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thiazoles and lg 100268

thiazoles has been researched along with lg 100268 in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (22.22)18.2507
2000's13 (72.22)29.6817
2010's1 (5.56)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bischoff, ED; Boehm, MF; Cesario, RM; Crombie, DL; Davies, PJ; Hamann, LG; Heyman, RA; Jow, L; Mondon, CE; Mukherjee, R; Nadzan, AM; Paterniti, JR1
Meier, CA1
Hirase, N; Mu, Y; Muta, K; Nawata, H; Takayanagi, R; Umemura, T; Yanase, T1
Mu, YM; Nawata, H; Nishi, Y; Oda, T; Takayanagi, R; Tanaka, A; Waseda, N; Yanase, T1
Breyer, MD; Breyer, RM; Davis, L; Guan, YF; Zhang, YH1
Cawthorne, MA; Crombie, DL; Heyman, RA; Hislop, DC; Liu, YL; Sennitt, MV1
Blanchard, SG; Gribble, GW; Honda, T; Leesnitzer, LM; Mangelsdorf, DJ; Plunket, KD; Porter, WW; Sporn, MB; Suh, N; Wang, Y; Willson, TM1
Cawthorne, MA; Emilsson, V; Heyman, R; Liu, YL; O'Dowd, J; Sennitt, M; Wang, S1
Boehm, M; Crombie, DL; Davies, PJ; Depre, C; Heyman, RA; Leibowitz, MD; Liu, S; Nagy, L; Singh Ahuja, H; Tontonoz, P1
Carter, L; Cha, BS; Ciaraldi, TP; Henry, RR; Mudaliar, S; Mukherjee, R; Nikoulina, SE; Paterniti, JR1
Goto, K; Mu, YM; Nawata, H; Nishi, Y; Takayanagi, R; Yanase, T1
Akanuma, Y; Ezaki, O; Fukayama, M; Hori, W; Ide, T; Itai, A; Kadowaki, T; Kagechika, H; Kamon, J; Kato, S; Kimura, S; Komeda, K; Kubota, N; Miki, H; Motojima, K; Murakami, K; Nagai, R; Shudo, K; Terauchi, Y; Tobe, K; Tsuboyama-Kasaoka, N; Tsuchida, A; Waki, H; Yamauchi, N; Yamauchi, T1
Charlton, SJ; Clapham, JC; Coxon, P; Macphee, CH; Marshall, IC; Moore, GB; Moores, K; Newman, SJ; Patel, L; Smith, SA1
Goto, K; Mu, YM; Nawata, H; Nishi, Y; Nomura, M; Okabe, T; Takayanagi, R; Yanase, T1
Blows, F; O'Rahilly, S; Sewter, CP; Vidal-Puig, A1
Domann, FE; Girnun, GD; Moore, SA; Robbins, ME1
Guo, SW; Wu, Y1
Decsi, T; Liebisch, G; Marosvölgyi, T; Mihály, J; Rühl, R; Schmitz, G; Weiss, K1

Reviews

1 review(s) available for thiazoles and lg 100268

ArticleYear
Novel pharmacological approaches to the prevention and treatment of non-insulin-dependent diabetes mellitus.
    European journal of endocrinology, 1997, Volume: 137, Issue:3

    Topics: Animals; Diabetes Mellitus, Type 2; Humans; Nicotinic Acids; Obesity; Tetrahydronaphthalenes; Thiazoles

1997

Other Studies

17 other study(ies) available for thiazoles and lg 100268

ArticleYear
Sensitization of diabetic and obese mice to insulin by retinoid X receptor agonists.
    Nature, 1997, Mar-27, Volume: 386, Issue:6623

    Topics: Animals; Bexarotene; Blood Glucose; Cells, Cultured; Diabetes Mellitus, Type 2; Female; Glucose Tolerance Test; Hypoglycemic Agents; Insulin; Insulin Resistance; Ligands; Mice; Mice, Inbred C57BL; Mice, Obese; Nicotinic Acids; Obesity; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Retinoid X Receptors; Rosiglitazone; Tetrahydronaphthalenes; Thiazoles; Thiazolidinediones; Transcription Factors; Transfection

1997
Thiazolidinedione induces apoptosis and monocytic differentiation in the promyelocytic leukemia cell line HL60.
    Oncology, 1999, Volume: 57 Suppl 2

    Topics: Antineoplastic Agents; Apoptosis; Blotting, Western; Cell Differentiation; Chromans; Drug Synergism; Gene Expression Regulation, Neoplastic; HL-60 Cells; Humans; Monocytes; Nicotinic Acids; Proto-Oncogene Proteins; Tetrahydronaphthalenes; Thiazoles; Thiazolidinediones; Troglitazone

1999
Insulin sensitizer, troglitazone, directly inhibits aromatase activity in human ovarian granulosa cells.
    Biochemical and biophysical research communications, 2000, May-19, Volume: 271, Issue:3

    Topics: Adult; Aromatase; Aromatase Inhibitors; Chromans; Dimerization; Enzyme Inhibitors; Estrogens; Female; Granulosa Cells; Humans; Nicotinic Acids; Ovary; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Retinoid X Receptors; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetrahydronaphthalenes; Thiazoles; Thiazolidinediones; Transcription Factors; Troglitazone

2000
Expression of peroxisome proliferator-activated receptor gamma (PPARgamma) in human transitional bladder cancer and its role in inducing cell death.
    Neoplasia (New York, N.Y.), 1999, Volume: 1, Issue:4

    Topics: Alitretinoin; Antineoplastic Agents; Apoptosis; Carcinoma, Transitional Cell; Carrier Proteins; Cell Death; Chromans; Cyclin D1; Cyclin-Dependent Kinase Inhibitor p16; Cyclin-Dependent Kinase Inhibitor p21; Cyclins; DNA; DNA, Complementary; Dose-Response Relationship, Drug; Fatty Acid-Binding Protein 7; Fatty Acid-Binding Proteins; G1 Phase; Humans; Immunoblotting; In Situ Hybridization; Ligands; Luciferases; Myelin P2 Protein; Neoplasm Proteins; Nicotinic Acids; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Retinoid X Receptors; Ribonucleases; Tetrahydronaphthalenes; Thiazoles; Thiazolidinediones; Transcription Factors; Transcriptional Activation; Transfection; Tretinoin; Troglitazone; Tumor Cells, Cultured; Tumor Suppressor Proteins; Urinary Bladder Neoplasms

1999
Retinoid X receptor agonists have anti-obesity effects and improve insulin sensitivity in Zucker fa/fa rats.
    International journal of obesity and related metabolic disorders : journal of the International Association for the Study of Obesity, 2000, Volume: 24, Issue:8

    Topics: Analysis of Variance; Animals; Blood Glucose; Body Weight; Eating; Hypoglycemic Agents; Insulin; Insulin Resistance; Male; Nicotinic Acids; Obesity; Rats; Rats, Zucker; Receptors, Retinoic Acid; Retinoid X Receptors; Rosiglitazone; Tetrahydronaphthalenes; Thiazoles; Thiazolidinediones; Transcription Factors

2000
A synthetic triterpenoid, 2-cyano-3,12-dioxooleana-1,9-dien-28-oic acid (CDDO), is a ligand for the peroxisome proliferator-activated receptor gamma.
    Molecular endocrinology (Baltimore, Md.), 2000, Volume: 14, Issue:10

    Topics: 3T3 Cells; Adipocytes; Animals; Cell Differentiation; CREB-Binding Protein; Drug Synergism; Ligands; Methylation; Mice; Nicotinic Acids; Nuclear Proteins; Nuclear Receptor Co-Repressor 1; Oleanolic Acid; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Repressor Proteins; Retinoid X Receptors; Rosiglitazone; Tetrahydronaphthalenes; Thiazoles; Thiazolidinediones; Trans-Activators; Transcription Factors; Transcriptional Activation

2000
The effects of rexinoids and rosiglitazone on body weight and uncoupling protein isoform expression in the Zucker fa/fa rat.
    Metabolism: clinical and experimental, 2000, Volume: 49, Issue:12

    Topics: Adipose Tissue, Brown; Animals; Body Weight; Carrier Proteins; Eating; Ion Channels; Membrane Proteins; Membrane Transport Proteins; Mitochondrial Proteins; Nicotinic Acids; Obesity; Proteins; Rats; Rats, Zucker; Receptors, Retinoic Acid; Retinoid X Receptors; RNA, Messenger; Rosiglitazone; Tetrahydronaphthalenes; Thiazoles; Thiazolidinediones; Transcription Factors; Uncoupling Protein 1; Uncoupling Protein 2; Uncoupling Protein 3; Weight Gain

2000
Differential effects of rexinoids and thiazolidinediones on metabolic gene expression in diabetic rodents.
    Molecular pharmacology, 2001, Volume: 59, Issue:4

    Topics: Adipose Tissue; Animals; Blood Glucose; Diabetes Mellitus; Diabetes Mellitus, Experimental; Disease Models, Animal; Gene Expression; Glucose Tolerance Test; Hyperglycemia; Hyperinsulinism; Hypoglycemic Agents; Liver; Male; Muscle, Skeletal; Nicotinic Acids; Obesity; Rats; Rats, Zucker; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Retinoid X Receptors; RNA, Messenger; Rosiglitazone; Tetrahydronaphthalenes; Thiazoles; Thiazolidinediones; Transcription Factors

2001
Peroxisome proliferator-activated receptor (PPAR) gamma and retinoid X receptor (RXR) agonists have complementary effects on glucose and lipid metabolism in human skeletal muscle.
    Diabetologia, 2001, Volume: 44, Issue:4

    Topics: CD36 Antigens; Chromans; Drug Synergism; Female; Glucose; Glycogen Synthase; Humans; Lipid Metabolism; Male; Middle Aged; Muscle, Skeletal; Nicotinic Acids; Oxidation-Reduction; Palmitic Acid; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Retinoid X Receptors; Tetrahydronaphthalenes; Thiazoles; Thiazolidinediones; Transcription Factors; Troglitazone

2001
Combined treatment with specific ligands for PPARgamma:RXR nuclear receptor system markedly inhibits the expression of cytochrome P450arom in human granulosa cancer cells.
    Molecular and cellular endocrinology, 2001, Jul-05, Volume: 181, Issue:1-2

    Topics: Aromatase; Cell Division; Chromans; Dactinomycin; Dose-Response Relationship, Drug; Down-Regulation; Enzyme Induction; Estrone; Female; Granulosa Cell Tumor; Humans; Ligands; Nicotinic Acids; Ovary; Promoter Regions, Genetic; Radioimmunoassay; Receptors, Cytoplasmic and Nuclear; Receptors, FSH; Receptors, Retinoic Acid; Retinoid X Receptors; RNA, Messenger; Tetrahydronaphthalenes; Thiazoles; Thiazolidinediones; Transcription Factors; Transcription, Genetic; Troglitazone; Tumor Cells, Cultured

2001
Inhibition of RXR and PPARgamma ameliorates diet-induced obesity and type 2 diabetes.
    The Journal of clinical investigation, 2001, Volume: 108, Issue:7

    Topics: 3T3 Cells; Adipose Tissue; Animals; Benzhydryl Compounds; Benzoates; Biphenyl Compounds; Diabetes Mellitus, Type 2; Epoxy Compounds; Fatty Acids; Hyperglycemia; Hypoglycemic Agents; Insulin Resistance; Leptin; Mice; Mice, Knockout; Nicotinic Acids; Obesity; Receptors, Adrenergic, beta-3; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Retinoid X Receptors; Rosiglitazone; Tetrahydronaphthalenes; Thiazoles; Thiazolidinediones; Transcription Factors

2001
PPARgamma is not a critical mediator of primary monocyte differentiation or foam cell formation.
    Biochemical and biophysical research communications, 2002, Jan-18, Volume: 290, Issue:2

    Topics: ATP Binding Cassette Transporter 1; ATP-Binding Cassette Transporters; CD36 Antigens; Cell Differentiation; Cells, Cultured; DNA-Binding Proteins; Dose-Response Relationship, Drug; Flow Cytometry; Foam Cells; Humans; Interleukin-6; Ligands; Light; Lipoproteins, LDL; Liver X Receptors; Macrophages; Matrix Metalloproteinase 9; Monocytes; Nicotinic Acids; Oligonucleotides, Antisense; Orphan Nuclear Receptors; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Retinoid X Receptors; RNA, Messenger; Rosiglitazone; Scattering, Radiation; Tetrahydronaphthalenes; Thiazoles; Thiazolidinediones; Transcription Factors

2002
Regulation of aromatase by nuclear receptors.
    The Journal of steroid biochemistry and molecular biology, 2001, Volume: 79, Issue:1-5

    Topics: Aromatase; Benzoates; Breast Neoplasms; Cholecalciferol; Chromans; Female; Gene Expression Regulation, Enzymologic; Gene Expression Regulation, Neoplastic; Granulosa Cells; Humans; Ligands; Nicotinic Acids; Receptors, Calcitriol; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Retinoid X Receptors; Retinoids; RNA, Messenger; RNA, Neoplasm; Tetrahydronaphthalenes; Thiazoles; Thiazolidinediones; Transcription Factors; Troglitazone; Tumor Cells, Cultured

2001
Regional differences in the response of human pre-adipocytes to PPARgamma and RXRalpha agonists.
    Diabetes, 2002, Volume: 51, Issue:3

    Topics: Adipocytes; Adult; Aged; Cell Differentiation; Female; Gene Expression; Humans; Hypoglycemic Agents; Ligands; Male; Middle Aged; Nicotinic Acids; Omentum; Polymerase Chain Reaction; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Retinoid X Receptors; RNA, Messenger; Rosiglitazone; Skin; Stem Cells; Tetrahydronaphthalenes; Thiazoles; Thiazolidinediones; Transcription Factors

2002
Identification of a functional peroxisome proliferator-activated receptor response element in the rat catalase promoter.
    Molecular endocrinology (Baltimore, Md.), 2002, Volume: 16, Issue:12

    Topics: Animals; Anticholesteremic Agents; Base Sequence; Catalase; Dimerization; Free Radical Scavengers; Gene Deletion; Gene Expression; Molecular Sequence Data; Mutagenesis; Organic Chemicals; Promoter Regions, Genetic; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Repetitive Sequences, Nucleic Acid; Response Elements; Retinoid X Receptors; RNA, Messenger; Rosiglitazone; Thiazoles; Thiazolidinediones; Transcription Factors; Transfection

2002
Peroxisome proliferator-activated receptor-gamma and retinoid X receptor agonists synergistically suppress proliferation of immortalized endometrial stromal cells.
    Fertility and sterility, 2009, Volume: 91, Issue:5 Suppl

    Topics: Cell Division; Cell Line; Endometrium; Estradiol; Female; Humans; Nicotinic Acids; PPAR gamma; Progesterone; Retinoid X Receptors; Stromal Cells; Tetrahydronaphthalenes; Tetrazolium Salts; Thiazoles; Thiazolidinediones

2009
Effect of synthetic ligands of PPAR α, β/δ, γ, RAR, RXR and LXR on the fatty acid composition of phospholipids in mice.
    Lipids, 2011, Volume: 46, Issue:11

    Topics: Acetyltransferases; Animals; Benzoates; Butyrates; Fatty Acid Elongases; Fatty Acids; Female; Gene Expression; Hydrocarbons, Fluorinated; Liver; Liver X Receptors; Mice; Mice, Inbred C57BL; Organic Chemicals; Orphan Nuclear Receptors; Peroxisome Proliferator-Activated Receptors; Phenylurea Compounds; Phospholipids; Receptors, Retinoic Acid; Rosiglitazone; Stearoyl-CoA Desaturase; Sulfonamides; Tetrahydronaphthalenes; Thiazoles; Thiazolidinediones

2011