Page last updated: 2024-08-21

thiazoles and cyclosporine

thiazoles has been researched along with cyclosporine in 47 studies

Research

Studies (47)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's14 (29.79)18.2507
2000's19 (40.43)29.6817
2010's13 (27.66)24.3611
2020's1 (2.13)2.80

Authors

AuthorsStudies
Claude, JR; Martin, C; Massicot, F; Pham Huy, C; Thevenin, M; Warnet, JM1
Cooper, MH; Gregory, SH; Starzl, TE; Wing, EJ1
Acosta, D; Jiang, T1
Cai, W; Foulkes, JG; Hu, L1
Chardonnet, Y; Lizard, G; Marionnet, AV; Schmitt, D1
Claude, JR; Duc, HT; Dutertre-Catella, H; Ellouk-Achard, S; Martin, C; Pham-Huy, C; Thevenin, M; Warnet, JM1
Claude, JR; Dutertre-Catella, H; Ellouk-Achard, S; Martin, C; Massicot, F; Pham-Huy, C; Rucay, P; Thevenin, M; Warnet, JM1
Borg, AG; Burgess, R; Fisher, A; Grey, M; Wood, P; Yin, JA1
Bonomini, L; DeFranco, P; Friedman, G; Jacobs, M; Kaplan, B; Lyman, N; Mulgaonkar, SP; Viscuso, R1
Brennan, DC; Burgess, SJ; Singer, GG1
Al Rayyes, O; Florén, CH1
Frantz, RP; Nguyen, TT1
Haug, MT; Park, MH; Pelegrin, D; Young, JB1
Downs, AM; Sansom, JE1
Kongkittingam, C; Vedejs, E1
Bal-Price, A; Brown, GC1
Calvo, M; Colell, A; Enrich, C; Fernández-Checa, JC; García-Ruiz, C; Morales, A1
Huang, ST; Lee, PN; Pang, JH; Yang, LJ; Yang, RC1
Davies, T; Kostrubsky, VE; Lodola, A; Rahbari, R1
Choy, YM; Fung, KP; Ko, S; Kong, SK; Kwok, TT; Lee, CY; Yuen, WF1
Evtodienko, YV; Kruglov, AG; Yaguzhinsky, LS; Yurkov, IS1
Cohen, RD; Ross, AS1
Liot, G; Lobner, D1
Gabryel, B; Małecki, A; Toborek, T1
Arakawa, K; Hirano, T; Saito, K; Saito, N; Satoh, H; Sugiyama, K; Takahashi, K1
Scheinfeld, N1
Jankowska, AM; Maciejewski, JP; Schade, AE; Schieven, GL; Susulic, V; Szpurka, H; Townsend, R; Zhang, R1
Cho, JY1
Abumrad, NA; Gaudel, C; Giordano, C; Grimaldi, PA; Schwartz, C1
de Boschero, MG; Giusto, NM; Zulian, SE1
Giordano, C; Gounon, P; Grimaldi, P; Hatem, SN; Jehl-Piétri, C; Lopez, P; Murdaca, J; Schwartz, C; Wagner, KD; Wagner, N1
Gaudel, C; Giordano, C; Grimaldi, PA; Jehl-Piétri, C; Lopez, P; Murdaca, J; Rousseau, AS; Sibille, B; Wagner, N1
Dannaoui, E; Lortholary, O; Schwarz, P1
Charkoftaki, G; Kytariolos, J; Macheras, P1
Chen, XX; Mao, YD; Sha, JH; Wang, H; Wang, LR; Zhou, ZM1
Benfica, PL; de Lima, AP; dos Santos, WB; Lacerda, Ede P; Mello, FM; Pavanin, LA; Pereira, Fde C; Ribeiro, Ade S; Valadares, MC; Vilanova-Costa, CA1
Alvarez-Calderon, F; Degregori, J; Druker, BJ; Eide, CA; Gregory, MA; Neviani, P; O'Hare, T; Perrotti, D; Phang, TL; Williams, RT; Zaberezhnyy, V1
Hirano, T; Isogai, K; Nakagawa, Y; Saito, K; Satoh, H; Sugiyama, K; Takahashi, K; Tasaki, M; Toyama, A1
Hokari, A1
Blake, SJ; Hughes, TP; Lyons, AB1
Carnovale, CE; Francés, DE; Marchissio, MJ; Marinelli, RA1
Bastide, C; Bruyere, F; Caremel, R; Castel-Lacanal, E; Cornu, JN; Guy, L; Karsenty, G; Kerdraon, J1
Baturin, D; Christians, U; DeGregori, J; Gardner, LA; Gore, L; Gregory, MA; Klawitter, J; Pollyea, DA; Porter, CC; Takebe, N; Zaberezhnyy, V1
Matsushima, N; Mendell, J; Parasrampuria, DA; Shi, M; Truitt, K; Zahir, H1
Huang, F; Rowland, L; Sabo, JP; Schultz, A; Trampisch, M; Voelk, C1
Blanco, MJ1
Fan, HH; Jing, LP; Li, JP; Li, Y; Peng, GX; Xiong, YZ; Yang, WR; Yang, Y; Ye, L; Zhang, FK; Zhang, L; Zhao, X; Zhou, K1

Reviews

5 review(s) available for thiazoles and cyclosporine

ArticleYear
Transcription-modulating drugs: mechanism and selectivity.
    Current opinion in biotechnology, 1996, Volume: 7, Issue:6

    Topics: Animals; Anti-Inflammatory Agents; Aspirin; Cyclosporine; Drug Design; Estrogen Antagonists; Humans; Hypoglycemic Agents; Immunosuppressive Agents; Polyenes; Sirolimus; Tacrolimus; Thiazoles; Transcription, Genetic

1996
Medical therapy for ulcerative colitis: the state of the art and beyond.
    Current gastroenterology reports, 2004, Volume: 6, Issue:6

    Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antimetabolites, Antineoplastic; Butyrates; Colitis, Ulcerative; Cyclosporine; Epidermal Growth Factor; Glucocorticoids; Humans; Immunosuppressive Agents; Infliximab; Interferons; Mercaptopurine; Plasmapheresis; Probiotics; Remission Induction; Thiazoles

2004
A review of deferasirox, bortezomib, dasatinib, and cyclosporine eye drops: possible uses and known side effects in cutaneous medicine.
    Journal of drugs in dermatology : JDD, 2007, Volume: 6, Issue:3

    Topics: Animals; Antineoplastic Agents; Benzoates; Boronic Acids; Bortezomib; Cyclosporine; Dasatinib; Deferasirox; Humans; Iron Chelating Agents; Ophthalmic Solutions; Protein Kinase Inhibitors; Pyrazines; Pyrimidines; Randomized Controlled Trials as Topic; Skin Diseases; Skin Neoplasms; Thiazoles; Triazoles

2007
[Improved virologic response in chronic hepatitis C treated with peginterferon, ribavirin and add-on drug].
    Nihon rinsho. Japanese journal of clinical medicine, 2011, Volume: 69 Suppl 4

    Topics: Antiviral Agents; Cyclosporine; Diterpenes; Drug Therapy, Combination; Fatty Acids, Monounsaturated; Fatty Alcohols; Female; Fluvastatin; Hepatitis C, Chronic; Humans; Indoles; Interferon-alpha; Male; Metformin; Nitro Compounds; Polyethylene Glycols; Recombinant Proteins; Ribavirin; Silybin; Silymarin; Thiazoles

2011
[Drug therapy of bladder dysfunction].
    Progres en urologie : journal de l'Association francaise d'urologie et de la Societe francaise d'urologie, 2013, Volume: 23, Issue:15

    Topics: Acetanilides; Anti-Inflammatory Agents; Botulinum Toxins, Type A; Cholinergic Antagonists; Cimetidine; Cyclosporine; Dimethyl Sulfoxide; Histamine H2 Antagonists; Humans; Immunosuppressive Agents; Muscarinic Antagonists; Neuromuscular Agents; Phosphodiesterase Inhibitors; Thiazoles; Urinary Bladder; Urinary Bladder Diseases; Urination; Urodynamics

2013

Trials

3 trial(s) available for thiazoles and cyclosporine

ArticleYear
Inhibition of calcineurin combined with dasatinib has direct and indirect anti-leukemia effects against BCR-ABL1(+) leukemia.
    American journal of hematology, 2014, Volume: 89, Issue:9

    Topics: Adult; Animals; Antineoplastic Combined Chemotherapy Protocols; Calcineurin Inhibitors; Cell Line, Tumor; Cyclosporine; Dasatinib; Drug Synergism; Female; Flow Cytometry; Fusion Proteins, bcr-abl; Humans; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Male; Mice; Mice, Inbred C57BL; Middle Aged; Protein Kinase Inhibitors; Pyrimidines; Thiazoles; Treatment Outcome

2014
Edoxaban drug-drug interactions with ketoconazole, erythromycin, and cyclosporine.
    British journal of clinical pharmacology, 2016, Volume: 82, Issue:6

    Topics: Administration, Oral; Adolescent; Adult; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cross-Over Studies; Cyclosporine; Cytochrome P-450 CYP3A; Drug Administration Schedule; Drug Interactions; Erythromycin; Factor Xa Inhibitors; Healthy Volunteers; Humans; Ketoconazole; Metabolic Clearance Rate; Middle Aged; Pyridines; Substrate Specificity; Thiazoles; Young Adult

2016
Pharmacokinetic Interaction between Faldaprevir and Cyclosporine or Tacrolimus in Healthy Volunteers: A Prospective, Open-Label, Fixed-Sequence, Crossover Study.
    Basic & clinical pharmacology & toxicology, 2018, Volume: 123, Issue:1

    Topics: Adolescent; Adult; Aminoisobutyric Acids; Antiviral Agents; Area Under Curve; Cross-Over Studies; Cyclosporine; Drug Interactions; Female; Graft Rejection; Healthy Volunteers; Hepatitis C; Humans; Immunosuppressive Agents; Leucine; Liver Transplantation; Male; Middle Aged; Oligopeptides; Proline; Prospective Studies; Quinolines; Secondary Prevention; Tacrolimus; Thiazoles; Young Adult

2018

Other Studies

39 other study(ies) available for thiazoles and cyclosporine

ArticleYear
Inhibitory effects of a platelet activating factor-antagonist 48740RP in cyclosporin-induced nephrotoxicity in the rat as assessed by renal glutathione metabolism parameters.
    Archives of toxicology. Supplement. = Archiv fur Toxikologie. Supplement, 1991, Volume: 14

    Topics: Aminopeptidases; Animals; Blood Urea Nitrogen; CD13 Antigens; Creatinine; Cyclosporine; Glutathione; Kidney; Kidney Cortex; Platelet Activating Factor; Pyridines; Rats; Thiazoles

1991
Rapamycin but not FK506 inhibits the proliferation of mononuclear phagocytes induced by colony-stimulating factors.
    Transplantation, 1994, Volume: 57, Issue:3

    Topics: Animals; Bone Marrow Cells; Cell Count; Cell Division; Colony-Stimulating Factors; Concanavalin A; Culture Media, Conditioned; Cyclosporine; Female; Lymphocyte Activation; Mice; Mice, Inbred C57BL; Phagocytes; Polyenes; Sirolimus; Spleen; T-Lymphocytes; Tacrolimus; Tetrazolium Salts; Thiazoles; Thymidine; Tritium

1994
An in vitro model of cyclosporine-induced nephrotoxicity.
    Fundamental and applied toxicology : official journal of the Society of Toxicology, 1993, Volume: 20, Issue:4

    Topics: Alkaline Phosphatase; Animals; Cell Survival; Cells, Cultured; Cyclosporine; Fluoresceins; Fluorescent Dyes; Kidney Cortex; Kidney Diseases; L-Lactate Dehydrogenase; Mitochondria; Neutral Red; Pharmaceutical Vehicles; Polyethylene Glycols; Propidium; Rats; Rats, Sprague-Dawley; Tetrazolium Salts; Thiazoles

1993
Comparative evaluation of the antiproliferative effect of cyclosporin A and gamma-interferon on normal and HPV-transformed keratinocytes by cell counting, MTT assay and tritiated thymidine incorporation.
    Cell biology and toxicology, 1997, Volume: 13, Issue:2

    Topics: Adult; Cell Count; Cell Division; Cell Line, Transformed; Cell Survival; Cells, Cultured; Coloring Agents; Cyclosporine; Growth Inhibitors; Humans; Interferon-gamma; Keratinocytes; Papillomaviridae; Reproducibility of Results; Tetrazolium Salts; Thiazoles; Thymidine; Tritium

1997
Implication of CYP 3A in the toxicity of cyclosporin G (CsG), cyclosporin A (CsA) and FK506 on rat hepatocytes in primary culture.
    Archives of toxicology, 1997, Volume: 71, Issue:7

    Topics: Animals; Aryl Hydrocarbon Hydroxylases; Calcium; Cell Survival; Cells, Cultured; Coloring Agents; Cyclosporine; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Flow Cytometry; Immunosuppressive Agents; Intracellular Fluid; Liver; Male; Oxidoreductases, N-Demethylating; Rats; Rats, Wistar; Tacrolimus; Tetrazolium Salts; Thiazoles

1997
Modulation of energy status and cytotoxicity induced by FK506 and cyclosporin A in a renal epithelial cell line.
    Archives of toxicology, 1997, Volume: 71, Issue:8

    Topics: Adenosine Triphosphate; Animals; Cell Survival; Cyclosporine; Energy Metabolism; Immunosuppressive Agents; Kidney; LLC-PK1 Cells; Nucleotides; Swine; Tacrolimus; Tetrazolium Salts; Thiazoles; Time Factors

1997
Effect on cell kill of addition of multidrug resistance modifiers cyclosporin A and PSC 833 to cytotoxic agents in acute myeloid leukaemia.
    Leukemia research, 1997, Volume: 21, Issue:9

    Topics: Acute Disease; Adolescent; Adult; Aged; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cell Survival; Coloring Agents; Cyclosporine; Cyclosporins; Cytarabine; Daunorubicin; Drug Resistance, Neoplasm; Drug Synergism; Etoposide; Female; Humans; Idarubicin; Leukemia, Myeloid; Male; Middle Aged; Mitoxantrone; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1997
Potential interaction of troglitazone and cyclosporine.
    Transplantation, 1998, May-27, Volume: 65, Issue:10

    Topics: Acute Disease; Chromans; Cyclosporine; Drug Interactions; Female; Graft Rejection; Humans; Hypoglycemic Agents; Immunosuppressive Agents; Middle Aged; Osmolar Concentration; Thiazoles; Thiazolidinediones; Troglitazone

1998
Effect of troglitazone on cyclosporine whole blood levels.
    Transplantation, 1998, Jul-27, Volume: 66, Issue:2

    Topics: Chromans; Cyclosporine; Drug Interactions; Humans; Hypoglycemic Agents; Immunosuppressive Agents; Kidney Transplantation; Thiazoles; Thiazolidinediones; Troglitazone

1998
Troglitazone upregulates LDL receptor activity in HepG2 cells.
    Diabetes, 1998, Volume: 47, Issue:8

    Topics: Chromans; Cyclosporine; Humans; Hypoglycemic Agents; Insulin; Lipoproteins, LDL; Liver; Receptors, LDL; RNA, Messenger; Thiazoles; Thiazolidinediones; Troglitazone; Tumor Cells, Cultured; Up-Regulation

1998
Rezulin (troglitazone) greatly increases cyclosporine metabolism.
    The Journal of heart and lung transplantation : the official publication of the International Society for Heart Transplantation, 1998, Volume: 17, Issue:10

    Topics: Chromans; Cyclosporine; Drug Interactions; Drug Therapy, Combination; Female; Heart Transplantation; Humans; Hypoglycemic Agents; Immunosuppressive Agents; Metabolic Clearance Rate; Middle Aged; Thiazoles; Thiazolidinediones; Troglitazone

1998
Troglitazone, a new antidiabetic agent, decreases cyclosporine level.
    The Journal of heart and lung transplantation : the official publication of the International Society for Heart Transplantation, 1998, Volume: 17, Issue:11

    Topics: Aged; Chromans; Cyclosporine; Diabetes Mellitus, Type 1; Drug Interactions; Heart Transplantation; Humans; Hypoglycemic Agents; Immunosuppressive Agents; Male; Middle Aged; Thiazoles; Thiazolidinediones; Troglitazone

1998
Severe contact allergy to footwear responding to handmade shoes.
    Contact dermatitis, 1999, Volume: 40, Issue:4

    Topics: Cyclosporine; Dermatitis, Allergic Contact; Foot Dermatoses; Humans; Immunosuppressive Agents; Male; Middle Aged; Patch Tests; Potassium Dichromate; Shoes; Thiazoles; Thiram

1999
Solution-phase synthesis of a hindered N-methylated tetrapeptide using Bts-protected amino acid chlorides: efficient coupling and methylation steps allow purification by extraction.
    The Journal of organic chemistry, 2000, Apr-21, Volume: 65, Issue:8

    Topics: Acylation; Amino Acids; Benzothiazoles; Chlorides; Cyclosporine; Methylation; Oligopeptides; Sulfones; Thiazoles

2000
Nitric-oxide-induced necrosis and apoptosis in PC12 cells mediated by mitochondria.
    Journal of neurochemistry, 2000, Volume: 75, Issue:4

    Topics: Adenosine Triphosphate; Animals; Apoptosis; Azides; Caspase Inhibitors; Caspases; Cell Respiration; Cyclosporine; Cytochrome c Group; Cytosol; Enzyme Inhibitors; Glucose; Lactic Acid; Membrane Potentials; Methacrylates; Mitochondria; Necrosis; Nitric Oxide; Nitric Oxide Donors; Oxygen Consumption; PC12 Cells; Rats; Thiazoles

2000
Trafficking of ganglioside GD3 to mitochondria by tumor necrosis factor-alpha.
    The Journal of biological chemistry, 2002, Sep-27, Volume: 277, Issue:39

    Topics: Actins; Animals; Apoptosis; Biological Transport; Bridged Bicyclo Compounds, Heterocyclic; Cell Death; Cell Membrane; Cholesterol; Cyclosporine; Cytoskeleton; Endosomes; Enzyme Inhibitors; Filipin; Gangliosides; Golgi Apparatus; Hepatocytes; Humans; Kinetics; Microscopy, Confocal; Microscopy, Immunoelectron; Mitochondria; Protein Binding; rab GTP-Binding Proteins; rab5 GTP-Binding Proteins; rab7 GTP-Binding Proteins; Rats; Signal Transduction; Thiazoles; Thiazolidines; Time Factors; Tumor Necrosis Factor-alpha

2002
Phyllanthus urinaria triggers the apoptosis and Bcl-2 down-regulation in Lewis lung carcinoma cells.
    Life sciences, 2003, Feb-28, Volume: 72, Issue:15

    Topics: Animals; Antineoplastic Agents, Phytogenic; Apoptosis; Carcinoma, Lewis Lung; Caspase 3; Caspases; Cell Survival; Cyclosporine; DNA Fragmentation; Down-Regulation; Flow Cytometry; Genes, bcl-2; Mice; Phyllanthus; Plant Extracts; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

2003
Agree that idiosyncratic hepatotoxicity in TRO-treated patients is uncertain, but concerned about the data.
    Toxicological sciences : an official journal of the Society of Toxicology, 2003, Volume: 71, Issue:2

    Topics: Apoptosis; Cell Survival; Chromans; Cyclosporine; Dose-Response Relationship, Drug; Drug Antagonism; Hepatocytes; Humans; Hypoglycemic Agents; Mitochondria, Liver; Thiazoles; Thiazolidinediones; Troglitazone; Tumor Cells, Cultured

2003
Hyperthermia and tumour necrosis factor-alpha induced apoptosis via mitochondrial damage.
    Life sciences, 2000, Jun-30, Volume: 67, Issue:6

    Topics: Animals; Apoptosis; Blotting, Western; Cell Line; Cyclosporine; Cytochrome c Group; Cytosol; Fever; Fluorescein-5-isothiocyanate; Fluorescent Dyes; Immunosuppressive Agents; Membranes; Mice; Mitochondria; Tetrazolium Salts; Thiazoles; Tumor Necrosis Factor-alpha

2000
Mechanism of superoxide anion generation in intact mitochondria in the presence of lucigenin and cyanide.
    Biochemistry. Biokhimiia, 2003, Volume: 68, Issue:12

    Topics: Acridines; Adenosine Triphosphate; Animals; Antimycin A; Carbonyl Cyanide p-Trifluoromethoxyphenylhydrazone; Cell Respiration; Cyanides; Cyclosporine; Kinetics; Luminescent Measurements; Methacrylates; Mitochondria, Liver; Oligomycins; Oxygen; Oxygen Consumption; Proton-Motive Force; Rats; Rats, Wistar; Spectrometry, Fluorescence; Succinic Acid; Superoxides; Thiazoles; Uncoupling Agents

2003
Role of MAPK/ERK in neurotrophin-4 potentiation of necrotic neuronal death.
    Neurochemical research, 2004, Volume: 29, Issue:12

    Topics: Animals; Butadienes; Cell Death; Cells, Cultured; Cyclosporine; Enzyme Activation; Flavonoids; Immunosuppressive Agents; L-Lactate Dehydrogenase; Mice; Mitogen-Activated Protein Kinases; Necrosis; Nerve Growth Factors; Neurons; Nitriles; Phosphorylation; Tetrazolium Salts; Thiazoles

2004
Immunosuppressive immunophilin ligands attenuate damage in cultured rat astrocytes depleted of glutathione and exposed to simulated ischemia in vitro. Comparison with N-acetylcysteine.
    Neurotoxicology, 2005, Volume: 26, Issue:3

    Topics: Acetylcysteine; Animals; Apoptosis; Astrocytes; Benzimidazoles; Brain Ischemia; Cell Separation; Cells, Cultured; Cyclosporine; Fluorescent Dyes; Free Radical Scavengers; Glutathione; Immunophilins; Immunosuppressive Agents; Ligands; Mitochondria; Oxidative Stress; Rats; Rats, Wistar; Reactive Oxygen Species; Tacrolimus; Tetrazolium Salts; Thiazoles

2005
Correlation between pharmacological efficacy of cyclosporine A and tacrolimus, evaluated by lymphocyte immunosuppressant-sensitivity test (LIST) with MTT assay procedure in renal transplant recipients.
    Journal of immunoassay & immunochemistry, 2006, Volume: 27, Issue:2

    Topics: Adult; Calcineurin Inhibitors; Cyclosporine; Female; Graft Rejection; Humans; Immunoassay; Immunosuppressive Agents; Kidney Transplantation; Lymphocyte Activation; Lymphocytes; Male; Middle Aged; Tacrolimus; Tetrazolium Salts; Thiazoles

2006
Dasatinib, a small-molecule protein tyrosine kinase inhibitor, inhibits T-cell activation and proliferation.
    Blood, 2008, Feb-01, Volume: 111, Issue:3

    Topics: Animals; Biomarkers; CD28 Antigens; CD3 Complex; Cell Proliferation; Cells, Cultured; Cyclosporine; Cytokines; Dasatinib; Humans; Lymphocyte Activation; Male; Mice; Protein Binding; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines; Receptors, Antigen, T-Cell; Signal Transduction; Sirolimus; T-Lymphocytes; Thiazoles

2008
Non-specific anti-proliferative effect of FTY720, a derivative of fungal metabolite from Iscaria sinclarii.
    Archives of pharmacal research, 2008, Volume: 31, Issue:2

    Topics: Aniline Compounds; Animals; Antibiotics, Antineoplastic; Cell Proliferation; Crotonates; Cyclosporine; Fingolimod Hydrochloride; Fungi; Hydroxybutyrates; Immunity, Cellular; Immunosuppressive Agents; Interleukin-2; Lipopolysaccharides; Macrophages; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Nitric Oxide; Nitriles; Propylene Glycols; Sphingosine; T-Lymphocytes; Tetrazolium Salts; Thiazoles; Toluidines; Tumor Necrosis Factor-alpha

2008
Pharmacological activation of PPARbeta promotes rapid and calcineurin-dependent fiber remodeling and angiogenesis in mouse skeletal muscle.
    American journal of physiology. Endocrinology and metabolism, 2008, Volume: 295, Issue:2

    Topics: Animals; Calcineurin; Calcineurin Inhibitors; Cyclosporine; Immunohistochemistry; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Muscle Fibers, Skeletal; Muscle, Skeletal; MyoD Protein; Myogenic Regulatory Factor 5; Neovascularization, Physiologic; Physical Conditioning, Animal; PPAR-beta; Succinate Dehydrogenase; Thiazoles

2008
Insulin action on polyunsaturated phosphatidic acid formation in rat brain: an "in vitro" model with synaptic endings from cerebral cortex and hippocampus.
    Neurochemical research, 2009, Volume: 34, Issue:7

    Topics: Animals; Cerebral Cortex; Chromones; Cyclosporine; Diacylglycerol Kinase; Diglycerides; Genistein; Guanosine 5'-O-(3-Thiotriphosphate); Hippocampus; Insulin; Insulin Antagonists; Morpholines; Okadaic Acid; Phosphatidic Acids; Phosphoprotein Phosphatases; Piperidines; Pyrimidinones; Quinazolinones; Rats; Rats, Wistar; Sodium Fluoride; Synaptosomes; Thiazoles; Vanadates

2009
Peroxisome proliferator-activated receptor beta stimulation induces rapid cardiac growth and angiogenesis via direct activation of calcineurin.
    Cardiovascular research, 2009, Jul-01, Volume: 83, Issue:1

    Topics: Animals; Calcineurin; Calcineurin Inhibitors; Cells, Cultured; Coronary Vessels; Cyclin-Dependent Kinase 9; Cyclosporine; Enzyme Inhibitors; Heart; Hypoxia-Inducible Factor 1, alpha Subunit; Male; Mice; Mice, Inbred C57BL; Models, Animal; Myocardium; Myocytes, Cardiac; Neovascularization, Physiologic; NFATC Transcription Factors; PPAR-beta; Thiazoles

2009
Peroxisome proliferator-activated receptor beta activation promotes myonuclear accretion in skeletal muscle of adult and aged mice.
    Pflugers Archiv : European journal of physiology, 2009, Volume: 458, Issue:5

    Topics: Aging; Animals; Calcineurin; Calcineurin Inhibitors; Cell Division; Cell Fusion; Cell Nucleus; Citrate (si)-Synthase; Cyclosporine; Male; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Mice, Transgenic; Muscle Fibers, Fast-Twitch; Muscle Fibers, Skeletal; Muscle, Skeletal; NFATC Transcription Factors; PPAR-beta; Proliferating Cell Nuclear Antigen; Satellite Cells, Skeletal Muscle; Succinate Dehydrogenase; Thiazoles

2009
In vitro interactions between antifungals and immunosuppressive drugs against zygomycetes.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:8

    Topics: Amphotericin B; Antifungal Agents; Azoles; Cyclosporine; Drug Interactions; Immunosuppressive Agents; Itraconazole; Microbial Sensitivity Tests; Mucorales; Rhizopus; Sirolimus; Tacrolimus; Thiazoles; Triazoles

2009
Novel milk-based oral formulations: proof of concept.
    International journal of pharmaceutics, 2010, May-10, Volume: 390, Issue:2

    Topics: Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Aspirin; Buffers; Chemistry, Pharmaceutical; Cyclosporine; Danazol; Ethanol; Humans; Male; Meloxicam; Milk; Solubility; Thiazines; Thiazoles

2010
AF-2364 is a prospective spermicide candidate.
    Asian journal of andrology, 2010, Volume: 12, Issue:3

    Topics: Adenosine Triphosphate; Animals; Cell Line, Tumor; Cell Survival; Cyclosporine; Drug Therapy, Combination; Humans; Hydrazines; Indazoles; Male; Mice; Mitochondria; Permeability; Seminal Plasma Proteins; Sperm Motility; Spermatocidal Agents; Spermatozoa; Tetrazolium Salts; Thiazoles

2010
The compound cis-(dichloro)tetrammineruthenium(III) chloride induces caspase-mediated apoptosis in K562 cells.
    Toxicology in vitro : an international journal published in association with BIBRA, 2010, Volume: 24, Issue:6

    Topics: Antineoplastic Agents; Apoptosis; Caspases; Cell Cycle; Cell Survival; Cyclosporine; Humans; K562 Cells; Leukemia, Erythroblastic, Acute; Ruthenium Compounds; Tetrazolium Salts; Thiazoles; Trypan Blue; Tumor Stem Cell Assay

2010
Wnt/Ca2+/NFAT signaling maintains survival of Ph+ leukemia cells upon inhibition of Bcr-Abl.
    Cancer cell, 2010, Jul-13, Volume: 18, Issue:1

    Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Benzamides; Blotting, Western; Calcium; Cell Proliferation; Cyclosporine; Cytokines; Dasatinib; Female; Flow Cytometry; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Immunosuppressive Agents; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Mice; Mice, Inbred C57BL; NFATC Transcription Factors; Philadelphia Chromosome; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; RNA, Small Interfering; Signal Transduction; Thiazoles; Tumor Cells, Cultured; Wnt Proteins

2010
Correlation between the pharmacological efficacy of cyclosporine and tacrolimus as evaluated by the lymphocyte immunosuppressant sensitivity test (LIST) and the MTT assay procedure in patients before and after renal transplantation.
    International journal of clinical pharmacology and therapeutics, 2011, Volume: 49, Issue:2

    Topics: Cyclosporine; Humans; Immunosuppressive Agents; Kidney Transplantation; Lymphocytes; Tacrolimus; Tetrazolium Salts; Thiazoles

2011
Drug-interaction studies evaluating T-cell proliferation reveal distinct activity of dasatinib and imatinib in combination with cyclosporine A.
    Experimental hematology, 2012, Volume: 40, Issue:8

    Topics: Benzamides; CD28 Antigens; CD3 Complex; Cyclosporine; Dasatinib; Drug Interactions; Humans; Imatinib Mesylate; Immunosuppressive Agents; Lymphocyte Activation; Piperazines; Protein Kinase Inhibitors; Pyrimidines; T-Lymphocytes; Thiazoles

2012
Mitochondrial aquaporin-8 knockdown in human hepatoma HepG2 cells causes ROS-induced mitochondrial depolarization and loss of viability.
    Toxicology and applied pharmacology, 2012, Oct-15, Volume: 264, Issue:2

    Topics: Adenosine Triphosphate; Aquaporins; Blotting, Western; Cell Survival; Cyclosporine; Hep G2 Cells; Humans; Hydrogen Peroxide; L-Lactate Dehydrogenase; Membrane Potential, Mitochondrial; Microscopy, Fluorescence; Mitochondria, Liver; Oxidants; Permeability; Reactive Oxygen Species; RNA, Small Interfering; Tetrazolium Salts; Thiazoles; Trypan Blue

2012
Building upon Nature's Framework: Overview of Key Strategies Toward Increasing Drug-Like Properties of Natural Product Cyclopeptides and Macrocycles.
    Methods in molecular biology (Clifton, N.J.), 2019, Volume: 2001

    Topics: Anthraquinones; Biological Availability; Biological Products; Chemistry, Pharmaceutical; Cyclosporine; Cyclotides; Daptomycin; Depsipeptides; Drug Design; Drug Discovery; Ethers, Cyclic; Gramicidin; Lipopeptides; Macrocyclic Compounds; Macrolides; omega-Conotoxins; Organophosphorus Compounds; Oxazoles; Peptides; Peptides, Cyclic; Thiazoles; Thiazolidines

2019
[Avatrombopag combined with standard immunosuppressive therapy in the treatment of severe aplastic anemia with hepatic impairment in six patients].
    Zhonghua xue ye xue za zhi = Zhonghua xueyexue zazhi, 2022, 11-14, Volume: 43, Issue:11

    Topics: Anemia, Aplastic; Antilymphocyte Serum; Cyclosporine; Humans; Immunosuppression Therapy; Immunosuppressive Agents; Thiazoles

2022