Page last updated: 2024-08-21

thiazoles and dimaprit

thiazoles has been researched along with dimaprit in 36 studies

Research

Studies (36)

TimeframeStudies, this research(%)All Research%
pre-199017 (47.22)18.7374
1990's17 (47.22)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's2 (5.56)2.80

Authors

AuthorsStudies
Bull, HA; Courtney, PF; Dowd, PM; Rustin, MH1
Nowak, JZ; Sek, B2
Mutafova-Yambolieva, V; Staneva-Stoytcheva, D; Todorov, S; Vassilev, P1
Madrid, JA; Pariente, JA; Salido, GM2
Raybould, HE; Yoneda, M1
Bordi, F; Catellani, PL; Impicciatore, M; Morini, G; Plazzi, PV; Silva, C; Vaona, G1
Rising, TJ; Steward, A1
Knigge, U; Matzen, S; Warberg, J2
Coruzzi, G; Noci, MT1
Bertaccini, G; Coruzzi, G; Dobrilla, G; Noci, MT1
Bertaccini, G; Coruzzi, G1
Franco, P; Guidobono, F; Netti, C; Pecile, A; Sibilia, V; Villa, I1
Akahori, H; Kamei, C; Kitazumi, K; Tasaka, K1
Barocelli, E; Bordi, F; Chiavarini, M; Impicciatore, M; Morini, G; Plazzi, PV; Vitali, F1
Maeno, H; Takagi, T; Takeda, M1
Guldvog, I; Linnestad, P; Schrumpf, E1
Badger, AM; Poste, G; Young, J1
Bordi, F; Chiavarini, M; Impicciatore, M; Morini, G1
Brooks, HL; Christensen, CW; Gross, GJ; Hardman, HF; Warltier, DC1
Daly, MJ; Humphray, JM; Stables, R1
Wong, CL1
Carson, CC; Davies, MG; Hagen, PO; Kim, YC; Lee, TH1
Iinuma, K; Onodera, K; Watanabe, T; Yokoyama, H1
Bertaccini, G; Coruzzi, G; Poli, E; Pozzoli, C; Timmerman, H2
Malinowska, B; Schlicker, E1
Davison, JS; Jennings, LJ; Lea, RW; Pozo, MJ; Salido, GM; Sharkey, KA; Singh, J1
Blandina, P; Cecchi, M; Giorgetti, M; Giovannini, MG; Leurs, R; Timmerman, H1
Bertaccini, G; Coruzzi, G; Gambarelli, E; Timmerman, H1
Meade, HM; Seeley, NA; Sturman, G1
Chen, Z; Fujii, Y; Kamei, C; Sugimoto, Y; Suzuki, G1
Gorog, DA1
Awane, H; Ezaki, M; Hishinuma, S; Inazuki, N; Michinaga, S; Mizuguchi, H; Shimizu, K; Sonoda, K1

Other Studies

36 other study(ies) available for thiazoles and dimaprit

ArticleYear
Characterization of histamine receptor sub-types regulating prostacyclin release from human endothelial cells.
    British journal of pharmacology, 1992, Volume: 107, Issue:2

    Topics: Cells, Cultured; Dimaprit; Endothelium, Vascular; Epoprostenol; Histamine; Histamine Agonists; Humans; Impromidine; Methylhistamines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Thiazoles; Umbilical Veins

1992
Cyclic AMP generating systems in vertebrate retina: effects of histamine and an established retinal modulator, dopamine.
    Agents and actions, 1991, Volume: 33, Issue:1-2

    Topics: Adenylyl Cyclases; Animals; Cerebral Cortex; Chickens; Cimetidine; Colforsin; Cyclic AMP; Dimaprit; Dopamine; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Retina; Thiazoles; Thiourea

1991
Involvement of calcium ions in the modulation of electrically-induced rat vas deferens contractions by histaminergic drugs.
    General pharmacology, 1991, Volume: 22, Issue:4

    Topics: Animals; Calcium; Cimetidine; Dimaprit; Diphenhydramine; Electric Stimulation; Histamine; In Vitro Techniques; Male; Muscle Contraction; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea; Vas Deferens; Verapamil

1991
Role of histamine receptors in rabbit pancreatic exocrine secretion stimulated by cholecystokinin and secretin.
    Experimental physiology, 1990, Volume: 75, Issue:5

    Topics: Animals; Chlorpheniramine; Cholecystokinin; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Female; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Pancreas; Rabbits; Receptors, Histamine H1; Receptors, Histamine H2; Secretin; Thiazoles; Thiourea

1990
Capsaicin-sensitive vagal afferent fibers do not contribute to histamine H2 receptor agonist-induced gastric acid secretion in anesthetized rats.
    European journal of pharmacology, 1990, Sep-21, Volume: 186, Issue:2-3

    Topics: Anesthesia; Animals; Capsaicin; Dimaprit; Dose-Response Relationship, Drug; Gastric Acid; Injections, Subcutaneous; Male; Neurons, Afferent; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea; Vagus Nerve

1990
Histamine receptors in unstimulated pancreatic exocrine secretion of the rabbit.
    Agents and actions, 1989, Volume: 28, Issue:1-2

    Topics: Animals; Chlorpheniramine; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Female; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; Kinetics; Male; Pancreas; Rabbits; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea

1989
H2-antagonists: synthesis and activity of 2-amino-5-thiazolyl derivatives.
    Farmaco (Societa chimica italiana : 1989), 1989, Volume: 44, Issue:11

    Topics: Amines; Animals; Cats; Chemical Phenomena; Chemistry; Dimaprit; Gastric Mucosa; Guinea Pigs; Heart; Histamine H2 Antagonists; In Vitro Techniques; Myocardial Contraction; Thiazoles; Thiourea

1989
The determination of receptor constants for histamine H2-agonists in the guinea-pig isolated right atrium using an irreversible H2-antagonist.
    British journal of pharmacology, 1986, Volume: 87, Issue:1

    Topics: Animals; Dimaprit; Dose-Response Relationship, Drug; Female; Guanidines; Guinea Pigs; Heart Rate; Histamine; Histamine H2 Antagonists; Imidazoles; Impromidine; In Vitro Techniques; Male; Methylhistamines; Receptors, Adrenergic, beta; Receptors, Histamine; Receptors, Histamine H2; Thiazoles; Thiourea

1986
Histaminergic stimulation of prolactin secretion mediated via H1- or H2-receptors: dependence on routes of administration.
    Neuroendocrinology, 1986, Volume: 44, Issue:1

    Topics: Animals; Cimetidine; Dimaprit; Histamine; Histamine H1 Antagonists; Male; Methylhistamines; Pituitary Gland, Anterior; Prolactin; Pyrilamine; Pyrimidinones; Rats; Receptors, Histamine; Thiazoles; Thiourea

1986
[Effect of a new H2 receptor antagonist, famotidine, on gastric secretion].
    Bollettino della Societa italiana di biologia sperimentale, 1986, Sep-30, Volume: 62, Issue:9

    Topics: Animals; Cats; Dimaprit; Dose-Response Relationship, Drug; Famotidine; Gastric Mucosa; Histamine; Histamine H2 Antagonists; Ranitidine; Rats; Thiazoles; Thiourea

1986
Inhibitory effect of famotidine on cat gastric secretion.
    Agents and actions, 1986, Volume: 19, Issue:3-4

    Topics: Animals; Cats; Dimaprit; Dose-Response Relationship, Drug; Famotidine; Female; Gastric Juice; Histamine H2 Antagonists; Ranitidine; Thiazoles; Thiourea

1986
Famotidine and ranitidine: any difference in the duration of action?
    Pharmacological research communications, 1987, Volume: 19, Issue:1

    Topics: Animals; Cats; Dimaprit; Famotidine; Gastric Acid; Gastric Juice; Histamine; Histamine H2 Antagonists; Ranitidine; Rats; Thiazoles; Thiourea; Time Factors

1987
Further evidence that brain histamine H2 receptors are stimulatory in the control of prolactin in the rat.
    Acta endocrinologica, 1988, Volume: 119, Issue:4

    Topics: Animals; Brain; Cimetidine; Dimaprit; Famotidine; Histamine H2 Antagonists; Injections, Intraventricular; Male; Methylhistamines; Prolactin; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Thiazoles; Thiourea

1988
The effects of histamine and some related compounds on conditioned avoidance response in rats.
    Life sciences, 1985, Nov-25, Volume: 37, Issue:21

    Topics: Acetylcholine; Animals; Avoidance Learning; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Hypothalamus; Injections, Intraventricular; Kinetics; Male; Methylhistamines; Pyrilamine; Rats; Rats, Inbred Strains; Scopolamine; Thiazoles; Thiourea

1985
Are histamine receptors involved in the stimulant activities of thiazolylethylamines supposed as cyclic models of dimaprit?
    Agents and actions, 1987, Volume: 20, Issue:3-4

    Topics: Animals; Cats; Dimaprit; Drug Evaluation, Preclinical; Gastric Acid; Gastrointestinal Motility; Guinea Pigs; In Vitro Techniques; Models, Chemical; Molecular Conformation; Receptors, Histamine H2; Structure-Activity Relationship; Thiazoles; Thiourea

1987
Histaminergic regulation of prolactin secretion: involvement of tuberoinfundibular dopaminergic neurons.
    Neuroendocrinology, 1988, Volume: 48, Issue:2

    Topics: Animals; Cerebral Ventricles; Dimaprit; Dopamine; Histamine; Infusions, Intra-Arterial; Injections, Intraventricular; Male; Neurons; Prolactin; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2; Reference Values; Thiazoles; Thiourea

1988
Kinetics of antisecretory action of a new H2-antagonist, YM-11170, in conscious dogs.
    European journal of pharmacology, 1983, Aug-05, Volume: 91, Issue:4

    Topics: Animals; Atropine; Cimetidine; Dimaprit; Dogs; Famotidine; Gastric Acid; Gastric Mucosa; Histamine H2 Antagonists; Kinetics; Male; Methacholine Chloride; Methacholine Compounds; Pentagastrin; Thiazoles; Thiourea

1983
The effect of histamine, H1 and H2 agonists, and H1 and H2 antagonists on postprandial pancreatic polypeptide release in dogs.
    Scandinavian journal of gastroenterology, 1983, Volume: 18, Issue:2

    Topics: Animals; Cimetidine; Dimaprit; Dogs; Food; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Pancreatic Polypeptide; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Secretory Rate; Thiazoles; Thiourea

1983
Inhibition of phytohaemagglutinin-induced proliferation of human peripheral blood lymphocytes by histamine and histamine H1 and H2 agonists.
    Clinical and experimental immunology, 1983, Volume: 51, Issue:1

    Topics: Cell Division; Cells, Cultured; Dimaprit; Dose-Response Relationship, Drug; Histamine; Humans; Imidazoles; Impromidine; Lymphocytes; Methylhistamines; Phytohemagglutinins; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea

1983
A possible physiological role of histamine H2-receptors in rat mesenteric circulation.
    European journal of pharmacology, 1983, Jun-03, Volume: 90, Issue:2-3

    Topics: Animals; Cimetidine; Dimaprit; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H2; Splanchnic Circulation; Thiazoles; Thiourea; Vasodilation

1983
Effects of histamine receptor stimulation on regional myocardial blood flow.
    The American journal of physiology, 1983, Volume: 245, Issue:3

    Topics: Animals; Blood Pressure; Cimetidine; Coronary Circulation; Dimaprit; Diphenhydramine; Dogs; Female; Heart Rate; Histamine; Male; Microspheres; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea

1983
Pharmacological interactions between ranitidine, cimetidine, metiamide and tiotidine at histamine H2-receptor sites in guinea-pig atria.
    Agents and actions, 1982, Volume: 12, Issue:1-2

    Topics: Animals; Cimetidine; Dimaprit; Drug Interactions; Furans; Guanidines; Guinea Pigs; Heart; Heart Rate; Histamine; In Vitro Techniques; Metiamide; Ranitidine; Receptors, Histamine; Receptors, Histamine H2; Thiazoles; Thiourea

1982
Stimulatory effect of histamine on cyclic AMP formation in chick pineal gland.
    Journal of neurochemistry, 1994, Volume: 63, Issue:4

    Topics: 1-Methyl-3-isobutylxanthine; Adenine; Analysis of Variance; Animals; Carbon Radioisotopes; Chickens; Colforsin; Cyclic AMP; Dimaprit; Guinea Pigs; Hippocampus; Histamine; Histamine Agonists; In Vitro Techniques; Kinetics; Male; Methylhistamines; Pineal Gland; Ranitidine; Rats; Rats, Wistar; Thiazoles; Tritium

1994
Effects of a histamine H2 receptor agonist and antagonist on restraint-induced antinociception in female mice.
    European journal of pharmacology, 1995, Jun-12, Volume: 279, Issue:2-3

    Topics: Animals; Benzothiazoles; Cimetidine; Dimaprit; Female; Histamine Agonists; Histamine H2 Antagonists; Mice; Mice, Inbred Strains; Pain Measurement; Phenoxypropanolamines; Piperidines; Reaction Time; Restraint, Physical; Stress, Psychological; Thiazoles

1995
Characterization and function of histamine receptors in corpus cavernosum.
    The Journal of urology, 1995, Volume: 153, Issue:2

    Topics: Acetylcholine; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Electric Stimulation; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Papaverine; Penis; Piperidines; Pyrilamine; Rabbits; Receptors, Histamine; Thiazoles

1995
2-Thiazolylethylamine, a selective histamine H1 agonist, decreases seizure susceptibility in mice.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 47, Issue:3

    Topics: Animals; Anticonvulsants; Dimaprit; Dose-Response Relationship, Drug; Electroshock; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Injections, Intraventricular; Male; Mice; Mice, Inbred Strains; Pentylenetetrazole; Receptors, Histamine H1; Seizures; Thiazoles

1994
In vitro cardiac pharmacology of the new histamine H2-receptor agonist amthamine: comparisons with histamine and dimaprit.
    Agents and actions, 1993, Volume: 40, Issue:1-2

    Topics: Animals; Atrial Function; Dimaprit; Electric Stimulation; Guinea Pigs; Heart; Heart Atria; Histamine; Histamine Agonists; Humans; In Vitro Techniques; Myocardial Contraction; Papillary Muscles; Rabbits; Ranitidine; Thiazoles

1993
Identification of endothelial H1, vascular H2 and cardiac presynaptic H3 receptors in the pithed rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 1993, Volume: 347, Issue:1

    Topics: Animals; Blood Pressure; Blood Vessels; Cardiovascular System; Dimaprit; Electric Stimulation; Endothelium, Vascular; Heart Rate; Histamine Agonists; Male; Methylhistamines; Myocardium; Rats; Rats, Wistar; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Thiazoles

1993
The source and action of histamine in the isolated guinea-pig gallbladder.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1995, Volume: 44, Issue:10

    Topics: Animals; Dimaprit; Electric Stimulation; Female; Gallbladder; Guinea Pigs; Histamine; Histamine Agonists; Histamine H2 Antagonists; Immunohistochemistry; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Ranitidine; Receptors, Histamine H3; Thiazoles

1995
Histamine H3 receptor inhibition of K(+)-evoked release of acetylcholine from rat cortex in vivo.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1996, Volume: 45 Suppl 1

    Topics: Acetylcholine; Analysis of Variance; Animals; Chromatography, High Pressure Liquid; Dimaprit; Histamine; Histamine Agonists; Histamine Antagonists; Male; Methylhistamines; Microdialysis; Neurons; Parietal Lobe; Piperidines; Potassium; Rats; Rats, Wistar; Receptors, Histamine H3; Thiazoles

1996
Cardiovascular effects of the novel histamine H2 receptor agonist amthamine: interaction with the adrenergic system.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cardiovascular System; Dimaprit; Dose-Response Relationship, Drug; Heart Rate; Histamine Agonists; Histamine H2 Antagonists; Male; Prazosin; Rats; Rats, Wistar; Tachycardia; Thiazoles

1996
Histamine receptor-independent muscle relaxation elicited by a series of histamine H2-receptor agonists on the isolated guinea pig duodenum: a study into the mechanism of action.
    General pharmacology, 1998, Volume: 31, Issue:4

    Topics: Animals; Dimaprit; Duodenum; Electric Stimulation; Guinea Pigs; Histamine Agonists; Impromidine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Structure-Activity Relationship; Thiazoles

1998
Histamine H2-receptor modulation in two mouse models of seizure susceptibility.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1999, Volume: 48 Suppl 1

    Topics: Acoustic Stimulation; Animals; Anticonvulsants; Benzothiazoles; Convulsants; Dimaprit; Female; Histamine Agonists; Histamine Antagonists; Male; Mice; Mice, Inbred DBA; Pentylenetetrazole; Phenoxypropanolamines; Piperidines; Receptors, Histamine H2; Seizures; Thiazoles

1999
Effects of histamine and related compounds on regional cerebral blood flow in rats.
    Methods and findings in experimental and clinical pharmacology, 1999, Volume: 21, Issue:9

    Topics: Animals; Benzothiazoles; Blood Pressure; Brain Chemistry; Dimaprit; Diphenhydramine; Drug Interactions; Hippocampus; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Male; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Rats, Wistar; Regional Blood Flow; Thiazoles; Time Factors

1999
Understanding the Effects of NOAC Combined with Antiplatelet Therapy on Clot Kinetics.
    Thrombosis and haemostasis, 2020, Volume: 120, Issue:1

    Topics: Anticoagulants; Aspirin; Clopidogrel; Coronary Artery Disease; Dimaprit; Humans; Kinetics; Platelet Aggregation Inhibitors; Pyridines; Thiazoles

2020
Selective histamine H
    Journal of pharmacological sciences, 2022, Volume: 150, Issue:3

    Topics: Angiopoietin-1; Animals; Blood-Brain Barrier; Brain Injuries, Traumatic; Dimaprit; Endothelial Cells; Evans Blue; Hedgehog Proteins; Histamine; Histamine Agonists; Male; Mice; Protective Factors; Ranitidine; Receptors, Histamine H2; RNA, Messenger; Thiazoles

2022