Page last updated: 2024-08-21

thiazoles and gw 610

thiazoles has been researched along with gw 610 in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bradshaw, TD; Choo, HL; Leong, CO; Muruhadas, A; Randhawa, N; Stevens, MF; Tan, BS; Tiong, KH1
Guengerich, FP; Wang, K1
Bradshaw, TD; Citossi, F; Farmer, PB; Gaskell, M; Hose, C; Kaur, B; Kellam, B; Leong, CO; Marlow, M; Monks, A; Singh, R; Stevens, MF; Stocks, M; Stone, EL1

Other Studies

3 other study(ies) available for thiazoles and gw 610

ArticleYear
CYP2S1 and CYP2W1 mediate 2-(3,4-dimethoxyphenyl)-5-fluorobenzothiazole (GW-610, NSC 721648) sensitivity in breast and colorectal cancer cells.
    Molecular cancer therapeutics, 2011, Volume: 10, Issue:10

    Topics: Antineoplastic Agents; Benzothiazoles; Breast Neoplasms; Cell Growth Processes; Cell Line, Tumor; Colorectal Neoplasms; Cytochrome P-450 CYP1A1; Cytochrome P-450 Enzyme System; Cytochrome P450 Family 2; Enzyme Induction; Female; Humans; Male; Thiazoles

2011
Bioactivation of fluorinated 2-aryl-benzothiazole antitumor molecules by human cytochrome P450s 1A1 and 2W1 and deactivation by cytochrome P450 2S1.
    Chemical research in toxicology, 2012, Aug-20, Volume: 25, Issue:8

    Topics: Antineoplastic Agents; Benzothiazoles; Biocatalysis; Chromatography, High Pressure Liquid; Cytochrome P-450 CYP1A1; Cytochrome P-450 Enzyme System; Cytochrome P450 Family 2; DNA Adducts; Humans; Kinetics; Microsomes, Liver; Oxidation-Reduction; Spectrometry, Mass, Electrospray Ionization; Thiazoles

2012
Antitumour benzothiazoles. Part 32: DNA adducts and double strand breaks correlate with activity; synthesis of 5F203 hydrogels for local delivery.
    Bioorganic & medicinal chemistry, 2015, Nov-01, Volume: 23, Issue:21

    Topics: Antineoplastic Agents; Benzothiazoles; Cell Line, Tumor; Cell Survival; Chromatography, High Pressure Liquid; Cytochrome P-450 CYP1A1; DNA Adducts; Drug Resistance, Neoplasm; Gene Expression Regulation; Histones; Humans; Hydrogels; Microscopy, Confocal; Prodrugs; Resveratrol; Stilbenes; Thiazoles

2015