Page last updated: 2024-08-21

thiazoles and glycine

thiazoles has been researched along with glycine in 80 studies

Research

Studies (80)

TimeframeStudies, this research(%)All Research%
pre-199019 (23.75)18.7374
1990's1 (1.25)18.2507
2000's22 (27.50)29.6817
2010's34 (42.50)24.3611
2020's4 (5.00)2.80

Authors

AuthorsStudies
Spenser, ID; White, RL1
Bellion, E; Faust, JR; Kirkley, DH1
Deutsch, HF; Fett, JW1
Burakowski, T; Muszyński, E; Pogorzelska-Lis, M1
Kumaoka, H; Morisaki, M; Saiki, K; Tazuya, K; Yamada, K1
de Waart, J; Knol, W1
Hatanaka, M; Ishimaru, T1
Herbertz, G; Reinauer, H1
Ellis, S; Fairwell, T; Lovins, RE1
Anderson, PJ; Gibson, D1
Iwashima, A; Kawasaki, T; Nakamura, M; Nose, Y1
Iwashima, A; Nose, Y2
Duggan, DE; Elfenbein, G; Pua, KH1
Linnett, PE; Walker, J2
Halpern, B; Westley, JW1
Diffey, BL; Hindson, TC1
Morimoto, Y; Nishikawa, K; Ohashi, M1
Kumaoka, H; Tanaka, K; Tazuya, K; Yamada, K1
Aukunuru, JV; Bandi, N; Kompella, UB; Sunkara, G; Thoreson, WB1
Dale, PJ; Moyes, C; Senior, IJ1
James, TL; Macdonald, JM; Schmidlin, O1
Du, HN; Hu, HY; Hu, J; Li, HT; Luo, XY; Tang, L; Zhou, JW1
Albrecht, J; Chlystun, M; Gozdz, A; Habas, A; Hetman, M; Jalili, A; Jaworski, J; Zielinska, M1
ROGERS, KT1
Bergeron, R; Gorfinkel, Y; Halman, S; Lowe, JA; Martina, M; Periyalwar, P; Schmidt, CJ1
Sebti, SM; Wang, DA1
Faden, AI; Lea, PM; Movsesyan, VA1
Sierra-Marcuño, G; Sierra-Paredes, G; Vázquez-López, A1
Keasling, JD; Muller, SJ; Wang, K1
Dong, LY; Lai, B; Sun, FY; Zhang, L; Zheng, P; Zhu, YH1
Alcaraz, L; Hughes, RA; Moody, CJ; Thompson, SP1
Ahmed, OA; Blagbrough, IS; Pourzand, C1
Ahmed, M; Aimoto, S; Constantinescu, SN; Elliott, JI; Kienlen-Campard, P; Li, H; Liu, W; Octave, JN; Sato, T; Smith, SO1
Cherney, MM; James, MN; Lemieux, MJ; Mahuran, DJ; Mark, BL; Withers, SG1
Baud, S; Keeley, FW; Miao, M; Pomès, R; Rauscher, S1
Gasparová, R; Lácová, M1
Lei, L; Li, Y; Liu, G; Liu, H; Ren, D; Wang, Y; Xu, J; Yang, H1
Chang, HY; King, CY; Lee, HC; Lin, JY; Wang, HL1
Clay, WC; Dean, DK; Michel, AD; Ng, SW; Roman, S; Walter, DS1
Carmi, C; Fu, J; King, AR; Lodola, A; Mor, M; Piomelli, D1
Butler, JD; Kurth, MJ; Mills, AD; Verkman, AS; Yang, B; Yoo, C1
Fukuda, S; Ito, M; Matsushita, M; Morinaga, H; Nakagawa, Y; Ohta, T; Sakata, S; Tanaka, M1
Albery-Larsdotter, S; Arlbrandt, S; Kjaer, MB; Ploj, K; Skantze, PM; Storlien, LH1
Beltramo, M; Brusa, R; Lozza, G; Mancini, I; Petrò, R; Reggiani, A; Scandroglio, P1
Ji, G; Li, Z; Neugebauer, V1
Ahemad, M; Khan, MS1
Chen, H; Gao, X; Guo, L; Jiang, X; Lai, R; Li, J; Qiu, M; Wu, H; Yan, X; Zhang, Q1
Steketee, JD; Timmer, KM1
Ludwig, C; Mootz, HD; Schwarzer, D; Thiel, IV1
McGinty, JF; Schwendt, M; Sigmon, SA1
Kalivas, PW; Knackstedt, L; Moussawi, K; Shen, H; Wang, X1
Byrnes, KR; Faden, AI; Loane, DJ; Stoica, BA; Zhang, J1
Christensen, MH; Kohlmeier, KA; Kristensen, MP; Kristiansen, U1
Conn, PJ; Kiritoshi, T; Lindsley, CW; Neugebauer, V; Ren, W; Stauffer, SR; Sun, H1
Bobermin, LD; de Souza, DF; Fontoura, JB; Gonçalves, CA; Hansen, F; Hoefel, AL; Leite, MC; Perry, ML; Silveira, Sda L; Tramontina, AC1
Ding, YH; Gong, J; Lan, R; Lin, G; Lu, F; Wang, J; Wang, Y; Xu, J; Yang, Z; Yin, F; Zhang, H; Zhang, X1
Chen, YR; Chiang, CH; Kuo, PH; Liang, JR; Shen, JC; Wang, S; Wang, YT; Yuan, HS1
Aras, P; Boily, M; Chagnon, M; Deblois, C; Sarrasin, B1
Charles, JR; Duva, MA; Lara, RL; Ramirez, GJ; Stanley, BG; Yang, CR1
Jones, HB; Martin, S; Page, C; Pickup, K; Rodrigues, A; Sarda, S; Wills, J; Wilson, I1
Arreola, AC; Kimmey, BA; Pierce, RC; Schmidt, HD1
Scheyer, AF; Tseng, KY; Wolf, ME1
Fukuda, S; Ito, M; Morinaga, H; Ohta, T; Sakata, S1
Chen, BP; Chen, W; Chern, Y; He, RY; Huang, JJ; Liu, GC; Sun, CS; Wang, CH; Wang, CY1
Akintola, T; Barrett, JP; Conn, PJ; Faden, AI; Kumar, A; Loane, DJ; Stoica, BA; Tchantchou, F; Xue, F1
Hayashi, M; Kijima, Y; Tazuya-Murayama, K; Yamada, K2
Ade, KK; Bhagat, S; Calakos, N; Conn, PJ; Dzirasa, K; Guo, W; Hamann, HC; Huber, KM; Kumar, S; O'Hare, JK; Quian, A; Rodriguiz, RM; Wan, Y; Wetsel, WC1
Abarca, J; Ferrada, C; Gysling, K; Sotomayor-Zárate, R1
Akasaka, R; Furukawa, A; Honda, K; Iwata, K; Kondo, M; Otsuki, K; Shimizu, K; Shinoda, M; Yonemoto, H1
Enkvist, E; Haljasorg, T; Lavogina, D; Mazina, O; Rahnel, H; Uri, A; Viht, K1
Bali, KK; Kuner, R1
Gong, G; Han, S; Hu, Y; Pan, J; Song, Z; Xie, L; Zhang, W1
Bargou, RC; Brünnert, D; Chatterjee, M; Driessen, C; Goyal, P; Heiden, R; Kirner, S; Kraus, M; Stühmer, T1
Gao, HY; Li, Y; Li, YT; Liu, MJ; Liu, P; Zhang, ZS; Zhao, SJ1
Khalesi, M; Saeb, M; Ziyaei Halimehjani, A1
Hayat, K; Ho, CT; Liu, M; Xu, H; Yu, J; Zhang, X; Zhou, T1
Brüning, T; Bury, D; Hayen, H; Käfferlein, HU; Koch, HM; Koslitz, S; Wrobel, SA1

Other Studies

80 other study(ies) available for thiazoles and glycine

ArticleYear
Thiamin biosynthesis in Saccharomyces cerevisiae. Origin of carbon-2 of the thiazole moiety.
    The Biochemical journal, 1979, May-01, Volume: 179, Issue:2

    Topics: Carbon Radioisotopes; Chemical Phenomena; Chemistry; Glycine; Methionine; Saccharomyces cerevisiae; Thiamine; Thiazoles; Tyrosine

1979
The biosynthesis of the thiazole moiety of thiamine in Salmonella Typhimurium.
    Biochimica et biophysica acta, 1976, Jun-23, Volume: 437, Issue:1

    Topics: Alanine; Glycine; Methionine; Salmonella typhimurium; Thiamine; Thiazoles; Tyrosine

1976
The variability of human lambda-chain constant regions and some relationships to V-regions sequences.
    Immunochemistry, 1976, Volume: 13, Issue:2

    Topics: Alanine; Amino Acid Sequence; Chromatography, Gel; Chromatography, Ion Exchange; Cystine; Electrophoresis, Paper; Glutamates; Glycine; Humans; Immunoglobulin lambda-Chains; Immunoglobulin Light Chains; Isoleucine; Leucine; Peptides; Proline; Serine; Thiazoles; Threonine; Valine

1976
[Synthesis of (N-(4-aminobenzenesulfonyl)-N-(2'-thiazolyl)-aminoacetic acid and some of its derivatives].
    Acta poloniae pharmaceutica, 1976, Volume: 33, Issue:1

    Topics: Aniline Compounds; Chemical Phenomena; Chemistry; Esters; Glycine; Thiazoles

1976
Biosynthesis of thiamin. Different biosynthetic routes of the thiazole moiety of thiamin in aerobic organisms and anaerobic organisms.
    Biochemistry international, 1987, Volume: 14, Issue:1

    Topics: Bacteria; Bacteria, Aerobic; Bacteria, Anaerobic; Glycine; Thiamine; Thiazoles; Tyrosine

1987
A comparative evaluation of Baird-Parker's ETGPA- and the KRANEP-medium for the selective enumeration of Staphylococcus aureus in foods.
    Zentralblatt fur Bakteriologie, Parasitenkunde, Infektionskrankheiten und Hygiene. Erste Abteilung Originale. Reihe A: Medizinische Mikrobiologie und Parasitologie, 1972, Volume: 219, Issue:2

    Topics: Azides; Bacteriological Techniques; Culture Media; Cycloheximide; Egg Yolk; Female; Food Microbiology; Glycine; Micrococcus; Pyruvates; Staphylococcus; Thiazoles

1972
Synthetic penicillins. Heterocyclic analogs of ampicillin. Structure-activity relationships.
    Journal of medicinal chemistry, 1973, Volume: 16, Issue:9

    Topics: Ampicillin; Bacillus subtilis; Chromatography, Paper; Escherichia coli; Glycine; Microbial Sensitivity Tests; Penicillins; Salmonella enteritidis; Shigella dysenteriae; Spectrophotometry, Infrared; Staphylococcus; Structure-Activity Relationship; Thiazoles; Thiophenes

1973
[Metabolism of chlormethiazol in the rat].
    Naunyn-Schmiedebergs Archiv fur Pharmakologie, 1971, Volume: 270, Issue:2

    Topics: Ammonia; Animals; Chlormethiazole; Chloroform; Chromatography, Thin Layer; Electrophoresis; Glycine; Methanol; Rats; Thiazoles

1971
Quantitative protein sequencing using mass spectrometry: N-terminal sequence analysis of small quantities of peptides from the mass spectral analysis of the N-methylthiourea derivatives.
    Biochemical and biophysical research communications, 1972, Dec-18, Volume: 49, Issue:6

    Topics: Alanine; Amino Acid Sequence; Amino Acids; Chemical Phenomena; Chemistry; Cyclization; Evaluation Studies as Topic; Fluoroacetates; Glutamates; Glycine; Hot Temperature; Hydantoins; Mass Spectrometry; Methods; Methylamines; Oligopeptides; Peptides; Phenylalanine; Proteins; Thiazoles; Thiocyanates; Thiourea; Volatilization

1972
Carboxyl group modification and amide assignments in automated sequencing of proteins.
    Biochemical and biophysical research communications, 1972, Oct-17, Volume: 49, Issue:2

    Topics: Amino Acid Sequence; Amino Acids; Asparagine; Aspartic Acid; Chemical Phenomena; Chemistry; Esters; Glutamates; Glutamine; Glycine; Hydrolysis; Imines; Methanol; Methods; Methylamines; Ribonucleases; Serine; Thiazoles

1972
Effect of amino acids and purine bases on thiamine synthesis by Escherichia coli.
    The Journal of vitaminology, 1968, Sep-10, Volume: 14, Issue:3

    Topics: Adenine; Amino Acids; Aspartic Acid; Culture Media; Cystine; Cytosine; Escherichia coli; Glutamates; Glycine; Guanine; Histidine; Hypoxanthines; Inositol; Isoleucine; Leucine; Methionine; Phenylalanine; Proline; Purines; Serine; Thiamine; Thiazoles; Threonine; Thymine; Tyrosine; Uracil; Valine

1968
Effect of glycine on thiazole biosynthesis in Escherichia coli.
    Journal of bacteriology, 1970, Volume: 101, Issue:3

    Topics: Escherichia coli; Genetics, Microbial; Glycine; Mutation; Thiamine; Thiazoles

1970
Incorporation of glycine in pyrimidine and thiazole moieties of thiamine in Escherichia coli.
    Biochimica et biophysica acta, 1971, Nov-12, Volume: 252, Issue:2

    Topics: Adenine; Alcohols; Carbon Isotopes; Chromatography, Ion Exchange; Escherichia coli; Genetics, Microbial; Glycine; Mutation; Phenylalanine; Pyrimidines; Thiamine; Thiazoles

1971
Purine metabolism in the chick embryo; effects of uricogenesis and xanthine oxidase inhibition.
    Molecular pharmacology, 1968, Volume: 4, Issue:1

    Topics: Adenine; Amines; Animals; Carbon Isotopes; Chick Embryo; Formates; Glycine; Guanine; Nucleic Acids; Nucleotides; Purines; Pyrazoles; Pyrimidines; Thiazoles; Uric Acid; Xanthine Oxidase

1968
Biosynthesis of thiamine. Incorporation experiments with 14C-labelled substrates and with (15N)glycine in Saccharomyces cerevisiae.
    The Biochemical journal, 1968, Volume: 109, Issue:2

    Topics: Acetates; Carbon Isotopes; Formates; Glycine; Methionine; Nitrogen; Pyrimidines; Radioisotopes; Saccharomyces; Serine; Thiamine; Thiazoles

1968
Biosynthesis of thiamin. IV. C-2 of glycine as the precursor of C-2 of the thiazole moiety in yeast.
    Biochimica et biophysica acta, 1969, Jul-30, Volume: 184, Issue:2

    Topics: Carbon Isotopes; Chemical Phenomena; Chemistry; Formaldehyde; Formates; Glycine; Methionine; Models, Biological; Saccharomyces; Serine; Sulfonic Acids; Thiamine; Thiazoles

1969
Optical resolution of D,L amino acids by gas chromatography and mass spectrometry.
    Biochemical and biophysical research communications, 1965, Sep-22, Volume: 20, Issue:6

    Topics: Alanine; Amino Acids; Aminobutyrates; Chemical Phenomena; Chemistry, Physical; Chromatography, Gas; Glycine; Leucine; Proline; Spectrum Analysis; Thiazoles

1965
Phototoxicity of a weedkiller: a correction.
    Contact dermatitis, 1984, Volume: 11, Issue:4

    Topics: Glycine; Glyphosate; Herbicides; Humans; Photosensitivity Disorders; Thiazoles

1984
KB-R7785, a novel matrix metalloproteinase inhibitor, exerts its antidiabetic effect by inhibiting tumor necrosis factor-alpha production.
    Life sciences, 1997, Volume: 61, Issue:8

    Topics: Animals; Blood Glucose; Body Weight; Glycine; Hydroxamic Acids; Hypoglycemic Agents; Insulin; Insulin Resistance; Male; Metalloendopeptidases; Mice; Mice, Inbred BALB C; Pioglitazone; Protease Inhibitors; Thiazoles; Thiazolidinediones; Tumor Necrosis Factor-alpha

1997
Biosynthesis of thiamin under anaerobic conditions in Saccharomyces cerevisiae.
    Biological & pharmaceutical bulletin, 2000, Volume: 23, Issue:1

    Topics: Aerobiosis; Anaerobiosis; Carbon Radioisotopes; Formates; Glycine; Mass Spectrometry; Nitrogen Isotopes; Oxygen; Pyridoxine; Pyrimidines; Saccharomyces cerevisiae; Thiamine; Thiazoles

2000
Expression of multidrug resistance-associated protein (MRP) in human retinal pigment epithelial cells and its interaction with BAPSG, a novel aldose reductase inhibitor.
    Pharmaceutical research, 2001, Volume: 18, Issue:5

    Topics: Aldehyde Reductase; Antimetabolites; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Cell Line; Cold Temperature; Enzyme Inhibitors; Epithelial Cells; Fluorescein; Glycine; Humans; Indicators and Reagents; Pigment Epithelium of Eye; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sulfones; Tetrazolium Salts; Thiazoles

2001
Herbicide sensitivity of transgenic multiple herbicide-tolerant oilseed rape.
    Pest management science, 2002, Volume: 58, Issue:4

    Topics: 2-Methyl-4-chlorophenoxyacetic Acid; Aminobutyrates; Arylsulfonates; Brassica napus; Glycine; Glyphosate; Herbicides; Paraquat; Plants, Genetically Modified; Risk Assessment; Thiazoles

2002
In vivo monitoring of hepatic glutathione in anesthetized rats by 13C NMR.
    Magnetic resonance in medicine, 2002, Volume: 48, Issue:3

    Topics: Animals; Carbon Isotopes; Female; Glutathione; Glycine; Liver; Magnetic Resonance Spectroscopy; Pyrrolidonecarboxylic Acid; Rats; Rats, Sprague-Dawley; Thiazoles; Thiazolidines

2002
A peptide motif consisting of glycine, alanine, and valine is required for the fibrillization and cytotoxicity of human alpha-synuclein.
    Biochemistry, 2003, Jul-29, Volume: 42, Issue:29

    Topics: Alanine; alpha-Synuclein; Amino Acid Motifs; Benzothiazoles; Circular Dichroism; Escherichia coli; Glycine; Humans; Microscopy, Atomic Force; Mutagenesis, Site-Directed; Mutation; Nerve Tissue Proteins; Peptides; Protein Binding; Protein Structure, Secondary; Protein Structure, Tertiary; Recombinant Proteins; Synucleins; Thiazoles; Time Factors; Valine

2003
Role of N-methyl-D-aspartate receptors in the neuroprotective activation of extracellular signal-regulated kinase 1/2 by cisplatin.
    The Journal of biological chemistry, 2003, Oct-31, Volume: 278, Issue:44

    Topics: Adenosine Triphosphate; Animals; Animals, Newborn; Antineoplastic Agents; Apoptosis; Blotting, Western; Brain; Caspases; Cells, Cultured; Cisplatin; Coloring Agents; DNA Fragmentation; Dose-Response Relationship, Drug; Enzyme Activation; Genes, Dominant; Glutamic Acid; Glycine; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Mutation; Neurons; Poly(ADP-ribose) Polymerases; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Signal Transduction; Tetrazolium Salts; Thiazoles; Time Factors; Transfection

2003
RODIOAUTOGRAPHIC ANALYSIS OF THE INCORPORATION OF PROTEIN AND NUCLEIC ACID PRECURSORS INTO VARIOUS TISSUES OF EARLY CHICK EMBRYOS CULTURED IN TOTO ON MEDIUM CONTAINING LICL.
    Developmental biology, 1964, Volume: 9

    Topics: Adenine; Autoradiography; Carbon Isotopes; Chick Embryo; Chlorides; Glycine; Lithium; Methionine; Nucleic Acid Precursors; Nucleosides; Proteins; Quinolinium Compounds; Research; RNA; Sodium Chloride; Spectrophotometry; Thiazoles; Tissue Culture Techniques; Tritium

1964
Glycine transporter type 1 blockade changes NMDA receptor-mediated responses and LTP in hippocampal CA1 pyramidal cells by altering extracellular glycine levels.
    The Journal of physiology, 2004, Jun-01, Volume: 557, Issue:Pt 2

    Topics: Acetates; Amino Acid Transport Systems, Neutral; Animals; Glycine; Glycine Plasma Membrane Transport Proteins; Hippocampus; In Vitro Techniques; Long-Term Potentiation; Male; Patch-Clamp Techniques; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Sarcosine; Thiazoles

2004
Palmitoylated cysteine 192 is required for RhoB tumor-suppressive and apoptotic activities.
    The Journal of biological chemistry, 2005, May-13, Volume: 280, Issue:19

    Topics: Alanine; Amino Acid Sequence; Apoptosis; Blotting, Western; Cell Cycle Proteins; Cell Line; Cell Line, Tumor; Cell Proliferation; Coloring Agents; Cyclin-Dependent Kinase Inhibitor p21; Cysteine; DNA Primers; Genes, Tumor Suppressor; Glycine; Humans; In Situ Nick-End Labeling; Molecular Sequence Data; Mutagenesis, Site-Directed; Mutation; Palmitic Acid; Promoter Regions, Genetic; Protein Biosynthesis; Protein Prenylation; rhoA GTP-Binding Protein; rhoB GTP-Binding Protein; Sequence Homology, Amino Acid; Serine; Tetrazolium Salts; Thiazoles; Transcription Factor AP-1; Transcription, Genetic; Transfection; Transforming Growth Factor beta

2005
Neuroprotective activity of the mGluR5 antagonists MPEP and MTEP against acute excitotoxicity differs and does not reflect actions at mGluR5 receptors.
    British journal of pharmacology, 2005, Volume: 145, Issue:4

    Topics: Animals; Apoptosis; Cell Survival; Cells, Cultured; Cerebral Cortex; Dizocilpine Maleate; Dose-Response Relationship, Drug; Etoposide; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Female; Glutamic Acid; Glycine; Hydrolysis; Male; Membrane Potentials; Mice; Mice, Knockout; N-Methylaspartate; Neurons; Neuroprotective Agents; Phenylacetates; Phosphatidylinositols; Pyridines; Rats; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Thiazoles

2005
Seizures induced by microperfusion of glutamate and glycine in the hippocampus of rats pretreated with latrunculin A.
    Neuroscience letters, 2005, Nov-11, Volume: 388, Issue:2

    Topics: Animals; Bridged Bicyclo Compounds, Heterocyclic; Dizocilpine Maleate; Drug Interactions; Epilepsy; Excitatory Amino Acid Antagonists; Glutamic Acid; Glycine; Hippocampus; Male; Microdialysis; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Thiazoles; Thiazolidines

2005
Effects of the sequence and size of non-polar residues on self-assembly of amphiphilic peptides.
    International journal of biological macromolecules, 2005, Sep-15, Volume: 36, Issue:4

    Topics: Alanine; Amino Acid Motifs; Amyloid; Benzothiazoles; Circular Dichroism; Congo Red; Gene Library; Glycine; Hydrogel, Polyethylene Glycol Dimethacrylate; Isoleucine; Leucine; Macromolecular Substances; Microscopy, Electron, Scanning; Microscopy, Electron, Transmission; Models, Molecular; Peptides; Phenylalanine; Protein Binding; Protein Conformation; Protein Folding; Protein Structure, Secondary; Temperature; Thiazoles; Ultraviolet Rays; Valine; X-Ray Diffraction

2005
Impact of inhibition of Qo site of mitochondrial complex III with myxothiazol on persistent sodium currents via superoxide and protein kinase C in rat hippocampal CA1 cells.
    Neurobiology of disease, 2006, Volume: 21, Issue:1

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Alkaloids; Animals; Antifungal Agents; Benzophenanthridines; Cyclic AMP-Dependent Protein Kinases; Electron Transport Complex I; Electron Transport Complex III; Enzyme Activation; Enzyme Inhibitors; Free Radical Scavengers; Glycine; Hippocampus; Hydroxyl Radical; Hypoxia, Brain; Isoquinolines; Metalloporphyrins; Methacrylates; Mitochondria; Patch-Clamp Techniques; Phenanthridines; Protein Kinase C; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Sodium; Sulfhydryl Compounds; Sulfonamides; Superoxides; Thiazoles

2006
Total synthesis of the thiopeptide antibiotic amythiamicin D.
    Journal of the American Chemical Society, 2005, Nov-09, Volume: 127, Issue:44

    Topics: Anti-Bacterial Agents; Cyclization; Glycine; Macrocyclic Compounds; Pyridines; Thiazoles

2005
Varying the unsaturation in N4,N9-dioctadecanoyl spermines: nonviral lipopolyamine vectors for more efficient plasmid DNA formulation.
    Pharmaceutical research, 2006, Volume: 23, Issue:1

    Topics: Cell Line; Cell Line, Tumor; Cell Survival; Cells, Cultured; Chemistry, Pharmaceutical; DNA; Drug Carriers; Electrochemistry; Fatty Acids; Glycine; Humans; Indicators and Reagents; Nanostructures; Particle Size; Plasmids; Skin; Spermine; Tetrazolium Salts; Thiazoles; Transfection

2006
Inhibitors of amyloid toxicity based on beta-sheet packing of Abeta40 and Abeta42.
    Biochemistry, 2006, May-02, Volume: 45, Issue:17

    Topics: Amino Acid Sequence; Amyloid; Amyloid beta-Peptides; Animals; Benzothiazoles; Fluorescent Dyes; Glycine; Humans; Methionine; Microscopy, Electron; Molecular Sequence Data; Neurons; Nuclear Magnetic Resonance, Biomolecular; Oligopeptides; Peptide Fragments; Protein Structure, Secondary; Protein Structure, Tertiary; Rats; Spectrometry, Fluorescence; Thiazoles

2006
Crystallographic structure of human beta-hexosaminidase A: interpretation of Tay-Sachs mutations and loss of GM2 ganglioside hydrolysis.
    Journal of molecular biology, 2006, Jun-16, Volume: 359, Issue:4

    Topics: Acetylglucosamine; Amino Acid Substitution; Arginine; Aspartic Acid; beta-N-Acetylhexosaminidases; Binding Sites; Crystallography, X-Ray; Dimerization; Gangliosidoses, GM2; Glycine; Glycosylation; Hexosaminidase A; Humans; Hydrolysis; Models, Molecular; Mutation; Protein Conformation; Protein Subunits; Tay-Sachs Disease; Thiazoles

2006
Proline and glycine control protein self-organization into elastomeric or amyloid fibrils.
    Structure (London, England : 1993), 2006, Volume: 14, Issue:11

    Topics: Alzheimer Disease; Amino Acid Sequence; Amyloid; Animals; Benzothiazoles; Chickens; Elastin; Entropy; Glycine; Humans; Insecta; Models, Molecular; Molecular Sequence Data; Peptides; Proline; Protein Conformation; Thiazoles; Triticum

2006
Reactions of 3-formylchromone with active methylene and methyl compounds and some subsequent reactions of the resulting condensation products.
    Molecules (Basel, Switzerland), 2005, Aug-31, Volume: 10, Issue:8

    Topics: Acetates; Acetonitriles; Barbiturates; Benzoates; Chromones; Dinitrobenzenes; Dioxanes; Glycine; Heterocyclic Compounds; Hippurates; Hydrocarbons; Models, Chemical; Pentanones; Phenylacetates; Propionates; Quinones; Sulfones; Thiazoles

2005
Activation of MAPK kinase 9 induces ethylene and camalexin biosynthesis and enhances sensitivity to salt stress in Arabidopsis.
    The Journal of biological chemistry, 2008, Oct-03, Volume: 283, Issue:40

    Topics: Arabidopsis; Arabidopsis Proteins; Ethylenes; Glycine; Hypocotyl; Indoles; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Seedlings; Silver; Sodium Chloride; Thiazoles

2008
Strain-specific sequences required for yeast [PSI+] prion propagation.
    Proceedings of the National Academy of Sciences of the United States of America, 2008, Sep-09, Volume: 105, Issue:36

    Topics: Amino Acid Sequence; Benzothiazoles; Glycine; Peptide Termination Factors; Prions; Proline; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Thiazoles

2008
Mechanism of action of species-selective P2X(7) receptor antagonists.
    British journal of pharmacology, 2009, Volume: 156, Issue:8

    Topics: Adamantane; Adenosine Triphosphate; Animals; Azabicyclo Compounds; Binding Sites; Cell Line, Tumor; Dogs; Dose-Response Relationship, Drug; Glycine; Guinea Pigs; Humans; Mice; Piperazines; Protein Conformation; Purinergic P2 Receptor Antagonists; Radioligand Assay; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2X7; Recombinant Fusion Proteins; Recombinant Proteins; Species Specificity; Structure-Activity Relationship; Temperature; Thiazoles; Transduction, Genetic; Vanadates

2009
A critical cysteine residue in monoacylglycerol lipase is targeted by a new class of isothiazolinone-based enzyme inhibitors.
    British journal of pharmacology, 2009, Volume: 157, Issue:6

    Topics: Amino Acid Sequence; Amino Acid Substitution; Animals; Cysteine; Drug Delivery Systems; Enzyme Inhibitors; Glycine; HeLa Cells; Humans; Molecular Sequence Data; Monoacylglycerol Lipases; Mutagenesis, Site-Directed; Rats; Structure-Activity Relationship; Substrate Specificity; Thiazoles; Thiazolidines

2009
Design and synthesis of a hybrid potentiator-corrector agonist of the cystic fibrosis mutant protein DeltaF508-CFTR.
    Bioorganic & medicinal chemistry letters, 2010, Jan-01, Volume: 20, Issue:1

    Topics: Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Drug Design; Glycine; Humans; Ion Channel Gating; Mutation; Protein Folding; Small Molecule Libraries; Structure-Activity Relationship; Thiazoles

2010
Pharmacological profiles of a novel protein tyrosine phosphatase 1B inhibitor, JTT-551.
    Diabetes, obesity & metabolism, 2010, Volume: 12, Issue:4

    Topics: Animals; Blood Glucose; Cell Line; Diabetes Mellitus, Type 2; Enzyme Inhibitors; Glycine; Hypoglycemic Agents; Liver; Male; Mice; Mice, Obese; Phosphorylation; Protein Tyrosine Phosphatase, Non-Receptor Type 1; Rats; Receptor, Insulin; Signal Transduction; Thiazoles

2010
The metabotropic glutamate mGluR5 receptor agonist CHPG stimulates food intake.
    Neuroreport, 2010, Jul-14, Volume: 21, Issue:10

    Topics: Animals; Catheterization; Dose-Response Relationship, Drug; Eating; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Fasting; Glycine; Injections, Intraperitoneal; Male; Phenylacetates; Pyridines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Thiazoles; Time Factors

2010
Evaluation of cannabinoid receptor 2 and metabotropic glutamate receptor 1 functional responses using a cell impedance-based technology.
    Journal of biomolecular screening, 2010, Volume: 15, Issue:10

    Topics: Analgesics; Animals; Benzimidazoles; Biological Assay; Calcium; Cannabinoids; CHO Cells; Chromones; Cricetinae; Cricetulus; Cyclic AMP; Cyclohexanols; Cycloleucine; Electric Impedance; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Glycine; Indoles; Naphthalenes; Neuroprotective Agents; Quinolines; Quisqualic Acid; Receptor, Cannabinoid, CB2; Receptors, Metabotropic Glutamate; Resorcinols; Signal Transduction; Thiazoles

2010
Mitochondrial reactive oxygen species are activated by mGluR5 through IP3 and activate ERK and PKA to increase excitability of amygdala neurons and pain behavior.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Jan-19, Volume: 31, Issue:3

    Topics: Amygdala; Analysis of Variance; Animals; Antioxidants; Benzoates; Cyclic AMP-Dependent Protein Kinases; Cyclic N-Oxides; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Extracellular Signal-Regulated MAP Kinases; Glycine; Inositol 1,4,5-Trisphosphate; Macrocyclic Compounds; Mitochondria; Neurons; NG-Nitroarginine Methyl Ester; Oxazoles; Pain; Pain Measurement; Pain Perception; Patch-Clamp Techniques; Pyridines; Reactive Oxygen Species; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Signal Transduction; Spin Labels; Superoxides; Thiazoles; Vocalization, Animal

2011
Effect of pesticides on plant growth promoting traits of greengram-symbiont, Bradyrhizobium sp. strain MRM6.
    Bulletin of environmental contamination and toxicology, 2011, Volume: 86, Issue:4

    Topics: Alanine; Bradyrhizobium; Dose-Response Relationship, Drug; Fabaceae; Fungicides, Industrial; Glycine; Glyphosate; Herbicides; Imidazoles; Insecticides; Neonicotinoids; Nitro Compounds; Organothiophosphorus Compounds; Oxazines; Symbiosis; Thiamethoxam; Thiazoles; Triazines; Triazoles

2011
A novel small Odorranalectin-bearing cubosomes: preparation, brain delivery and pharmacodynamic study on amyloid-β₂₅₋₃₅-treated rats following intranasal administration.
    European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V, 2012, Volume: 80, Issue:2

    Topics: Administration, Intranasal; Alzheimer Disease; Amyloid beta-Peptides; Animals; Brain; Coumarins; Disease Models, Animal; Drug Carriers; Drug Delivery Systems; Glycine; Intracellular Signaling Peptides and Proteins; Lectins; Maze Learning; Peptide Fragments; Rats; Rats, Sprague-Dawley; Streptavidin; Thiazoles; Tissue Distribution

2012
Examination of a role for metabotropic glutamate receptor 5 in the medial prefrontal cortex in cocaine sensitization in rats.
    Psychopharmacology, 2012, Volume: 221, Issue:1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzimidazoles; Central Nervous System Sensitization; Cocaine; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Male; Microinjections; Motor Activity; Prefrontal Cortex; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, AMPA; Receptors, Metabotropic Glutamate; Resorcinols; Thiazoles; Ventral Tegmental Area

2012
Probing intein-catalyzed thioester formation by unnatural amino acid substitutions in the active site.
    Biochemistry, 2012, Jan-10, Volume: 51, Issue:1

    Topics: Amino Acid Substitution; Bacterial Proteins; Catalysis; Catalytic Domain; Cysteine; DnaB Helicases; Esters; Genetic Variation; Glycine; Homocysteine; Inteins; Molecular Sequence Data; Peptide Fragments; Protein Precursors; Protein Processing, Post-Translational; Protein Splicing; Signal Transduction; Sulfhydryl Compounds; Synechocystis; Thiazoles

2012
RGS4 overexpression in the rat dorsal striatum modulates mGluR5- and amphetamine-mediated behavior and signaling.
    Psychopharmacology, 2012, Volume: 221, Issue:4

    Topics: Amphetamine; Animals; Behavior, Animal; Central Nervous System Stimulants; Corpus Striatum; Excitatory Amino Acid Agonists; Glycine; Male; MAP Kinase Signaling System; Proto-Oncogene Proteins c-akt; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; RGS Proteins; Thiazoles

2012
Role of mGluR5 neurotransmission in reinstated cocaine-seeking.
    Addiction biology, 2013, Volume: 18, Issue:1

    Topics: Analysis of Variance; Animals; Biotinylation; Blotting, Western; Carrier Proteins; Cocaine; Cocaine-Related Disorders; Cues; Disease Models, Animal; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Excitatory Amino Acid Agonists; Extinction, Psychological; Glycine; Homer Scaffolding Proteins; Male; Microinjections; Nucleus Accumbens; Phenylacetates; Protein Binding; Protein Transport; Pyridines; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Recurrence; Self Administration; Synaptic Transmission; Thiazoles

2013
Delayed mGluR5 activation limits neuroinflammation and neurodegeneration after traumatic brain injury.
    Journal of neuroinflammation, 2012, Feb-28, Volume: 9

    Topics: Animals; Brain Injuries; Calcium-Binding Proteins; Cognition Disorders; Diffusion Tensor Imaging; Disease Models, Animal; Ectodysplasins; Encephalitis; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Gene Expression Regulation; Glycine; Hippocampus; Magnetic Resonance Imaging; Male; Mice; Mice, Inbred C57BL; Microfilament Proteins; Microglia; Movement Disorders; Neurodegenerative Diseases; Neurons; Phenylacetates; Pyridines; Receptor, Metabotropic Glutamate 5; Receptors, Immunologic; Receptors, Metabotropic Glutamate; Recovery of Function; Statistics, Nonparametric; Thiazoles; Time Factors

2012
Pharmacological evidence of functional inhibitory metabotrophic glutamate receptors on mouse arousal-related cholinergic laterodorsal tegmental neurons.
    Neuropharmacology, 2013, Volume: 66

    Topics: Amino Acids; Animals; Animals, Outbred Strains; Arousal; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Cholinergic Neurons; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glycine; Mesencephalon; Mice; Neural Inhibition; Peptides; Phenylacetates; Potassium Channel Blockers; Pyridines; Receptors, Metabotropic Glutamate; Thiazoles

2013
Modulation of pyramidal cell output in the medial prefrontal cortex by mGluR5 interacting with CB1.
    Neuropharmacology, 2013, Volume: 66

    Topics: Animals; Arachidonic Acids; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glycine; Inhibitory Postsynaptic Potentials; Male; Morpholines; Neural Inhibition; Niacinamide; Phenylacetates; Prefrontal Cortex; Pyramidal Cells; Pyrazoles; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Synaptic Transmission; Thiazoles

2013
Methylglyoxal alters glucose metabolism and increases AGEs content in C6 glioma cells.
    Metabolic brain disease, 2012, Volume: 27, Issue:4

    Topics: Cell Line, Tumor; Coloring Agents; Energy Metabolism; Glioma; Glucose; Glycation End Products, Advanced; Glycine; Humans; Lactic Acid; Lactoylglutathione Lyase; Neutral Red; Oxidation-Reduction; Propidium; Pyruvaldehyde; Tetrazolium Salts; Thiazoles; Thiolester Hydrolases

2012
Dissecting the phenotypes of Plk1 inhibition in cancer cells using novel kinase inhibitory chemical CBB2001.
    Laboratory investigation; a journal of technical methods and pathology, 2012, Volume: 92, Issue:10

    Topics: Amides; Animals; Aurora Kinase A; Aurora Kinases; Benzimidazoles; Cell Cycle Proteins; Cell Division; Cell Line, Tumor; Cell Proliferation; Cyclin B1; Female; Geminin; Glycine; Humans; Inhibitory Concentration 50; Mice; Mice, Inbred BALB C; Mice, Nude; Neoplasms; Nitriles; Polo-Like Kinase 1; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Sulfones; Thiazoles

2012
The truncated C-terminal RNA recognition motif of TDP-43 protein plays a key role in forming proteinaceous aggregates.
    The Journal of biological chemistry, 2013, Mar-29, Volume: 288, Issue:13

    Topics: Amino Acid Motifs; Amyloidogenic Proteins; Amyotrophic Lateral Sclerosis; Benzothiazoles; Chromatography; Circular Dichroism; Dimerization; DNA-Binding Proteins; DNA, Complementary; Frontotemporal Lobar Degeneration; Glutathione Transferase; Glycine; Humans; Neurodegenerative Diseases; Peptides; Protein Binding; Protein Denaturation; Protein Folding; Protein Structure, Secondary; Protein Structure, Tertiary; Scattering, Radiation; Thiazoles; X-Rays

2013
Acetylcholinesterase in honey bees (Apis mellifera) exposed to neonicotinoids, atrazine and glyphosate: laboratory and field experiments.
    Environmental science and pollution research international, 2013, Volume: 20, Issue:8

    Topics: Acetylcholinesterase; Animals; Atrazine; Bees; Glycine; Glyphosate; Guanidines; Herbicides; Imidazoles; Insecticides; Neonicotinoids; Nitro Compounds; Pollen; Quebec; Thiazoles; Zea mays

2013
Activation of lateral hypothalamic mGlu1 and mGlu5 receptors elicits feeding in rats.
    Neuropharmacology, 2014, Volume: 79

    Topics: Animals; Benzimidazoles; Benzopyrans; Cycloleucine; Dose-Response Relationship, Drug; Eating; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Hypothalamus; Male; Phenylacetates; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; Thiazoles; Time Factors

2014
The metabolic fate of [14C]-fenclozic acid in the hepatic reductase null (HRN) mouse.
    Xenobiotica; the fate of foreign compounds in biological systems, 2014, Volume: 44, Issue:2

    Topics: Animals; Autoradiography; Carbon Radioisotopes; Feces; Glycine; Inactivation, Metabolic; Liver; Male; Mice; Mice, Knockout; Oxidoreductases; Taurine; Thiazoles; Tissue Distribution

2014
Group I metabotropic glutamate receptor-mediated activation of PKC gamma in the nucleus accumbens core promotes the reinstatement of cocaine seeking.
    Addiction biology, 2015, Volume: 20, Issue:2

    Topics: Animals; Benzimidazoles; Cocaine; Cocaine-Related Disorders; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Nucleus Accumbens; Phosphorylation; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-alpha; Pyridines; Rats; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; Thiazoles

2015
A protein synthesis-dependent mechanism sustains calcium-permeable AMPA receptor transmission in nucleus accumbens synapses during withdrawal from cocaine self-administration.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2014, Feb-19, Volume: 34, Issue:8

    Topics: Animals; Benzoates; Calcium; Cocaine-Related Disorders; Cycloheximide; Excitatory Amino Acid Antagonists; Glycine; Male; Methoxyhydroxyphenylglycol; Nucleus Accumbens; Patch-Clamp Techniques; Protein Biosynthesis; Protein Synthesis Inhibitors; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Self Administration; Substance Withdrawal Syndrome; Synapses; Synaptic Transmission; Thiazoles; Ventral Tegmental Area

2014
Pharmacological effects of JTT-551, a novel protein tyrosine phosphatase 1B inhibitor, in diet-induced obesity mice.
    Journal of diabetes research, 2014, Volume: 2014

    Topics: Animals; Blood Glucose; Body Weight; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 2; Glucose; Glycine; Hypothalamus; Leptin; Lipid Metabolism; Male; Mice; Mice, Inbred C57BL; Mice, Obese; Obesity; Protein Tyrosine Phosphatase, Non-Receptor Type 1; Protein Tyrosine Phosphatases; Signal Transduction; STAT3 Transcription Factor; Thiazoles

2014
The influence of pathological mutations and proline substitutions in TDP-43 glycine-rich peptides on its amyloid properties and cellular toxicity.
    PloS one, 2014, Volume: 9, Issue:8

    Topics: Amino Acid Sequence; Amino Acid Substitution; Amyloid; Animals; Benzothiazoles; Cell Membrane; DNA-Binding Proteins; Glycine; Mice; Molecular Sequence Data; Mutant Proteins; Mutation; Peptides; Proline; Protein Aggregates; Protein Multimerization; Protein Structure, Secondary; Spectrum Analysis, Raman; Thiazoles; Time Factors

2014
Novel mGluR5 positive allosteric modulator improves functional recovery, attenuates neurodegeneration, and alters microglial polarization after experimental traumatic brain injury.
    Neurotherapeutics : the journal of the American Society for Experimental NeuroTherapeutics, 2014, Volume: 11, Issue:4

    Topics: Allosteric Regulation; Animals; Brain Injuries; Cell Count; Cerebral Cortex; Disease Models, Animal; Glycine; Hippocampus; Male; Membrane Glycoproteins; Mice; Mice, Inbred C57BL; Microglia; Motor Activity; NADPH Oxidase 2; NADPH Oxidases; Neuroprotective Agents; Nitric Oxide Synthase Type II; Phenylacetates; Pyridines; Receptor, Metabotropic Glutamate 5; Recovery of Function; Thiazoles

2014
The Biosynthesis of the Thiazole Moiety of Thiamin in the Archaeon Halobacterium salinarum.
    Journal of nutritional science and vitaminology, 2015, Volume: 61, Issue:3

    Topics: Biosynthetic Pathways; Glycine; Halobacterium salinarum; Pyrimidines; Thiamine; Thiazoles

2015
The Biosynthesis of the Pyrimidine Moiety of Thiamin in Halobacterium salinarum.
    Journal of nutritional science and vitaminology, 2016, Volume: 62, Issue:2

    Topics: Biosynthetic Pathways; Escherichia coli; Glycine; Halobacterium salinarum; Histidine; Purines; Pyridoxine; Pyrimidines; Ribonucleotides; Saccharomyces cerevisiae; Thiamine; Thiazoles

2016
Increased Metabotropic Glutamate Receptor 5 Signaling Underlies Obsessive-Compulsive Disorder-like Behavioral and Striatal Circuit Abnormalities in Mice.
    Biological psychiatry, 2016, 10-01, Volume: 80, Issue:7

    Topics: Animals; Behavior, Animal; Corpus Striatum; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Grooming; Mice; Mice, Knockout; Mice, Transgenic; Nerve Tissue Proteins; Niacinamide; Obsessive-Compulsive Disorder; Pyridines; Receptor, Metabotropic Glutamate 5; Signal Transduction; Thiazoles

2016
The activation of metabotropic glutamate 5 receptors in the rat ventral tegmental area increases dopamine extracellular levels.
    Neuroreport, 2017, Jan-01, Volume: 28, Issue:1

    Topics: Animals; Dopamine; Excitatory Amino Acid Agents; Extracellular Fluid; Glutamic Acid; Glycine; Kynurenic Acid; Male; Microdialysis; Phenylacetates; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Thiazoles; Ventral Tegmental Area

2017
Sensitization of TRPV1 and TRPA1 via peripheral mGluR5 signaling contributes to thermal and mechanical hypersensitivity.
    Pain, 2017, Volume: 158, Issue:9

    Topics: Acetanilides; Animals; Disease Models, Animal; Enzyme Inhibitors; Freund's Adjuvant; Glutamic Acid; Glycine; Hyperalgesia; Male; Neurons; Pain; Pain Threshold; Phenylacetates; Physical Stimulation; Purines; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Signal Transduction; Skin; Thiazoles; Trigeminal Ganglion; TRPA1 Cation Channel; TRPV Cation Channels

2017
A Selective Biligand Inhibitor of CK2 Increases Caspase-3 Activity in Cancer Cells and Inhibits Platelet Aggregation.
    ChemMedChem, 2017, 10-20, Volume: 12, Issue:20

    Topics: Antineoplastic Agents; Casein Kinase II; Caspase 3; Cell Cycle Proteins; Chaperonins; Enzyme Activation; Gene Expression Regulation, Neoplastic; Glycine; HeLa Cells; Humans; Molecular Structure; Phosphorylation; Platelet Aggregation; Thiazoles

2017
Therapeutic potential for leukocyte elastase in chronic pain states harboring a neuropathic component.
    Pain, 2017, Volume: 158, Issue:11

    Topics: Analgesics; Animals; Cancer Pain; Chronic Pain; Cyclic S-Oxides; Disease Models, Animal; Female; Glycine; Hyperalgesia; Leukocyte Elastase; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Motor Activity; Neuralgia; Pain Measurement; Pain Threshold; Pregabalin; Serine Proteinase Inhibitors; Sulfonamides; Thiazoles

2017
Expression, Purification, and Activity of ActhiS, a Thiazole Biosynthesis Enzyme from Acremonium chrysogenum.
    Biochemistry. Biokhimiia, 2017, Volume: 82, Issue:7

    Topics: Acremonium; Adenosine Diphosphate; Amino Acid Sequence; Chromatography, High Pressure Liquid; Fungal Proteins; Glycine; Ligands; Magnetic Resonance Spectroscopy; Mass Spectrometry; Mutagenesis, Site-Directed; NAD; Recombinant Proteins; Sequence Alignment; Thiamine Pyrophosphate; Thiazoles

2017
Novel cell line models to study mechanisms and overcoming strategies of proteasome inhibitor resistance in multiple myeloma.
    Biochimica et biophysica acta. Molecular basis of disease, 2019, 06-01, Volume: 1865, Issue:6

    Topics: A549 Cells; Amino Acid Substitution; Antineoplastic Agents; Boron Compounds; Bortezomib; Cell Line, Tumor; Cell Survival; Dose-Response Relationship, Drug; Drug Resistance, Neoplasm; Gene Expression; Glycine; Histone Deacetylases; Humans; Indoles; Models, Biological; Multiple Myeloma; Mutation; Oligopeptides; Panobinostat; Phosphatidylinositol 3-Kinase; Proteasome Endopeptidase Complex; Proteasome Inhibitors; Pyrimidines; Thiazoles

2019
Photoprotection by mitochondrial alternative pathway is enhanced at heat but disabled at chilling.
    The Plant journal : for cell and molecular biology, 2020, Volume: 104, Issue:2

    Topics: Arabidopsis; Chlorophyll A; Cold Temperature; Glycine; Hot Temperature; Light; Methacrylates; Mitochondria; Mitochondrial Proteins; Mutation; NADP; Oxidoreductases; Photosynthesis; Plant Leaves; Plant Proteins; Serine; Thiazoles

2020
Multicomponent synthesis of fully substituted thiazoles using glycine-based dithiocarbamates, acetic anhydride and nitroalkenes.
    Organic & biomolecular chemistry, 2022, 05-11, Volume: 20, Issue:18

    Topics: Acetic Anhydrides; Alkenes; Glycine; Molecular Structure; Nitro Compounds; Thiazoles

2022
Formation Priority of Pyrazines and 2-Acetylthiazole Dependent on the Added Cysteine and Fragments of Deoxyosones during the Thermal Process of the Glycine-Ribose Amadori Compound.
    Journal of agricultural and food chemistry, 2022, Sep-21, Volume: 70, Issue:37

    Topics: Cysteamine; Cysteine; Glycine; Glyoxal; Magnesium Oxide; Maillard Reaction; Pyrazines; Pyruvaldehyde; Ribose; Thiazoles

2022
Quantitative Metabolism and Urinary Elimination Kinetics of Seven Neonicotinoids and Neonicotinoid-Like Compounds in Humans.
    Environmental science & technology, 2023, Dec-05, Volume: 57, Issue:48

    Topics: Glycine; Humans; Insecticides; Male; Neonicotinoids; Nitro Compounds; Thiazoles

2023