thiazoles has been researched along with cyclosporine in 47 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 14 (29.79) | 18.2507 |
2000's | 19 (40.43) | 29.6817 |
2010's | 13 (27.66) | 24.3611 |
2020's | 1 (2.13) | 2.80 |
Authors | Studies |
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Claude, JR; Martin, C; Massicot, F; Pham Huy, C; Thevenin, M; Warnet, JM | 1 |
Cooper, MH; Gregory, SH; Starzl, TE; Wing, EJ | 1 |
Acosta, D; Jiang, T | 1 |
Cai, W; Foulkes, JG; Hu, L | 1 |
Chardonnet, Y; Lizard, G; Marionnet, AV; Schmitt, D | 1 |
Claude, JR; Duc, HT; Dutertre-Catella, H; Ellouk-Achard, S; Martin, C; Pham-Huy, C; Thevenin, M; Warnet, JM | 1 |
Claude, JR; Dutertre-Catella, H; Ellouk-Achard, S; Martin, C; Massicot, F; Pham-Huy, C; Rucay, P; Thevenin, M; Warnet, JM | 1 |
Borg, AG; Burgess, R; Fisher, A; Grey, M; Wood, P; Yin, JA | 1 |
Bonomini, L; DeFranco, P; Friedman, G; Jacobs, M; Kaplan, B; Lyman, N; Mulgaonkar, SP; Viscuso, R | 1 |
Brennan, DC; Burgess, SJ; Singer, GG | 1 |
Al Rayyes, O; Florén, CH | 1 |
Frantz, RP; Nguyen, TT | 1 |
Haug, MT; Park, MH; Pelegrin, D; Young, JB | 1 |
Downs, AM; Sansom, JE | 1 |
Kongkittingam, C; Vedejs, E | 1 |
Bal-Price, A; Brown, GC | 1 |
Calvo, M; Colell, A; Enrich, C; Fernández-Checa, JC; García-Ruiz, C; Morales, A | 1 |
Huang, ST; Lee, PN; Pang, JH; Yang, LJ; Yang, RC | 1 |
Davies, T; Kostrubsky, VE; Lodola, A; Rahbari, R | 1 |
Choy, YM; Fung, KP; Ko, S; Kong, SK; Kwok, TT; Lee, CY; Yuen, WF | 1 |
Evtodienko, YV; Kruglov, AG; Yaguzhinsky, LS; Yurkov, IS | 1 |
Cohen, RD; Ross, AS | 1 |
Liot, G; Lobner, D | 1 |
Gabryel, B; Małecki, A; Toborek, T | 1 |
Arakawa, K; Hirano, T; Saito, K; Saito, N; Satoh, H; Sugiyama, K; Takahashi, K | 1 |
Scheinfeld, N | 1 |
Jankowska, AM; Maciejewski, JP; Schade, AE; Schieven, GL; Susulic, V; Szpurka, H; Townsend, R; Zhang, R | 1 |
Cho, JY | 1 |
Abumrad, NA; Gaudel, C; Giordano, C; Grimaldi, PA; Schwartz, C | 1 |
de Boschero, MG; Giusto, NM; Zulian, SE | 1 |
Giordano, C; Gounon, P; Grimaldi, P; Hatem, SN; Jehl-Piétri, C; Lopez, P; Murdaca, J; Schwartz, C; Wagner, KD; Wagner, N | 1 |
Gaudel, C; Giordano, C; Grimaldi, PA; Jehl-Piétri, C; Lopez, P; Murdaca, J; Rousseau, AS; Sibille, B; Wagner, N | 1 |
Dannaoui, E; Lortholary, O; Schwarz, P | 1 |
Charkoftaki, G; Kytariolos, J; Macheras, P | 1 |
Chen, XX; Mao, YD; Sha, JH; Wang, H; Wang, LR; Zhou, ZM | 1 |
Benfica, PL; de Lima, AP; dos Santos, WB; Lacerda, Ede P; Mello, FM; Pavanin, LA; Pereira, Fde C; Ribeiro, Ade S; Valadares, MC; Vilanova-Costa, CA | 1 |
Alvarez-Calderon, F; Degregori, J; Druker, BJ; Eide, CA; Gregory, MA; Neviani, P; O'Hare, T; Perrotti, D; Phang, TL; Williams, RT; Zaberezhnyy, V | 1 |
Hirano, T; Isogai, K; Nakagawa, Y; Saito, K; Satoh, H; Sugiyama, K; Takahashi, K; Tasaki, M; Toyama, A | 1 |
Hokari, A | 1 |
Blake, SJ; Hughes, TP; Lyons, AB | 1 |
Carnovale, CE; Francés, DE; Marchissio, MJ; Marinelli, RA | 1 |
Bastide, C; Bruyere, F; Caremel, R; Castel-Lacanal, E; Cornu, JN; Guy, L; Karsenty, G; Kerdraon, J | 1 |
Baturin, D; Christians, U; DeGregori, J; Gardner, LA; Gore, L; Gregory, MA; Klawitter, J; Pollyea, DA; Porter, CC; Takebe, N; Zaberezhnyy, V | 1 |
Matsushima, N; Mendell, J; Parasrampuria, DA; Shi, M; Truitt, K; Zahir, H | 1 |
Huang, F; Rowland, L; Sabo, JP; Schultz, A; Trampisch, M; Voelk, C | 1 |
Blanco, MJ | 1 |
Fan, HH; Jing, LP; Li, JP; Li, Y; Peng, GX; Xiong, YZ; Yang, WR; Yang, Y; Ye, L; Zhang, FK; Zhang, L; Zhao, X; Zhou, K | 1 |
5 review(s) available for thiazoles and cyclosporine
Article | Year |
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Transcription-modulating drugs: mechanism and selectivity.
Topics: Animals; Anti-Inflammatory Agents; Aspirin; Cyclosporine; Drug Design; Estrogen Antagonists; Humans; Hypoglycemic Agents; Immunosuppressive Agents; Polyenes; Sirolimus; Tacrolimus; Thiazoles; Transcription, Genetic | 1996 |
Medical therapy for ulcerative colitis: the state of the art and beyond.
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antimetabolites, Antineoplastic; Butyrates; Colitis, Ulcerative; Cyclosporine; Epidermal Growth Factor; Glucocorticoids; Humans; Immunosuppressive Agents; Infliximab; Interferons; Mercaptopurine; Plasmapheresis; Probiotics; Remission Induction; Thiazoles | 2004 |
A review of deferasirox, bortezomib, dasatinib, and cyclosporine eye drops: possible uses and known side effects in cutaneous medicine.
Topics: Animals; Antineoplastic Agents; Benzoates; Boronic Acids; Bortezomib; Cyclosporine; Dasatinib; Deferasirox; Humans; Iron Chelating Agents; Ophthalmic Solutions; Protein Kinase Inhibitors; Pyrazines; Pyrimidines; Randomized Controlled Trials as Topic; Skin Diseases; Skin Neoplasms; Thiazoles; Triazoles | 2007 |
[Improved virologic response in chronic hepatitis C treated with peginterferon, ribavirin and add-on drug].
Topics: Antiviral Agents; Cyclosporine; Diterpenes; Drug Therapy, Combination; Fatty Acids, Monounsaturated; Fatty Alcohols; Female; Fluvastatin; Hepatitis C, Chronic; Humans; Indoles; Interferon-alpha; Male; Metformin; Nitro Compounds; Polyethylene Glycols; Recombinant Proteins; Ribavirin; Silybin; Silymarin; Thiazoles | 2011 |
[Drug therapy of bladder dysfunction].
Topics: Acetanilides; Anti-Inflammatory Agents; Botulinum Toxins, Type A; Cholinergic Antagonists; Cimetidine; Cyclosporine; Dimethyl Sulfoxide; Histamine H2 Antagonists; Humans; Immunosuppressive Agents; Muscarinic Antagonists; Neuromuscular Agents; Phosphodiesterase Inhibitors; Thiazoles; Urinary Bladder; Urinary Bladder Diseases; Urination; Urodynamics | 2013 |
3 trial(s) available for thiazoles and cyclosporine
Article | Year |
---|---|
Inhibition of calcineurin combined with dasatinib has direct and indirect anti-leukemia effects against BCR-ABL1(+) leukemia.
Topics: Adult; Animals; Antineoplastic Combined Chemotherapy Protocols; Calcineurin Inhibitors; Cell Line, Tumor; Cyclosporine; Dasatinib; Drug Synergism; Female; Flow Cytometry; Fusion Proteins, bcr-abl; Humans; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Male; Mice; Mice, Inbred C57BL; Middle Aged; Protein Kinase Inhibitors; Pyrimidines; Thiazoles; Treatment Outcome | 2014 |
Edoxaban drug-drug interactions with ketoconazole, erythromycin, and cyclosporine.
Topics: Administration, Oral; Adolescent; Adult; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cross-Over Studies; Cyclosporine; Cytochrome P-450 CYP3A; Drug Administration Schedule; Drug Interactions; Erythromycin; Factor Xa Inhibitors; Healthy Volunteers; Humans; Ketoconazole; Metabolic Clearance Rate; Middle Aged; Pyridines; Substrate Specificity; Thiazoles; Young Adult | 2016 |
Pharmacokinetic Interaction between Faldaprevir and Cyclosporine or Tacrolimus in Healthy Volunteers: A Prospective, Open-Label, Fixed-Sequence, Crossover Study.
Topics: Adolescent; Adult; Aminoisobutyric Acids; Antiviral Agents; Area Under Curve; Cross-Over Studies; Cyclosporine; Drug Interactions; Female; Graft Rejection; Healthy Volunteers; Hepatitis C; Humans; Immunosuppressive Agents; Leucine; Liver Transplantation; Male; Middle Aged; Oligopeptides; Proline; Prospective Studies; Quinolines; Secondary Prevention; Tacrolimus; Thiazoles; Young Adult | 2018 |
39 other study(ies) available for thiazoles and cyclosporine
Article | Year |
---|---|
Inhibitory effects of a platelet activating factor-antagonist 48740RP in cyclosporin-induced nephrotoxicity in the rat as assessed by renal glutathione metabolism parameters.
Topics: Aminopeptidases; Animals; Blood Urea Nitrogen; CD13 Antigens; Creatinine; Cyclosporine; Glutathione; Kidney; Kidney Cortex; Platelet Activating Factor; Pyridines; Rats; Thiazoles | 1991 |
Rapamycin but not FK506 inhibits the proliferation of mononuclear phagocytes induced by colony-stimulating factors.
Topics: Animals; Bone Marrow Cells; Cell Count; Cell Division; Colony-Stimulating Factors; Concanavalin A; Culture Media, Conditioned; Cyclosporine; Female; Lymphocyte Activation; Mice; Mice, Inbred C57BL; Phagocytes; Polyenes; Sirolimus; Spleen; T-Lymphocytes; Tacrolimus; Tetrazolium Salts; Thiazoles; Thymidine; Tritium | 1994 |
An in vitro model of cyclosporine-induced nephrotoxicity.
Topics: Alkaline Phosphatase; Animals; Cell Survival; Cells, Cultured; Cyclosporine; Fluoresceins; Fluorescent Dyes; Kidney Cortex; Kidney Diseases; L-Lactate Dehydrogenase; Mitochondria; Neutral Red; Pharmaceutical Vehicles; Polyethylene Glycols; Propidium; Rats; Rats, Sprague-Dawley; Tetrazolium Salts; Thiazoles | 1993 |
Comparative evaluation of the antiproliferative effect of cyclosporin A and gamma-interferon on normal and HPV-transformed keratinocytes by cell counting, MTT assay and tritiated thymidine incorporation.
Topics: Adult; Cell Count; Cell Division; Cell Line, Transformed; Cell Survival; Cells, Cultured; Coloring Agents; Cyclosporine; Growth Inhibitors; Humans; Interferon-gamma; Keratinocytes; Papillomaviridae; Reproducibility of Results; Tetrazolium Salts; Thiazoles; Thymidine; Tritium | 1997 |
Implication of CYP 3A in the toxicity of cyclosporin G (CsG), cyclosporin A (CsA) and FK506 on rat hepatocytes in primary culture.
Topics: Animals; Aryl Hydrocarbon Hydroxylases; Calcium; Cell Survival; Cells, Cultured; Coloring Agents; Cyclosporine; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Flow Cytometry; Immunosuppressive Agents; Intracellular Fluid; Liver; Male; Oxidoreductases, N-Demethylating; Rats; Rats, Wistar; Tacrolimus; Tetrazolium Salts; Thiazoles | 1997 |
Modulation of energy status and cytotoxicity induced by FK506 and cyclosporin A in a renal epithelial cell line.
Topics: Adenosine Triphosphate; Animals; Cell Survival; Cyclosporine; Energy Metabolism; Immunosuppressive Agents; Kidney; LLC-PK1 Cells; Nucleotides; Swine; Tacrolimus; Tetrazolium Salts; Thiazoles; Time Factors | 1997 |
Effect on cell kill of addition of multidrug resistance modifiers cyclosporin A and PSC 833 to cytotoxic agents in acute myeloid leukaemia.
Topics: Acute Disease; Adolescent; Adult; Aged; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cell Survival; Coloring Agents; Cyclosporine; Cyclosporins; Cytarabine; Daunorubicin; Drug Resistance, Neoplasm; Drug Synergism; Etoposide; Female; Humans; Idarubicin; Leukemia, Myeloid; Male; Middle Aged; Mitoxantrone; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured | 1997 |
Potential interaction of troglitazone and cyclosporine.
Topics: Acute Disease; Chromans; Cyclosporine; Drug Interactions; Female; Graft Rejection; Humans; Hypoglycemic Agents; Immunosuppressive Agents; Middle Aged; Osmolar Concentration; Thiazoles; Thiazolidinediones; Troglitazone | 1998 |
Effect of troglitazone on cyclosporine whole blood levels.
Topics: Chromans; Cyclosporine; Drug Interactions; Humans; Hypoglycemic Agents; Immunosuppressive Agents; Kidney Transplantation; Thiazoles; Thiazolidinediones; Troglitazone | 1998 |
Troglitazone upregulates LDL receptor activity in HepG2 cells.
Topics: Chromans; Cyclosporine; Humans; Hypoglycemic Agents; Insulin; Lipoproteins, LDL; Liver; Receptors, LDL; RNA, Messenger; Thiazoles; Thiazolidinediones; Troglitazone; Tumor Cells, Cultured; Up-Regulation | 1998 |
Rezulin (troglitazone) greatly increases cyclosporine metabolism.
Topics: Chromans; Cyclosporine; Drug Interactions; Drug Therapy, Combination; Female; Heart Transplantation; Humans; Hypoglycemic Agents; Immunosuppressive Agents; Metabolic Clearance Rate; Middle Aged; Thiazoles; Thiazolidinediones; Troglitazone | 1998 |
Troglitazone, a new antidiabetic agent, decreases cyclosporine level.
Topics: Aged; Chromans; Cyclosporine; Diabetes Mellitus, Type 1; Drug Interactions; Heart Transplantation; Humans; Hypoglycemic Agents; Immunosuppressive Agents; Male; Middle Aged; Thiazoles; Thiazolidinediones; Troglitazone | 1998 |
Severe contact allergy to footwear responding to handmade shoes.
Topics: Cyclosporine; Dermatitis, Allergic Contact; Foot Dermatoses; Humans; Immunosuppressive Agents; Male; Middle Aged; Patch Tests; Potassium Dichromate; Shoes; Thiazoles; Thiram | 1999 |
Solution-phase synthesis of a hindered N-methylated tetrapeptide using Bts-protected amino acid chlorides: efficient coupling and methylation steps allow purification by extraction.
Topics: Acylation; Amino Acids; Benzothiazoles; Chlorides; Cyclosporine; Methylation; Oligopeptides; Sulfones; Thiazoles | 2000 |
Nitric-oxide-induced necrosis and apoptosis in PC12 cells mediated by mitochondria.
Topics: Adenosine Triphosphate; Animals; Apoptosis; Azides; Caspase Inhibitors; Caspases; Cell Respiration; Cyclosporine; Cytochrome c Group; Cytosol; Enzyme Inhibitors; Glucose; Lactic Acid; Membrane Potentials; Methacrylates; Mitochondria; Necrosis; Nitric Oxide; Nitric Oxide Donors; Oxygen Consumption; PC12 Cells; Rats; Thiazoles | 2000 |
Trafficking of ganglioside GD3 to mitochondria by tumor necrosis factor-alpha.
Topics: Actins; Animals; Apoptosis; Biological Transport; Bridged Bicyclo Compounds, Heterocyclic; Cell Death; Cell Membrane; Cholesterol; Cyclosporine; Cytoskeleton; Endosomes; Enzyme Inhibitors; Filipin; Gangliosides; Golgi Apparatus; Hepatocytes; Humans; Kinetics; Microscopy, Confocal; Microscopy, Immunoelectron; Mitochondria; Protein Binding; rab GTP-Binding Proteins; rab5 GTP-Binding Proteins; rab7 GTP-Binding Proteins; Rats; Signal Transduction; Thiazoles; Thiazolidines; Time Factors; Tumor Necrosis Factor-alpha | 2002 |
Phyllanthus urinaria triggers the apoptosis and Bcl-2 down-regulation in Lewis lung carcinoma cells.
Topics: Animals; Antineoplastic Agents, Phytogenic; Apoptosis; Carcinoma, Lewis Lung; Caspase 3; Caspases; Cell Survival; Cyclosporine; DNA Fragmentation; Down-Regulation; Flow Cytometry; Genes, bcl-2; Mice; Phyllanthus; Plant Extracts; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured | 2003 |
Agree that idiosyncratic hepatotoxicity in TRO-treated patients is uncertain, but concerned about the data.
Topics: Apoptosis; Cell Survival; Chromans; Cyclosporine; Dose-Response Relationship, Drug; Drug Antagonism; Hepatocytes; Humans; Hypoglycemic Agents; Mitochondria, Liver; Thiazoles; Thiazolidinediones; Troglitazone; Tumor Cells, Cultured | 2003 |
Hyperthermia and tumour necrosis factor-alpha induced apoptosis via mitochondrial damage.
Topics: Animals; Apoptosis; Blotting, Western; Cell Line; Cyclosporine; Cytochrome c Group; Cytosol; Fever; Fluorescein-5-isothiocyanate; Fluorescent Dyes; Immunosuppressive Agents; Membranes; Mice; Mitochondria; Tetrazolium Salts; Thiazoles; Tumor Necrosis Factor-alpha | 2000 |
Mechanism of superoxide anion generation in intact mitochondria in the presence of lucigenin and cyanide.
Topics: Acridines; Adenosine Triphosphate; Animals; Antimycin A; Carbonyl Cyanide p-Trifluoromethoxyphenylhydrazone; Cell Respiration; Cyanides; Cyclosporine; Kinetics; Luminescent Measurements; Methacrylates; Mitochondria, Liver; Oligomycins; Oxygen; Oxygen Consumption; Proton-Motive Force; Rats; Rats, Wistar; Spectrometry, Fluorescence; Succinic Acid; Superoxides; Thiazoles; Uncoupling Agents | 2003 |
Role of MAPK/ERK in neurotrophin-4 potentiation of necrotic neuronal death.
Topics: Animals; Butadienes; Cell Death; Cells, Cultured; Cyclosporine; Enzyme Activation; Flavonoids; Immunosuppressive Agents; L-Lactate Dehydrogenase; Mice; Mitogen-Activated Protein Kinases; Necrosis; Nerve Growth Factors; Neurons; Nitriles; Phosphorylation; Tetrazolium Salts; Thiazoles | 2004 |
Immunosuppressive immunophilin ligands attenuate damage in cultured rat astrocytes depleted of glutathione and exposed to simulated ischemia in vitro. Comparison with N-acetylcysteine.
Topics: Acetylcysteine; Animals; Apoptosis; Astrocytes; Benzimidazoles; Brain Ischemia; Cell Separation; Cells, Cultured; Cyclosporine; Fluorescent Dyes; Free Radical Scavengers; Glutathione; Immunophilins; Immunosuppressive Agents; Ligands; Mitochondria; Oxidative Stress; Rats; Rats, Wistar; Reactive Oxygen Species; Tacrolimus; Tetrazolium Salts; Thiazoles | 2005 |
Correlation between pharmacological efficacy of cyclosporine A and tacrolimus, evaluated by lymphocyte immunosuppressant-sensitivity test (LIST) with MTT assay procedure in renal transplant recipients.
Topics: Adult; Calcineurin Inhibitors; Cyclosporine; Female; Graft Rejection; Humans; Immunoassay; Immunosuppressive Agents; Kidney Transplantation; Lymphocyte Activation; Lymphocytes; Male; Middle Aged; Tacrolimus; Tetrazolium Salts; Thiazoles | 2006 |
Dasatinib, a small-molecule protein tyrosine kinase inhibitor, inhibits T-cell activation and proliferation.
Topics: Animals; Biomarkers; CD28 Antigens; CD3 Complex; Cell Proliferation; Cells, Cultured; Cyclosporine; Cytokines; Dasatinib; Humans; Lymphocyte Activation; Male; Mice; Protein Binding; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines; Receptors, Antigen, T-Cell; Signal Transduction; Sirolimus; T-Lymphocytes; Thiazoles | 2008 |
Non-specific anti-proliferative effect of FTY720, a derivative of fungal metabolite from Iscaria sinclarii.
Topics: Aniline Compounds; Animals; Antibiotics, Antineoplastic; Cell Proliferation; Crotonates; Cyclosporine; Fingolimod Hydrochloride; Fungi; Hydroxybutyrates; Immunity, Cellular; Immunosuppressive Agents; Interleukin-2; Lipopolysaccharides; Macrophages; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Nitric Oxide; Nitriles; Propylene Glycols; Sphingosine; T-Lymphocytes; Tetrazolium Salts; Thiazoles; Toluidines; Tumor Necrosis Factor-alpha | 2008 |
Pharmacological activation of PPARbeta promotes rapid and calcineurin-dependent fiber remodeling and angiogenesis in mouse skeletal muscle.
Topics: Animals; Calcineurin; Calcineurin Inhibitors; Cyclosporine; Immunohistochemistry; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Muscle Fibers, Skeletal; Muscle, Skeletal; MyoD Protein; Myogenic Regulatory Factor 5; Neovascularization, Physiologic; Physical Conditioning, Animal; PPAR-beta; Succinate Dehydrogenase; Thiazoles | 2008 |
Insulin action on polyunsaturated phosphatidic acid formation in rat brain: an "in vitro" model with synaptic endings from cerebral cortex and hippocampus.
Topics: Animals; Cerebral Cortex; Chromones; Cyclosporine; Diacylglycerol Kinase; Diglycerides; Genistein; Guanosine 5'-O-(3-Thiotriphosphate); Hippocampus; Insulin; Insulin Antagonists; Morpholines; Okadaic Acid; Phosphatidic Acids; Phosphoprotein Phosphatases; Piperidines; Pyrimidinones; Quinazolinones; Rats; Rats, Wistar; Sodium Fluoride; Synaptosomes; Thiazoles; Vanadates | 2009 |
Peroxisome proliferator-activated receptor beta stimulation induces rapid cardiac growth and angiogenesis via direct activation of calcineurin.
Topics: Animals; Calcineurin; Calcineurin Inhibitors; Cells, Cultured; Coronary Vessels; Cyclin-Dependent Kinase 9; Cyclosporine; Enzyme Inhibitors; Heart; Hypoxia-Inducible Factor 1, alpha Subunit; Male; Mice; Mice, Inbred C57BL; Models, Animal; Myocardium; Myocytes, Cardiac; Neovascularization, Physiologic; NFATC Transcription Factors; PPAR-beta; Thiazoles | 2009 |
Peroxisome proliferator-activated receptor beta activation promotes myonuclear accretion in skeletal muscle of adult and aged mice.
Topics: Aging; Animals; Calcineurin; Calcineurin Inhibitors; Cell Division; Cell Fusion; Cell Nucleus; Citrate (si)-Synthase; Cyclosporine; Male; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Mice, Transgenic; Muscle Fibers, Fast-Twitch; Muscle Fibers, Skeletal; Muscle, Skeletal; NFATC Transcription Factors; PPAR-beta; Proliferating Cell Nuclear Antigen; Satellite Cells, Skeletal Muscle; Succinate Dehydrogenase; Thiazoles | 2009 |
In vitro interactions between antifungals and immunosuppressive drugs against zygomycetes.
Topics: Amphotericin B; Antifungal Agents; Azoles; Cyclosporine; Drug Interactions; Immunosuppressive Agents; Itraconazole; Microbial Sensitivity Tests; Mucorales; Rhizopus; Sirolimus; Tacrolimus; Thiazoles; Triazoles | 2009 |
Novel milk-based oral formulations: proof of concept.
Topics: Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Aspirin; Buffers; Chemistry, Pharmaceutical; Cyclosporine; Danazol; Ethanol; Humans; Male; Meloxicam; Milk; Solubility; Thiazines; Thiazoles | 2010 |
AF-2364 is a prospective spermicide candidate.
Topics: Adenosine Triphosphate; Animals; Cell Line, Tumor; Cell Survival; Cyclosporine; Drug Therapy, Combination; Humans; Hydrazines; Indazoles; Male; Mice; Mitochondria; Permeability; Seminal Plasma Proteins; Sperm Motility; Spermatocidal Agents; Spermatozoa; Tetrazolium Salts; Thiazoles | 2010 |
The compound cis-(dichloro)tetrammineruthenium(III) chloride induces caspase-mediated apoptosis in K562 cells.
Topics: Antineoplastic Agents; Apoptosis; Caspases; Cell Cycle; Cell Survival; Cyclosporine; Humans; K562 Cells; Leukemia, Erythroblastic, Acute; Ruthenium Compounds; Tetrazolium Salts; Thiazoles; Trypan Blue; Tumor Stem Cell Assay | 2010 |
Wnt/Ca2+/NFAT signaling maintains survival of Ph+ leukemia cells upon inhibition of Bcr-Abl.
Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Benzamides; Blotting, Western; Calcium; Cell Proliferation; Cyclosporine; Cytokines; Dasatinib; Female; Flow Cytometry; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Immunosuppressive Agents; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Mice; Mice, Inbred C57BL; NFATC Transcription Factors; Philadelphia Chromosome; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; RNA, Small Interfering; Signal Transduction; Thiazoles; Tumor Cells, Cultured; Wnt Proteins | 2010 |
Correlation between the pharmacological efficacy of cyclosporine and tacrolimus as evaluated by the lymphocyte immunosuppressant sensitivity test (LIST) and the MTT assay procedure in patients before and after renal transplantation.
Topics: Cyclosporine; Humans; Immunosuppressive Agents; Kidney Transplantation; Lymphocytes; Tacrolimus; Tetrazolium Salts; Thiazoles | 2011 |
Drug-interaction studies evaluating T-cell proliferation reveal distinct activity of dasatinib and imatinib in combination with cyclosporine A.
Topics: Benzamides; CD28 Antigens; CD3 Complex; Cyclosporine; Dasatinib; Drug Interactions; Humans; Imatinib Mesylate; Immunosuppressive Agents; Lymphocyte Activation; Piperazines; Protein Kinase Inhibitors; Pyrimidines; T-Lymphocytes; Thiazoles | 2012 |
Mitochondrial aquaporin-8 knockdown in human hepatoma HepG2 cells causes ROS-induced mitochondrial depolarization and loss of viability.
Topics: Adenosine Triphosphate; Aquaporins; Blotting, Western; Cell Survival; Cyclosporine; Hep G2 Cells; Humans; Hydrogen Peroxide; L-Lactate Dehydrogenase; Membrane Potential, Mitochondrial; Microscopy, Fluorescence; Mitochondria, Liver; Oxidants; Permeability; Reactive Oxygen Species; RNA, Small Interfering; Tetrazolium Salts; Thiazoles; Trypan Blue | 2012 |
Building upon Nature's Framework: Overview of Key Strategies Toward Increasing Drug-Like Properties of Natural Product Cyclopeptides and Macrocycles.
Topics: Anthraquinones; Biological Availability; Biological Products; Chemistry, Pharmaceutical; Cyclosporine; Cyclotides; Daptomycin; Depsipeptides; Drug Design; Drug Discovery; Ethers, Cyclic; Gramicidin; Lipopeptides; Macrocyclic Compounds; Macrolides; omega-Conotoxins; Organophosphorus Compounds; Oxazoles; Peptides; Peptides, Cyclic; Thiazoles; Thiazolidines | 2019 |
[Avatrombopag combined with standard immunosuppressive therapy in the treatment of severe aplastic anemia with hepatic impairment in six patients].
Topics: Anemia, Aplastic; Antilymphocyte Serum; Cyclosporine; Humans; Immunosuppression Therapy; Immunosuppressive Agents; Thiazoles | 2022 |