thiazoles has been researched along with dimaprit in 36 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 17 (47.22) | 18.7374 |
1990's | 17 (47.22) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 2 (5.56) | 2.80 |
Authors | Studies |
---|---|
Bull, HA; Courtney, PF; Dowd, PM; Rustin, MH | 1 |
Nowak, JZ; Sek, B | 2 |
Mutafova-Yambolieva, V; Staneva-Stoytcheva, D; Todorov, S; Vassilev, P | 1 |
Madrid, JA; Pariente, JA; Salido, GM | 2 |
Raybould, HE; Yoneda, M | 1 |
Bordi, F; Catellani, PL; Impicciatore, M; Morini, G; Plazzi, PV; Silva, C; Vaona, G | 1 |
Rising, TJ; Steward, A | 1 |
Knigge, U; Matzen, S; Warberg, J | 2 |
Coruzzi, G; Noci, MT | 1 |
Bertaccini, G; Coruzzi, G; Dobrilla, G; Noci, MT | 1 |
Bertaccini, G; Coruzzi, G | 1 |
Franco, P; Guidobono, F; Netti, C; Pecile, A; Sibilia, V; Villa, I | 1 |
Akahori, H; Kamei, C; Kitazumi, K; Tasaka, K | 1 |
Barocelli, E; Bordi, F; Chiavarini, M; Impicciatore, M; Morini, G; Plazzi, PV; Vitali, F | 1 |
Maeno, H; Takagi, T; Takeda, M | 1 |
Guldvog, I; Linnestad, P; Schrumpf, E | 1 |
Badger, AM; Poste, G; Young, J | 1 |
Bordi, F; Chiavarini, M; Impicciatore, M; Morini, G | 1 |
Brooks, HL; Christensen, CW; Gross, GJ; Hardman, HF; Warltier, DC | 1 |
Daly, MJ; Humphray, JM; Stables, R | 1 |
Wong, CL | 1 |
Carson, CC; Davies, MG; Hagen, PO; Kim, YC; Lee, TH | 1 |
Iinuma, K; Onodera, K; Watanabe, T; Yokoyama, H | 1 |
Bertaccini, G; Coruzzi, G; Poli, E; Pozzoli, C; Timmerman, H | 2 |
Malinowska, B; Schlicker, E | 1 |
Davison, JS; Jennings, LJ; Lea, RW; Pozo, MJ; Salido, GM; Sharkey, KA; Singh, J | 1 |
Blandina, P; Cecchi, M; Giorgetti, M; Giovannini, MG; Leurs, R; Timmerman, H | 1 |
Bertaccini, G; Coruzzi, G; Gambarelli, E; Timmerman, H | 1 |
Meade, HM; Seeley, NA; Sturman, G | 1 |
Chen, Z; Fujii, Y; Kamei, C; Sugimoto, Y; Suzuki, G | 1 |
Gorog, DA | 1 |
Awane, H; Ezaki, M; Hishinuma, S; Inazuki, N; Michinaga, S; Mizuguchi, H; Shimizu, K; Sonoda, K | 1 |
36 other study(ies) available for thiazoles and dimaprit
Article | Year |
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Characterization of histamine receptor sub-types regulating prostacyclin release from human endothelial cells.
Topics: Cells, Cultured; Dimaprit; Endothelium, Vascular; Epoprostenol; Histamine; Histamine Agonists; Humans; Impromidine; Methylhistamines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Thiazoles; Umbilical Veins | 1992 |
Cyclic AMP generating systems in vertebrate retina: effects of histamine and an established retinal modulator, dopamine.
Topics: Adenylyl Cyclases; Animals; Cerebral Cortex; Chickens; Cimetidine; Colforsin; Cyclic AMP; Dimaprit; Dopamine; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Retina; Thiazoles; Thiourea | 1991 |
Involvement of calcium ions in the modulation of electrically-induced rat vas deferens contractions by histaminergic drugs.
Topics: Animals; Calcium; Cimetidine; Dimaprit; Diphenhydramine; Electric Stimulation; Histamine; In Vitro Techniques; Male; Muscle Contraction; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea; Vas Deferens; Verapamil | 1991 |
Role of histamine receptors in rabbit pancreatic exocrine secretion stimulated by cholecystokinin and secretin.
Topics: Animals; Chlorpheniramine; Cholecystokinin; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Female; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Pancreas; Rabbits; Receptors, Histamine H1; Receptors, Histamine H2; Secretin; Thiazoles; Thiourea | 1990 |
Capsaicin-sensitive vagal afferent fibers do not contribute to histamine H2 receptor agonist-induced gastric acid secretion in anesthetized rats.
Topics: Anesthesia; Animals; Capsaicin; Dimaprit; Dose-Response Relationship, Drug; Gastric Acid; Injections, Subcutaneous; Male; Neurons, Afferent; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea; Vagus Nerve | 1990 |
Histamine receptors in unstimulated pancreatic exocrine secretion of the rabbit.
Topics: Animals; Chlorpheniramine; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Female; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; Kinetics; Male; Pancreas; Rabbits; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea | 1989 |
H2-antagonists: synthesis and activity of 2-amino-5-thiazolyl derivatives.
Topics: Amines; Animals; Cats; Chemical Phenomena; Chemistry; Dimaprit; Gastric Mucosa; Guinea Pigs; Heart; Histamine H2 Antagonists; In Vitro Techniques; Myocardial Contraction; Thiazoles; Thiourea | 1989 |
The determination of receptor constants for histamine H2-agonists in the guinea-pig isolated right atrium using an irreversible H2-antagonist.
Topics: Animals; Dimaprit; Dose-Response Relationship, Drug; Female; Guanidines; Guinea Pigs; Heart Rate; Histamine; Histamine H2 Antagonists; Imidazoles; Impromidine; In Vitro Techniques; Male; Methylhistamines; Receptors, Adrenergic, beta; Receptors, Histamine; Receptors, Histamine H2; Thiazoles; Thiourea | 1986 |
Histaminergic stimulation of prolactin secretion mediated via H1- or H2-receptors: dependence on routes of administration.
Topics: Animals; Cimetidine; Dimaprit; Histamine; Histamine H1 Antagonists; Male; Methylhistamines; Pituitary Gland, Anterior; Prolactin; Pyrilamine; Pyrimidinones; Rats; Receptors, Histamine; Thiazoles; Thiourea | 1986 |
[Effect of a new H2 receptor antagonist, famotidine, on gastric secretion].
Topics: Animals; Cats; Dimaprit; Dose-Response Relationship, Drug; Famotidine; Gastric Mucosa; Histamine; Histamine H2 Antagonists; Ranitidine; Rats; Thiazoles; Thiourea | 1986 |
Inhibitory effect of famotidine on cat gastric secretion.
Topics: Animals; Cats; Dimaprit; Dose-Response Relationship, Drug; Famotidine; Female; Gastric Juice; Histamine H2 Antagonists; Ranitidine; Thiazoles; Thiourea | 1986 |
Famotidine and ranitidine: any difference in the duration of action?
Topics: Animals; Cats; Dimaprit; Famotidine; Gastric Acid; Gastric Juice; Histamine; Histamine H2 Antagonists; Ranitidine; Rats; Thiazoles; Thiourea; Time Factors | 1987 |
Further evidence that brain histamine H2 receptors are stimulatory in the control of prolactin in the rat.
Topics: Animals; Brain; Cimetidine; Dimaprit; Famotidine; Histamine H2 Antagonists; Injections, Intraventricular; Male; Methylhistamines; Prolactin; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Thiazoles; Thiourea | 1988 |
The effects of histamine and some related compounds on conditioned avoidance response in rats.
Topics: Acetylcholine; Animals; Avoidance Learning; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Hypothalamus; Injections, Intraventricular; Kinetics; Male; Methylhistamines; Pyrilamine; Rats; Rats, Inbred Strains; Scopolamine; Thiazoles; Thiourea | 1985 |
Are histamine receptors involved in the stimulant activities of thiazolylethylamines supposed as cyclic models of dimaprit?
Topics: Animals; Cats; Dimaprit; Drug Evaluation, Preclinical; Gastric Acid; Gastrointestinal Motility; Guinea Pigs; In Vitro Techniques; Models, Chemical; Molecular Conformation; Receptors, Histamine H2; Structure-Activity Relationship; Thiazoles; Thiourea | 1987 |
Histaminergic regulation of prolactin secretion: involvement of tuberoinfundibular dopaminergic neurons.
Topics: Animals; Cerebral Ventricles; Dimaprit; Dopamine; Histamine; Infusions, Intra-Arterial; Injections, Intraventricular; Male; Neurons; Prolactin; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2; Reference Values; Thiazoles; Thiourea | 1988 |
Kinetics of antisecretory action of a new H2-antagonist, YM-11170, in conscious dogs.
Topics: Animals; Atropine; Cimetidine; Dimaprit; Dogs; Famotidine; Gastric Acid; Gastric Mucosa; Histamine H2 Antagonists; Kinetics; Male; Methacholine Chloride; Methacholine Compounds; Pentagastrin; Thiazoles; Thiourea | 1983 |
The effect of histamine, H1 and H2 agonists, and H1 and H2 antagonists on postprandial pancreatic polypeptide release in dogs.
Topics: Animals; Cimetidine; Dimaprit; Dogs; Food; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Pancreatic Polypeptide; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Secretory Rate; Thiazoles; Thiourea | 1983 |
Inhibition of phytohaemagglutinin-induced proliferation of human peripheral blood lymphocytes by histamine and histamine H1 and H2 agonists.
Topics: Cell Division; Cells, Cultured; Dimaprit; Dose-Response Relationship, Drug; Histamine; Humans; Imidazoles; Impromidine; Lymphocytes; Methylhistamines; Phytohemagglutinins; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea | 1983 |
A possible physiological role of histamine H2-receptors in rat mesenteric circulation.
Topics: Animals; Cimetidine; Dimaprit; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H2; Splanchnic Circulation; Thiazoles; Thiourea; Vasodilation | 1983 |
Effects of histamine receptor stimulation on regional myocardial blood flow.
Topics: Animals; Blood Pressure; Cimetidine; Coronary Circulation; Dimaprit; Diphenhydramine; Dogs; Female; Heart Rate; Histamine; Male; Microspheres; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea | 1983 |
Pharmacological interactions between ranitidine, cimetidine, metiamide and tiotidine at histamine H2-receptor sites in guinea-pig atria.
Topics: Animals; Cimetidine; Dimaprit; Drug Interactions; Furans; Guanidines; Guinea Pigs; Heart; Heart Rate; Histamine; In Vitro Techniques; Metiamide; Ranitidine; Receptors, Histamine; Receptors, Histamine H2; Thiazoles; Thiourea | 1982 |
Stimulatory effect of histamine on cyclic AMP formation in chick pineal gland.
Topics: 1-Methyl-3-isobutylxanthine; Adenine; Analysis of Variance; Animals; Carbon Radioisotopes; Chickens; Colforsin; Cyclic AMP; Dimaprit; Guinea Pigs; Hippocampus; Histamine; Histamine Agonists; In Vitro Techniques; Kinetics; Male; Methylhistamines; Pineal Gland; Ranitidine; Rats; Rats, Wistar; Thiazoles; Tritium | 1994 |
Effects of a histamine H2 receptor agonist and antagonist on restraint-induced antinociception in female mice.
Topics: Animals; Benzothiazoles; Cimetidine; Dimaprit; Female; Histamine Agonists; Histamine H2 Antagonists; Mice; Mice, Inbred Strains; Pain Measurement; Phenoxypropanolamines; Piperidines; Reaction Time; Restraint, Physical; Stress, Psychological; Thiazoles | 1995 |
Characterization and function of histamine receptors in corpus cavernosum.
Topics: Acetylcholine; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Electric Stimulation; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Papaverine; Penis; Piperidines; Pyrilamine; Rabbits; Receptors, Histamine; Thiazoles | 1995 |
2-Thiazolylethylamine, a selective histamine H1 agonist, decreases seizure susceptibility in mice.
Topics: Animals; Anticonvulsants; Dimaprit; Dose-Response Relationship, Drug; Electroshock; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Injections, Intraventricular; Male; Mice; Mice, Inbred Strains; Pentylenetetrazole; Receptors, Histamine H1; Seizures; Thiazoles | 1994 |
In vitro cardiac pharmacology of the new histamine H2-receptor agonist amthamine: comparisons with histamine and dimaprit.
Topics: Animals; Atrial Function; Dimaprit; Electric Stimulation; Guinea Pigs; Heart; Heart Atria; Histamine; Histamine Agonists; Humans; In Vitro Techniques; Myocardial Contraction; Papillary Muscles; Rabbits; Ranitidine; Thiazoles | 1993 |
Identification of endothelial H1, vascular H2 and cardiac presynaptic H3 receptors in the pithed rat.
Topics: Animals; Blood Pressure; Blood Vessels; Cardiovascular System; Dimaprit; Electric Stimulation; Endothelium, Vascular; Heart Rate; Histamine Agonists; Male; Methylhistamines; Myocardium; Rats; Rats, Wistar; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Thiazoles | 1993 |
The source and action of histamine in the isolated guinea-pig gallbladder.
Topics: Animals; Dimaprit; Electric Stimulation; Female; Gallbladder; Guinea Pigs; Histamine; Histamine Agonists; Histamine H2 Antagonists; Immunohistochemistry; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Ranitidine; Receptors, Histamine H3; Thiazoles | 1995 |
Histamine H3 receptor inhibition of K(+)-evoked release of acetylcholine from rat cortex in vivo.
Topics: Acetylcholine; Analysis of Variance; Animals; Chromatography, High Pressure Liquid; Dimaprit; Histamine; Histamine Agonists; Histamine Antagonists; Male; Methylhistamines; Microdialysis; Neurons; Parietal Lobe; Piperidines; Potassium; Rats; Rats, Wistar; Receptors, Histamine H3; Thiazoles | 1996 |
Cardiovascular effects of the novel histamine H2 receptor agonist amthamine: interaction with the adrenergic system.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cardiovascular System; Dimaprit; Dose-Response Relationship, Drug; Heart Rate; Histamine Agonists; Histamine H2 Antagonists; Male; Prazosin; Rats; Rats, Wistar; Tachycardia; Thiazoles | 1996 |
Histamine receptor-independent muscle relaxation elicited by a series of histamine H2-receptor agonists on the isolated guinea pig duodenum: a study into the mechanism of action.
Topics: Animals; Dimaprit; Duodenum; Electric Stimulation; Guinea Pigs; Histamine Agonists; Impromidine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Structure-Activity Relationship; Thiazoles | 1998 |
Histamine H2-receptor modulation in two mouse models of seizure susceptibility.
Topics: Acoustic Stimulation; Animals; Anticonvulsants; Benzothiazoles; Convulsants; Dimaprit; Female; Histamine Agonists; Histamine Antagonists; Male; Mice; Mice, Inbred DBA; Pentylenetetrazole; Phenoxypropanolamines; Piperidines; Receptors, Histamine H2; Seizures; Thiazoles | 1999 |
Effects of histamine and related compounds on regional cerebral blood flow in rats.
Topics: Animals; Benzothiazoles; Blood Pressure; Brain Chemistry; Dimaprit; Diphenhydramine; Drug Interactions; Hippocampus; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Male; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Rats, Wistar; Regional Blood Flow; Thiazoles; Time Factors | 1999 |
Understanding the Effects of NOAC Combined with Antiplatelet Therapy on Clot Kinetics.
Topics: Anticoagulants; Aspirin; Clopidogrel; Coronary Artery Disease; Dimaprit; Humans; Kinetics; Platelet Aggregation Inhibitors; Pyridines; Thiazoles | 2020 |
Selective histamine H
Topics: Angiopoietin-1; Animals; Blood-Brain Barrier; Brain Injuries, Traumatic; Dimaprit; Endothelial Cells; Evans Blue; Hedgehog Proteins; Histamine; Histamine Agonists; Male; Mice; Protective Factors; Ranitidine; Receptors, Histamine H2; RNA, Messenger; Thiazoles | 2022 |