thiazoles has been researched along with fenobam in 6 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 1 (16.67) | 29.6817 |
| 2010's | 5 (83.33) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Fischer, C; Gerber, PR; Jaeschke, G; Kratochwil, N; Malherbe, P; Mühlemann, A; Porter, RH; Stahl, M; Zenner, MT | 1 |
| Bi, GH; Gardner, EL; Keck, TM; Newman, AH; Srivastava, R; Wang, XF; Xi, ZX; Yang, HJ; Zhang, HY; Zou, MF | 1 |
| Ellgren, M; Raboisson, P; Swedberg, MD | 1 |
| Hosseini, SA; Iman, M; Jafari, R; Javidan, A; Taghizadeh, MJ | 1 |
| Berardo, C; Di Pasqua, LG; Ferrigno, A; Nicoletti, F; Richelmi, P; Siciliano, V; Vairetti, M | 1 |
| Christopher, JA; Congreve, M; Doré, AS; Errey, JC; Ferenczy, GG; Keserű, GM; Marshall, FH; Mason, JS; Okrasa, K; Orgován, Z; Rucktooa, P; Serrano-Vega, MJ | 1 |
6 other study(ies) available for thiazoles and fenobam
| Article | Year |
|---|---|
Comparison of the binding pockets of two chemically unrelated allosteric antagonists of the mGlu5 receptor and identification of crucial residues involved in the inverse agonism of MPEP.
Topics: Binding Sites; Calcium; Cell Line; Cell Membrane; Cells, Cultured; Excitatory Amino Acid Antagonists; Fluorometry; Humans; Imidazoles; Inositol Phosphates; Models, Molecular; Mutation; Plasmids; Pyridines; Quisqualic Acid; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Thiazoles | 2006 |
A novel mGluR5 antagonist, MFZ 10-7, inhibits cocaine-taking and cocaine-seeking behavior in rats.
Topics: Allosteric Regulation; Analysis of Variance; Animals; Binding, Competitive; Cocaine; Cues; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Enzyme-Linked Immunosorbent Assay; Excitatory Amino Acid Antagonists; HEK293 Cells; Humans; Imidazoles; In Vitro Techniques; Infusions, Intravenous; Inhibitory Concentration 50; Male; Motor Activity; Nitriles; Piperidines; Pyridines; Random Allocation; Rats; Receptor, Metabotropic Glutamate 5; Reinforcement Schedule; Reward; Secondary Prevention; Self Administration; Sucrose; Thiazoles | 2014 |
mGluR5 antagonist-induced psychoactive properties: MTEP drug discrimination, a pharmacologically selective non-NMDA effect with apparent lack of reinforcing properties.
Topics: Animals; Behavior, Animal; Discrimination, Psychological; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Imidazoles; Male; Phencyclidine; Psychotropic Drugs; Pyridines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, N-Methyl-D-Aspartate; Reinforcement, Psychology; Self Administration; Thiazoles | 2014 |
Docking, Molecular Dynamics Simulation and Synthesis of New Fenobam Analogues as mGlu5 Receptor Antagonists.
Topics: Anti-Anxiety Agents; Computer Simulation; Humans; Imidazoles; Molecular Docking Simulation; Molecular Dynamics Simulation; Molecular Structure; Receptor, Metabotropic Glutamate 5; Thiazoles | 2016 |
Selective Blockade of the Metabotropic Glutamate Receptor mGluR5 Protects Mouse Livers in In Vitro and Ex Vivo Models of Ischemia Reperfusion Injury.
Topics: Adenosine Triphosphate; Animals; Cell Hypoxia; Disease Models, Animal; Hepatocytes; Imidazoles; Liver; Mice; Mitochondria, Liver; Piperidines; Pyridines; Rats; Receptor, Metabotropic Glutamate 5; Reperfusion Injury; Thiazoles; Tumor Necrosis Factor-alpha | 2018 |
Structure-Based Optimization Strategies for G Protein-Coupled Receptor (GPCR) Allosteric Modulators: A Case Study from Analyses of New Metabotropic Glutamate Receptor 5 (mGlu
Topics: Allosteric Regulation; Allosteric Site; Crystallography, X-Ray; Drug Design; Humans; Imidazoles; Indoles; Ligands; Molecular Docking Simulation; Protein Structure, Tertiary; Pyridines; Receptor, Metabotropic Glutamate 5; Thiazoles; Water | 2019 |