Page last updated: 2024-08-21

thiazoles and gamma-aminobutyric acid

thiazoles has been researched along with gamma-aminobutyric acid in 45 studies

Research

Studies (45)

TimeframeStudies, this research(%)All Research%
pre-19902 (4.44)18.7374
1990's10 (22.22)18.2507
2000's15 (33.33)29.6817
2010's18 (40.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Blin, O; Dusticier, N; Nieoullon, A; Samuel, D1
Becquet, D; Faudon, M; Hery, F1
Ferko, AP1
Baruch, P; Chéramy, A; Glowinski, J; Godeheu, G; Romo, R1
Benavides, J; Camelin, JC; Flamand, F; Gueremy, C; Le Fur, G; Legrand, JJ; Mitrani, N; Uzan, A1
Hefti, F; Widmer, HR2
Martin, D; Nadler, JV; Thompson, MA1
Amagasu, SM; MacIver, MB; Mikulec, AA; Monroe, FA1
Andrus, PK; Cutting, FB; Doble, A; Gurney, ME; Hall, ED; Taylor, CP; Zhai, P1
Damgaard, I; Rodríguez-Farré, E; Schousboe, A; Suñol, C; Vale, C1
Oliveira, CR; Rego, AC1
Hernández-Pech, X; Merchant-Larios, H; Morán, J; Pasantes-Morales, H1
Fisher, M; Schaebitz, W1
Cross, AJ; Gabrielsson, J; Green, AR; Hainsworth, AH; Jones, JA; Lambert, DG; Murray, TK; Nelson, RM; Richards, DA1
Freeman, MP; Gelenberg, AJ; Gnanadesikan, M1
Ciraulo, DA; Hennen, J; Jensen, JE; Ke, Y; Knapp, C; Kwak, T; Meyer, AA; Nassar, LE; Renshaw, PF; Sarid-Segal, O; Streeter, CC1
Höfner, G; Kragler, A; Wanner, KT1
Ducray, A; Krebs, SH; Meyer, M; Schaller, B; Seiler, RW; Widmer, HR1
Batlle, A; Battah, S; Casas, A; Di Venosa, G; Dobbin, P; Macrobert, AJ; Rodriguez, L1
Molnar, MZ; Mucsi, I; Novak, M1
Di Monte, DA; Johnston, LC; Langston, WJ; Reaney, SH1
Andres, RH; Ducray, AD; Qualls, R; Schläppi, JA; Schlattner, U; Seiler, RW; Wallimann, T; Widmer, HR1
Klein, S; Nicolas, LB; Prinssen, EP1
Bernotas, RC; Beyer, CE; Boikess, S; Cole, DC; Coupet, J; Dawson, LA; Ellingboe, JW; Feng, X; Galante, R; Huang, P; Kelly, MF; Lennox, WJ; Leung, L; Marquis, K; Rosenzweig-Lipson, S; Schechter, LE; Smith, DL; Stock, JR; Zhang, GM1
Bond, D; Gilron, I; Mercer, CD; Orr, E; Tu, D1
Marcy, VR; Marino, MJ; Schaffhauser, H; West, PJ1
Akaike, H; Akaike, N; Hori, N; Ito, Y; Jang, II; Ogawa, S1
Newman, M1
Coetzee, JF; Cull, CA; Kelly, LL; Kohake, LE; KuKanich, B; Mosher, RA; Mueting, SL1
Coetzee, JF; Gehring, R; Kukanich, B; Malreddy, PR1
Dzhala, V; Glykys, J; Khazipov, R; Staley, K; Valeeva, G1
Allen, K; Badino, P; Bergamasco, L; Bertolotti, L; Coetzee, JF; Dockweiler, J; Edwards-Callaway, LN; Fraccaro, E; Glynn, H; Kukanich, B; Odore, R1
Allen, KA; Bergamasco, LL; Coetzee, JF; Dockweiler, JC; Edwards-Callaway, LN; Fraccaro, E; Glynn, HD; Jones, M; KuKanich, B; Lubbers, B1
Aoki, Y; Eguchi, Y; Inage, K; Inoue, G; Ishikawa, T; Kamoda, H; Kishida, S; Kubota, G; Kuniyoshi, K; Miyagi, M; Nakamura, J; Ochiai, N; Ohtori, S; Oikawa, Y; Orita, S; Sainoh, T; Sakuma, Y; Suzkuki, M; Takahashi, K; Takaso, M; Toyone, T; Yamauchi, K1
Deng, XQ; Liu, DC; Quan, ZS; Wang, SB1
Anderson, DE; Coetzee, JF; Gehring, R; Kohake, LE; Kukanich, B; Mosher, RA; Robert, B; Wang, C; White, BJ1
Brazhe, A; Jensen, K; Jessen, SB; Lauritzen, M; Lind, BL; Mathiesen, C; Thomsen, K1
Duggan, S; Dumerton-Shore, D; Gilron, I; McGrath, M; Orr, E; Rooney, R; Tu, D1
Avoli, M; D'Antuono, M; Hamidi, S1
Castonguay, A; Chen, Z; Cottet, M; De Koninck, Y; Doyle, T; Egan, TM; Ford, A; Jacobson, KA; Little, JW; Salvemini, D; Symons-Liguori, AM; Tosh, DK; Vanderah, TW1
Burrell, BD; Miiller, E; Peterson, W; Summers, T; Wang, Y1
Baur, R; Maldifassi, MC; Middendorp, SJ; Sigel, E1
Corona-Ramos, JN; Espinosa-Juárez, JV; Jaramillo-Morales, OA; López-Muñoz, FJ; Medina-López, JR1
Buck, A; Gietl, A; Henning, A; Hock, C; Kirchner, T; Leh, SE; Nitsch, RM; Preti, MG; Pruessmann, KP; Quevenco, FC; Schreiner, SJ; Steininger, SC; Unschuld, PG; van Bergen, JMG; Van De Ville, D; Wyss, M1

Reviews

3 review(s) available for thiazoles and gamma-aminobutyric acid

ArticleYear
An overview of acute stroke therapy: past, present, and future.
    Archives of internal medicine, 2000, Nov-27, Volume: 160, Issue:21

    Topics: Acute Disease; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Antibodies; Brain Ischemia; Calcium Channel Blockers; Cardiovascular Agents; Cell Adhesion Molecules; Clinical Trials as Topic; Cytidine Diphosphate Choline; Cytokines; Drug Therapy, Combination; Fibrinolytic Agents; Free Radical Scavengers; gamma-Aminobutyric Acid; Growth Substances; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; N-Methylaspartate; Neuroprotective Agents; Nootropic Agents; Piperidines; Stroke; Thiazoles; Thrombolytic Therapy

2000
Alternatives to lithium and divalproex in the maintenance treatment of bipolar disorder.
    Bipolar disorders, 2003, Volume: 5, Issue:3

    Topics: Acetates; Amines; Anticonvulsants; Antimanic Agents; Antipsychotic Agents; Benzodiazepines; Bipolar Disorder; Calcium Channel Blockers; Carbamazepine; Clozapine; Cyclohexanecarboxylic Acids; Dibenzothiazepines; Donepezil; Fatty Acids, Omega-3; Fructose; Gabapentin; gamma-Aminobutyric Acid; Humans; Indans; Lamotrigine; Lithium Carbonate; Olanzapine; Piperazines; Piperidines; Pirenzepine; Quetiapine Fumarate; Risperidone; Thiazoles; Topiramate; Treatment Outcome; Triazines; Valproic Acid

2003
Management of restless legs syndrome in patients on dialysis.
    Drugs, 2006, Volume: 66, Issue:5

    Topics: Amines; Anticonvulsants; Benzothiazoles; Clonazepam; Cyclohexanecarboxylic Acids; Dopamine Agents; Gabapentin; gamma-Aminobutyric Acid; Humans; Kidney Failure, Chronic; Levodopa; Narcotics; Pramipexole; Renal Dialysis; Restless Legs Syndrome; Thiazoles; Uremia

2006

Trials

5 trial(s) available for thiazoles and gamma-aminobutyric acid

ArticleYear
Prefrontal GABA levels in cocaine-dependent subjects increase with pramipexole and venlafaxine treatment.
    Psychopharmacology, 2005, Volume: 182, Issue:4

    Topics: Adult; Antidepressive Agents, Second-Generation; Antioxidants; Benzothiazoles; Cocaine-Related Disorders; Cyclohexanols; Double-Blind Method; Female; gamma-Aminobutyric Acid; Humans; Magnetic Resonance Spectroscopy; Male; Middle Aged; Nicotine; Pramipexole; Prefrontal Cortex; Protons; Retrospective Studies; Thiazoles; Time Factors; Venlafaxine Hydrochloride

2005
A randomized, double-blind, controlled trial of perioperative administration of gabapentin, meloxicam and their combination for spontaneous and movement-evoked pain after ambulatory laparoscopic cholecystectomy.
    Anesthesia and analgesia, 2009, Volume: 108, Issue:2

    Topics: Adult; Aged; Aged, 80 and over; Ambulatory Surgical Procedures; Amines; Analgesics, Non-Narcotic; Analgesics, Opioid; Cholecystectomy, Laparoscopic; Cyclohexanecarboxylic Acids; Double-Blind Method; Drug Therapy, Combination; Female; Gabapentin; gamma-Aminobutyric Acid; Humans; Male; Meloxicam; Middle Aged; Movement; Oxygen Inhalation Therapy; Pain Measurement; Pain, Postoperative; Patient Satisfaction; Spirometry; Thiazines; Thiazoles; Treatment Outcome; Young Adult

2009
The pharmacokinetics and effects of meloxicam, gabapentin, and flunixin in postweaning dairy calves following dehorning with local anesthesia.
    Journal of veterinary pharmacology and therapeutics, 2013, Volume: 36, Issue:6

    Topics: Amines; Anesthetics, Local; Animals; Anti-Inflammatory Agents, Non-Steroidal; Cattle; Cattle Diseases; Clonixin; Cyclohexanecarboxylic Acids; Dairying; Gabapentin; gamma-Aminobutyric Acid; Horns; Male; Meloxicam; Pain Measurement; Pain, Postoperative; Thiazines; Thiazoles

2013
Efficacy of combination of meloxicam and pregabalin for pain in knee osteoarthritis.
    Yonsei medical journal, 2013, Volume: 54, Issue:5

    Topics: Aged; Aged, 80 and over; Drug Therapy, Combination; Female; gamma-Aminobutyric Acid; Humans; Male; Meloxicam; Middle Aged; Osteoarthritis, Knee; Pain Measurement; Pregabalin; Thiazines; Thiazoles

2013
The effect of triple vs. double nonopioid therapy on postoperative pain and functional outcome after abdominal hysterectomy: a randomised double-blind control trial.
    European journal of anaesthesiology, 2015, Volume: 32, Issue:4

    Topics: Acetaminophen; Adult; Amines; Analgesia, Patient-Controlled; Analgesics, Opioid; Cyclohexanecarboxylic Acids; Double-Blind Method; Drug Therapy, Combination; Early Termination of Clinical Trials; Female; Gabapentin; gamma-Aminobutyric Acid; Humans; Hysterectomy; Meloxicam; Middle Aged; Morphine; Ontario; Pain Measurement; Pain, Postoperative; Recovery of Function; Thiazines; Thiazoles; Time Factors; Treatment Outcome

2015

Other Studies

37 other study(ies) available for thiazoles and gamma-aminobutyric acid

ArticleYear
Effects of riluzole (2-amino-6-trifluoromethoxy benzothiazole) on striatal neurochemical markers in the rat, with special reference to the dopamine, choline, GABA and glutamate synaptosomal high affinity uptake systems.
    Fundamental & clinical pharmacology, 1992, Volume: 6, Issue:4-5

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Aspartic Acid; Biomarkers; Choline; Corpus Striatum; Culture Media; Dopamine; Female; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Hydroxyindoleacetic Acid; Neurotransmitter Uptake Inhibitors; Rats; Rats, Wistar; Riluzole; Serotonin; Synaptic Transmission; Synaptosomes; Thiazoles; Tritium

1992
In vivo evidence for an inhibitory glutamatergic control of serotonin release in the cat caudate nucleus: involvement of GABA neurons.
    Brain research, 1990, Jun-11, Volume: 519, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; Animals; Aspartic Acid; Bicuculline; Cats; Caudate Nucleus; Female; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Male; N-Methylaspartate; Neurons; Riluzole; Serotonin; Spinal Cord; Synaptic Transmission; Tetrodotoxin; Thiazoles

1990
The interaction between ethanol and cysteine on the central depressant effects of ethanol in mice.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:3

    Topics: Animals; Cysteine; Drug Synergism; Ethanol; gamma-Aminobutyric Acid; Injections, Intraventricular; Isethionic Acid; Male; Mice; Posture; Pyrrolidonecarboxylic Acid; Reflex; Thiazoles; Thiazolidines

1990
In vivo presynaptic control of dopamine release in the cat caudate nucleus--II. Facilitatory or inhibitory influence of L-glutamate.
    Neuroscience, 1986, Volume: 19, Issue:4

    Topics: Animals; Caudate Nucleus; Cerebral Cortex; Dopamine; Female; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Male; Neural Pathways; Rats; Receptors, Glutamate; Receptors, Neurotransmitter; Riluzole; Synaptic Transmission; Tetrodotoxin; Thiazoles

1986
2-Amino-6-trifluoromethoxy benzothiazole, a possible antagonist of excitatory amino acid neurotransmission--II. Biochemical properties.
    Neuropharmacology, 1985, Volume: 24, Issue:11

    Topics: Acetylcholine; Amino Acids; Animals; Anticonvulsants; Apomorphine; Cerebellum; Chlordiazepoxide; Cyclic GMP; Diazepam; gamma-Aminobutyric Acid; Harmaline; In Vitro Techniques; Injections, Intraventricular; Isoniazid; Male; Rats; Rats, Inbred Strains; Riluzole; Synaptic Transmission; Thiazoles

1985
Neurotrophin-4/5 promotes survival and differentiation of rat striatal neurons developing in culture.
    The European journal of neuroscience, 1994, Nov-01, Volume: 6, Issue:11

    Topics: Animals; Blotting, Western; Calbindin 2; Cell Differentiation; Cell Survival; Cells, Cultured; DNA; gamma-Aminobutyric Acid; Humans; Immunohistochemistry; Neostriatum; Nerve Growth Factors; Neurons; Phosphatidylinositols; Rats; Recombinant Proteins; S100 Calcium Binding Protein G; Tetrazolium Salts; Thiazoles

1994
Stimulation of GABAergic neuron differentiation by NT-4/5 in cultures of rat cerebral cortex.
    Brain research. Developmental brain research, 1994, Jul-15, Volume: 80, Issue:1-2

    Topics: Animals; Blotting, Western; Brain-Derived Neurotrophic Factor; Calbindins; Cell Differentiation; Cells, Cultured; Cerebral Cortex; Excitatory Amino Acids; gamma-Aminobutyric Acid; Glutamic Acid; Immunohistochemistry; Nerve Growth Factors; Nerve Tissue Proteins; Neurons; Rats; S100 Calcium Binding Protein G; Stimulation, Chemical; Tetrazolium Salts; Thiazoles

1994
The neuroprotective agent riluzole inhibits release of glutamate and aspartate from slices of hippocampal area CA1.
    European journal of pharmacology, 1993, Dec-21, Volume: 250, Issue:3

    Topics: Animals; Aspartic Acid; Excitatory Amino Acid Antagonists; Female; gamma-Aminobutyric Acid; Glutamates; Hippocampus; Potassium; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Riluzole; Thiazoles

1993
Riluzole anesthesia: use-dependent block of presynaptic glutamate fibers.
    Anesthesiology, 1996, Volume: 85, Issue:3

    Topics: Action Potentials; Anesthetics; Animals; gamma-Aminobutyric Acid; Glutamic Acid; In Vitro Techniques; Male; Rats; Rats, Sprague-Dawley; Riluzole; Sodium Channel Blockers; Synaptic Transmission; Thiazoles

1996
Benefit of vitamin E, riluzole, and gabapentin in a transgenic model of familial amyotrophic lateral sclerosis.
    Annals of neurology, 1996, Volume: 39, Issue:2

    Topics: Acetates; Amines; Amyotrophic Lateral Sclerosis; Animals; Brain; Cyclohexanecarboxylic Acids; Diet; Disease Progression; Gabapentin; gamma-Aminobutyric Acid; Humans; Mice; Mice, Transgenic; Oxidative Stress; Riluzole; Spinal Cord; Superoxide Dismutase; Survival Analysis; Thiazoles; Vitamin E

1996
Cytotoxic action of lindane in neocortical GABAergic neurons is primarily mediated by interaction with flunitrazepam-sensitive GABA(A) receptors.
    Journal of neuroscience research, 1998, May-01, Volume: 52, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Cell Survival; Cells, Cultured; Coloring Agents; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Flunitrazepam; GABA Agonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Hexachlorocyclohexane; Insecticides; Mice; Mitochondria; Neocortex; Neurons; Receptors, GABA-A; Tetrazolium Salts; Thiazoles; Time Factors

1998
Influence of gamma-aminobutyric acid on retinal cells excitotoxicity upon glucose deprivation.
    Neuroscience research, 1999, Volume: 34, Issue:1

    Topics: Animals; Bicuculline; Cells, Cultured; Chick Embryo; Coloring Agents; Dose-Response Relationship, Drug; GABA Agents; GABA Antagonists; gamma-Aminobutyric Acid; Glucose; Neurons; Nipecotic Acids; Retina; Tetrazolium Salts; Thiazoles

1999
Release of taurine in apoptotic cerebellar granule neurons in culture.
    Pflugers Archiv : European journal of physiology, 2000, Volume: 439, Issue:3

    Topics: Animals; Apoptosis; Caspase 3; Caspases; Cell Size; Cell Survival; Cells, Cultured; Cerebellum; Chloride Channels; Coloring Agents; Diffusion; Enzyme Precursors; gamma-Aminobutyric Acid; Glutamic Acid; Membrane Potentials; Neurons; Potassium Chloride; Rats; Sodium; Taurine; Tetrazolium Salts; Thiazoles

2000
Neuroprotective efficacy of AR-A008055, a clomethiazole analogue, in a global model of acute ischaemic stroke and its effect on ischaemia-induced glutamate and GABA efflux in vitro.
    Neuropharmacology, 2001, Volume: 41, Issue:2

    Topics: Animals; Brain Ischemia; Chlormethiazole; Female; gamma-Aminobutyric Acid; Gerbillinae; Glutamic Acid; Hippocampus; Male; Methylamines; Neuroprotective Agents; Rats; Rats, Wistar; Stroke; Thiazoles

2001
Novel parent structures for inhibitors of the murine GABA transporters mGAT3 and mGAT4.
    European journal of pharmacology, 2005, Sep-05, Volume: 519, Issue:1-2

    Topics: Acetates; Animals; beta-Alanine; Cell Line; Chlorocebus aethiops; COS Cells; Dose-Response Relationship, Drug; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Guanidines; Humans; Membrane Transport Modulators; Membrane Transport Proteins; Mice; Molecular Structure; Neurotransmitter Uptake Inhibitors; Plasmids; Propionates; Serine; Structure-Activity Relationship; Thiazoles; Transfection; Tritium

2005
GDNF family ligands display distinct action profiles on cultured GABAergic and serotonergic neurons of rat ventral mesencephalon.
    Brain research, 2006, Jan-19, Volume: 1069, Issue:1

    Topics: Analysis of Variance; Animals; Cell Count; Cells, Cultured; Embryo, Mammalian; gamma-Aminobutyric Acid; Glial Cell Line-Derived Neurotrophic Factors; Immunohistochemistry; Mesencephalon; Neurites; Neurons; Phosphopyruvate Hydratase; Rats; Serotonin; Tetrazolium Salts; Thiazoles

2006
Mechanisms of 5-aminolevulinic acid ester uptake in mammalian cells.
    British journal of pharmacology, 2006, Volume: 147, Issue:7

    Topics: Aminolevulinic Acid; Animals; Biological Transport, Active; Cell Line; Cell Line, Tumor; Cell Membrane; Cytoplasm; Diffusion; Female; GABA Antagonists; gamma-Aminobutyric Acid; Mice; Porphyrins; Succinic Acid; Temperature; Tetrazolium Salts; Thiazoles

2006
Comparison of the neurotoxic effects of proteasomal inhibitors in primary mesencephalic cultures.
    Experimental neurology, 2006, Volume: 202, Issue:2

    Topics: Acetylcysteine; Analysis of Variance; Animals; Cell Count; Cells, Cultured; Dopamine; Dose-Response Relationship, Drug; Embryo, Mammalian; Enzyme Inhibitors; gamma-Aminobutyric Acid; Immunohistochemistry; Mesencephalon; Neurons; Neurotoxins; Proteasome Inhibitors; Rats; Rats, Sprague-Dawley; Tetrazolium Salts; Thiazoles; Time Factors; Tritium

2006
Creatine treatment promotes differentiation of GABA-ergic neuronal precursors in cultured fetal rat spinal cord.
    Journal of neuroscience research, 2007, Volume: 85, Issue:9

    Topics: Animals; Blotting, Western; Cell Differentiation; Cell Survival; Cells, Cultured; Choline O-Acetyltransferase; Creatine; Creatine Kinase; Energy Metabolism; Female; gamma-Aminobutyric Acid; Immunohistochemistry; Mitogen-Activated Protein Kinase 1; Neurons; Nitro Compounds; Pregnancy; Propionates; Rats; Spinal Cord; Stem Cells; Tetrazolium Salts; Thiazoles; Tubulin

2007
Defensive-like behaviors induced by ultrasound: further pharmacological characterization in Lister-hooded rats.
    Psychopharmacology, 2007, Volume: 194, Issue:2

    Topics: Amines; Analgesics, Opioid; Animals; Anti-Anxiety Agents; Bridged Bicyclo Compounds; Buspirone; Calcium Channel Blockers; Cyclohexanecarboxylic Acids; Diazepam; Dose-Response Relationship, Drug; Escape Reaction; Fear; Freezing Reaction, Cataleptic; Gabapentin; gamma-Aminobutyric Acid; Haloperidol; Imidazoles; Male; Morphine; Motor Activity; Nociceptin Receptor; Pregabalin; Pyridines; Rats; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Receptors, Opioid; Spiro Compounds; Thiazoles; Ultrasonics

2007
Discovery of N1-(6-chloroimidazo[2,1-b][1,3]thiazole-5-sulfonyl)tryptamine as a potent, selective, and orally active 5-HT(6) receptor agonist.
    Journal of medicinal chemistry, 2007, Nov-15, Volume: 50, Issue:23

    Topics: Administration, Oral; Animals; Biological Availability; CHO Cells; Cricetinae; Cricetulus; Dogs; Frontal Lobe; gamma-Aminobutyric Acid; Haplorhini; Humans; In Vitro Techniques; Mice; Microdialysis; Microsomes, Liver; Radioligand Assay; Rats; Receptors, Serotonin; Serotonin Receptor Agonists; Solubility; Structure-Activity Relationship; Thiazoles; Tryptamines

2007
Activation of the 5-HT(6) receptor attenuates long-term potentiation and facilitates GABAergic neurotransmission in rat hippocampus.
    Neuroscience, 2009, Dec-01, Volume: 164, Issue:2

    Topics: Animals; CA1 Region, Hippocampal; Dose-Response Relationship, Drug; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Long-Term Potentiation; Male; Piperazines; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulfonamides; Synaptic Transmission; Theta Rhythm; Thiazoles; Tryptamines

2009
Effects of Z-338, a novel gastroprokinetic agent, on the actions of excitatory and inhibitory neurotransmitters on neurons in area postrema.
    Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi, 2010, Volume: 46, Issue:1

    Topics: Adenosine Triphosphate; Animals; Area Postrema; Benzamides; Excitatory Amino Acid Agonists; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; Ganglionic Stimulants; Gastrointestinal Agents; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Kainic Acid; Male; N-Methylaspartate; Neurons; Nicotine; Patch-Clamp Techniques; Rats; Rats, Wistar; Thiazoles; Vagus Nerve

2010
Bitter pills for drug companies.
    BMJ (Clinical research ed.), 2010, Sep-17, Volume: 341

    Topics: Acetamides; Drug Approval; Drug Industry; Fraud; gamma-Aminobutyric Acid; Isoxazoles; Linezolid; Motivation; Off-Label Use; Oxazolidinones; Piperazines; Pregabalin; Sulfonamides; Thiazoles; United States

2010
Pharmacokinetics of oral gabapentin alone or co-administered with meloxicam in ruminant beef calves.
    Veterinary journal (London, England : 1997), 2011, Volume: 190, Issue:1

    Topics: Administration, Oral; Amines; Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Area Under Curve; Cattle; Cyclohexanecarboxylic Acids; Drug Therapy, Combination; Gabapentin; gamma-Aminobutyric Acid; Half-Life; Kinetics; Male; Meloxicam; Thiazines; Thiazoles

2011
Pharmacokinetics and milk secretion of gabapentin and meloxicam co-administered orally in Holstein-Friesian cows.
    Journal of veterinary pharmacology and therapeutics, 2013, Volume: 36, Issue:1

    Topics: Administration, Oral; Amines; Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Cattle; Cyclohexanecarboxylic Acids; Drug Therapy, Combination; Female; Gabapentin; gamma-Aminobutyric Acid; Meloxicam; Milk; Thiazines; Thiazoles

2013
Traumatic alterations in GABA signaling disrupt hippocampal network activity in the developing brain.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2012, Mar-21, Volume: 32, Issue:12

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Age Factors; Animals; Animals, Newborn; Antigens, Surface; Brain Injuries; Bumetanide; Caspases; Cell Count; Choline; Excitatory Amino Acid Antagonists; Female; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Humans; Imaging, Three-Dimensional; In Vitro Techniques; Luminescent Proteins; Male; Membrane Glycoproteins; Mice; Mice, Transgenic; Microscopy, Confocal; Nerve Net; Neurons; Phosphinic Acids; Propanolamines; Rats; Rats, Sprague-Dawley; Recombinant Fusion Proteins; Regression Analysis; Signal Transduction; Sodium Potassium Chloride Symporter Inhibitors; Statistics, Nonparametric; Thiazoles; Thioglycolates; Time Factors; Valine

2012
A study to compare circulating flunixin, meloxicam and gabapentin concentrations with prostaglandin E₂ levels in calves undergoing dehorning.
    Research in veterinary science, 2013, Volume: 95, Issue:1

    Topics: Amines; Analgesics; Animals; Area Under Curve; Cattle; Clonixin; Cyclohexanecarboxylic Acids; Dinoprostone; Gabapentin; gamma-Aminobutyric Acid; Half-Life; Horns; Male; Meloxicam; Pain; Random Allocation; Statistics, Nonparametric; Thiazines; Thiazoles

2013
Synthesis and anticonvulsant activity evaluation of 7-alkoxy[1,2,4]triazolo[3,4-b]benzothiazol-3(2H)-ones.
    Archiv der Pharmazie, 2014, Volume: 347, Issue:4

    Topics: Administration, Oral; Animals; Anticonvulsants; Disease Models, Animal; Electroshock; gamma-Aminobutyric Acid; Mice; Neurotoxicity Syndromes; Seizures; Structure-Activity Relationship; Thiazoles

2014
Impact of oral meloxicam administered alone or in combination with gabapentin on experimentally induced lameness in beef calves.
    Journal of animal science, 2014, Volume: 92, Issue:2

    Topics: Amines; Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Cattle; Cattle Diseases; Cyclohexanecarboxylic Acids; Gabapentin; gamma-Aminobutyric Acid; Lameness, Animal; Male; Meloxicam; Thiazines; Thiazoles

2014
GABAA Receptor-Mediated Bidirectional Control of Synaptic Activity, Intracellular Ca2+, Cerebral Blood Flow, and Oxygen Consumption in Mouse Somatosensory Cortex In Vivo.
    Cerebral cortex (New York, N.Y. : 1991), 2015, Volume: 25, Issue:9

    Topics: Action Potentials; Animals; Biophysics; Calcium; Cerebrovascular Circulation; Dose-Response Relationship, Drug; Egtazic Acid; Electric Stimulation; Functional Laterality; GABA Agonists; gamma-Aminobutyric Acid; Isoxazoles; Mice; Oxygen Consumption; Partial Pressure; Pyridines; Receptors, GABA-A; Somatosensory Cortex; Sulfonamides; Thiazoles; Vibrissae; Zolpidem

2015
On the contribution of KCC2 and carbonic anhydrase to two types of in vitro interictal discharge.
    Pflugers Archiv : European journal of physiology, 2015, Volume: 467, Issue:11

    Topics: Acetazolamide; Animals; CA3 Region, Hippocampal; Carbonic Anhydrase Inhibitors; Carbonic Anhydrases; gamma-Aminobutyric Acid; Male; Membrane Potentials; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Seizures; Solute Carrier Family 12, Member 1; Thiazoles; Thioglycolates

2015
Engagement of the GABA to KCC2 signaling pathway contributes to the analgesic effects of A3AR agonists in neuropathic pain.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2015, 04-15, Volume: 35, Issue:15

    Topics: Adenosine; Adenosine A3 Receptor Agonists; Analgesics; Animals; Disease Models, Animal; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; HEK293 Cells; Humans; Hyperalgesia; K Cl- Cotransporters; Male; Mice; Pain Threshold; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sciatica; Signal Transduction; Spinal Nerve Roots; Symporters; Thiazoles; Thioglycolates

2015
Differential effects of GABA in modulating nociceptive vs. non-nociceptive synapses.
    Neuroscience, 2015, Jul-09, Volume: 298

    Topics: Acetylcholine; Animals; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Postsynaptic Potentials; GABA Agents; gamma-Aminobutyric Acid; Ganglia, Invertebrate; Leeches; Membrane Potentials; Neostigmine; Nociceptors; Patch-Clamp Techniques; Physical Stimulation; Pressure; Sodium Potassium Chloride Symporter Inhibitors; Synapses; Synaptic Transmission; Thiazoles; Thioglycolates

2015
Positive modulation of synaptic and extrasynaptic GABAA receptors by an antagonist of the high affinity benzodiazepine binding site.
    Neuropharmacology, 2015, Volume: 95

    Topics: Allosteric Regulation; Animals; Benzodiazepines; Binding Sites; Diazepam; Flumazenil; GABA Agents; gamma-Aminobutyric Acid; HEK293 Cells; Humans; Membrane Potentials; Mutation; Neurons; Oocytes; Patch-Clamp Techniques; Protein Isoforms; Quinolines; Radioligand Assay; Receptors, GABA-A; Recombinant Proteins; Thiazoles; Transfection; Xenopus laevis

2015
Antinociceptive Interactions Between Meloxicam and Gabapentin in Neuropathic Pain Depend on the Ratio used in Combination in Rats.
    Drug development research, 2016, Volume: 77, Issue:3

    Topics: Amines; Analgesics; Animals; Area Under Curve; Cyclohexanecarboxylic Acids; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Synergism; Drug Therapy, Combination; Gabapentin; gamma-Aminobutyric Acid; Male; Meloxicam; Neuralgia; Rats; Thiazines; Thiazoles; Treatment Outcome

2016
GABA and glutamate moderate beta-amyloid related functional connectivity in cognitively unimpaired old-aged adults.
    NeuroImage. Clinical, 2019, Volume: 22

    Topics: Aged; Aging; Amyloid beta-Peptides; Aniline Compounds; Cerebellum; Cerebral Cortex; Connectome; Female; gamma-Aminobutyric Acid; Glutamic Acid; Gray Matter; Humans; Magnetic Resonance Imaging; Magnetic Resonance Spectroscopy; Male; Neuroimaging; Positron-Emission Tomography; Thiazoles

2019