thiazoles has been researched along with isomethyleugenol in 62 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 7 (11.29) | 18.7374 |
1990's | 8 (12.90) | 18.2507 |
2000's | 19 (30.65) | 29.6817 |
2010's | 26 (41.94) | 24.3611 |
2020's | 2 (3.23) | 2.80 |
Authors | Studies |
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Ankenbauer, RG; Cox, CD; Rinehart, KL; Staley, AL | 1 |
Fujiwara, M; Kobayashi, T; Shibata, K; Takayanagi, N; Yamamoto, I | 1 |
Bakke, JE; Feil, VJ; Huwe, JK; Larsen, GL | 1 |
Davis, WM; Khalsa, JH | 1 |
Jackson, JR; Stoodley, RJ | 1 |
Fennessy, MR; Gaff, GA; Heimans, RL | 1 |
Nohta, H; Noma, S; Ohkura, Y; Yoo, BT | 1 |
Cundliffe, E; Thompson, J | 1 |
Bortolan-Gianese, P; Dubini, F; Falchi, M; Ferrario, F; Marcucci, A | 1 |
Belajová, E; Bujdáková, H; Farkas, P; Kuchta, T; Léka, C; Russell, NJ | 1 |
Andreani, A; Benelli, B; Degli Esposti, M; Ghelli, A; Leoni, A; Locatelli, A; Rambaldi, M; Ratta, M | 1 |
Iinuma, H; Naganawa, H; Shimanaka, K; Takahashi, Y; Takeuchi, T | 1 |
D'Souza, T; Dryer, SE; Nowak, JZ; Sek, B | 1 |
Horie, T; Kakiki, M; Kozaki, T; Mishima, M; Naitoh, T; Yuzuriha, T | 1 |
Agúndez, JA; Albet, C; Benítez, J; Carrillo, JA; Herrero, E; Márquez, M; Martínez, C; Ortiz, JA | 1 |
Kongkittingam, C; Vedejs, E | 1 |
Burke, RM; Doig, AJ; Hughes, E | 1 |
Blanchard, SG; Gribble, GW; Honda, T; Leesnitzer, LM; Mangelsdorf, DJ; Plunket, KD; Porter, WW; Sporn, MB; Suh, N; Wang, Y; Willson, TM | 1 |
Gordon, DJ; Meredith, SC; Sciarretta, KL | 1 |
Häring, HU; Kausch, C; Machicao, F; Rett, K; Stumvoll, M; Wahl, HG | 1 |
Gastaldo, L; Marinelli, F | 1 |
Tang, W; Yao, Y | 1 |
Aboul-ela, F; Klinck, R; Lentzen, G; Matassova, N; Murchie, AI | 1 |
Abdel Aleem, AH; Abdel-Aal, MT; El Ashry, ES; El-Sayed, WA | 1 |
Colwell, LF; Gonzalez, EJ; Habulihaz, B; He, H; Leiting, B; Lyons, KA; Marsilio, F; Ok, HO; Parmee, ER; Patel, RA; Thornberry, NA; Weber, AE; Wu, JK; Xu, J | 1 |
Gnirss, R; Jekel, M; Kloepfer, A; Reemtsma, T | 1 |
Boltze, C; Diab-Assef, M; Foltzer-Jourdainne, C; Gali-Muhtasib, H; Hartig, R; Roessner, A; Rohrbeck, A; Schneider-Stock, R; Schönfeld, P | 1 |
Badis, M; Gauthier-Manuel, B; Heck, R; Marsura, A; Rogalska, E; Van der Heyden, A; Zywocinski, A | 1 |
Berliner, MA; Clark, MP; Nag, PP; Stroup, BW; Williams, DR | 1 |
Berg, M; de la Nava, EM; Dodge, JA; Evers, B; Hankotius, D; Hary, U; Jungheim, LN; Mest, HJ; Mohr, M; Muehl, BS; Petersen, S; Riedel-Herold, G; Ruehter, G; Sommer, B; Tebbe, MJ; Thrasher, KJ; Voelkers, S | 1 |
Berscheit, HL; Huang, AJ; Yuan, C | 1 |
Bacskay, I; Feher, P; Fenyvesi, E; Fenyvesi, F; Kiss, T; Kocsan, R; Pasztor, N; Szabo, G; Szente, L; Varadi, J; Vecsernyes, M | 1 |
Charro, N; Florencio, MH; Justino, GC; Mira, L; Rodríguez-Gómez, MJ; Santos, MR | 1 |
Apirakaramwong, A; Kowapradit, J; Ngawhiranpat, T; Opanasopit, P; Rojanarata, T; Ruktanonchai, U; Sajomsang, W | 1 |
Chen, D; Gong, R; Jia, X; Li, Z; Murchie, AI; Shen, Y; Wang, P; Wang, Z; Xu, Y; Yang, H; Yang, Y; Zhao, L; Zhou, P | 1 |
Alioua, A; Berr, A; Heintz, D; Heitz, T; McCallum, EJ; Shen, WH | 1 |
Almy, J; de Revel, G; Marchand, S | 1 |
Gómez-Vallejo, V; Llop, J | 1 |
Barré, P; Eliezer, D; Huster, D; Künze, G; Scheidt, HA; Thomas, L | 1 |
Kamel, AM; Obach, RS; Prakash, C | 1 |
Boateng, AA; Nsimba, RY; West, N | 1 |
Gong, T; Jia, SJ; Lai, YQ; Zhang, BK; Zhao, M | 1 |
Lawrence, HR; Lawrence, NJ; Mahajan, K; Mahajan, NP | 1 |
Deng, K; Katz, L; Keasling, JD; Petzold, CJ; Phelan, RM; Poust, S | 1 |
Bagdi, AK; Ghosh, M; Hajra, A; Monir, K | 1 |
Attanzio, A; Barraja, P; Carbone, A; Ciancimino, C; Cirrincione, G; Di Vita, G; Diana, P; Livrea, MA; Montalbano, A; Parrino, B; Spanò, V; Tesoriere, L | 1 |
Chen, D; Jiang, H; Murchie, AI; Yin, S | 1 |
Bednarek, MA; Bockus, AT; Lokey, RS; Pye, CR; Schwochert, JA; Sok, V; Townsend, CE | 1 |
Chen, F; Gao, AH; Gong, CJ; Li, J; Li, JY; Nan, FJ; Sheng, L; Su, MB; Zhang, YM; Zhou, YB | 1 |
Beijnen, JH; Fox, JA; Jamieson, G; Lucas, L; Nijenhuis, CM; Rosing, H; Schellens, JH | 1 |
Cao, LL; Ji, J; Sun, XL; Yang, DD; Zeng, XN; Zhang, L; Zhao, Z | 1 |
Chen, F; Deng, Z; Ding, W; Ji, X; Li, Y; Mo, T; Qianzhu, H; Tu, T; Yu, Y; Zhang, Q; Zhao, J | 1 |
Harada, A; Komatsu, T; Kudou, K; Maehara, K; Maehara, Y; Nogami, J; Ohkawa, Y; Oki, E; Saeki, H | 1 |
Badding, ED; Booker, SJ; Gadsby, LK; Grove, TL; LaMattina, JW; Wang, B | 2 |
Brigaud, T; Chaume, G; Lensen, N; Miclet, E; Pytkowicz, J; Simon, J | 1 |
Hudson, GA; Mahanta, N; Mitchell, DA; van der Donk, WA; Zhang, Z | 1 |
Cantu, EJ; Forester, SC; Grimes, KL; Kaur, B; McCarthy, JJ; Stuart, CM | 1 |
Booker, SJ; Lamb, AL; McFarlane, JS; Prisinzano, TE; Ronnebaum, TA | 1 |
Jin, WB; Tang, GL; Wu, S; Xu, YF; Yuan, H | 1 |
Brigaud, T; Chaume, G; Lensen, N; Malquin, N; Miclet, E; Rahgoshay, K | 1 |
Cowling, VH; Fordyce, EAF; Gray, DW; Green, CJ; Pearson, LA; Petit, AP | 1 |
1 review(s) available for thiazoles and isomethyleugenol
Article | Year |
---|---|
Recent advances in HemN-like radical S-adenosyl-l-methionine enzyme-catalyzed reactions.
Topics: Bacterial Proteins; Coproporphyrinogen Oxidase; Duocarmycins; Enzymes; Escherichia coli Proteins; Heme; Hydrogen; Methylation; Peptides, Cyclic; Polyketides; Protein Methyltransferases; S-Adenosylmethionine; Thiazoles | 2020 |
1 trial(s) available for thiazoles and isomethyleugenol
Article | Year |
---|---|
Comparative in vitro and in vivo inhibition of cytochrome P450 CYP1A2, CYP2D6, and CYP3A by H2-receptor antagonists.
Topics: Adult; Anti-Anxiety Agents; Antitussive Agents; Aryl Hydrocarbon Hydroxylases; Benzenesulfonates; Caffeine; Central Nervous System Stimulants; Cimetidine; Cytochrome P-450 CYP1A2 Inhibitors; Cytochrome P-450 CYP2D6 Inhibitors; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Dextromethorphan; Double-Blind Method; Histamine H2 Antagonists; Humans; In Vitro Techniques; Male; Methylation; Microsomes, Liver; Midazolam; Oxidoreductases, N-Demethylating; Psychomotor Performance; Ranitidine; Thiazoles | 1999 |
60 other study(ies) available for thiazoles and isomethyleugenol
Article | Year |
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Mutasynthesis of siderophore analogues by Pseudomonas aeruginosa.
Topics: Indicators and Reagents; Iron; Iron Chelating Agents; Magnetic Resonance Spectroscopy; Methylation; Molecular Structure; Phenols; Pseudomonas aeruginosa; Spectrophotometry, Infrared; Structure-Activity Relationship; Thiazoles | 1991 |
Immunomodulatory effect of a newly synthesized compound, TOK-8801 (N-(2-phenylethyl)-3,6,6-trimethyl-5,6-dihydroimidazo [2,1-b]thiazole-2-carboxamide) on antibody production in vivo and delayed-type hypersensitivity in mice.
Topics: Adjuvants, Immunologic; Animals; Antibody Formation; Antigens; Erythrocytes; Female; Humans; Hypersensitivity, Delayed; Imidazoles; Male; Methylation; Mice; Mice, Inbred C57BL; Mice, Inbred ICR; Serum Albumin; Sheep; Thiazoles | 1990 |
In vitro metabolism of the methylthio group of 2-methylthiobenzothiazole by rat liver.
Topics: Animals; Benzothiazoles; Chromatography, High Pressure Liquid; Chromatography, Thin Layer; Gas Chromatography-Mass Spectrometry; Glutathione; Glutathione Transferase; In Vitro Techniques; Liver; Methylation; Oxidation-Reduction; Rats; Sulfhydryl Compounds; Thiazoles | 1988 |
Morphine lethality in rats: effects of inhibitors of brain catecholamine synthesis and methylation.
Topics: Alcohols; Animals; Brain; Catechol O-Methyltransferase Inhibitors; Catecholamines; Cycloheptanes; Dopamine beta-Hydroxylase; Drug Synergism; Lethal Dose 50; Male; Methylation; Methyltyrosines; Morphine; Rats; Thiazoles; Thiourea; Time Factors; Tyrosine 3-Monooxygenase | 1973 |
Studies related to penicillins. VII. The structure of the epimers derived from 6 -substituted penicillanic acids.
Topics: Chemical Phenomena; Chemistry; Methylation; Nitriles; Penicillanic Acid; Penicillins; Stereoisomerism; Thiazoles | 1972 |
Some aspects of the metabolism of morphine-N-oxide.
Topics: Acridines; Analgesics; Animals; Codeine; Cyclic N-Oxides; In Vitro Techniques; Injections, Intraperitoneal; Liver; Male; Methylation; Morphinans; Morphine; Rats; Thiazoles | 1971 |
Assay for catechol-O-methyltransferase in erythrocytes using a new fluorogenic substrate, 2-(3,4-dihydroxyphenyl)naphtho[1,2-d]thiazole.
Topics: Benzothiazoles; Catechol O-Methyltransferase; Catechol O-Methyltransferase Inhibitors; Chromatography, High Pressure Liquid; Erythrocytes; Fluorescent Dyes; Humans; Hydrogen-Ion Concentration; In Vitro Techniques; Methylation; Pyrogallol; Spectrometry, Fluorescence; Thiazoles | 1984 |
The mode of action of nosiheptide (multhiomycin) and the mechanism of resistance in the producing organism.
Topics: Anti-Bacterial Agents; Bacterial Proteins; Drug Resistance, Microbial; Escherichia coli; Methylation; Pentoses; Peptide Elongation Factors; Ribosomes; Streptomyces; Thiazoles; Thiostrepton | 1981 |
[Transmethylating activity of arginine thiazolidinecarboxylate (ATCA) in acute CCL4 poisoning and diet-induced steatosis in the rat].
Topics: Animals; Arginine; Carbon Tetrachloride Poisoning; Chemical and Drug Induced Liver Injury; Diet; Fatty Liver; Male; Methylation; Rats; Thiazoles; Thiazolidines | 1980 |
Inhibition of sterol 4-demethylation in Candida albicans by 6-amino-2-n-pentylthiobenzothiazole, a novel mechanism of action for an antifungal agent.
Topics: Antifungal Agents; Candida albicans; Ergosterol; Methylation; Saccharomyces cerevisiae; Thiazoles | 1995 |
Thienylimidazo[2,1-b]thiazoles as inhibitors of mitochondrial NADH dehydrogenase.
Topics: Animals; Ascaridoidea; Cattle; Magnetic Resonance Spectroscopy; Methylation; Mitochondria; NADH Dehydrogenase; Structure-Activity Relationship; Thiazoles | 1995 |
Novel antibiotics, amythiamicins. II. Structure elucidation of amythiamicin D.
Topics: Acetylation; Anti-Bacterial Agents; Chemical Phenomena; Chemistry, Physical; Hydrochloric Acid; Hydrolysis; Macrocyclic Compounds; Magnetic Resonance Spectroscopy; Methylation; Molecular Structure; Spectrometry, Mass, Fast Atom Bombardment; Thiazoles | 1994 |
Does histamine stimulate cyclic AMP formation in the avian pineal gland via a novel (non-H1, non-H2, non-H3) histamine receptor subtype.
Topics: Animals; Benzothiazoles; Chickens; Cyclic AMP; Ducks; Histamine; Histamine Agonists; Histamine H2 Antagonists; Ion Channels; Male; Methylation; Phenoxypropanolamines; Pineal Gland; Piperidines; Receptors, Histamine; Stimulation, Chemical; Thiazoles | 1995 |
Identification of the metabolites of a new oxazolidinone MAO-A inhibitor in rat.
Topics: Animals; Benzothiazoles; Carbon Radioisotopes; Chromatography, High Pressure Liquid; Hydroxylation; Magnetic Resonance Spectroscopy; Male; Methylation; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Oxazoles; Oxazolidinones; Rats; Rats, Sprague-Dawley; Spectrometry, Mass, Fast Atom Bombardment; Thiazoles | 1997 |
Solution-phase synthesis of a hindered N-methylated tetrapeptide using Bts-protected amino acid chlorides: efficient coupling and methylation steps allow purification by extraction.
Topics: Acylation; Amino Acids; Benzothiazoles; Chlorides; Cyclosporine; Methylation; Oligopeptides; Sulfones; Thiazoles | 2000 |
Inhibition of toxicity in the beta-amyloid peptide fragment beta -(25-35) using N-methylated derivatives: a general strategy to prevent amyloid formation.
Topics: Amyloid beta-Peptides; Animals; Benzothiazoles; Cell Death; Coloring Agents; Congo Red; Dose-Response Relationship, Drug; Fluorescent Dyes; Methylation; Microscopy, Electron; PC12 Cells; Peptide Biosynthesis; Peptide Fragments; Protein Binding; Protein Conformation; Protein Folding; Protein Structure, Secondary; Rats; Spectrophotometry; Tetrazolium Salts; Thiazoles | 2000 |
A synthetic triterpenoid, 2-cyano-3,12-dioxooleana-1,9-dien-28-oic acid (CDDO), is a ligand for the peroxisome proliferator-activated receptor gamma.
Topics: 3T3 Cells; Adipocytes; Animals; Cell Differentiation; CREB-Binding Protein; Drug Synergism; Ligands; Methylation; Mice; Nicotinic Acids; Nuclear Proteins; Nuclear Receptor Co-Repressor 1; Oleanolic Acid; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Repressor Proteins; Retinoid X Receptors; Rosiglitazone; Tetrahydronaphthalenes; Thiazoles; Thiazolidinediones; Trans-Activators; Transcription Factors; Transcriptional Activation | 2000 |
Inhibition of beta-amyloid(40) fibrillogenesis and disassembly of beta-amyloid(40) fibrils by short beta-amyloid congeners containing N-methyl amino acids at alternate residues.
Topics: Alzheimer Disease; Amino Acid Sequence; Amino Acids; Amyloid beta-Peptides; Benzothiazoles; Chymotrypsin; Drug Resistance; Humans; Methylation; Microscopy, Fluorescence; Molecular Sequence Data; Peptide Fragments; Protein Structure, Secondary; Protein Structure, Tertiary; Thiazoles; Ultracentrifugation | 2001 |
Troglitazone downregulates delta-6 desaturase gene expression in human skeletal muscle cell cultures.
Topics: Adult; Cells, Cultured; Cholesterol Esters; Chromans; Dose-Response Relationship, Drug; Fatty Acid Desaturases; Female; Gene Amplification; Gene Expression Regulation, Enzymologic; Humans; Hypoglycemic Agents; Kinetics; Linoleoyl-CoA Desaturase; Male; Methylation; Muscle, Skeletal; Receptors, Cytoplasmic and Nuclear; Reference Values; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiazoles; Thiazolidinediones; Transcription Factors; Transcription, Genetic; Troglitazone | 2002 |
Changes in GE2270 antibiotic production in Planobispora rosea through modulation of methylation metabolism.
Topics: Actinomycetales; Adenosine; Anti-Bacterial Agents; Culture Media; Drug Interactions; Fermentation; Methionine; Methylation; Molecular Structure; Peptides; Peptides, Cyclic; Thiazoles; Vitamin B 12 | 2003 |
NMR investigation of the alkaline-like conformational transition of horse heart cytochrome c in the presence of exogenous thiazole.
Topics: Alkalies; Animals; Cytochromes c; Heart; Heme; Horses; Hydrogen-Ion Concentration; Isomerism; Ligands; Magnetic Resonance Spectroscopy; Methylation; Molecular Structure; Protein Conformation; Protons; Thiazoles; Titrimetry | 2003 |
Structural basis for contrasting activities of ribosome binding thiazole antibiotics.
Topics: Anti-Bacterial Agents; Bacteriocins; Base Sequence; Binding Sites; Guanosine Triphosphate; Hydrolysis; Magnetic Resonance Spectroscopy; Methylation; Methyltransferases; Models, Molecular; Molecular Sequence Data; Peptides; Protein Binding; Ribosomes; RNA, Ribosomal, 23S; Thiazoles; Thiostrepton | 2003 |
Synthesis of some functionalized arylaminomethyl-1 ,2,4-triazoles, 1,3,4-oxa- and thiadiazoles.
Topics: Antiviral Agents; Cell Line; Cell Survival; Drug Screening Assays, Antitumor; Enzyme-Linked Immunosorbent Assay; Hepatitis B virus; Humans; Indicators and Reagents; Magnetic Resonance Spectroscopy; Methylation; Oxazoles; Reverse Transcriptase Polymerase Chain Reaction; Thiazoles; Triazoles | 2003 |
Discovery of potent and selective beta-homophenylalanine based dipeptidyl peptidase IV inhibitors.
Topics: Aminobutyrates; Animals; Biological Availability; Dipeptidyl Peptidase 4; Half-Life; Methylation; Protease Inhibitors; Rats; Structure-Activity Relationship; Thiazoles | 2004 |
Occurrence of benzothiazoles in municipal wastewater and their fate in biological treatment.
Topics: Benzothiazoles; Bioreactors; Cities; Mass Spectrometry; Membranes, Artificial; Methylation; Sewage; Thiazoles; Time Factors; Waste Disposal, Fluid; Water Purification | 2004 |
5-Aza-cytidine is a potent inhibitor of DNA methyltransferase 3a and induces apoptosis in HCT-116 colon cancer cells via Gadd45- and p53-dependent mechanisms.
Topics: Annexin A5; Apoptosis; Azacitidine; Benzothiazoles; Blotting, Western; Cell Cycle Proteins; Cell Line, Tumor; Cell Proliferation; Cyclin-Dependent Kinase Inhibitor p21; DNA (Cytosine-5-)-Methyltransferases; DNA Methyltransferase 3A; DNA, Complementary; DNA, Neoplasm; Down-Regulation; Enzyme Inhibitors; Flow Cytometry; G2 Phase; GADD45 Proteins; Humans; In Situ Nick-End Labeling; Intracellular Signaling Peptides and Proteins; Methylation; Proteins; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiazoles; Toluene; Tumor Suppressor Protein p53 | 2005 |
Formation of Langmuir layers and surface modification using new upper-rim fully tethered bipyridinyl or bithiazolyl cyclodextrins and their fluorescent metal complexes.
Topics: Cyclodextrins; Fluorescence; Isomerism; Ligands; Metals; Methylation; Microscopy; Molecular Structure; Optical Devices; Pyridines; Thiazoles | 2004 |
Samarium Barbier reactions of alpha-iodomethyloxazoles and thiazoles with aliphatic aldehydes.
Topics: Aldehydes; Heterocyclic Compounds, 4 or More Rings; Iodine; Methylation; Molecular Structure; Oxazoles; Samarium; Thiazoles | 2005 |
Structure activity studies of the serine-AIB dipeptide domain in 2,3-dihydroisothiazole based growth hormone secretagogues.
Topics: Aminobutyrates; Animals; Carboxylic Acids; Cells, Cultured; Cross-Linking Reagents; Dipeptides; Growth Hormone; Male; Methylation; Molecular Structure; Phenanthrenes; Pituitary Gland; Rats; Rats, Sprague-Dawley; Serine; Structure-Activity Relationship; Thiazoles | 2005 |
Identification of an amyloidogenic region on keratoepithelin via synthetic peptides.
Topics: Amino Acid Sequence; Amyloid; Benzothiazoles; Circular Dichroism; Congo Red; Extracellular Matrix Proteins; Fluorescence; Humans; Methylation; Molecular Sequence Data; Mutation; Peptides; Protein Structure, Secondary; Thiazoles; Transforming Growth Factor beta | 2007 |
Cytotoxicity of different types of methylated beta-cyclodextrins and ionic derivatives.
Topics: Antineoplastic Agents; beta-Cyclodextrins; Cell Line, Tumor; Cell Survival; HeLa Cells; Humans; Indicators and Reagents; Methylation; Tetrazolium Salts; Thiazoles | 2007 |
Influence of the metabolic profile on the in vivo antioxidant activity of quercetin under a low dosage oral regimen in rats.
Topics: Animals; Antioxidants; Benzothiazoles; Chromatography, High Pressure Liquid; Glucuronides; Male; Methylation; Quercetin; Rats; Rats, Sprague-Dawley; Spectrometry, Mass, Electrospray Ionization; Sulfates; Sulfonic Acids; Thiazoles | 2008 |
Methylated N-(4-N,N-dimethylaminobenzyl) chitosan, a novel chitosan derivative, enhances paracellular permeability across intestinal epithelial cells (Caco-2).
Topics: Caco-2 Cells; Chitosan; Dextrans; Fluorescein-5-isothiocyanate; Humans; Hydrogen-Ion Concentration; Intestinal Absorption; Magnetic Resonance Spectroscopy; Methylation; Spectroscopy, Fourier Transform Infrared; Tetrazolium Salts; Thiazoles; Tight Junctions | 2008 |
Crystal structure of the nosiheptide-resistance methyltransferase of Streptomyces actuosus.
Topics: Binding Sites; Catalysis; Crystallography, X-Ray; Drug Resistance, Bacterial; Methylation; Methyltransferases; Protein Multimerization; RNA; Streptomyces; Substrate Specificity; Thiazoles | 2010 |
Arabidopsis histone methyltransferase SET DOMAIN GROUP8 mediates induction of the jasmonate/ethylene pathway genes in plant defense response to necrotrophic fungi.
Topics: Alternaria; Arabidopsis; Arabidopsis Proteins; Botrytis; Cyclopentanes; Ethylenes; Gene Expression Regulation, Plant; Histone Methyltransferases; Histone-Lysine N-Methyltransferase; Histones; Indoles; Methylation; Oxylipins; Plant Diseases; Plant Growth Regulators; Plant Immunity; Promoter Regions, Genetic; RNA, Plant; Thiazoles | 2010 |
The cysteine reaction with diacetyl under wine-like conditions: proposed mechanisms for mixed origins of 2-methylthiazole, 2-methyl-3-thiazoline, 2-methylthiazolidine, and 2,4,5-trimethyloxazole.
Topics: Acetaldehyde; Cysteine; Databases, Factual; Diacetyl; Gas Chromatography-Mass Spectrometry; Hexanones; Methylation; Models, Chemical; Oxazoles; Thiazoles; Volatile Organic Compounds; Wine | 2011 |
Fully automated and reproducible radiosynthesis of high specific activity [¹¹C]raclopride and [¹¹C]Pittsburgh compound-B using the combination of two commercial synthesizers.
Topics: Aniline Compounds; Carbon Radioisotopes; Hydrocarbons, Iodinated; Isotope Labeling; Mesylates; Methylation; Raclopride; Radiochemistry; Radiopharmaceuticals; Reproducibility of Results; Thiazoles | 2011 |
Binding of the three-repeat domain of tau to phospholipid membranes induces an aggregated-like state of the protein.
Topics: Alzheimer Disease; Amino Acid Sequence; Benzothiazoles; Biophysics; Circular Dichroism; Humans; Lipid Bilayers; Lipids; Liposomes; Lysine; Magnetic Resonance Spectroscopy; Methylation; Molecular Sequence Data; Phosphatidylcholines; Phosphatidylserines; Phospholipids; Protein Binding; Protein Conformation; Protein Structure, Secondary; Protein Structure, Tertiary; Static Electricity; tau Proteins; Thiazoles; Unilamellar Liposomes | 2012 |
Reduction and methylation of ziprasidone by glutathione, aldehyde oxidase, and thiol S-methyltransferase in humans: an in vitro study.
Topics: Aldehyde Oxidase; Antipsychotic Agents; Cytosol; Glutathione; Humans; Liver; Methylation; Methyltransferases; Microsomes, Liver; Oxidation-Reduction; Piperazines; Thiazoles | 2012 |
Structure and radical scavenging activity relationships of pyrolytic lignins.
Topics: Acetylation; Antioxidants; Benzothiazoles; Biphenyl Compounds; Free Radical Scavengers; Hot Temperature; Lignans; Magnetic Resonance Spectroscopy; Methylation; Picrates; Structure-Activity Relationship; Sulfonic Acids; Thiazoles | 2012 |
Homocysteine-induced hypermethylation of DDAH2 promoter contributes to apoptosis of endothelial cells.
Topics: Amidohydrolases; Annexin A5; Antimetabolites, Antineoplastic; Apoptosis; Azacitidine; Cell Survival; Coloring Agents; Endothelial Cells; Homocysteine; Methylation; Promoter Regions, Genetic; Real-Time Polymerase Chain Reaction; Repressor Proteins; Tetrazolium Salts; Thiazoles | 2013 |
ACK1 tyrosine kinase interacts with histone demethylase KDM3A to regulate the mammary tumor oncogene HOXA1.
Topics: Adaptor Proteins, Signal Transducing; Adaptor Proteins, Vesicular Transport; Amino Acid Sequence; Animals; Binding Sites; Cell Line, Tumor; Dasatinib; Drug Resistance, Neoplasm; Epigenesis, Genetic; Gene Expression Regulation, Neoplastic; Genes, Reporter; Humans; Jumonji Domain-Containing Histone Demethylases; Luciferases; Mammary Glands, Human; Methylation; Models, Molecular; Molecular Sequence Data; Neuregulin-1; Protein Binding; Protein-Tyrosine Kinases; Pyrimidines; Receptor, ErbB-2; Signal Transduction; Tamoxifen; Thiazoles; Transcription, Genetic | 2014 |
Divergent mechanistic routes for the formation of gem-dimethyl groups in the biosynthesis of complex polyketides.
Topics: Acyl Carrier Protein; Epothilones; Mass Spectrometry; Methylation; Phenols; Polyketide Synthases; Polyketides; Thiazoles | 2015 |
Regioselective oxidative trifluoromethylation of imidazoheterocycles via C(sp2)-H bond functionalization.
Topics: Catalysis; Hydrogen Bonding; Imidazoles; Methylation; Molecular Structure; Oxidation-Reduction; Pyridines; Stereoisomerism; Thiazoles | 2015 |
3-[4-(1H-indol-3-yl)-1,3-thiazol-2-yl]-1H-pyrrolo[2,3-b]pyridines, nortopsentin analogues with antiproliferative activity.
Topics: Alkaloids; Antineoplastic Agents; Apoptosis; Cell Line, Tumor; Cell Proliferation; Drug Design; G2 Phase; Halogenation; Humans; Imidazoles; Indoles; Membrane Potential, Mitochondrial; Methylation; Mitochondria; Molecular Structure; Neoplasms; Pyridines; Pyrroles; Resting Phase, Cell Cycle; Thiazoles | 2015 |
Substrate recognition and modification by the nosiheptide resistance methyltransferase.
Topics: Anti-Bacterial Agents; Binding Sites; Drug Resistance, Bacterial; Enzyme Activation; Methylation; Methyltransferases; Mutation; Nucleic Acid Conformation; Protein Binding; Protein Multimerization; RNA; Substrate Specificity; Thiazoles | 2015 |
Going Out on a Limb: Delineating The Effects of β-Branching, N-Methylation, and Side Chain Size on the Passive Permeability, Solubility, and Flexibility of Sanguinamide A Analogues.
Topics: Caco-2 Cells; Humans; Membranes, Artificial; Methylation; Molecular Dynamics Simulation; Peptides, Cyclic; Permeability; Solubility; Structure-Activity Relationship; Thiazoles; Water | 2015 |
Design, synthesis and biological evaluation of bisthiazole-based trifluoromethyl ketone derivatives as potent HDAC inhibitors with improved cellular efficacy.
Topics: Antineoplastic Agents; Cell Line, Tumor; Drug Design; Drug Screening Assays, Antitumor; Halogenation; Histone Deacetylase Inhibitors; Humans; Ketones; Methylation; Neoplasms; Structure-Activity Relationship; Thiazoles; Zinc | 2016 |
Quantification of vosaroxin and its metabolites N-desmethylvosaroxin and O-desmethylvosaroxin in human plasma and urine using high-performance liquid chromatography-tandem mass spectrometry.
Topics: Antineoplastic Agents; Body Fluids; Chemical Precipitation; Chromatography, High Pressure Liquid; Humans; Limit of Detection; Methylation; Naphthyridines; Reproducibility of Results; Tandem Mass Spectrometry; Thiazoles | 2016 |
PPARβ/δ activation protects against corticosterone-induced ER stress in astrocytes by inhibiting the CpG hypermethylation of microRNA-181a.
Topics: Animals; Astrocytes; Cell Survival; Cells, Cultured; Corticosterone; CpG Islands; Endoplasmic Reticulum Stress; Methylation; MicroRNAs; PPAR delta; PPAR-beta; Rats; Rats, Sprague-Dawley; Thiazoles | 2017 |
The Catalytic Mechanism of the Class C Radical S-Adenosylmethionine Methyltransferase NosN.
Topics: Anti-Bacterial Agents; Catalysis; Free Radicals; Methylation; Methyltransferases; Molecular Structure; S-Adenosylmethionine; Thiazoles | 2017 |
The requirement of Mettl3-promoted
Topics: 5' Untranslated Regions; Adenosine; Animals; Cell Differentiation; Cell Line; Cell Proliferation; ELAV-Like Protein 1; G2 Phase; Gene Expression Regulation; Methylation; Methyltransferases; Mice; Muscle Development; Muscle, Skeletal; Myoblasts; MyoD Protein; Quinolines; RNA, Small Interfering; S Phase; Signal Transduction; Thiazoles; Thymidine | 2017 |
NosN, a Radical S-Adenosylmethionine Methylase, Catalyzes Both C1 Transfer and Formation of the Ester Linkage of the Side-Ring System during the Biosynthesis of Nosiheptide.
Topics: Methylation; Methyltransferases; S-Adenosylhomocysteine; S-Adenosylmethionine; Thiazoles | 2017 |
Homochiral versus Heterochiral Trifluoromethylated Pseudoproline Containing Dipeptides: A Powerful Tool to Switch the Prolyl-Amide Bond Conformation.
Topics: Amides; Dipeptides; Fluorine; Methylation; Molecular Structure; Proline; Stereoisomerism; Thiazoles | 2017 |
Mechanism of a Class C Radical S-Adenosyl-l-methionine Thiazole Methyl Transferase.
Topics: Anti-Bacterial Agents; Deoxyadenosines; Hydrogen; Methylation; Methyltransferases; Peptides, Cyclic; Protons; S-Adenosylhomocysteine; S-Adenosylmethionine; Solvents; Thiazoles | 2017 |
Enhancing the Cancer Cell Growth Inhibitory Effects of Table Grape Anthocyanins.
Topics: Anthocyanins; Antineoplastic Agents, Phytogenic; Breast Neoplasms; Caco-2 Cells; Catechol O-Methyltransferase; Catechol O-Methyltransferase Inhibitors; Catechols; Cell Proliferation; Colonic Neoplasms; Drug Synergism; Female; Fruit; Glucosides; HT29 Cells; Humans; Methylation; Nitriles; Oxidative Stress; Phytotherapy; Plant Extracts; Tetrazolium Salts; Thiazoles; Vitis | 2018 |
Using Peptide Mimics to Study the Biosynthesis of the Side-Ring System of Nosiheptide.
Topics: Bacterial Proteins; Biosynthetic Pathways; Enzyme Assays; Methylation; Methyltransferases; Peptides; Recombinant Proteins; S-Adenosylmethionine; Streptomyces; Thiazoles | 2018 |
Stuffed Methyltransferase Catalyzes the Penultimate Step of Pyochelin Biosynthesis.
Topics: Bacterial Proteins; Catalysis; Catechol O-Methyltransferase; Escherichia coli; Kinetics; Methanocaldococcus; Methionine Adenosyltransferase; Methylation; Methyltransferases; Peptide Synthases; Phenols; Protein Domains; Pseudomonas aeruginosa; S-Adenosylmethionine; Thiazoles | 2019 |
CF
Topics: Hydrogen Bonding; Methylation; Molecular Conformation; Peptides; Proline; Stereoisomerism; Thiazoles; Toluene | 2019 |
Development of a High-Throughput Screening Assay to Identify Inhibitors of the SARS-CoV-2 Guanine-N7-Methyltransferase Using RapidFire Mass Spectrometry.
Topics: Antiparasitic Agents; Antiviral Agents; Cloning, Molecular; COVID-19; Drug Repositioning; Enzyme Assays; Enzyme Inhibitors; Escherichia coli; Exoribonucleases; Gene Expression; Genetic Vectors; High-Throughput Screening Assays; Humans; Kinetics; Mass Spectrometry; Methylation; Nitro Compounds; Prescription Drugs; Recombinant Fusion Proteins; RNA Caps; RNA, Viral; SARS-CoV-2; Small Molecule Libraries; Thiazoles; Viral Nonstructural Proteins; Virus Replication | 2021 |