thiazoles has been researched along with isatin in 12 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (8.33) | 18.2507 |
2000's | 2 (16.67) | 29.6817 |
2010's | 6 (50.00) | 24.3611 |
2020's | 3 (25.00) | 2.80 |
Authors | Studies |
---|---|
Gürsoy, A; Karali, N | 1 |
Glover, V; Igosheva, N; Lorz, C; Mehmet, H; O'Conner, E | 1 |
Hu, C; Lee, H; Solomon, VR | 1 |
Duan, W; Liu, L; Lou, G; Ma, S; Wang, W; Xue, F; Zhang, H; Zhang, S | 1 |
Ahmed, EM; Khalil, NA; Taher, AT | 1 |
Calvo, TR; Cândido-Bacani, Pde M; Cólus, IM; Mori, MP; Varanda, EA; Vilegas, W | 1 |
Farag, AA | 1 |
Bianco, G; Corona, A; Cottiglia, F; Distinto, S; Maccioni, E; Meleddu, R; Melis, C; Tramontano, E | 1 |
Chen, M; Chen, S; Deng, B; Li, L; Li, W; Peng, Y; Wang, G; Wang, J; Xie, Z | 1 |
Alberto de Simone, C; Alves Pereira, VR; Alves, LC; Barros Freitas, LA; Brayner, FA; Caroline da Silva Santos, A; de Cássia Silva, G; de Moraes Gomes, PAT; Lima Leite, AC; Nayara do Nascimento Albuquerque, F; Silva, ED | 1 |
Bhatia, S; Chigurupati, S; Felemban, SG; Jabeen, A; Khan, KM; Perveen, S; Qureshi, U; Saleem, F; Solangi, M; Taha, M; Ul-Haq, Z; Zafar, F | 1 |
Abouzid, KAM; Al-Hussain, SA; Albohy, A; Elleboudy, NS; Kassab, RM; Muhammad, ZA; Zaki, MEA | 1 |
12 other study(ies) available for thiazoles and isatin
Article | Year |
---|---|
Synthesis and anticonvulsant activity of some new thiosemicarbazone and 4-thiazolidone derivatives bearing an isatin moiety.
Topics: Animals; Anticonvulsants; Isatin; Magnetic Resonance Spectroscopy; Mice; Structure-Activity Relationship; Thiazoles; Thiosemicarbazones | 1994 |
Isatin, an endogenous monoamine oxidase inhibitor, triggers a dose- and time-dependent switch from apoptosis to necrosis in human neuroblastoma cells.
Topics: Annexin A5; Antiparkinson Agents; Apoptosis; Cell Cycle; Cell Line, Tumor; Cell Membrane Permeability; Cell Proliferation; Cell Survival; Dopamine; Dose-Response Relationship, Drug; Energy Metabolism; Humans; Isatin; Monoamine Oxidase Inhibitors; Necrosis; Neuroblastoma; Neurons; Neurotoxins; Parkinson Disease; Propidium; Tetrazolium Salts; Thiazoles; Time Factors | 2005 |
Hybrid pharmacophore design and synthesis of isatin-benzothiazole analogs for their anti-breast cancer activity.
Topics: Antineoplastic Agents; Benzothiazoles; Breast Neoplasms; Drug Design; Drug Screening Assays, Antitumor; Female; Humans; Indoles; Isatin; Thiazoles | 2009 |
Catalytic enantioselective Henry reactions of isatins: application in the concise synthesis of (S)-(-)-spirobrassinin.
Topics: Biological Products; Catalysis; Isatin; Molecular Structure; Spiro Compounds; Stereoisomerism; Thiazoles | 2011 |
Synthesis of novel isatin-thiazoline and isatin-benzimidazole conjugates as anti-breast cancer agents.
Topics: Antineoplastic Agents; Benzimidazoles; Breast Neoplasms; Cell Line, Tumor; Chromatography, Thin Layer; Drug Screening Assays, Antitumor; Female; Humans; Indicators and Reagents; Isatin; MCF-7 Cells; Spectrophotometry, Infrared; Spectrophotometry, Ultraviolet; Thiazoles | 2011 |
In vitro assessment of the cytotoxic, apoptotic, and mutagenic potentials of isatin.
Topics: Animals; Apoptosis; Cell Division; Cell Nucleus; Cell Survival; CHO Cells; Cricetinae; Cricetulus; DNA, Neoplasm; Dose-Response Relationship, Drug; Female; HeLa Cells; Humans; Isatin; Micronuclei, Chromosome-Defective; Micronucleus Tests; Mutagens; Plant Extracts; Plants, Medicinal; Tetrazolium Salts; Thiazoles | 2013 |
Synthesis and Antimicrobial Activity of 5-(morpholinosulfonyl)isatin Derivatives Incorporating a Thiazole Moiety.
Topics: Anti-Bacterial Agents; Antifungal Agents; Isatin; Microbial Sensitivity Tests; Structure-Activity Relationship; Thiazoles | 2015 |
Isatin thiazoline hybrids as dual inhibitors of HIV-1 reverse transcriptase.
Topics: Anti-HIV Agents; Dose-Response Relationship, Drug; HIV Reverse Transcriptase; HIV-1; Humans; Isatin; Microbial Sensitivity Tests; Models, Molecular; Molecular Structure; Reverse Transcriptase Inhibitors; Structure-Activity Relationship; Thiazoles | 2017 |
Synthesis, Biological Evaluation, and Molecular Docking Studies of Novel Isatin-Thiazole Derivatives as α-Glucosidase Inhibitors.
Topics: alpha-Glucosidases; Binding Sites; Glycoside Hydrolase Inhibitors; Isatin; Molecular Docking Simulation; Molecular Dynamics Simulation; Molecular Structure; Protein Binding; Structure-Activity Relationship; Thiazoles | 2017 |
Structural improvement of new thiazolyl-isatin derivatives produces potent and selective trypanocidal and leishmanicidal compounds.
Topics: Drug Design; Inhibitory Concentration 50; Isatin; Leishmania; Structure-Activity Relationship; Thiazoles; Trypanocidal Agents | 2021 |
Isatin thiazoles as antidiabetic: Synthesis, in vitro enzyme inhibitory activities, kinetics, and in silico studies.
Topics: alpha-Amylases; alpha-Glucosidases; Diabetes Mellitus; Glycoside Hydrolase Inhibitors; Humans; Hypoglycemic Agents; Isatin; Kinetics; Molecular Docking Simulation; Molecular Structure; Structure-Activity Relationship; Thiazoles | 2022 |
Tackling Microbial Resistance with Isatin-Decorated Thiazole Derivatives: Design, Synthesis, and in vitro Evaluation of Antimicrobial and Antibiofilm Activity.
Topics: Anti-Bacterial Agents; Anti-Infective Agents; Antifungal Agents; Biofilms; Escherichia coli; Isatin; Methicillin-Resistant Staphylococcus aureus; Microbial Sensitivity Tests; Molecular Docking Simulation; Staphylococcus aureus; Thiazoles | 2022 |