Page last updated: 2024-08-21

thiazoles and fluorobenzenes

thiazoles has been researched along with fluorobenzenes in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (50.00)29.6817
2010's4 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Adell, A; Amargós-Bosch, M; Artigas, F; Bortolozzi, A; Díaz-Mataix, L; Pons, S; Serrats, J1
Hazemann, I; Joachimiak, A; Karplus, M; Mitschler, A; Podjarny, A; Ruiz, F; Schneider, T1
Hirano, T; Iseki, K; Itagaki, S; Kagawa, T; Kobayashi, M; Takano, R1
An, X; Guo, CC; Li, X; Tan, Z; Wang, S; Xie, K; Yang, Z; Zhou, X1
Aznar, S; El-Sayed, M; Elvang, AB; Ettrup, A; Holm, P; Klein, AB; Knudsen, GM; Mikkelsen, JD; Santini, MA; Stensbøl, TB1
Andrews, J; Cheng, A; Custodio, JM; Hao, J; Kearney, BP; Lepist, EI; Ling, KH; Ramanathan, S; Ray, AS; Wang, H1
Amar, E; Dolkart, O; Marmor, S; Shapira, S; Steinberg, EL; Weinbroum, AA1

Trials

1 trial(s) available for thiazoles and fluorobenzenes

ArticleYear
Pharmacokinetics of cobicistat boosted-elvitegravir administered in combination with rosuvastatin.
    Journal of clinical pharmacology, 2014, Volume: 54, Issue:6

    Topics: Adult; Animals; Anti-HIV Agents; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Carbamates; CHO Cells; Cobicistat; Cricetulus; Dogs; Drug Combinations; Drug Interactions; Drug Therapy, Combination; Female; Fluorobenzenes; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Liver-Specific Organic Anion Transporter 1; Madin Darby Canine Kidney Cells; Male; Neoplasm Proteins; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Pyrimidines; Quinolones; Rosuvastatin Calcium; Solute Carrier Organic Anion Transporter Family Member 1B3; Sulfonamides; Thiazoles

2014

Other Studies

7 other study(ies) available for thiazoles and fluorobenzenes

ArticleYear
In vivo modulation of 5-hydroxytryptamine release in mouse prefrontal cortex by local 5-HT(2A) receptors: effect of antipsychotic drugs.
    The European journal of neuroscience, 2003, Volume: 18, Issue:5

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Aminopyridines; Anesthetics, Local; Animals; Antipsychotic Agents; Benzopyrans; Blotting, Western; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Fluorobenzenes; Immunohistochemistry; In Situ Hybridization; Indoles; Indophenol; Male; Mice; Mice, Inbred C57BL; Microdialysis; Piperidines; Prazosin; Prefrontal Cortex; Quinoxalines; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Thiazoles; Time Factors

2003
New drugs and dosage forms.
    American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists, 2003, Oct-01, Volume: 60, Issue:19

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Clobetasol; Dosage Forms; Drug Combinations; Fluorobenzenes; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hypoglycemic Agents; Imidazoles; Metformin; Pharmaceutical Preparations; Phosphodiesterase Inhibitors; Piperazines; Pyrimidines; Rosuvastatin Calcium; Sulfonamides; Sulfones; Thiazoles; Triazines; United States; United States Food and Drug Administration; Vardenafil Dihydrochloride

2003
The crystallographic structure of the aldose reductase-IDD552 complex shows direct proton donation from tyrosine 48.
    Acta crystallographica. Section D, Biological crystallography, 2004, Volume: 60, Issue:Pt 8

    Topics: Aldehyde Reductase; Binding Sites; Carboxylic Acids; Crystallography, X-Ray; Enzyme Inhibitors; Fluorobenzenes; Humans; Hydrogen-Ion Concentration; Models, Molecular; Molecular Structure; NADP; Protein Structure, Tertiary; Protons; Thiazoles; Tyrosine

2004
Effect of medium pH on the cytotoxicity of hydrophilic statins.
    Journal of pharmacy & pharmaceutical sciences : a publication of the Canadian Society for Pharmaceutical Sciences, Societe canadienne des sciences pharmaceutiques, 2007, Volume: 10, Issue:3

    Topics: Animals; Apoptosis; Caspases; Cell Line; Cell Survival; Chromatography, High Pressure Liquid; Fluorobenzenes; Humans; Hydrogen-Ion Concentration; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Muscle, Skeletal; Myoblasts; Pravastatin; Pyrimidines; Rats; Rhabdomyosarcoma, Embryonal; Rosuvastatin Calcium; Sulfonamides; Tetrazolium Salts; Thiazoles; Toxicity Tests

2007
Pd-catalyzed decarboxylative arylation of thiazole, benzoxazole, and polyfluorobenzene with substituted benzoic acids.
    Organic letters, 2010, Apr-02, Volume: 12, Issue:7

    Topics: Benzoates; Benzoxazoles; Catalysis; Decarboxylation; Fluorobenzenes; Molecular Structure; Palladium; Stereoisomerism; Thiazoles

2010
Plaque deposition dependent decrease in 5-HT2A serotonin receptor in AbetaPPswe/PS1dE9 amyloid overexpressing mice.
    Journal of Alzheimer's disease : JAD, 2010, Volume: 20, Issue:4

    Topics: Aging; Amphetamines; Amyloid beta-Protein Precursor; Aniline Compounds; Animals; Autoradiography; Citalopram; Data Interpretation, Statistical; Fluorobenzenes; Genes, fos; Head Movements; Humans; In Situ Hybridization; Indicators and Reagents; Male; Mice; Mice, Transgenic; Piperidines; Plaque, Amyloid; Receptor, Serotonin, 5-HT2A; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Serotonin Receptor Agonists; Thiazoles

2010
Protective effects of rosuvastatin in a rat model of lung contusion: Stimulation of the cyclooxygenase 2-prostaglandin E-2 pathway.
    Surgery, 2015, Volume: 157, Issue:5

    Topics: Acute Lung Injury; Animals; Bronchoalveolar Lavage Fluid; Contusions; Cyclooxygenase 2; Dinoprostone; Disease Models, Animal; Drug Evaluation, Preclinical; Fluorobenzenes; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Lung; Male; Meloxicam; Pyrimidines; Random Allocation; Rats; Rosuvastatin Calcium; Sulfonamides; Thiazines; Thiazoles

2015