; Melphalan; Methionine Sulfoximine; Neoplasms; Pyrrolidonecarboxylic Acid; Thiazoles; Thiazolidines; Zinostatin

1986
Evaluation of a tetrazolium-based semiautomated colorimetric assay: assessment of chemosensitivity testing.
    Cancer research, 1987, Feb-15, Volume: 47, Issue:4

    Topics: Animals; Antineoplastic Agents; Autoanalysis; Cell Line; Cisplatin; Clone Cells; Colorimetry; Coloring Agents; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Doxorubicin; Drug Resistance; Humans; In Vitro Techniques; Lung Neoplasms; Melphalan; Tetrazolium Salts; Thiazoles; Vinblastine

1987
[Quantitative determination of alkylating cytostatics on TLC plate with 4-pyridinecarboxaldehyde-2-benzothiazolylhydrazone].
    Arzneimittel-Forschung, 1973, Volume: 23, Issue:11

    Topics: Acetophenones; Alkylating Agents; Chromatography, Thin Layer; Cyclophosphamide; Hydrazones; Indicators and Reagents; Mannomustine; Melphalan; Methods; Nitrogen Mustard Compounds; Pyridines; Spectrophotometry; Temperature; Thiazoles

1973
Nitrogen mustard drug resistant B-cell chronic lymphocytic leukemia as an in vivo model for crosslinking agent resistance.
    Mutation research, 1995, Volume: 336, Issue:3

    Topics: B-Lymphocytes; Chlorambucil; Cisplatin; Cross-Linking Reagents; DNA Adducts; DNA Damage; DNA Repair; DNA, Neoplasm; Drug Resistance; Humans; Inactivation, Metabolic; Leukemia, Lymphocytic, Chronic, B-Cell; Melphalan; Methyl Methanesulfonate; Mitomycin; Nitrogen Mustard Compounds; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1995
Sensitization effect of L-2-oxothiazolidine-4-carboxylate on tumor cells to melphalan and the role of 5-oxo-L-prolinase in glutathione modulation in tumor cells.
    Biochemical pharmacology, 1998, Sep-15, Volume: 56, Issue:6

    Topics: Antineoplastic Agents, Phytogenic; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Drug Synergism; Glutathione; Humans; Melphalan; Pyroglutamate Hydrolase; Pyrrolidonecarboxylic Acid; Thiazoles; Thiazolidines; Tumor Cells, Cultured

1998
Coexpression of rat glutathione S-transferase A3 and human cytidine deaminase by a bicistronic retroviral vector confers in vitro resistance to nitrogen mustards and cytosine arabinoside in murine fibroblasts.
    Cancer gene therapy, 2000, Volume: 7, Issue:5

    Topics: 3T3 Cells; Animals; Antimetabolites, Antineoplastic; Antineoplastic Agents, Alkylating; Blotting, Southern; Cell Division; Cytarabine; Cytidine Deaminase; DNA, Complementary; Drug Resistance, Neoplasm; Fibroblasts; Gene Transfer Techniques; Genetic Vectors; Glutathione Transferase; Humans; Mechlorethamine; Melphalan; Mice; Protein Biosynthesis; Rats; Retroviridae; Tetrazolium Salts; Thiazoles; Transduction, Genetic

2000
The proteasome inhibitor PS-341 markedly enhances sensitivity of multiple myeloma tumor cells to chemotherapeutic agents.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2003, Volume: 9, Issue:3

    Topics: Active Transport, Cell Nucleus; Adenoviridae; Antineoplastic Agents; Apoptosis; Blotting, Western; Boronic Acids; Bortezomib; Cell Division; Cell Nucleus; Cell Survival; Cysteine Endopeptidases; Cytosol; Dose-Response Relationship, Drug; Genes, Dominant; Humans; I-kappa B Proteins; Melphalan; Microscopy, Fluorescence; Multienzyme Complexes; Multiple Myeloma; NF-kappa B; NF-KappaB Inhibitor alpha; Phosphorylation; Proteasome Endopeptidase Complex; Pyrazines; Tetrazolium Salts; Thiazoles; Time Factors; Transfection; Tumor Cells, Cultured; Ubiquitin

2003
The design, synthesis and anticancer activity of new nitrogen mustard derivatives of natural indole phytoalexin 1-methoxyspirobrassinol.
    Neoplasma, 2009, Volume: 56, Issue:4

    Topics: Antineoplastic Agents; Apoptosis; Caspases; Cell Differentiation; Cell Proliferation; DNA Damage; Drug Design; Drug Screening Assays, Antitumor; Female; Glutathione; Humans; Indoles; Inhibitory Concentration 50; Melphalan; Molecular Structure; Phytoalexins; Sesquiterpenes; Structure-Activity Relationship; Terpenes; Thiazoles; Tumor Cells, Cultured

2009
Reduced-intensity conditioning followed by peripheral blood stem cell transplantation for adult patients with high-risk acute lymphoblastic leukemia.
    Biology of blood and marrow transplantation : journal of the American Society for Blood and Marrow Transplantation, 2009, Volume: 15, Issue:11

    Topics: Adult; Aged; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Combined Modality Therapy; Dasatinib; Disease-Free Survival; Drug Administration Schedule; Female; Follow-Up Studies; Graft Survival; Graft vs Host Disease; Humans; Imatinib Mesylate; Male; Melphalan; Middle Aged; Myeloablative Agonists; Neoplasms, Second Primary; Peripheral Blood Stem Cell Transplantation; Piperazines; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Pyrimidines; Reoperation; Retrospective Studies; Risk; Thiazoles; Transplantation Conditioning; Transplantation, Homologous; Vidarabine; Young Adult

2009
The novel, proteasome-independent NF-kappaB inhibitor V1810 induces apoptosis and cell cycle arrest in multiple myeloma and overcomes NF-kappaB-mediated drug resistance.
    Molecular cancer therapeutics, 2010, Volume: 9, Issue:2

    Topics: Animals; Antineoplastic Agents; Apoptosis; Benzimidazoles; Cell Cycle; Cell Survival; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Humans; Inhibitory Concentration 50; Melphalan; Mice; Multiple Myeloma; NF-kappa B; Phosphorylation; Proteasome Endopeptidase Complex; Proteasome Inhibitors; Thiazoles

2010
By inhibiting Src, verapamil and dasatinib overcome multidrug resistance via increased expression of Bim and decreased expressions of MDR1 and survivin in human multidrug-resistant myeloma cells.
    Leukemia research, 2014, Volume: 38, Issue:1

    Topics: Animals; Antineoplastic Agents; Apoptosis Regulatory Proteins; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bcl-2-Like Protein 11; Blotting, Western; Cell Line; Cell Line, Tumor; Cell Survival; Dasatinib; Dexamethasone; Down-Regulation; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Synergism; Enzyme Activation; Humans; Inhibitor of Apoptosis Proteins; Melphalan; Membrane Proteins; Multiple Myeloma; Protein Kinase Inhibitors; Proto-Oncogene Proteins; Pyrimidines; src-Family Kinases; Survivin; Thiazoles; Up-Regulation; Verapamil

2014
SRC family kinase inhibition as a novel strategy to augment melphalan-based regional chemotherapy of advanced extremity melanoma.
    Annals of surgical oncology, 2014, Volume: 21, Issue:3

    Topics: Animals; Antineoplastic Agents, Alkylating; Apoptosis; Blotting, Western; Cell Proliferation; Dasatinib; Female; Humans; Melanoma; Melphalan; Mutation; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-kit; Pyrimidines; Rats; Rats, Nude; Real-Time Polymerase Chain Reaction; src-Family Kinases; Thiazoles; Tumor Cells, Cultured; Xenograft Model Antitumor Assays

2014
Surface-Modified Melphalan Nanoparticles for Intravitreal Chemotherapy of Retinoblastoma.
    Investigative ophthalmology & visual science, 2019, 04-01, Volume: 60, Issue:5

    Topics: Antineoplastic Agents, Alkylating; Coumarins; Drug Delivery Systems; Flow Cytometry; Humans; Intravitreal Injections; Melphalan; Microscopy, Electron, Scanning; Nanoparticles; Particle Size; Polylactic Acid-Polyglycolic Acid Copolymer; Retinal Neoplasms; Retinoblastoma; Thiazoles; Tumor Cells, Cultured

2019