Page last updated: 2024-08-21

thiazoles and daunorubicin

thiazoles has been researched along with daunorubicin in 36 studies

Research

Studies (36)

TimeframeStudies, this research(%)All Research%
pre-19902 (5.56)18.7374
1990's12 (33.33)18.2507
2000's18 (50.00)29.6817
2010's4 (11.11)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Rosazza, JP; Smith, RV1
Belov, L; Davey, MW; Davey, RA; Kidman, AD; Marks, DC1
Hählen, K; Huismans, DR; Loonen, AH; Pieters, R; van der Does-van den Berg, A; van Wering, ER; Veerman, AJ1
Broekema, GJ; Dirven, MW; Hählen, K; Heyenbrok, MW; Huismans, DR; Loonen, AH; Pieters, R; Veerman, AJ1
Bejaoui, N; Cinq-Mars, B; Lemieux, P; Pagé, M1
Efferth, T; Fabry, U; Glatte, P; Osieka, R1
Hählen, K; Kaspers, GJ; Pieters, R; Van Wering, ER; Van Zantwijk, I; Veerman, AJ1
Barrand, MA; Rhodes, T; Twentyman, PR1
Chen, LM; Huang, SH; Hwang, WS; Tseng, MT; Wang, CC1
Hählen, K; Huismans, DR; Kaspers, GJ; Loonen, AH; Pieters, R; van Wering, ER; Veerman, AJ1
Efferth, T; Fabry, U; Osieka, R1
Chiba, P; Ecker, G; Schaper, KJ1
Borg, AG; Burgess, R; Fisher, A; Grey, M; Wood, P; Yin, JA1
George, AR; Howlett, DR; Markwell, RE; Owen, DE; Ward, RV1
Iffert, T; Maser, E; Moeller, A; Soldan, M1
Chauvier, D; Kegelaer, G; Manfait, M; Morjani, H1
Balcerska, A; Balwierz, W; Chybicka, A; Debski, R; Kowalczyk, J; Kurylak, A; Matysiak, M; Rokicka-Milewska, R; Sońta-Jakimczyk, D; Styczyński, J; Wachowiak, J; Wysocki, M1
Barbier, M; Boumendjel, A; Boutonnat, J; Hadjeri, M; Mariotte, AM; Ronot, X1
Blazek, B; Hajduch, M; Janostakova, A; Kouzmina, G; Mihal, V; Noskova, V; Orel, M; Pospisilova, D; Safarova, M; Stary, J1
Schinköthe, T; Staib, P; Strunk, T; Tiehen, J1
Cooper, JM; Gu, M; Hartley, JA; Hochhauser, D; Lo, S; Schapira, AH; Taanman, JW; Tolner, B1
Asselin, B; Buck, S; Hamre, M; Ozdemir, O; Pullen, J; Ravindranath, Y; Savaşan, S1
Hu, X; Lu, Q; Qiangrong, P; Wang, T1
Jekerle, V; Klinkhammer, W; Piquette-Miller, M; Reilly, RM; Wiese, M1
Ainoon, O; Cheong, SK; Fazlina, N; Hamidah, H; Hamidah, NH; Jamal, R; Maha, A; Zarina, AL; Zulkifli, SZ1
Hungerer, C; Koch, L; Maser, E; Plebuch, M; Soldan, M1
Enokita, M; Hashimoto, T; Hori, Y; Iwatsubo, T; Kato, M; Kinoshita, H; Toyo'oka, T1
Chi, HS; Choi, SJ; Im, HJ; Jang, S; Jun, KR; Lee, JH; Lee, KH; Moon, HN; Park, CJ; Seo, JJ1
Beverloo, HB; Cornelissen, JJ; Deenik, W; Valk, PJ; van der Poel-van de Luytgaarde, SC; van Esser, JW; Wattel, MM1
Tallman, M1
Chen, B; Guo, D; Hu, H; Li, X; Wang, X; Wu, C1
Baumert, D; Jacobs, A; Möllmann, L; Sterz, K; Wiese, M1
Breydo, L; Dutta, S; Fekry, MI; Gates, KS; Szekely, J; Zang, H1
Bhatia, R; Dos Santos, C; Forman, SJ; Ho, YW; Kuo, YH; Lin, A; Liu, H; McDonald, T1
Hatta, Y1
McElligott, F; O'Marcaigh, A; O'Rafferty, C; Smith, O; Storey, L1

Reviews

2 review(s) available for thiazoles and daunorubicin

ArticleYear
Microbial models for drug metabolism.
    Advances in applied microbiology, 1979, Volume: 25

    Topics: Acronine; Animals; Aporphines; Bacteria; Biotransformation; Cannabinoids; Chemical Phenomena; Chemistry; Cytochrome P-450 Enzyme System; Danazol; Daunorubicin; Ellipticines; Fungi; Indans; Mammals; Models, Biological; Oxidation-Reduction; Oxygenases; Papaverine; Pharmaceutical Preparations; Prostaglandins; Species Specificity; Spironolactone; Thiazoles; Yeasts

1979
[Acute lymphoblastic leukemia].
    [Rinsho ketsueki] The Japanese journal of clinical hematology, 2014, Volume: 55, Issue:2

    Topics: Adolescent; Adult; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Cyclophosphamide; Dasatinib; Daunorubicin; Doxorubicin; Enzyme Inhibitors; Humans; Imatinib Mesylate; Methotrexate; Middle Aged; Philadelphia Chromosome; Piperazines; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prognosis; Protein-Tyrosine Kinases; Pyrimidines; Thiazoles; Young Adult

2014

Other Studies

34 other study(ies) available for thiazoles and daunorubicin

ArticleYear
The MTT cell viability assay for cytotoxicity testing in multidrug-resistant human leukemic cells.
    Leukemia research, 1992, Volume: 16, Issue:12

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Survival; Coloring Agents; Daunorubicin; Drug Resistance; Drug Screening Assays, Antitumor; Epirubicin; Humans; Membrane Glycoproteins; Tetrazolium Salts; Thiazoles; Trypan Blue; Verapamil; Vinblastine

1992
Relation of cellular drug resistance to long-term clinical outcome in childhood acute lymphoblastic leukaemia.
    Lancet (London, England), 1991, Aug-17, Volume: 338, Issue:8764

    Topics: Antineoplastic Agents; Asparaginase; Chi-Square Distribution; Child; Coloring Agents; Daunorubicin; Drug Resistance; Drug Screening Assays, Antitumor; Female; Humans; Male; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prednisolone; Prognosis; Remission Induction; Tetrazolium Salts; Thiazoles; Thioguanine; Tumor Cells, Cultured; Vincristine

1991
In vitro drug sensitivity of cells from children with leukemia using the MTT assay with improved culture conditions.
    Blood, 1990, Dec-01, Volume: 76, Issue:11

    Topics: Asparaginase; Cells, Cultured; Child; Coloring Agents; Culture Media; Cyclophosphamide; Cytarabine; Daunorubicin; Dose-Response Relationship, Drug; Drug Resistance; Drug Screening Assays, Antitumor; Humans; Mechlorethamine; Mercaptopurine; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prednisolone; Tetrazolium Salts; Thiazoles; Thioguanine; Vincristine

1990
Optimization of the tetrazolium-based colorimetric assay for the measurement of cell number and cytotoxicity.
    International journal of immunopharmacology, 1988, Volume: 10, Issue:7

    Topics: Animals; Cell Count; Cell Survival; Colorimetry; Daunorubicin; Humans; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1988
Expression of apoptosis-related oncoproteins and modulation of apoptosis by caffeine in human leukemic cells.
    Journal of cancer research and clinical oncology, 1995, Volume: 121, Issue:11

    Topics: Apoptosis; Caffeine; Carboplatin; Cluster Analysis; Coloring Agents; Daunorubicin; Drug Resistance, Neoplasm; Flow Cytometry; G2 Phase; Gamma Rays; Gene Expression Regulation, Leukemic; Glutathione; GTP-Binding Proteins; HL-60 Cells; Humans; Immunohistochemistry; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid; Leukemia, Myeloid, Acute; Leukemia, Promyelocytic, Acute; Lymphoma, Non-Hodgkin; Multivariate Analysis; Oncogene Proteins v-fos; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-bcl-2; Radiation Tolerance; ras Proteins; S Phase; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured; Tumor Suppressor Protein p53

1995
Drug combination testing in acute lymphoblastic leukemia using the MTT assay.
    Leukemia research, 1995, Volume: 19, Issue:3

    Topics: Antineoplastic Combined Chemotherapy Protocols; Cyclophosphamide; Daunorubicin; Drug Interactions; Drug Resistance; Humans; In Vitro Techniques; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prednisolone; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured; Vincristine

1995
Modification by brefeldin A, bafilomycin A1 and 7-chloro-4-nitrobenz-2-oxa-1,3-diazole (NBD) of cellular accumulation and intracellular distribution of anthracyclines in the non-P-glycoprotein-mediated multidrug-resistant cell line COR-L23/R.
    British journal of cancer, 1994, Volume: 70, Issue:1

    Topics: 4-Chloro-7-nitrobenzofurazan; Anti-Bacterial Agents; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Brefeldin A; Carcinoma, Non-Small-Cell Lung; Carrier Proteins; Cell Nucleus; Cyclopentanes; Cytoplasm; Daunorubicin; Doxorubicin; Drug Interactions; Drug Resistance; Drug Screening Assays, Antitumor; Golgi Apparatus; Humans; Lung Neoplasms; Macrolides; Membrane Glycoproteins; Protein Synthesis Inhibitors; Proton-Translocating ATPases; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1994
Prediction of chemotherapy response in human leukemia using in vitro chemosensitivity test.
    Leukemia research, 1993, Volume: 17, Issue:8

    Topics: Adult; Aged; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Bone Marrow; Coloring Agents; Cytarabine; Daunorubicin; Drug Screening Assays, Antitumor; Female; Humans; Leukemia, Myeloid, Acute; Male; Middle Aged; Mitoxantrone; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prednisolone; Prognosis; Tetrazolium Salts; Thiazoles

1993
Cellular drug resistance profiles that might explain the prognostic value of immunophenotype and age in childhood acute lymphoblastic leukemia.
    Leukemia, 1993, Volume: 7, Issue:3

    Topics: Aging; Antineoplastic Agents; Child; Child, Preschool; Daunorubicin; Drug Resistance; Drug Screening Assays, Antitumor; Humans; Immunophenotyping; Infant; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Predictive Value of Tests; Prognosis; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured; Vincristine

1993
Apoptosis and resistance to daunorubicin in human leukemic cells.
    Leukemia, 1997, Volume: 11, Issue:7

    Topics: Antibiotics, Antineoplastic; Apoptosis; Daunorubicin; Drug Resistance; Humans; Leukemia; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1997
Estimation of the chemosensitizing activity of modulators of multi-drug resistance via combined simultaneous analysis of sigmoidal dose-response curves.
    The Journal of pharmacy and pharmacology, 1997, Volume: 49, Issue:3

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Survival; Daunorubicin; Dose-Response Relationship, Drug; Drug Interactions; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Propafenone; Structure-Activity Relationship; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1997
Effect on cell kill of addition of multidrug resistance modifiers cyclosporin A and PSC 833 to cytotoxic agents in acute myeloid leukaemia.
    Leukemia research, 1997, Volume: 21, Issue:9

    Topics: Acute Disease; Adolescent; Adult; Aged; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cell Survival; Coloring Agents; Cyclosporine; Cyclosporins; Cytarabine; Daunorubicin; Drug Resistance, Neoplasm; Drug Synergism; Etoposide; Female; Humans; Idarubicin; Leukemia, Myeloid; Male; Middle Aged; Mitoxantrone; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1997
Common structural features determine the effectiveness of carvedilol, daunomycin and rolitetracycline as inhibitors of Alzheimer beta-amyloid fibril formation.
    The Biochemical journal, 1999, Oct-15, Volume: 343 Pt 2

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Carbazoles; Carvedilol; Cell Survival; Daunorubicin; Humans; Inhibitory Concentration 50; Microscopy, Electron; Models, Chemical; Molecular Structure; Neurons; Polymers; Propanolamines; Protein Binding; Rolitetracycline; Structure-Activity Relationship; Tetrazolium Salts; Thermodynamics; Thiazoles; Tumor Cells, Cultured

1999
Modulation of daunorubicin toxicity by liposomal encapsulation and use of specific inhibitors in vitro.
    Toxicology, 2000, Apr-03, Volume: 144, Issue:1-3

    Topics: Antibiotics, Antineoplastic; Breast Neoplasms; Daunorubicin; Drug Carriers; Drug Compounding; Drug Resistance, Neoplasm; Humans; Liposomes; Rutin; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

2000
Reversal of multidrug resistance-associated protein-mediated daunorubicin resistance by camptothecin.
    Journal of pharmaceutical sciences, 2002, Volume: 91, Issue:8

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents, Phytogenic; Breast Neoplasms; Camptothecin; Cell Line; Cell Nucleus; Chemokines, CC; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Fluorescent Antibody Technique; Gene Expression Regulation, Neoplastic; Humans; Leukemia; Microscopy, Confocal; Reverse Transcriptase Polymerase Chain Reaction; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

2002
The influence of intracellular idarubicin and daunorubicin levels on drug cytotoxicity in childhood acute leukemia.
    Acta biochimica Polonica, 2002, Volume: 49, Issue:1

    Topics: Adolescent; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Child; Child, Preschool; Daunorubicin; Flow Cytometry; Humans; Idarubicin; Infant; Leukemia, Myeloid, Acute; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Tetrazolium Salts; Thiazoles

2002
Modulation of P-glycoprotein-mediated multidrug resistance by flavonoid derivatives and analogues.
    Journal of medicinal chemistry, 2003, May-22, Volume: 46, Issue:11

    Topics: Antineoplastic Agents; Apoptosis; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Division; Chromones; Daunorubicin; Drug Resistance, Multiple; Drug Synergism; Flavonoids; Fluorescent Dyes; Humans; Necrosis; Piperazines; Quinolinium Compounds; Rhodamine 123; Thiazoles; Tumor Cells, Cultured

2003
The analysis of correlations between drug resistance and clinical/laboratory measures found in a group of children with all treated by ALL-BFM 90 protocol.
    Bulletin du cancer, 2004, Volume: 91, Issue:4

    Topics: Adolescent; Age Factors; Antineoplastic Combined Chemotherapy Protocols; Asparaginase; Child; Child, Preschool; Coloring Agents; Cyclophosphamide; Cytarabine; Daunorubicin; Drug Resistance, Neoplasm; Female; Humans; In Vitro Techniques; Male; Mercaptopurine; Methotrexate; Multivariate Analysis; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Predictive Value of Tests; Prednisone; Remission Induction; Sex Factors; Tetrazolium Salts; Thiazoles; Vincristine

2004
Determination of caspase-3 activation fails to predict chemosensitivity in primary acute myeloid leukemia blasts.
    BMC cancer, 2005, Jun-11, Volume: 5

    Topics: Adult; Aged; Antineoplastic Agents; Apoptosis; Bone Marrow Cells; Caspase 3; Caspases; Cell Death; Cell Line, Tumor; Cytarabine; Daunorubicin; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Enzyme Activation; Female; Humans; Kinetics; Leukemia, Myeloid, Acute; Male; Middle Aged; Spectrometry, Fluorescence; Tetrazolium Salts; Thiazoles

2005
Assessment of the significance of mitochondrial DNA damage by chemotherapeutic agents.
    International journal of oncology, 2005, Volume: 27, Issue:2

    Topics: Antigens, Neoplasm; Antineoplastic Agents; Apoptosis; ATP Binding Cassette Transporter, Subfamily B; Blotting, Southern; Cell Cycle; Cell Line, Tumor; Cell Proliferation; Cytochromes c; Daunorubicin; DNA Damage; DNA Topoisomerases, Type II; DNA-Binding Proteins; DNA, Mitochondrial; Dose-Response Relationship, Drug; Flow Cytometry; Humans; Immunoblotting; Inhibitory Concentration 50; Intracellular Membranes; Membrane Potentials; Pyridines; Thiazoles; Tumor Suppressor Protein p53

2005
Evaluation of cytotoxicity by flow cytometric drug sensitivity assay in childhood T-cell acute lymphoblastic leukemia.
    Leukemia & lymphoma, 2005, Volume: 46, Issue:6

    Topics: Apoptosis; Bone Marrow Cells; Child; Daunorubicin; Drug Screening Assays, Antitumor; Flow Cytometry; Humans; Immunophenotyping; Inhibitory Concentration 50; Leukemia, T-Cell; Medical Oncology; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Reproducibility of Results; Sensitivity and Specificity; Tetrazolium Salts; Thiazoles

2005
Schisandrin B--a novel inhibitor of P-glycoprotein.
    Biochemical and biophysical research communications, 2005, Sep-23, Volume: 335, Issue:2

    Topics: Affinity Labels; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cell Line, Tumor; Cell Proliferation; Cyclooctanes; Daunorubicin; Dihydropyridines; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Humans; Inhibitory Concentration 50; K562 Cells; Lignans; Models, Chemical; Neoplasms; Polycyclic Compounds; Protein Binding; Tetrazolium Salts; Thiazoles; Time Factors

2005
Novel tetrahydroisoquinolin-ethyl-phenylamine based multidrug resistance inhibitors with broad-spectrum modulating properties.
    Cancer chemotherapy and pharmacology, 2007, Volume: 59, Issue:1

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Benzamides; Cell Line, Tumor; Cell Survival; Daunorubicin; Drug Design; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Humans; Isoquinolines; Mitoxantrone; Neoplasm Proteins; ortho-Aminobenzoates; Phthalic Acids; Quinolines; Reverse Transcriptase Polymerase Chain Reaction; Tetrazolium Salts; Thiazoles

2007
Expression of multidrug resistance (MDR) proteins and in vitro drug resistance in acute leukemias.
    Hematology (Amsterdam, Netherlands), 2007, Volume: 12, Issue:1

    Topics: Acute Disease; Adolescent; Adult; Age Factors; Aged; Aged, 80 and over; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; Cell Survival; Child; Child, Preschool; Coloring Agents; Cytarabine; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Humans; Infant; Inhibitory Concentration 50; Leukemia; Leukemia, Myeloid; Male; Methylphenazonium Methosulfate; Middle Aged; Neoplasm Proteins; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Recurrence; Staining and Labeling; Tetrazolium Salts; Thiazoles; Treatment Outcome; Tumor Cells, Cultured

2007
Increased resistance of tumor cells to daunorubicin after transfection of cDNAs coding for anthracycline inactivating enzymes.
    Cancer letters, 2007, Sep-18, Volume: 255, Issue:1

    Topics: Alcohol Oxidoreductases; Aldehyde Reductase; Aldo-Keto Reductases; Antibiotics, Antineoplastic; Cell Line, Tumor; Cloning, Molecular; Daunorubicin; DNA, Complementary; Drug Resistance; Humans; Inhibitory Concentration 50; Pancreatic Neoplasms; Tetrazolium Salts; Thiazoles; Transfection

2007
Analytical method for beta-amyloid fibrils using CE-laser induced fluorescence and its application to screening for inhibitors of beta-amyloid protein aggregation.
    Analytical chemistry, 2007, Jul-01, Volume: 79, Issue:13

    Topics: Alzheimer Disease; Amino Acid Sequence; Amyloid beta-Peptides; Benzothiazoles; Daunorubicin; Fluorescence; Fluorescent Dyes; Humans; Indoles; Lasers; Mass Screening; Melatonin; Molecular Sequence Data; Propionates; Sensitivity and Specificity; Thiazoles; Time Factors

2007
Relationship between in vitro chemosensitivity assessed with MTT assay and clinical outcomes in 103 patients with acute leukemia.
    The Korean journal of laboratory medicine, 2007, Volume: 27, Issue:2

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Antibiotics, Antineoplastic; Child; Child, Preschool; Coloring Agents; Cytarabine; Daunorubicin; Drug Evaluation, Preclinical; Drug Resistance, Neoplasm; Female; Humans; Infant; Leukemia, Biphenotypic, Acute; Leukemia, Myeloid, Acute; Male; Middle Aged; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Tetrazolium Salts; Thiazoles; Treatment Outcome

2007
Rapid complete cytogenetic remission after upfront dasatinib monotherapy in a patient with a NUP214-ABL1-positive T-cell acute lymphoblastic leukemia.
    Leukemia, 2009, Volume: 23, Issue:3

    Topics: Antineoplastic Combined Chemotherapy Protocols; Asparaginase; Combined Modality Therapy; Cytarabine; Dasatinib; Daunorubicin; Granulocyte Colony-Stimulating Factor; Humans; In Situ Hybridization, Fluorescence; Male; Methotrexate; Mitoxantrone; Neoplasm Proteins; Neutropenia; Oncogene Proteins, Fusion; Peripheral Blood Stem Cell Transplantation; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; Prednisone; Pyrimidines; Remission Induction; Splenic Rupture; Thiazoles; Vincristine; Young Adult

2009
Existing and emerging therapeutic options for the treatment of acute myeloid leukemia.
    Clinical advances in hematology & oncology : H&O, 2008, Volume: 6, Issue:11

    Topics: Adenine; Adenine Nucleotides; Aminoglycosides; Anti-Inflammatory Agents, Non-Steroidal; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Arabinonucleosides; Carbazoles; Clofarabine; Cytarabine; Dasatinib; Daunorubicin; fms-Like Tyrosine Kinase 3; Furans; Gemtuzumab; Humans; Leukemia, Myeloid, Acute; Naphthalimides; Organophosphonates; Prognosis; Protein Kinase Inhibitors; Pyrimidines; Sesquiterpenes; Staurosporine; Stem Cell Transplantation; Thiazoles; Tretinoin

2008
Study on the enhanced cellular uptake effect of daunorubicin on leukemia cells mediated via functionalized nickel nanoparticles.
    Biomedical materials (Bristol, England), 2009, Volume: 4, Issue:2

    Topics: Antineoplastic Agents; Biocompatible Materials; Cell Line, Tumor; Daunorubicin; Electrochemistry; Humans; K562 Cells; Leukemia; Metal Nanoparticles; Microscopy, Atomic Force; Microscopy, Fluorescence; Nanotechnology; Nickel; Permeability; Tetrazolium Salts; Thiazoles

2009
Activators of P-glycoprotein: Structure-activity relationships and investigation of their mode of action.
    ChemMedChem, 2009, Volume: 4, Issue:11

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Benzothiazoles; Cell Line, Tumor; Daunorubicin; Drug Resistance, Neoplasm; Humans; Imidazoles; Rhodamine 123; Structure-Activity Relationship; Thiazoles

2009
Noncovalent DNA binding drives DNA alkylation by leinamycin: evidence that the Z,E-5-(thiazol-4-yl)-penta-2,4-dienone moiety of the natural product serves as an atypical DNA intercalator.
    Journal of the American Chemical Society, 2011, Nov-09, Volume: 133, Issue:44

    Topics: Alkylation; Binding Sites; Biological Products; Daunorubicin; DNA; Lactams; Macrolides; Models, Molecular; Molecular Conformation; Structure-Activity Relationship; Thiazoles; Thiones

2011
The Src and c-Kit kinase inhibitor dasatinib enhances p53-mediated targeting of human acute myeloid leukemia stem cells by chemotherapeutic agents.
    Blood, 2013, Sep-12, Volume: 122, Issue:11

    Topics: Adult; Aged; Aged, 80 and over; Animals; Antineoplastic Combined Chemotherapy Protocols; Dasatinib; Daunorubicin; Female; Humans; Leukemia, Myeloid, Acute; Male; Mice; Mice, Inbred C57BL; Mice, SCID; Middle Aged; Neoplastic Stem Cells; Phosphorylation; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-kit; Pyrimidines; RNA Interference; src-Family Kinases; Thiazoles; Tumor Cells, Cultured; Tumor Suppressor Protein p53; Xenograft Model Antitumor Assays; Young Adult

2013
Pneumatosis intestinalis and imatinib mesylate.
    Annals of hematology, 2014, Volume: 93, Issue:10

    Topics: Antineoplastic Combined Chemotherapy Protocols; Asparaginase; Benzamides; Child, Preschool; Dasatinib; Daunorubicin; Dexamethasone; Drug Substitution; Female; Humans; Imatinib Mesylate; Parenteral Nutrition, Total; Piperazines; Pneumatosis Cystoides Intestinalis; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Protein Kinase Inhibitors; Pyrimidines; Recurrence; Thiazoles; Vincristine

2014