Page last updated: 2024-08-21

thiazoles and fluorine

thiazoles has been researched along with fluorine in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-19903 (13.64)18.7374
1990's2 (9.09)18.2507
2000's7 (31.82)29.6817
2010's10 (45.45)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Berry, WK; Davies, DR; Gordon, JJ1
Colby, TD; Goldstein, BM; Jones, JP; Pankiewicz, KW; Zatorski, A1
Goldstein, BM; Lipka, P; Mollova, N; Pankiewicz, KW; Schram, KH; Watanabe, KA; Zatorski, A1
Li, Z; Liu, Z; Qian, X; Song, G1
Eckelman, WC; Huang, BX; Jagoda, EM; Kiesewetter, DO; Ma, Y1
BAHEL, SC; GIRI, S; JOSHI, KC1
INOUE, S; NAGANO, H; NODIFF, EA; SAGGIOMO, AJ1
Amir, E; Rozen, S1
Ballard, P; Bradbury, RH; Harris, CS; Hennequin, LF; Hickinson, M; Kendrew, J; Kettle, JG; Klinowska, T; Ogilvie, DJ; Pearson, SE; Williams, EJ; Wilson, I1
Askew, B; Bartberger, MD; Cai, L; Chen, M; Cupples, R; Emery, M; Fotsch, C; Hale, C; Han, N; Hungate, RW; Johansson, L; Jordan, S; Li, A; Liu, Q; Moniz, G; Pyring, D; St Jean, DJ; Sun, Y; Tedenborg, L; Wang, M; Williams, M; Yuan, C; Zhang, J1
d'Agostino, R; D'Aloia, E; Favia, P; Gristina, R; Milella, A; Nardulli, M; Sardella, E; Senesi, GS1
Camilleri, J1
Barbeau, O; Brigaud, T; Chaume, G; Lesot, P1
Jiang, XQ; Yu, WQ; Zhang, FQ; Zhang, YL1
Fisker, E; Jacobsen, CB; Jørgensen, KA; Nielsen, M; Worgull, D; Zweifel, T1
Brender, JR; Hartman, K; Marsh, EN; Ramamoorthy, A; Suzuki, Y1
Durga Prasad, K; Pavan, MS; Row, TN1
Gao, YQ; Mou, W; Wang, P; Wu, K; Xu, S; Zhang, S1
Aonuma, M; Fukutake, S; Kawato, H; Kitagawa, M; Miyazaki, M; Naito, H; Okayama, T; Seki, T; Soga, T; Sugimoto, Y; Uoto, K; Yoshida, K1
Camenisch, G; James, AD; Luneau, A; Marvalin, C; Meissner, A1
Brigaud, T; Chaume, G; Lensen, N; Miclet, E; Pytkowicz, J; Simon, J1
Coogan, MP; Griffin, JM; Hughes, E; Middleton, DA1

Other Studies

22 other study(ies) available for thiazoles and fluorine

ArticleYear
Protection of animals against soman (1,2,2-trimethylpropyl methylphosphono-fluoridate) by pretreatment with some other organophosphorus compounds, followed by oxime and atropine.
    Biochemical pharmacology, 1971, Volume: 20, Issue:1

    Topics: Amitriptyline; Animals; Atropine; Bromides; Carbamates; Cholinesterase Inhibitors; Diphosphates; Drug Antagonism; Female; Fluorine; Guinea Pigs; Hydroxamic Acids; Isoflurophate; Lethal Dose 50; Nitrates; Nitrophenols; Nitroso Compounds; Organophosphonates; Organophosphorus Compounds; Orphenadrine; Oximes; Parasympatholytics; Physostigmine; Poisoning; Pyridinium Compounds; Rabbits; Rats; Salicylates; Scopolamine; Species Specificity; Sulfonic Acids; Sulfuric Acids; Thiazoles; Time Factors

1971
Potent inhibitors of human inosine monophosphate dehydrogenase type II. Fluorine-substituted analogues of thiazole-4-carboxamide adenine dinucleotide.
    Journal of medicinal chemistry, 1995, Mar-31, Volume: 38, Issue:7

    Topics: Adenine Nucleotides; Adenosine Diphosphate; Animals; Fluorine; Horses; Humans; IMP Dehydrogenase; NAD; Recombinant Proteins; Thiazoles

1995
Synthesis of thiazole-4-carboxamide-adenine difluoromethylenediphosphonates substituted with fluorine at C-2' of the adenosine.
    Carbohydrate research, 1993, Oct-18, Volume: 249, Issue:1

    Topics: Adenine Nucleotides; Adenosine; Fluorine; Indicators and Reagents; Magnetic Resonance Spectroscopy; Molecular Structure; Spectrometry, Mass, Fast Atom Bombardment; Thiazoles

1993
Synthesis and quantitative structure-activity relationships of fluorine-containing 4,4-dihydroxylmethyl-2-aryliminooxazo(thiazo)lidines as trehalase inhibitors.
    Journal of agricultural and food chemistry, 2001, Volume: 49, Issue:11

    Topics: Animals; Drosophila melanogaster; Enzyme Inhibitors; Fluorine; Quantitative Structure-Activity Relationship; Thiazoles; Trehalase

2001
Identification of metabolites of fluorine-18-labeled M2 muscarinic receptor agonist, 3-(3-[(3-fluoropropyl)thio]-1,2,5-thiadiazol-4-yl)-1,2,5,6-tetrahydro-1-methylpyridine, produced by human and rat hepatocytes.
    Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 2002, Jan-25, Volume: 766, Issue:2

    Topics: Animals; Chromatography, High Pressure Liquid; Fluorine; Hepatocytes; Humans; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Muscarinic Agonists; Pyridines; Rats; Rats, Sprague-Dawley; Thiazoles; Tomography, Emission-Computed

2002
Fungicidal & insecticidal activity of some organic fluorine compounds containing aryloxy, benzamido, acetamido & thiazole ring systems.
    Journal of scientific & industrial research. C, Biological sciences, 1962, Volume: 21C

    Topics: Antifungal Agents; Fluorine; Fluorine Compounds; Fungicides, Industrial; Insecticides; Thiazoles

1962
FLUORINE-CONTAINING POTENTIAL ANTICANCER AGENTS. II. SYNTHESES OF SOME TRIFLUOROMETHYLPURINES AND TRIFLUOROMETHYLTHIAZOLOPYRIMIDINES.
    Journal of medicinal chemistry, 1964, Volume: 7

    Topics: Antineoplastic Agents; Chemistry, Pharmaceutical; Fluorine; Mice; Neoplasms; Neoplasms, Experimental; Pharmacology; Purines; Pyrimidines; Research; Thiazoles

1964
Easy access to the family of thiazole N-oxides using HOF x CH3CN.
    Chemical communications (Cambridge, England), 2006, Jun-04, Issue:21

    Topics: Acetonitriles; Fluorine; Hydrogen; Molecular Structure; Oxides; Thiazoles; Water; X-Ray Diffraction

2006
Inhibitors of epidermal growth factor receptor tyrosine kinase: optimisation of potency and in vivo pharmacokinetics.
    Bioorganic & medicinal chemistry letters, 2006, Sep-15, Volume: 16, Issue:18

    Topics: Animals; Antineoplastic Agents; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; ErbB Receptors; Fluorine; Gefitinib; Humans; Inhibitory Concentration 50; Mice; Molecular Structure; Neoplasms; Protein Kinase Inhibitors; Quinazolines; Rats; Structure-Activity Relationship; Thiazoles; Xenograft Model Antitumor Assays

2006
The discovery of 2-anilinothiazolones as 11beta-HSD1 inhibitors.
    Bioorganic & medicinal chemistry letters, 2007, Nov-15, Volume: 17, Issue:22

    Topics: 11-beta-Hydroxysteroid Dehydrogenase Type 1; Animals; Chlorine; CHO Cells; Cricetinae; Cricetulus; Crystallography, X-Ray; Fluorine; Humans; Molecular Structure; Rats; Structure-Activity Relationship; Thiazoles

2007
Increasing cell adhesion on plasma deposited fluorocarbon coatings by changing the surface topography.
    Journal of biomedical materials research. Part B, Applied biomaterials, 2009, Volume: 88, Issue:1

    Topics: 3T3 Cells; Animals; Biocompatible Materials; Carbon; Cell Adhesion; Cell Membrane; Colloids; Extracellular Matrix; Fluorine; Fluorocarbons; Humans; Mice; Microscopy, Electron, Scanning; Surface Properties; Tetrazolium Salts; Thiazoles

2009
The biocompatibility of modified experimental Portland cements with potential for use in dentistry.
    International endodontic journal, 2008, Volume: 41, Issue:12

    Topics: Aluminum; Aluminum Compounds; Biocompatible Materials; Calcium Compounds; Cell Line, Tumor; Cell Survival; Coloring Agents; Dental Cements; Fluorine; Glass Ionomer Cements; Humans; Humidity; Indicators and Reagents; Materials Testing; Oxazines; Sulfur Compounds; Temperature; Tetrazolium Salts; Thiazoles; Time Factors; Xanthenes

2008
Synthesis of 2-trifluoromethyl-1,3-oxazolidines as hydrolytically stable pseudoprolines.
    The Journal of organic chemistry, 2010, Jun-18, Volume: 75, Issue:12

    Topics: Acylation; Esters; Fluorine; Methane; Molecular Structure; Oxazoles; Proline; Thiazoles

2010
In vitro behavior of MC3T3-E1 preosteoblast with different annealing temperature titania nanotubes.
    Oral diseases, 2010, Volume: 16, Issue:7

    Topics: 3T3 Cells; Animals; Anthraquinones; Biocompatible Materials; Calcification, Physiologic; Cell Adhesion; Cell Culture Techniques; Cell Proliferation; Cell Shape; Cell Survival; Coloring Agents; Crystallization; Crystallography; Fluorine; Hot Temperature; Materials Testing; Mice; Microscopy, Atomic Force; Microscopy, Confocal; Microscopy, Electron, Scanning; Nanotubes; Osteoblasts; Photoelectron Spectroscopy; Surface Properties; Tetrazolium Salts; Thiazoles; Titanium; X-Ray Diffraction

2010
Asymmetric organocatalytic monofluorovinylations.
    Journal of the American Chemical Society, 2011, May-18, Volume: 133, Issue:19

    Topics: Catalysis; Fluorine; Molecular Structure; Peptides; Stereoisomerism; Sulfones; Thiazoles; Vinyl Compounds

2011
Alternative pathways of human islet amyloid polypeptide aggregation distinguished by (19)f nuclear magnetic resonance-detected kinetics of monomer consumption.
    Biochemistry, 2012, Oct-16, Volume: 51, Issue:41

    Topics: Benzothiazoles; Catechin; Circular Dichroism; Fluorine; Humans; Islet Amyloid Polypeptide; Kinetics; Nuclear Magnetic Resonance, Biomolecular; Protein Binding; Spectrometry, Fluorescence; Thiazoles

2012
Halogen bonding in fluorine: experimental charge density study on intermolecular F···F and F···S donor-acceptor contacts.
    Chemical communications (Cambridge, England), 2013, Sep-04, Volume: 49, Issue:68

    Topics: Binding Sites; Fluorine; Models, Molecular; Molecular Structure; Sulfur; Thiazoles

2013
Construction and characterization on composite electrospinning fibers doped with iridium complex owing fluorine atoms in its auxiliary ligand.
    Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy, 2014, Oct-15, Volume: 131

    Topics: Coordination Complexes; Crystallization; Crystallography, X-Ray; Electrochemical Techniques; Fluorine; Halogenation; Iridium; Ligands; Luminescence; Microtechnology; Models, Molecular; Pentanes; Povidone; Thiazoles

2014
Discovery of DS-5272 as a promising candidate: A potent and orally active p53-MDM2 interaction inhibitor.
    Bioorganic & medicinal chemistry, 2015, May-15, Volume: 23, Issue:10

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Bone Neoplasms; Cell Line, Tumor; Cell Proliferation; Drug Discovery; Fluorine; Gene Expression; Humans; Imidazoles; Male; Mice; Mice, Inbred BALB C; Mice, Nude; Protein Binding; Proto-Oncogene Proteins c-mdm2; Pyrrolidines; Sarcoma; Thiazoles; Tumor Suppressor Protein p53; Xenograft Model Antitumor Assays

2015
Comparison of
    Drug metabolism and disposition: the biological fate of chemicals, 2017, Volume: 45, Issue:8

    Topics: Carbon Radioisotopes; Chromatography, Liquid; Fluorine; Humans; Magnetic Resonance Imaging; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Thiazoles

2017
Homochiral versus Heterochiral Trifluoromethylated Pseudoproline Containing Dipeptides: A Powerful Tool to Switch the Prolyl-Amide Bond Conformation.
    The Journal of organic chemistry, 2017, 12-15, Volume: 82, Issue:24

    Topics: Amides; Dipeptides; Fluorine; Methylation; Molecular Structure; Proline; Stereoisomerism; Thiazoles

2017
Average orientation of a fluoroaromatic molecule in lipid bilayers from DFT-informed NMR measurements of
    Physical chemistry chemical physics : PCCP, 2018, Jul-11, Volume: 20, Issue:27

    Topics: Aniline Compounds; Anisotropy; Diffusion; Dimyristoylphosphatidylcholine; Fluorine; Hydrogen; Hydrophobic and Hydrophilic Interactions; Lipid Bilayers; Magnetic Resonance Spectroscopy; Models, Molecular; Molecular Structure; Organic Chemicals; Thiazoles

2018