Page last updated: 2024-08-21

thiazoles and flumazenil

thiazoles has been researched along with flumazenil in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (25.00)18.2507
2000's2 (50.00)29.6817
2010's1 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chimirri, A; DeSarro, A; DeSarro, GB; Grasso, S; Zappalà, M1
Ai, J; Fomum, ZT; Nielsen, M; Sterner, O; Wahe, H; Wang, X; Witt, MR1
Chojnacka-Wójcik, E; Cosford, ND; Klodzinska, A; Nowak, G; Pilc, A; Tatarczyńska, E1
Baur, R; Maldifassi, MC; Middendorp, SJ; Sigel, E1

Other Studies

4 other study(ies) available for thiazoles and flumazenil

ArticleYear
Molecular requirement for anticonvulsant activity in a series of thiazolo-1,4-benzodiazepine derivatives and comparison with classical benzodiazepines.
    General pharmacology, 1993, Volume: 24, Issue:4

    Topics: Acoustic Stimulation; Animals; Anticonvulsants; Benzodiazepines; Binding, Competitive; Body Temperature; Flumazenil; Flunitrazepam; In Vitro Techniques; Injections, Intraperitoneal; Male; Mice; Mice, Inbred DBA; Molecular Weight; Pentylenetetrazole; Rats; Rats, Sprague-Dawley; Seizures; Structure-Activity Relationship; Thiazoles

1993
2-Oxo-2H-Pyrimido[2,1-b]benzothiazoles inhibit brain benzodiazepine receptor binding in vitro.
    Pharmacology, 2000, Volume: 60, Issue:4

    Topics: Animals; Benzothiazoles; Brain; Flumazenil; GABA Modulators; Humans; Male; Rats; Rats, Wistar; Receptors, GABA-A; Thiazoles

2000
Anxiolytic-like effects of MTEP, a potent and selective mGlu5 receptor agonist does not involve GABA(A) signaling.
    Neuropharmacology, 2004, Volume: 47, Issue:3

    Topics: Animals; Behavior, Animal; Diazepam; Dose-Response Relationship, Drug; Drinking; Drinking Behavior; Drug Interactions; Electroshock; Exploratory Behavior; Flumazenil; GABA Modulators; Male; Maze Learning; Mice; Pyridines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, GABA-A; Receptors, Metabotropic Glutamate; Sensory Thresholds; Signal Transduction; Thiazoles

2004
Positive modulation of synaptic and extrasynaptic GABAA receptors by an antagonist of the high affinity benzodiazepine binding site.
    Neuropharmacology, 2015, Volume: 95

    Topics: Allosteric Regulation; Animals; Benzodiazepines; Binding Sites; Diazepam; Flumazenil; GABA Agents; gamma-Aminobutyric Acid; HEK293 Cells; Humans; Membrane Potentials; Mutation; Neurons; Oocytes; Patch-Clamp Techniques; Protein Isoforms; Quinolines; Radioligand Assay; Receptors, GABA-A; Recombinant Proteins; Thiazoles; Transfection; Xenopus laevis

2015