thiazoles has been researched along with leukotriene d4 in 9 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 5 (55.56) | 18.2507 |
2000's | 4 (44.44) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Renzetti, LM; Wasserman, MA; Welton, AF | 1 |
Kadowaki, S; Nakao, E; Takahashi, K; Umezu, K; Yamada, K; Yamada, N | 1 |
Carlson, RP; Gray, WB; Grimes, D; Hartman, DA; Howell, RE; Jenkins, LP; Kreft, AF; Kubrak, D | 1 |
Maehr, H; Yang, R | 1 |
Arakida, Y; Honda, K; Miyata, K; Ohga, K; Suwa, K; Yamada, T; Yokota, M | 1 |
Kislalioglu, MS; Malick, AW; Mehta, KA; Phuapradit, W; Shah, NH | 2 |
Arakida, Y; Honda, K; Miyata, K; Morio, H; Ohga, K; Okada, Y; Suwa, K; Yamada, T; Yokota, M | 1 |
Hiyama, Y; Ishimura, M; Kataoka, S; Kurokawa, S; Maeda, T; Morizumi, K; Suda, M | 1 |
9 other study(ies) available for thiazoles and leukotriene d4
Article | Year |
---|---|
Synergism exhibited by LTD4 and PAF receptor antagonists in decreasing antigen-induced airway microvascular leakage.
Topics: Animals; Bronchi; Bronchodilator Agents; Drug Synergism; Guinea Pigs; Immunization; Leukotriene D4; Lung; Male; Microcirculation; Ovalbumin; Phenanthridines; Platelet Membrane Glycoproteins; Pulmonary Circulation; Receptors, Cell Surface; Receptors, G-Protein-Coupled; SRS-A; Thiazoles; Trachea; Triazines | 1995 |
Pharmacological profile of the novel, potent and selective peptide leukotriene antagonist (E)-2,2-diethyl-3'-[2-[2-(4-isopropyl)thiazolyl]ethenyl]succinanilic acid.
Topics: Acetylcholine; Animals; Bronchodilator Agents; Dose-Response Relationship, Drug; Guinea Pigs; Histamine Antagonists; Ileum; In Vitro Techniques; Leukotriene Antagonists; Leukotriene C4; Leukotriene D4; Male; Muscle Contraction; Muscle, Smooth; Penicillin G; Pyrilamine; Thiazoles; Trachea | 1994 |
Pulmonary pharmacology of WAY-126299A: a dual-acting 5-lipoxygenase inhibitor and leukotriene D4 antagonist.
Topics: Acetamides; Anesthesia; Animals; Benzothiazoles; Bronchoconstriction; Guinea Pigs; Humans; Hydroxyurea; In Vitro Techniques; Leukotriene D4; Lipoxygenase Inhibitors; Lung; Naphthaleneacetic Acids; Quinolines; Respiration, Artificial; Thiazoles | 1995 |
Structure optimization of a leukotriene D4 antagonist by combinatorial chemistry in solution.
Topics: Animals; Anti-Asthmatic Agents; Chemistry, Pharmaceutical; Guinea Pigs; Leukotriene D4; Muscle Contraction; Muscle, Smooth; Solutions; Thiazoles | 1997 |
In vitro pharmacologic profile of YM158, a new dual antagonist for LTD4 and TXA2 receptors.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Carbachol; Dinoprost; Guinea Pigs; Humans; In Vitro Techniques; Leukotriene Antagonists; Leukotriene D4; Male; Membrane Proteins; Muscle Contraction; Platelet Aggregation; Platelet Aggregation Inhibitors; Prostaglandin D2; Receptors, Leukotriene; Receptors, Thromboxane; Tetrazoles; Thiazoles; Trachea | 1998 |
Effect of formulation and process variables on porosity parameters and release rates from a multi unit erosion matrix of a poorly soluble drug.
Topics: Chemistry, Pharmaceutical; Delayed-Action Preparations; Drug Compounding; Leukotriene D4; Mercury; Polymethacrylic Acids; Porosity; Powders; Solubility; Surface Properties; Tablets; Thiazoles; Wettability | 2000 |
In vivo pharmacologic profile of YM158, a new dual antagonist for leukotriene D4 and thromboxane A2 receptors.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Airway Resistance; Animals; Anti-Asthmatic Agents; Dose-Response Relationship, Drug; Guinea Pigs; Leukotriene Antagonists; Leukotriene D4; Male; Receptors, Thromboxane; Tetrazoles; Thiazoles | 2000 |
Release performance of a poorly soluble drug from a novel, Eudragit-based multi-unit erosion matrix.
Topics: Acrylic Resins; Algorithms; Diffusion; Excipients; Leukotriene D4; Osmosis; Particle Size; Plasticizers; Polymethacrylic Acids; Solubility; Surface Properties; Temperature; Thiazoles | 2001 |
Effects of KP-496, a novel dual antagonist at the cysteinyl leukotriene receptor 1 and the thromboxane A(2) receptor, on airway obstruction in guinea pigs.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetates; Administration, Inhalation; Administration, Oral; Airway Obstruction; Animals; Anti-Asthmatic Agents; Benzoates; Benzoquinones; Bronchoconstriction; Cyclopropanes; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Therapy, Combination; Guinea Pigs; Heptanoic Acids; Leukotriene Antagonists; Leukotriene D4; Lung; Male; Membrane Proteins; Ovalbumin; Prostaglandin Antagonists; Quinolines; Receptors, Leukotriene; Receptors, Thromboxane A2, Prostaglandin H2; Respiratory Hypersensitivity; Sulfides; Thiazoles; Time Factors | 2008 |