thiazoles has been researched along with cyclic gmp in 36 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 5 (13.89) | 18.7374 |
1990's | 13 (36.11) | 18.2507 |
2000's | 10 (27.78) | 29.6817 |
2010's | 5 (13.89) | 24.3611 |
2020's | 3 (8.33) | 2.80 |
Authors | Studies |
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Rozmysłowicz, T | 2 |
el-Fakahany, EE; Lai, WS | 1 |
Dickinson, KE; Hirschowitz, BI; Hokin, LE; Pruitt, RE; Sekar, MC | 1 |
Francis, LP; Singh, J | 1 |
Butler, RD; Evans, RL; McCrohan, CR | 1 |
Benavides, J; Camelin, JC; Flamand, F; Gueremy, C; Le Fur, G; Legrand, JJ; Mitrani, N; Uzan, A | 1 |
Caciacli, F; Ciancetta, S; Ciccarelli, R | 1 |
Kazarov, AR; Sobolev, AS; Tertov, VV | 1 |
Alkon, DL; Inoue, H; Kouchi, T; Sakakibara, M; Yoshioka, T | 1 |
Bacon, ER; Bode, DC; Buchholz, RA; Dundore, RL; Lesher, GY; Pagani, ED; Silver, PJ; Singh, B | 1 |
Jensen, RT; Johnson, BE; Le, PT; Ohsaki, Y; Yang, HK | 1 |
Arnone, M; Gonalons, N; Gueudet, C; Gully, D; Heaulme, M; Keane, P; Le Fur, G; Poncelet, M; Santucci, V; Thurneyssen, O | 1 |
Lesage, AS; Leysen, JE; Peeters, L | 1 |
Bansinath, M; Nivarthi, RN; Turndorf, H | 1 |
Hall, ED; Oostveen, JA; Sethy, VH; Wu, H | 1 |
Alonso, R; Arnone, M; Bignon, E; Boigegrain, R; Brodin, R; Gueudet, C; Héaulme, M; Keane, P; Landi, M; Le Fur, G; Maffrand, JP; Molimard, JC; Olliero, D; Pascal, M; Poncelet, M; Seban, E; Simiand, J; Soubrié, P | 1 |
Hamad, AM; Johnson, SR; Knox, AJ | 1 |
Aguirre-Bañuelos, P; Granados-Soto, V | 1 |
Borda, E; Sterin-Borda, L; Stranieri, G | 1 |
Belinsky, MG; Chen, ZS; Guo, Y; Hopper-Borge, E; Kotova, E; Kruh, GD; Lee, K | 1 |
Antunes, E; De Nucci, G; Marcondes, S; Moreira, J; Thomazzi, SM | 1 |
Broadbent, T; Hsieh, E; Thiagarajah, JR; Verkman, AS | 1 |
Severina, IS | 1 |
Chan, SL; Chan, SS; Fiscus, RR; Fraser, M; Tsang, BK | 1 |
Danoff, TM; Johnson, AG; Pearce, GL | 1 |
Brahmachari, S; Fung, YK; Pahan, K | 1 |
Mejía-García, TA; Paes-de-Carvalho, R | 1 |
Carniglia, L; Caruso, C; Durand, D; Lasaga, M | 1 |
Cámara, M; Frangipani, E; Heeb, S; Imperi, F; Kaever, V; Visaggio, D; Visca, P | 1 |
Balligand, JL | 1 |
Chao, YC; Fleischer, J; Yang, RB | 1 |
Antunes, E; Bertollotto, GM; Candido, TZ; De Nucci, G; de Oliveira, MG; Kiguti, LRA; Mónica, FZ; Pupo, AS; Rojas-Moscoso, JA | 1 |
Allard, PM; Gdaniec, BG; Köhler, T; Queiroz, EF; van Delden, C; Wolfender, JL | 1 |
Abdel-Rady, M; Abou-Salim, MA; Atalla, AA; Barakat, A; El-Adasy, AA; Elshaier, YAMM; Hassan, MIA; Hussein, AHM; Khames, AA | 1 |
Bai, H; Chen, H; Gao, L; Jia, L; Liu, L; Lv, L; Ma, T; Song, X; Wang, X; Wu, Y; Xu, X; Yu, Y; Zhang, Z; Zhao, M | 1 |
2 review(s) available for thiazoles and cyclic gmp
Article | Year |
---|---|
[No: a new look on the mechanism of action of old drugs].
Topics: Animals; Antiprotozoal Agents; Cyclic GMP; Guanylate Cyclase; Humans; Nitric Oxide; Nitric Oxide Donors; Signal Transduction; Thiazoles | 2005 |
Cardiac salvage by tweaking with beta-3-adrenergic receptors.
Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Animals; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Endothelial Cells; Heart Diseases; Humans; Myocardial Contraction; Myocytes, Cardiac; Nitric Oxide; Nitric Oxide Synthase Type I; Nitric Oxide Synthase Type III; Receptors, Adrenergic, beta-3; Signal Transduction; Thiazoles; Ventricular Remodeling | 2016 |
1 trial(s) available for thiazoles and cyclic gmp
Article | Year |
---|---|
A randomized, double-blind, placebo-controlled, parallel-group study to assess the efficacy and safety of dual ACE/NEP inhibitor GW660511X in mild-to-moderate hypertensive patients.
Topics: Adolescent; Adult; Aged; Angiotensin-Converting Enzyme Inhibitors; Antihypertensive Agents; Atrial Natriuretic Factor; Blood Pressure; Cyclic GMP; Dizziness; Double-Blind Method; Female; Headache; Humans; Hypertension; Male; Middle Aged; Neprilysin; Peptidyl-Dipeptidase A; Placebos; Thiazoles; Treatment Outcome | 2006 |
33 other study(ies) available for thiazoles and cyclic gmp
Article | Year |
---|---|
[Effect of thioproline in vitro on selected functions of peripheral blood lymphocytes from healthy persons and patients with lympho- proliferative syndromes].
Topics: Adolescent; Adult; Aged; Antineoplastic Agents; B-Lymphocytes; Blood Donors; Cyclic AMP; Cyclic GMP; Cytotoxicity, Immunologic; DNA; Dose-Response Relationship, Drug; Female; Humans; In Vitro Techniques; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphoma, Non-Hodgkin; Male; Middle Aged; Models, Biological; T-Lymphocytes; Thiazoles; Thiazolidines | 1991 |
Antagonism by the diacylglycerol kinase inhibitor R59 022 of muscarinic receptor-mediated cyclic GMP formation and binding of [3H]N-methylscopolamine.
Topics: Animals; Binding, Competitive; Carbachol; Cyclic GMP; Diacylglycerol Kinase; Mice; Muscarinic Antagonists; N-Methylscopolamine; Phosphotransferases; Pyrimidinones; Receptors, Muscarinic; Scopolamine Derivatives; Thiazoles; Tumor Cells, Cultured | 1990 |
Muscarinic receptor antagonist activity of diacylglycerol lipase and kinase inhibitors.
Topics: Animals; Brain; Cells, Cultured; Cyclic GMP; Cyclohexanes; Cyclohexanones; Guinea Pigs; Heart; Lipoprotein Lipase; Myocardium; N-Methylscopolamine; Pancreas; Parasympatholytics; Platelet Activating Factor; Pyrimidinones; Rats; Receptors, Muscarinic; Scopolamine Derivatives; Thiazoles; Tritium | 1990 |
Effects of phorbol ester and related compounds on acetylcholine-evoked [3H]leucine-labelled protein secretion in permeabilized rat pancreatic acini.
Topics: Acetylcholine; Animals; Calcium; Cell Membrane Permeability; Cyclic GMP; Female; In Vitro Techniques; Inositol Phosphates; Male; Pancreas; Phospholipid Ethers; Polymyxin B; Proteins; Pyrimidinones; Rats; Tetradecanoylphorbol Acetate; Thiazoles | 1990 |
Tentacle contraction in Heliophrya erhardi (Suctoria): the role of inositol phospholipid metabolites and cyclic nucleotides in stimulus-response coupling.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Bucladesine; Chlorides; Ciliophora; Cyclic AMP; Cyclic GMP; Dibutyryl Cyclic GMP; Inositol Phosphates; Lithium; Lithium Chloride; Muscle Contraction; Pyrimidinones; Sugar Phosphates; Tetradecanoylphorbol Acetate; Thiazoles | 1988 |
Cytostatic influence of thioproline on peripheral lymphocytes of healthy persons and non-Hodgkin's lymphoma patients.
Topics: Adolescent; Adult; Antineoplastic Agents; Cyclic AMP; Cyclic GMP; Humans; In Vitro Techniques; Lymphocytes; Lymphoma, Non-Hodgkin; Reference Values; Thiazoles; Thiazolidines; Thymidine | 1989 |
2-Amino-6-trifluoromethoxy benzothiazole, a possible antagonist of excitatory amino acid neurotransmission--II. Biochemical properties.
Topics: Acetylcholine; Amino Acids; Animals; Anticonvulsants; Apomorphine; Cerebellum; Chlordiazepoxide; Cyclic GMP; Diazepam; gamma-Aminobutyric Acid; Harmaline; In Vitro Techniques; Injections, Intraventricular; Isoniazid; Male; Rats; Rats, Inbred Strains; Riluzole; Synaptic Transmission; Thiazoles | 1985 |
Effect of arginine salt of thioproline (thiazolidine carboxylate) on cyclic nucleotides of cerebral tumour.
Topics: Arginine; Brain Chemistry; Brain Neoplasms; Cyclic AMP; Cyclic GMP; Humans; Thiazoles; Thiazolidines | 1980 |
Effects of radioprotectors on the cAMP and cGMP systems.
Topics: Adenylyl Cyclases; Animals; beta-Aminoethyl Isothiourea; Biogenic Amines; Cyclic AMP; Cyclic GMP; Enzyme Activation; Guanylate Cyclase; Male; Mercaptoethylamines; Mice; Phosphoric Diester Hydrolases; Protein Kinases; Radiation-Protective Agents; Rats; Rats, Inbred Strains; Thiazoles; Thiourea | 1984 |
Induction of photoresponse by the hydrolysis of polyphosphoinositides in the Hermissenda type B photoreceptor.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Cyclic AMP; Cyclic GMP; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Hydrolysis; Inositol 1,4,5-Trisphosphate; Kinetics; Lithium Chloride; Models, Biological; Neomycin; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositol Phosphates; Photoreceptor Cells, Invertebrate; Platelet Activating Factor; Pyrimidinones; Snails; Spermine; Thiazoles; Thionucleotides; Type C Phospholipases | 1994 |
Species-dependent pharmacodynamic effects of the selective low Km cyclic AMP phosphodiesterase III inhibitors WIN 58993 and WIN 62005.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Administration, Oral; Animals; Aorta; Blood Pressure; Cardiotonic Agents; Cyclic GMP; Cyclic Nucleotide Phosphodiesterases, Type 3; Dogs; Dose-Response Relationship, Drug; Female; Heart Rate; Imidazoles; Injections, Intravenous; Isoenzymes; Male; Milrinone; Myocardial Contraction; Myocardium; Phosphodiesterase Inhibitors; Pyridines; Pyridones; Rats; Rats, Sprague-Dawley; Species Specificity; Structure-Activity Relationship; Thiazoles; Vasodilator Agents; Ventricular Function, Left | 1995 |
Human small cell lung cancer cell lines express functional atrial natriuretic peptide receptors.
Topics: Atrial Natriuretic Factor; Base Sequence; Blotting, Southern; Carcinoma, Small Cell; Cell Division; Cyclic GMP; HeLa Cells; Humans; Iodine Radioisotopes; Lung Neoplasms; Molecular Sequence Data; Polymerase Chain Reaction; Radioimmunoassay; Receptors, Atrial Natriuretic Factor; Ribonucleases; RNA, Messenger; Stimulation, Chemical; Tetrazolium Salts; Thiazoles; Thymidine; Tritium; Tumor Cells, Cultured | 1993 |
Neurobehavioural effects of SR 27897, a selective cholecystokinin type A (CCK-A) receptor antagonist.
Topics: Animals; Apomorphine; Brain; Cyclic GMP; Dose-Response Relationship, Drug; Female; Indoleacetic Acids; Male; Mice; Motor Activity; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Cholecystokinin; Thiazoles | 1993 |
Lubeluzole, a novel long-term neuroprotectant, inhibits the glutamate-activated nitric oxide synthase pathway.
Topics: Animals; Arginine; Cells, Cultured; Cyclic GMP; Glutamic Acid; Guanylate Cyclase; Hippocampus; Interferon-gamma; Lipopolysaccharides; Neuroprotective Agents; Nitric Oxide Synthase; Piperidines; Rats; Stereoisomerism; Thiazoles | 1996 |
Role of nitric oxide-mediated signal transduction in hypothermia induced by intravenous anesthetics.
Topics: Anesthetics, Intravenous; Animals; Cerebellum; Cyclic GMP; Hypothermia; Ketamine; Mice; Nitric Oxide; Nitric Oxide Synthase; Pentobarbital; Proto-Oncogene Proteins c-fos; Riluzole; Signal Transduction; Thiazoles | 1997 |
Neuroprotective effects of the dopamine agonists pramipexole and bromocriptine in 3-acetylpyridine-treated rats.
Topics: Adenosine Triphosphate; Animals; Benzothiazoles; Body Temperature; Bromocriptine; Cerebellum; Cyclic GMP; Dopamine Agonists; Male; Motor Activity; Neurons; Neuroprotective Agents; Neurotoxins; Olivary Nucleus; Pramipexole; Pyridines; Rats; Rats, Wistar; Thiazoles | 1997 |
SR146131: a new potent, orally active, and selective nonpeptide cholecystokinin subtype 1 receptor agonist. II. In vivo pharmacological characterization.
Topics: Animals; Appetite Stimulants; Callithrix; Cerebellum; Cyclic GMP; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Eating; Female; Gallbladder Emptying; Gastric Acid; Gastric Emptying; Gerbillinae; Indoles; Male; Mice; Motor Activity; Neuropeptide Y; Paraventricular Hypothalamic Nucleus; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Species Specificity; Stereotyped Behavior; Thiazoles | 1999 |
Antiproliferative effects of NO and ANP in cultured human airway smooth muscle.
Topics: Asthma; Atrial Natriuretic Factor; Blood Proteins; Cell Division; Cells, Cultured; Coloring Agents; Cyclic GMP; Diuretics; Hemoglobins; Hemostatics; Humans; Hyperplasia; Lung; Mitogens; Muscle, Smooth; Nitric Oxide; Nitric Oxide Donors; Nitroprusside; Penicillamine; Peptide Fragments; Phosphodiesterase Inhibitors; Purinones; Tetrazolium Salts; Thiazoles; Thrombin; Vasodilator Agents | 1999 |
Evidence for the participation of the nitric oxide-cyclic GMP pathway in the antinociceptive action of meloxicam in the formalin test.
Topics: Analgesics, Non-Narcotic; Animals; Cyclic GMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Formaldehyde; Guanylate Cyclase; Meloxicam; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Oxadiazoles; Pain; Pain Measurement; Quinoxalines; Rats; Rats, Wistar; Thiazines; Thiazoles | 2000 |
H(1)-Receptor activation triggers the endogenous nitric oxide signalling system in the rat submandibular gland.
Topics: Amylases; Animals; Cyclic GMP; Histamine Agonists; In Vitro Techniques; Nitric Oxide; Nitric Oxide Synthase; Phosphatidylinositols; Rats; Receptors, Histamine H1; Signal Transduction; Submandibular Gland; Thiazoles; Type C Phospholipases | 2002 |
MRP8, ATP-binding cassette C11 (ABCC11), is a cyclic nucleotide efflux pump and a resistance factor for fluoropyrimidines 2',3'-dideoxycytidine and 9'-(2'-phosphonylmethoxyethyl)adenine.
Topics: Adenine; Adenosine Triphosphate; Animals; Antineoplastic Agents; Antiviral Agents; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Cell Membrane; Colforsin; Coloring Agents; Cyclic AMP; Cyclic GMP; DNA, Complementary; Dose-Response Relationship, Drug; Drug Resistance; Floxuridine; Fluorouracil; Genetic Vectors; Growth Inhibitors; Immunoblotting; Inhibitory Concentration 50; Insecta; Models, Biological; Nitrosamines; Nucleotides; Organophosphonates; Swine; Tetrazolium Salts; Thiazoles; Time Factors; Transfection; Zalcitabine | 2003 |
Role of cyclic GMP on inhibition by nitric oxide donors of human eosinophil chemotaxis in vitro.
Topics: Adolescent; Adult; Blotting, Western; Cell Survival; Chemotaxis, Leukocyte; Cyclic GMP; Eosinophils; Female; Humans; In Vitro Techniques; Male; Middle Aged; Molsidomine; N-Formylmethionine Leucyl-Phenylalanine; Nitric Oxide Donors; Nitroprusside; Penicillamine; Tetrazolium Salts; Thiazoles; Tyrosine | 2004 |
Prevention of toxin-induced intestinal ion and fluid secretion by a small-molecule CFTR inhibitor.
Topics: Administration, Oral; Animals; Bacterial Toxins; Benzoates; Body Fluids; Cell Line; Chlorides; Cholera Toxin; Cyclic AMP; Cyclic GMP; Electric Conductivity; Enterotoxins; Escherichia coli Proteins; Humans; Injections, Intraperitoneal; Intestinal Mucosa; Intestines; Ion Channels; Male; Mice; Mice, Inbred Strains; Mice, Mutant Strains; Rats; Rats, Wistar; Thiazoles; Thiazolidines; Tissue Distribution | 2004 |
Regulation of p53 and suppression of apoptosis by the soluble guanylyl cyclase/cGMP pathway in human ovarian cancer cells.
Topics: Adenoviridae; Apoptosis; Atrial Natriuretic Factor; bcl-2-Associated X Protein; Benzothiazoles; Caspase 3; Caspases; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Cyclin-Dependent Kinase Inhibitor p21; Enzyme Activation; Enzyme Inhibitors; Female; Gene Expression Regulation, Neoplastic; Guanylate Cyclase; Half-Life; Humans; Mutation; Ovarian Neoplasms; Oxadiazoles; Phosphorylation; Proto-Oncogene Proteins c-mdm2; Quinoxalines; RNA, Small Interfering; Serine; Signal Transduction; Thiazoles; Toluene; Tumor Cells, Cultured; Tumor Suppressor Protein p53; X-Linked Inhibitor of Apoptosis Protein | 2006 |
Induction of glial fibrillary acidic protein expression in astrocytes by nitric oxide.
Topics: Animals; Animals, Newborn; Astrocytes; Cell Survival; Cells, Cultured; Cerebral Cortex; Corpus Striatum; Cyclic GMP; Cyclic N-Oxides; Cytokines; Dose-Response Relationship, Drug; Drug Interactions; Electrophoretic Mobility Shift Assay; Enzyme Inhibitors; Fluorescent Antibody Technique; Free Radical Scavengers; Gene Expression; Glial Fibrillary Acidic Protein; HIV Envelope Protein gp120; Imidazoles; Lipopolysaccharides; Lysine; Male; Mice; Mice, Inbred C57BL; Nitric Oxide; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetrazolium Salts; Thiazoles; Thionucleotides; Time Factors | 2006 |
Nitric oxide regulates cell survival in purified cultures of avian retinal neurons: involvement of multiple transduction pathways.
Topics: Adenosine; Aminoquinolines; Analysis of Variance; Animals; Cell Survival; Cells, Cultured; Chick Embryo; Cyclic GMP; Cyclic N-Oxides; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Free Radical Scavengers; Imidazoles; Neurons; Nitrates; Nitric Oxide; Nitric Oxide Donors; Nitrites; Penicillamine; Retina; Signal Transduction; Tetrazolium Salts; Thiazoles; Tritium | 2007 |
Metabotropic glutamate receptor 3 activation prevents nitric oxide-induced death in cultured rat astrocytes.
Topics: 1-Methyl-3-isobutylxanthine; Amino Acids; Animals; Animals, Newborn; Astrocytes; Bridged Bicyclo Compounds, Heterocyclic; Caspase 3; Cell Death; Cells, Cultured; Cerebral Cortex; Cyclic AMP; Cyclic GMP; Cytochromes c; DNA Fragmentation; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Gene Expression Regulation; In Situ Nick-End Labeling; Interferon-gamma; Neurotransmitter Agents; Nitric Oxide; Nitric Oxide Donors; Phosphatidylserines; Phosphodiesterase Inhibitors; Polyamines; Polysaccharides; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Tetrazolium Salts; Thiazoles | 2010 |
The Gac/Rsm and cyclic-di-GMP signalling networks coordinately regulate iron uptake in Pseudomonas aeruginosa.
Topics: Bacterial Proteins; Cyclic GMP; Gene Expression Regulation, Bacterial; Iron; Oligopeptides; Phenols; Pseudomonas aeruginosa; Repressor Proteins; RNA-Binding Proteins; Siderophores; Sigma Factor; Thiazoles; Virulence Factors | 2014 |
Guanylyl cyclase-G is an alarm pheromone receptor in mice.
Topics: Animals; Behavior, Animal; Cyclic GMP; Ganglia, Sensory; Guanylate Cyclase; Male; Membrane Proteins; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons; Nose; Pheromones; Signal Transduction; Thiazoles | 2018 |
Mirabegron elicits rat corpus cavernosum relaxation and increases in vivo erectile response.
Topics: Acetanilides; Animals; Arterial Pressure; Cyclic AMP; Cyclic GMP; Gene Expression Regulation; Intracellular Space; Male; Muscle Contraction; Muscle Relaxation; Penile Erection; Penis; Rats; Rats, Wistar; Receptors, Adrenergic, beta; RNA, Messenger; Thiazoles | 2019 |
Surface sensing triggers a broad-spectrum antimicrobial response in Pseudomonas aeruginosa.
Topics: Anti-Bacterial Agents; Antibiosis; Biofilms; Cyclic GMP; Glycolipids; Oligopeptides; Phenols; Pseudomonas aeruginosa; Quinolines; Quorum Sensing; Siderophores; Staphylococcus aureus; Thiazoles | 2020 |
Multifunctional Isosteric Pyridine Analogs-Based 2-Aminothiazole: Design, Synthesis, and Potential Phosphodiesterase-5 Inhibitory Activity.
Topics: Cyclic GMP; Cyclic Nucleotide Phosphodiesterases, Type 5; Drug Design; Humans; Phosphodiesterase 5 Inhibitors; Pyridines; Structure-Activity Relationship; Thiazoles | 2021 |
Xylazole inhibits NO-cGMP pathway in fetal rat nerve cells.
Topics: Adenosine Triphosphatases; Animals; Animals, Newborn; Cells, Cultured; Cyclic GMP; Neurons; Nitric Oxide; Rats; Signal Transduction; Thiazoles | 2022 |