Page last updated: 2024-08-21

thiazoles and indole

thiazoles has been researched along with indole in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (5.88)18.2507
2000's3 (17.65)29.6817
2010's10 (58.82)24.3611
2020's3 (17.65)2.80

Authors

AuthorsStudies
Zook, M1
Bullington, JL; Jackson, PF1
Androsov, DA; Neckers, DC1
Billinton, A; Brown, SH; Chowdhury, A; Giblin, GM; Goldsmith, P; Hall, A; Hurst, DN; Naylor, A; Patel, S; Scoccitti, T; Theobald, PJ1
Dahal, BK; Ghofrani, HA; Grimminger, F; Kast, R; Kosanovic, D; Lai, YJ; Pamarthi, PK; Schermuly, RT; Schirok, H; Seeger, W; Stasch, JP; Sydykov, A; Weissmann, N1
Adam, JM; Baker, J; Bursi, R; Campbell, R; Clark, JK; Cottney, JE; Deehan, M; Easson, AM; Ecker, D; Edwards, D; Epemolu, O; Evans, L; Fields, R; Francis, S; Harradine, P; Jeremiah, F; Kiyoi, T; McArthur, D; Morrison, A; Passier, P; Pick, J; Ratcliffe, P; Schnabel, PG; Schulz, J; Steinbrede, H; Udo de Haes, J; Walker, G; Westwood, P; Wishart, G1
Angelucci, A; Botta, M; Brullo, C; Christopher, RS; Crespan, E; Delle Monache, S; Kissova, M; Maga, G; Mori, M; Musumeci, F; Radi, M; Sanità, P; Schenone, S; Tintori, C1
Diezel, C; Roth, C; Schön, M; Somssich, IE; Töller, A; Westphal, L; Wiermer, M1
Banothu, J; Bavantula, R; Crooks, PA; Gali, R; Gondru, R; Velivela, Y1
Cai, C; Gigolashvili, T; Guo, R; Jia, C; Liu, Y; Miao, H; Shao, Z; Sun, B; Wang, J; Wang, Q; Zhang, L; Zhao, Y1
Choi, SP; Jung, CK; Jung, SH; Kim, GT; Kim, TH; Lee, JY; Song, JU1
Attanzio, A; Barraja, P; Carbone, A; Cascioferro, S; Cirrincione, G; Diana, P; Montalbano, A; Parrino, B; Spanò, V; Tesoriere, L1
Deng, Z; Ding, W; Ji, W; Liu, WQ; Ma, X; Mo, T; Tang, B; Wu, R; Wu, Y; Xu, P; Yu, Y; Zhang, Q; Zhang, W; Zhao, J1
Awadallah, FM; Bua, S; Mahmoud, WR; Nada, HH; Nocentini, A; Supuran, CT1
Alves de Lima, MDC; Alves, JEF; de Almeida, SMV; de Carvalho Júnior, LB; de Lima Souza, TRC; de Moura, RO; de Oliveira, JF1
Finiuk, N; Garazd, M; Kashchak, N; Kryshchyshyn-Dylevych, A; Lesyk, R; Niemczuk, K; Posyniak, A; Radko, L; Stoika, R1
Acharya, SS; Bhaumick, P; Choudhury, LH; Kumar, R; Parvin, T1

Reviews

1 review(s) available for thiazoles and indole

ArticleYear
Pyridinylimidazole based p38 MAP kinase inhibitors.
    Current topics in medicinal chemistry, 2002, Volume: 2, Issue:9

    Topics: Animals; Antirheumatic Agents; Arthritis, Experimental; Drug Design; Enzyme Inhibitors; Humans; Imidazoles; Indoles; Mitogen-Activated Protein Kinases; Oxazoles; p38 Mitogen-Activated Protein Kinases; Pyridines; Structure-Activity Relationship; Thiazoles; Tumor Cells, Cultured

2002

Other Studies

16 other study(ies) available for thiazoles and indole

ArticleYear
Biosynthesis of camalexin from tryptophan pathway intermediates in cell-suspension cultures of Arabidopsis.
    Plant physiology, 1998, Volume: 118, Issue:4

    Topics: Arabidopsis; Ascomycota; Cells, Cultured; Indoles; Kinetics; ortho-Aminobenzoates; Plant Diseases; Thiazoles; Tryptophan

1998
Synthesis and reactivity of 4-(2-chloro-5-nitrophenyl)-1,2,3-thiadiazole. A novel one-pot synthesis of N-substituted indole-2-thiols.
    The Journal of organic chemistry, 2007, Jul-06, Volume: 72, Issue:14

    Topics: Indoles; Molecular Structure; Nitro Compounds; Sulfhydryl Compounds; Thiazoles

2007
Discovery of a novel indole series of EP1 receptor antagonists by scaffold hopping.
    Bioorganic & medicinal chemistry letters, 2008, Apr-15, Volume: 18, Issue:8

    Topics: Animals; Humans; Hydrogen Bonding; Indoles; Microsomes, Liver; Models, Molecular; Molecular Structure; Rats; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP1 Subtype; Structure-Activity Relationship; Thiazoles

2008
Therapeutic efficacy of azaindole-1 in experimental pulmonary hypertension.
    The European respiratory journal, 2010, Volume: 36, Issue:4

    Topics: Animals; Azabicyclo Compounds; Cell Proliferation; Disease Models, Animal; Enzyme Inhibitors; Hemodynamics; Hypertension, Pulmonary; Indoles; Lung; Male; Mice; Rats; Rats, Sprague-Dawley; rho-Associated Kinases; Telemetry; Tetrazolium Salts; Thiazoles; Thymidine; Treatment Outcome

2010
Design, synthesis and structure-activity relationships of (indo-3-yl) heterocyclic derivatives as agonists of the CB1 receptor. Discovery of a clinical candidate.
    Bioorganic & medicinal chemistry letters, 2011, Apr-15, Volume: 21, Issue:8

    Topics: Animals; Cytochrome P-450 Enzyme System; Dogs; Drug Design; Drug Evaluation, Preclinical; Heterocyclic Compounds; Indoles; Mice; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Structure-Activity Relationship; Thiazoles

2011
A combination strategy to inhibit Pim-1: synergism between noncompetitive and ATP-competitive inhibitors.
    ChemMedChem, 2013, Volume: 8, Issue:3

    Topics: Adenosine Triphosphate; Antineoplastic Agents; Binding Sites; Binding, Competitive; Cell Line, Tumor; Cell Survival; Crystallography, X-Ray; Humans; Indoles; Kinetics; Molecular Docking Simulation; Protein Binding; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-pim-1; Pyrroles; Recombinant Proteins; Structure-Activity Relationship; Thiazoles

2013
Analyses of wrky18 wrky40 plants reveal critical roles of SA/EDS1 signaling and indole-glucosinolate biosynthesis for Golovinomyces orontii resistance and a loss-of resistance towards Pseudomonas syringae pv. tomato AvrRPS4.
    Molecular plant-microbe interactions : MPMI, 2013, Volume: 26, Issue:7

    Topics: Arabidopsis; Arabidopsis Proteins; Ascomycota; Botrytis; Cyclopentanes; Disease Resistance; DNA-Binding Proteins; Gene Expression Regulation, Plant; Glucosinolates; Indoles; Mutation; Oomycetes; Oxylipins; Plant Diseases; Plant Growth Regulators; Plant Leaves; Plants, Genetically Modified; Pseudomonas syringae; Salicylic Acid; Signal Transduction; Thiazoles; Transcription Factors

2013
One-pot multicomponent synthesis of indole incorporated thiazolylcoumarins and their antibacterial, anticancer and DNA cleavage studies.
    Bioorganic & medicinal chemistry letters, 2015, Jan-01, Volume: 25, Issue:1

    Topics: Anti-Bacterial Agents; Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Coumarins; DNA Cleavage; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Humans; Indoles; Thiazoles

2015
Classic myrosinase-dependent degradation of indole glucosinolate attenuates fumonisin B1-induced programmed cell death in Arabidopsis.
    The Plant journal : for cell and molecular biology, 2015, Volume: 81, Issue:6

    Topics: Arabidopsis; Arabidopsis Proteins; Cell Death; Cytochrome P-450 Enzyme System; Fumonisins; Glucosinolates; Glycoside Hydrolases; Indoleacetic Acids; Indoles; Mutation; Thiazoles

2015
Design and synthesis of novel 2-(indol-5-yl)thiazole derivatives as xanthine oxidase inhibitors.
    Bioorganic & medicinal chemistry letters, 2015, Mar-15, Volume: 25, Issue:6

    Topics: Animals; Binding Sites; Drug Design; Enzyme Inhibitors; Half-Life; Hydrophobic and Hydrophilic Interactions; Indoles; Microsomes, Liver; Molecular Docking Simulation; Protein Binding; Protein Structure, Tertiary; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship; Thiazoles; Uric Acid; Xanthine Oxidase

2015
Synthesis and Antitumor Activity of New Thiazole Nortopsentin Analogs.
    Marine drugs, 2016, Dec-14, Volume: 14, Issue:12

    Topics: Antineoplastic Agents; Apoptosis; Cell Cycle; Cell Line, Tumor; Drug Screening Assays, Antitumor; HCT116 Cells; Humans; Imidazoles; Indoles; MCF-7 Cells; Thiazoles

2016
Biosynthesis of the nosiheptide indole side ring centers on a cryptic carrier protein NosJ.
    Nature communications, 2017, 09-05, Volume: 8, Issue:1

    Topics: Bacterial Proteins; Biosynthetic Pathways; Carrier Proteins; Indoles; Kinetics; Protein Binding; Streptomyces; Surface Plasmon Resonance; Thiazoles

2017
Inhibition studies on a panel of human carbonic anhydrases with N1-substituted secondary sulfonamides incorporating thiazolinone or imidazolone-indole tails.
    Journal of enzyme inhibition and medicinal chemistry, 2018, Volume: 33, Issue:1

    Topics: Carbonic Anhydrase Inhibitors; Carbonic Anhydrases; Dose-Response Relationship, Drug; Humans; Imidazoles; Indoles; Molecular Structure; Structure-Activity Relationship; Sulfonamides; Thiazoles

2018
Novel indole-thiazole and indole-thiazolidinone derivatives as DNA groove binders.
    International journal of biological macromolecules, 2021, Feb-15, Volume: 170

    Topics: Circular Dichroism; DNA; Ethidium; Fluorescent Dyes; Indoles; Molecular Docking Simulation; Spectrometry, Fluorescence; Thermodynamics; Thiazoles

2021
Synthesis of novel indole-thiazolidinone hybrid structures as promising scaffold with anticancer potential.
    Bioorganic & medicinal chemistry, 2021, 11-15, Volume: 50

    Topics: Animals; Antineoplastic Agents; Apoptosis; Cell Proliferation; Cells, Cultured; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Humans; Indoles; Mice; Mice, Inbred BALB C; Molecular Structure; Structure-Activity Relationship; Thiazoles

2021
Multicomponent Synthesis of Fluorescent Thiazole-Indole Hybrids and Thiazole-Based Novel Polymers.
    The Journal of organic chemistry, 2022, 09-02, Volume: 87, Issue:17

    Topics: Acetates; Indoles; Polymers; Thiazoles

2022