Page last updated: 2024-08-21

thiazoles and curcumin

thiazoles has been researched along with curcumin in 53 studies

Research

Studies (53)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (1.89)18.2507
2000's18 (33.96)29.6817
2010's32 (60.38)24.3611
2020's2 (3.77)2.80

Authors

AuthorsStudies
Aggarwal, BB; McQueen, T; Mehta, K; Pantazis, P1
Atherton, K; Campbell, FC; Daly, AK; Harbottle, A1
Kang, HJ; Kim, MS; Moon, A1
Chen, A; Fu, Y; Xu, J1
Hasegawa, K; Naiki, H; Ono, K; Yamada, M1
Chen, A; Zheng, S1
Ambegaokar, SS; Begum, AN; Chen, PP; Cole, GM; Frautschy, SA; Glabe, CG; Kayed, R; Lim, GP; Simmons, MR; Ubeda, OJ; Yang, F1
Dubiel, W; Dumdey, R; Frommel, C; Füllbeck, M; Huang, X; Preissner, R1
Chakrabarti, R; Cohen, AN; LoTempio, MM; Ramalingam, TS; Ramamurthy, B; Srivatsan, ES; Steele, HL; Veena, MS; Wang, MB1
Anuchapreeda, S; Chanarat, P; Limtrakul, P; Sittipreechacharn, S; Thanarattanakorn, P1
Campbell, FC; Collett, GP1
Kowdley, KV; Messner, DJ; Sivam, G1
Chen, X; Han, Y; Li, W; Lin, R; Liu, P; Pi, R1
Byun, JH; Kim, DJ; Kim, H; Kim, Y; Lee, WK; Mook-Jung, I; Yoo, KH1
Cao, C; Di, W; Hu, G; Kivlin, R; Lu, S; Pan, W; Song, X; Wallin, B; Wan, Y; Yang, H1
Lohiya, NK; Pal, R; Talwar, GP; Vishwakarma, R; Vyas, HK1
Dubey, VK; Sarkar, N; Singh, AN1
Anantharam, V; Bravosanpedro, JM; Fuentes, JM; González-Polo, RA; Kanthasamy, AG; Morán, JM; Niso-Santano, M; Ortiz-Ortiz, MA; Soler, G1
Carver, JA; Ecroyd, H; Hudson, SA; Kee, TW1
Kwon, TK; Lim, JH1
Bresjanac, M; Kovacs, GG; Mohorko, N; Popović, M; Repovs, G1
Banerjee, S; Kanwar, SS; Majumdar, AP; Nautiyal, J; Patel, BB; Sarkar, FH; Yu, Y1
Camacho-Alonso, F; Gómez-Garcia, F; López-Jornet, P1
Hirao, K; Shirai, N; Taguchi, H; Tooyama, I; Yamamoto, A; Yanagisawa, D1
Alavez, S; Klang, IM; Lithgow, GJ; Vantipalli, MC; Zucker, DJ1
Nahar, U; Nehru, B; Sood, PK1
Chen, A; Feng, Y; Kang, Q; Lin, J; Tang, Y1
Jiang, T; Pan, LF; Zhang, YH; Zhi, XL; Zhou, P1
Han, H; Kim, HY; Kim, Y; Lee, YS; Roh, EJ; Seo, JH; Shin, KJ1
Basir, SF; Bharti, AC; Das, BC; Mahata, S; Pandey, A; Shishodia, G; Shukla, S; Tyagi, A; Vishnoi, K1
Chereddy, KK; Coco, R; des Rieux, A; Memvanga, PB; Préat, V; Ucakar, B; Vandermeulen, G1
Cao, R; Chen, J; Chen, Q; Gong, L; Liu, Y; Lv, J; Qu, W; Shi, H; Wang, Z; Xiao, J; Zhang, H1
Bouillaguet, S; Bulit, F; Feki, A; Filieri, A; Grad, I; Lange, N; Manoil, D; Schrenzel, J; Simon, S; Wataha, JC1
Gong, Y; Guo, Y; Lin, J; Shan, Q; Shi, F; Shi, R; Yang, X1
Bonnat, L; Chierici, S; Dufour, E; Garcia, J; Moni, L1
Bose, A; Chowdhury, PK; Gautam, S; Karmakar, S1
Arya, P; Kundu, B; Mishra, P; Mukherjee, G; Srivastava, A; Vasaikar, SV1
Chen, C; Chen, G; Chen, QH; Wang, G; Wang, R; Zhang, C; Zhang, Q; Zhang, X; Zheng, S; Zhong, Q1
Khodagholi, F; Mazaheri, M; Moosavi-Movahedi, AA; Saboury, AA; Shaerzadeh, F; Sheibani, N1
Ahmad, B; Kale, A; Mothi, N; Muthu, SA1
Chojnacki, JE; Liu, K; Saathoff, JM; Zhang, S1
Hu, YH; Ren, WM; Tang, XC; Xu, MM; Zhang, HY1
Kim, SY; Lee, JW; Moon, EY; Park, S; Um, SH1
Jia, Y; Liu, S; Liu, X; Pan, W; Tian, C; Wang, H; Wang, Y; Yan, J1
Huang, CF; Liu, HS; Ramesh, C; Su, CL; Tseng, CL; Yao, CF1
Cui, M; Fu, H1
Aguilera-Garrido, A; Boulaiz, H; Galisteo-González, F; Marchal, JA; Molina-Bolívar, JA; Navarro, SA; Ramírez, A1
Hassani, L; Mahmudian, A; Moeeni, M; Mohammadi, F1
Duan, D; Jiang, Y; Li, Y; Mu, H; Ni, L; Sun, K; Wang, A; Wu, Z; Yan, X; Zhang, L1
Patel, B; Patel, MM; Rawal, S1
Jain, VK; Kumar, R; Kumar, V; Nagpal, S1
Chen, Z; Kong, LY; Wang, JS; Wei, DD; Yang, L1
Abd Malek, SN; Abdul Wahab, N; Ahmed Hamdi, OA; Awang, K; Looi, CY; Syed Abdul Rahman, SN; Thomas, NF1

Reviews

2 review(s) available for thiazoles and curcumin

ArticleYear
Advances in development of fluorescent probes for detecting amyloid-β aggregates.
    Acta pharmacologica Sinica, 2016, Volume: 37, Issue:6

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Animals; Benzothiazoles; Boron Compounds; Curcumin; Fluorescent Dyes; Humans; Optical Imaging; Stilbenes; Thiazoles; Thiophenes

2016
Fluorescent Imaging of Amyloid-β Deposits in Brain: An Overview of Probe Development and a Highlight of the Applications for In Vivo Imaging.
    Current medicinal chemistry, 2018, Volume: 25, Issue:23

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Benzothiazoles; Brain; Congo Red; Curcumin; Fluorescent Dyes; Humans; Microscopy, Fluorescence, Multiphoton; Positron Emission Tomography Computed Tomography; Thiazoles

2018

Other Studies

51 other study(ies) available for thiazoles and curcumin

ArticleYear
Antiproliferative effect of curcumin (diferuloylmethane) against human breast tumor cell lines.
    Anti-cancer drugs, 1997, Volume: 8, Issue:5

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; Blotting, Western; Breast Neoplasms; Cell Cycle; Cell Division; Cell Line; Curcumin; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Humans; Ornithine Decarboxylase; Tetrazolium Salts; Thiazoles

1997
Role of glutathione S-transferase P1, P-glycoprotein and multidrug resistance-associated protein 1 in acquired doxorubicin resistance.
    International journal of cancer, 2001, Jun-15, Volume: 92, Issue:6

    Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Calcium Channel Blockers; Coloring Agents; Curcumin; Cytosol; Dose-Response Relationship, Drug; Doxorubicin; Drug Resistance, Neoplasm; Genetic Vectors; Glutathione S-Transferase pi; Glutathione Transferase; Humans; Immunoblotting; Inhibitory Concentration 50; Isoenzymes; Liver; Multidrug Resistance-Associated Proteins; Phenotype; Protein Transport; Rats; Reverse Transcriptase Polymerase Chain Reaction; Tetrazolium Salts; Thiazoles; Transfection; Tumor Cells, Cultured; Verapamil

2001
Inhibition of invasion and induction of apoptosis by curcumin in H-ras-transformed MCF10A human breast epithelial cells.
    Archives of pharmacal research, 2001, Volume: 24, Issue:4

    Topics: Antineoplastic Agents, Phytogenic; Apoptosis; Breast; Caspase 3; Caspases; Curcumin; DNA Fragmentation; Enzyme Activation; Epithelial Cells; Female; Gene Expression Regulation; Genes, bcl-2; Genes, ras; Humans; Immunoblotting; Oxidation-Reduction; Reactive Oxygen Species; Signal Transduction; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

2001
Activation of peroxisome proliferator-activated receptor-gamma contributes to the inhibitory effects of curcumin on rat hepatic stellate cell growth.
    American journal of physiology. Gastrointestinal and liver physiology, 2003, Volume: 285, Issue:1

    Topics: Actins; Animals; Antineoplastic Agents; Antioxidants; Cell Division; Chromans; Collagen Type I; Curcumin; Dose-Response Relationship, Drug; Drug Synergism; Fibronectins; Gene Expression; Hepatocytes; Male; NF-kappa B; Rats; Rats, Sprague-Dawley; Receptors, Cytoplasmic and Nuclear; RNA, Messenger; Thiazoles; Thiazolidinediones; Transcription Factors; Troglitazone

2003
Curcumin has potent anti-amyloidogenic effects for Alzheimer's beta-amyloid fibrils in vitro.
    Journal of neuroscience research, 2004, Mar-15, Volume: 75, Issue:6

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Anti-Inflammatory Agents, Non-Steroidal; Benzothiazoles; Cinnamates; Curcumin; Depsides; Dose-Response Relationship, Drug; In Vitro Techniques; Kinetics; Lipoxygenase Inhibitors; Masoprocol; Microscopy, Electron; Microscopy, Polarization; Neurofibrillary Tangles; Peptide Fragments; Platelet Aggregation Inhibitors; Rosmarinic Acid; Spectrometry, Fluorescence; Thiazoles; Time Factors

2004
Activation of PPARgamma is required for curcumin to induce apoptosis and to inhibit the expression of extracellular matrix genes in hepatic stellate cells in vitro.
    The Biochemical journal, 2004, Nov-15, Volume: 384, Issue:Pt 1

    Topics: Animals; Apoptosis; Cell Proliferation; Curcumin; Cyclin D1; Enzyme Inhibitors; Extracellular Matrix; Flow Cytometry; Gene Expression Regulation; Liver; Male; Nitro Compounds; PPAR gamma; Rats; Rats, Sprague-Dawley; Receptors, Transforming Growth Factor beta; Signal Transduction; Thiazoles; Transforming Growth Factor beta; Transforming Growth Factor beta1

2004
Curcumin inhibits formation of amyloid beta oligomers and fibrils, binds plaques, and reduces amyloid in vivo.
    The Journal of biological chemistry, 2005, Feb-18, Volume: 280, Issue:7

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzoates; Benzothiazoles; Biphenyl Compounds; Blood-Brain Barrier; Brain; Cell Line, Tumor; Congo Red; Curcumin; Diamines; Humans; Ibuprofen; Mice; Mice, Transgenic; Naproxen; Peptide Fragments; Plaque, Amyloid; Protein Binding; Protein Denaturation; Protein Structure, Quaternary; Pyridazines; Solubility; Thiazoles

2005
Novel curcumin- and emodin-related compounds identified by in silico 2D/3D conformer screening induce apoptosis in tumor cells.
    BMC cancer, 2005, Aug-05, Volume: 5

    Topics: Annexin A5; Antineoplastic Agents; Apoptosis; Caspase 3; Caspase 7; Caspases; Cell Line, Tumor; Cell Survival; COP9 Signalosome Complex; Curcumin; DNA Fragmentation; Drug Design; Drug Screening Assays, Antitumor; Emodin; Enzyme Inhibitors; Gene Expression Regulation, Neoplastic; HeLa Cells; Humans; Models, Chemical; Models, Statistical; Multiprotein Complexes; Peptide Hydrolases; Propidium; Proto-Oncogene Proteins c-jun; Signal Transduction; Software; Tetrazolium Salts; Thiazoles; Tumor Suppressor Protein p53

2005
Curcumin suppresses growth of head and neck squamous cell carcinoma.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2005, Oct-01, Volume: 11, Issue:19 Pt 1

    Topics: Animals; Annexin A5; Antineoplastic Agents; Blotting, Western; Carcinoma, Squamous Cell; Cell Line, Tumor; Cell Nucleus; Cell Separation; Cell Survival; Curcumin; Cyclin D1; Dose-Response Relationship, Drug; Female; Flow Cytometry; Head and Neck Neoplasms; Humans; I-kappa B Proteins; In Vitro Techniques; Mice; Mice, Nude; Microscopy, Fluorescence; Neoplasm Transplantation; NF-kappa B; NF-KappaB Inhibitor alpha; Phosphorylation; Tetrazolium Salts; Thiazoles

2005
Inhibitory effect of curcumin on WT1 gene expression in patient leukemic cells.
    Archives of pharmacal research, 2006, Volume: 29, Issue:1

    Topics: Adolescent; Antineoplastic Agents; Cell Line, Tumor; Child; Child, Preschool; Curcumin; Electrophoresis, Polyacrylamide Gel; Female; Gene Expression Regulation, Neoplastic; Genes, Wilms Tumor; Humans; Infant; K562 Cells; Leukemia; Male; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetrazolium Salts; Thiazoles

2006
Overexpression of p65/RelA potentiates curcumin-induced apoptosis in HCT116 human colon cancer cells.
    Carcinogenesis, 2006, Volume: 27, Issue:6

    Topics: Apoptosis; Cell Line, Tumor; Cell Survival; Curcumin; Gene Expression Regulation, Neoplastic; Humans; NF-kappa B; Poly(ADP-ribose) Polymerases; Tetrazolium Salts; Thiazoles; Transcription Factor RelA; Transfection; X-Linked Inhibitor of Apoptosis Protein

2006
Curcumin reduces the toxic effects of iron loading in rat liver epithelial cells.
    Liver international : official journal of the International Association for the Study of the Liver, 2009, Volume: 29, Issue:1

    Topics: Animals; Cells, Cultured; Curcumin; Deferoxamine; Epithelial Cells; Ferric Compounds; Inhibitory Concentration 50; Liver; Oxidative Stress; Quaternary Ammonium Compounds; Rats; Reactive Oxygen Species; Signal Transduction; Tetrazolium Salts; Thiazoles

2009
Exposure to metal ions regulates mRNA levels of APP and BACE1 in PC12 cells: blockage by curcumin.
    Neuroscience letters, 2008, Aug-08, Volume: 440, Issue:3

    Topics: Amyloid beta-Protein Precursor; Amyloid Precursor Protein Secretases; Analysis of Variance; Animals; Curcumin; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gene Expression Regulation; Metals; PC12 Cells; Rats; RNA, Messenger; Tetrazolium Salts; Thiazoles; Time Factors

2008
Aminostyrylbenzofuran derivatives as potent inhibitors for Abeta fibril formation.
    Bioorganic & medicinal chemistry letters, 2008, Oct-15, Volume: 18, Issue:20

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Benzofurans; Benzothiazoles; Benzoxazoles; Chemistry, Pharmaceutical; Curcumin; Drug Design; Electrons; Humans; Inhibitory Concentration 50; Models, Chemical; Peptide Fragments; Structure-Activity Relationship; Styrenes; Thiazoles

2008
AMPK mediates curcumin-induced cell death in CaOV3 ovarian cancer cells.
    Oncology reports, 2008, Volume: 20, Issue:6

    Topics: AMP-Activated Protein Kinases; Antineoplastic Agents; Cell Death; Cell Line, Tumor; Cell Survival; Curcumin; Enzyme Inhibitors; Female; Gene Expression Regulation, Enzymologic; Gene Expression Regulation, Neoplastic; Humans; Ovarian Neoplasms; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Tetrazolium Salts; Thiazoles

2008
Selective killing of leukemia and lymphoma cells ectopically expressing hCGbeta by a conjugate of curcumin with an antibody against hCGbeta subunit.
    Oncology, 2009, Volume: 76, Issue:2

    Topics: Aged; Antigens, CD; Antigens, Differentiation, Myelomonocytic; Cell Separation; Chorionic Gonadotropin, beta Subunit, Human; Curcumin; Drug Design; Female; Humans; Leukemia; Leukemia, Myeloid, Acute; Leukocytes, Mononuclear; Lymphoma; Male; Middle Aged; Sialic Acid Binding Ig-like Lectin 3; Tetrazolium Salts; Thiazoles; U937 Cells

2009
Effect of curcumin on amyloidogenic property of molten globule-like intermediate state of 2,5-diketo-D-gluconate reductase A.
    Biological chemistry, 2009, Volume: 390, Issue:10

    Topics: Amyloid; Amyloidosis; Benzothiazoles; Biological Assay; Circular Dichroism; Curcumin; Hydrogen-Ion Concentration; Microscopy, Atomic Force; Protein Folding; Protein Structure, Secondary; Spectrometry, Fluorescence; Spectrophotometry, Ultraviolet; Sugar Alcohol Dehydrogenases; Thiazoles; Time Factors

2009
Curcumin enhances paraquat-induced apoptosis of N27 mesencephalic cells via the generation of reactive oxygen species.
    Neurotoxicology, 2009, Volume: 30, Issue:6

    Topics: Acetylcysteine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Apoptosis; Caspase 3; Cell Line, Transformed; Curcumin; Dose-Response Relationship, Drug; Drug Synergism; Flow Cytometry; Gene Expression Regulation; Herbicides; Hydrogen Peroxide; Mesencephalon; Neurons; Nitric Oxide Synthase Type I; Nitric Oxide Synthase Type II; Paraquat; Rats; Reactive Oxygen Species; Tetrazolium Salts; Thiazoles; Tyrosine; Vitamin E

2009
The thioflavin T fluorescence assay for amyloid fibril detection can be biased by the presence of exogenous compounds.
    The FEBS journal, 2009, Volume: 276, Issue:20

    Topics: Amyloid; Benzothiazoles; Biological Assay; Curcumin; Fluorescent Dyes; Quercetin; Reproducibility of Results; Resveratrol; Spectrometry, Fluorescence; Stilbenes; Thiazoles

2009
Curcumin inhibits phorbol myristate acetate (PMA)-induced MCP-1 expression by inhibiting ERK and NF-kappaB transcriptional activity.
    Food and chemical toxicology : an international journal published for the British Industrial Biological Research Association, 2010, Volume: 48, Issue:1

    Topics: Antineoplastic Agents; Blotting, Western; Cell Nucleus; Chemokine CCL2; Coloring Agents; Curcumin; Electrophoretic Mobility Shift Assay; Enzyme-Linked Immunosorbent Assay; Extracellular Signal-Regulated MAP Kinases; Humans; Luciferases; NF-kappa B; Promoter Regions, Genetic; Reverse Transcriptase Polymerase Chain Reaction; RNA; Tetradecanoylphorbol Acetate; Tetrazolium Salts; Thiazoles; Transcription Factor AP-1; Transcription, Genetic; Transfection; U937 Cells

2010
Curcumin labeling of neuronal fibrillar tau inclusions in human brain samples.
    Journal of neuropathology and experimental neurology, 2010, Volume: 69, Issue:4

    Topics: Alzheimer Disease; Benzothiazoles; Brain Diseases; Curcumin; Humans; Neurofibrillary Tangles; Neurons; Pick Disease of the Brain; Silver Staining; Supranuclear Palsy, Progressive; tau Proteins; Tauopathies; Thiazoles

2010
Curcumin enhances dasatinib-induced inhibition of growth and transformation of colon cancer cells.
    International journal of cancer, 2011, Feb-15, Volume: 128, Issue:4

    Topics: Adenoma; Adenomatous Polyposis Coli Protein; Animals; Antineoplastic Agents; Blotting, Western; Cell Adhesion; Cell Movement; Cell Proliferation; Cell Transformation, Neoplastic; Cells, Cultured; Colonic Neoplasms; CSK Tyrosine-Protein Kinase; Curcumin; Dasatinib; Drug Synergism; Electrophoretic Mobility Shift Assay; Endothelium, Vascular; ErbB Receptors; Female; Humans; Immunoenzyme Techniques; Intestinal Neoplasms; Mice; Mice, Knockout; Neoplasm Invasiveness; Neovascularization, Pathologic; NF-kappa B; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines; Receptor, IGF Type 1; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; src-Family Kinases; Thiazoles; Umbilical Veins

2011
Effect of curcumin and irradiation in PE/CA-PJ15 oral squamous cell carcinoma.
    Acta odontologica Scandinavica, 2011, Volume: 69, Issue:5

    Topics: Antineoplastic Agents; Carcinoma, Squamous Cell; Cell Line, Tumor; Cell Survival; Colorimetry; Coloring Agents; Curcumin; Humans; Mouth Neoplasms; Neoadjuvant Therapy; Radiation-Sensitizing Agents; Radiotherapy Dosage; Tetrazolium Salts; Thiazoles; Time Factors

2011
Curcuminoid binds to amyloid-β1-42 oligomer and fibril.
    Journal of Alzheimer's disease : JAD, 2011, Volume: 24 Suppl 2

    Topics: Amyloid; Amyloid beta-Peptides; Analysis of Variance; Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzothiazoles; Curcumin; Dose-Response Relationship, Drug; Fluorescent Dyes; Humans; Microscopy, Electron, Scanning Transmission; Peptide Fragments; Protein Binding; Thiazoles; Time Factors

2011
Amyloid-binding compounds maintain protein homeostasis during ageing and extend lifespan.
    Nature, 2011, Apr-14, Volume: 472, Issue:7342

    Topics: Aging; Amyloid; Amyloid beta-Peptides; Animals; Autophagy; Benzothiazoles; Caenorhabditis elegans; Caenorhabditis elegans Proteins; Curcumin; DNA-Binding Proteins; Dose-Response Relationship, Drug; Forkhead Transcription Factors; Homeostasis; Humans; Longevity; Molecular Chaperones; Paralysis; Phenotype; Proteasome Endopeptidase Complex; Protein Binding; Proteins; Survival Analysis; Thiazoles; Transcription Factors

2011
Curcumin attenuates aluminum-induced oxidative stress and mitochondrial dysfunction in rat brain.
    Neurotoxicity research, 2011, Volume: 20, Issue:4

    Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Aluminum; Animals; Anti-Inflammatory Agents, Non-Steroidal; Brain; Curcumin; Electron Transport Complex IV; Gene Expression Regulation; Glutathione; HSP72 Heat-Shock Proteins; Mitochondria; NADH Dehydrogenase; Oxidative Stress; Rats; Rats, Sprague-Dawley; RNA, Messenger; Succinate Dehydrogenase; Tetrazolium Salts; Thiazoles

2011
Curcumin inhibits gene expression of receptor for advanced glycation end-products (RAGE) in hepatic stellate cells in vitro by elevating PPARγ activity and attenuating oxidative stress.
    British journal of pharmacology, 2012, Volume: 166, Issue:8

    Topics: Animals; Curcumin; Gene Expression Regulation; Gene Knockdown Techniques; Glutathione; Hepatic Stellate Cells; Lipid Peroxidation; Male; Mice; Mice, Inbred C57BL; Nitro Compounds; Oxidative Stress; PPAR gamma; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Real-Time Polymerase Chain Reaction; Receptor for Advanced Glycation End Products; Receptors, Immunologic; RNA; RNA, Small Interfering; Thiazoles

2012
Inhibitory effect of curcumin on the Al(III)-induced Aβ₄₂ aggregation and neurotoxicity in vitro.
    Biochimica et biophysica acta, 2012, Volume: 1822, Issue:8

    Topics: Aluminum; Alzheimer Disease; Amyloid beta-Peptides; Animals; Benzothiazoles; Circular Dichroism; Curcumin; Microscopy, Atomic Force; Neurotoxicity Syndromes; PC12 Cells; Peptide Fragments; Rats; Thiazoles

2012
Small molecules that protect against β-amyloid-induced cytotoxicity by inhibiting aggregation of β-amyloid.
    Bioorganic & medicinal chemistry, 2012, Aug-15, Volume: 20, Issue:16

    Topics: Amyloid beta-Peptides; Animals; Benzene Derivatives; Benzothiazoles; Cells, Cultured; Coumaric Acids; Curcumin; Disease Models, Animal; Dose-Response Relationship, Drug; Male; Mice; Mice, Inbred ICR; Molecular Structure; Molecular Weight; Peptide Fragments; Resveratrol; Stilbenes; Thiazoles

2012
Functional regulatory role of STAT3 in HPV16-mediated cervical carcinogenesis.
    PloS one, 2013, Volume: 8, Issue:7

    Topics: Carcinogenesis; Caspase 3; Cell Line, Tumor; Curcumin; Electrophoretic Mobility Shift Assay; Female; Flow Cytometry; Gene Expression Regulation, Viral; Human papillomavirus 16; Humans; Immunoblotting; Immunohistochemistry; Oncogene Proteins, Viral; RNA, Small Interfering; STAT3 Transcription Factor; Tetrazolium Salts; Thiazoles; Tyrphostins; Uterine Cervical Neoplasms

2013
Combined effect of PLGA and curcumin on wound healing activity.
    Journal of controlled release : official journal of the Controlled Release Society, 2013, Oct-28, Volume: 171, Issue:2

    Topics: Animals; Anti-Inflammatory Agents; Cell Line, Tumor; Cell Survival; Collagen; Curcumin; Female; Glutathione Peroxidase; Keratinocytes; L-Lactate Dehydrogenase; Lactic Acid; Mice; Nanoparticles; NF-kappa B; Peroxidase; Polyglycolic Acid; Polylactic Acid-Polyglycolic Acid Copolymer; Skin; Tetrazolium Salts; Thiazoles; Wound Healing

2013
B19, a novel monocarbonyl analogue of curcumin, induces human ovarian cancer cell apoptosis via activation of endoplasmic reticulum stress and the autophagy signaling pathway.
    International journal of biological sciences, 2013, Volume: 9, Issue:8

    Topics: Analysis of Variance; Apoptosis; Autophagy; Blotting, Western; Cell Line, Tumor; Curcumin; Dose-Response Relationship, Drug; Endoplasmic Reticulum Stress; Female; Flow Cytometry; Fluorescent Antibody Technique; Humans; Microscopy, Electron; Signal Transduction; Tetrazolium Salts; Thiazoles

2013
Antimicrobial activity and cytotoxicity of 3 photosensitizers activated with blue light.
    Journal of endodontics, 2014, Volume: 40, Issue:3

    Topics: Animals; Anti-Infective Agents; Cell Line; Cell Survival; Coloring Agents; Curcumin; Dental Pulp; Embryonic Stem Cells; Eosine Yellowish-(YS); Humans; Lactobacillus; Light; Mice; Microbial Viability; Mitochondria; Odontoblasts; Photosensitizing Agents; Rose Bengal; Tetrazolium Salts; Thiazoles

2014
Curcumin induces apoptosis via simultaneously targeting AKT/mTOR and RAF/MEK/ERK survival signaling pathways in human leukemia THP-1 cells.
    Die Pharmazie, 2014, Volume: 69, Issue:3

    Topics: Annexin A5; Antineoplastic Agents; Apoptosis; Blotting, Western; Cell Line, Tumor; Cell Proliferation; Coloring Agents; Curcumin; Enzyme Activation; Fluorescein-5-isothiocyanate; Fluorescent Dyes; Humans; Leukemia, Myeloid, Acute; MAP Kinase Kinase Kinases; MAP Kinase Signaling System; Oncogene Protein v-akt; raf Kinases; Tetrazolium Salts; Thiazoles; TOR Serine-Threonine Kinases

2014
'Clickable' 2,5-diketopiperazines as scaffolds for ligation of biomolecules: their use in Aβ inhibitor assembly.
    Organic & biomolecular chemistry, 2014, Jul-21, Volume: 12, Issue:27

    Topics: Amyloid beta-Peptides; Benzothiazoles; Curcumin; Diketopiperazines; Ligation; Thiazoles

2014
β-cyclodextrin and curcumin, a potent cocktail for disaggregating and/or inhibiting amyloids: a case study with α-synuclein.
    Biochemistry, 2014, Jul-01, Volume: 53, Issue:25

    Topics: alpha-Synuclein; Amyloid; Benzothiazoles; beta-Cyclodextrins; Circular Dichroism; Curcumin; Drug Synergism; Fluorescent Dyes; Thiazoles

2014
Selective interception of gelsolin amyloidogenic stretch results in conformationally distinct aggregates with reduced toxicity.
    ACS chemical neuroscience, 2014, Oct-15, Volume: 5, Issue:10

    Topics: Amyloid; Benzothiazoles; Curcumin; Emetine; Fluorescence; Gelsolin; Hydrophobic and Hydrophilic Interactions; Kinetics; Light; Microscopy, Atomic Force; Molecular Docking Simulation; Particle Size; Peptides; Scattering, Radiation; Spectroscopy, Fourier Transform Infrared; Thiazoles

2014
Structure-Activity Relationship and Pharmacokinetic Studies of 1,5-Diheteroarylpenta-1,4-dien-3-ones: A Class of Promising Curcumin-Based Anticancer Agents.
    Journal of medicinal chemistry, 2015, Jun-11, Volume: 58, Issue:11

    Topics: Animals; Antineoplastic Agents; Cell Proliferation; Chromatography, High Pressure Liquid; Curcumin; Drug Design; Female; Humans; Male; Mice; Mice, Inbred C57BL; Models, Molecular; Molecular Structure; Pentanones; Prostatic Neoplasms; Structure-Activity Relationship; Tandem Mass Spectrometry; Thiazoles; Tissue Distribution; Tumor Cells, Cultured; Uterine Cervical Neoplasms

2015
Curcumin Protects β-Lactoglobulin Fibril Formation and Fibril-Induced Neurotoxicity in PC12 Cells.
    PloS one, 2015, Volume: 10, Issue:7

    Topics: Aflatoxin M1; Animals; Benzothiazoles; Cattle; Cell Death; Cell Differentiation; Circular Dichroism; Curcumin; Hydrogen-Ion Concentration; Lactoglobulins; Lead; Microscopy, Atomic Force; Microscopy, Fluorescence; Neurites; Neuroprotection; Neuroprotective Agents; Neurotoxins; PC12 Cells; Protein Structure, Secondary; Rats; Reactive Oxygen Species; Spectrometry, Fluorescence; Thiazoles

2015
Curcumin promotes fibril formation in F isomer of human serum albumin via amorphous aggregation.
    Biophysical chemistry, 2015, Volume: 207

    Topics: Amyloid; Benzothiazoles; Circular Dichroism; Curcumin; Humans; Isomerism; Kinetics; Microscopy, Electron, Transmission; Protein Binding; Protein Stability; Protein Structure, Secondary; Protein Structure, Tertiary; Serum Albumin; Temperature; Thiazoles

2015
Bivalent ligands incorporating curcumin and diosgenin as multifunctional compounds against Alzheimer's disease.
    Bioorganic & medicinal chemistry, 2015, Nov-15, Volume: 23, Issue:22

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Benzothiazoles; Cell Line, Tumor; Cell Survival; Curcumin; Diosgenin; Drug Design; Humans; Ligands; Neuroprotective Agents; Reactive Oxygen Species; Thiazoles

2015
Curcumin hampers the antitumor effect of vinblastine via the inhibition of microtubule dynamics and mitochondrial membrane potential in HeLa cervical cancer cells.
    Phytomedicine : international journal of phytotherapy and phytopharmacology, 2016, Jun-15, Volume: 23, Issue:7

    Topics: Animals; Antineoplastic Agents, Phytogenic; Apoptosis; Caspase 3; Cell Survival; Curcumin; Drug Synergism; Female; HeLa Cells; Humans; Male; Membrane Potential, Mitochondrial; Mice, Inbred C57BL; Microtubules; Reactive Oxygen Species; Tetrazolium Salts; Thiazoles; Vinblastine

2016
Co-delivery of docetaxel and curcumin prodrug via dual-targeted nanoparticles with synergistic antitumor activity against prostate cancer.
    Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie, 2017, Volume: 88

    Topics: Aconitic Acid; Animals; Antineoplastic Agents; Cell Death; Cell Line, Tumor; Coumarins; Curcumin; Docetaxel; Drug Delivery Systems; Drug Liberation; Drug Stability; Drug Synergism; Endocytosis; Humans; Inhibitory Concentration 50; Lactic Acid; Male; Mice, Inbred BALB C; Mice, Nude; Nanoparticles; Particle Size; Peptides; Polyethylene Glycols; Polyglycolic Acid; Polylactic Acid-Polyglycolic Acid Copolymer; Prodrugs; Prostatic Neoplasms; Proton Magnetic Resonance Spectroscopy; Taxoids; Thiazoles

2017
Using gene expression database to uncover biology functions of 1,4-disubstituted 1,2,3-triazole analogues synthesized via a copper (I)-catalyzed reaction.
    European journal of medicinal chemistry, 2017, May-26, Volume: 132

    Topics: Antineoplastic Agents; Apoptosis; Autophagy; Carcinoma, Hepatocellular; Cell Line, Tumor; Copper; Curcumin; Databases, Genetic; Glycogen Synthase Kinase 3; Humans; Liver Neoplasms; Structure-Activity Relationship; Thiazoles; Triazoles; Urea

2017
Albumin-covered lipid nanocapsules exhibit enhanced uptake performance by breast-tumor cells.
    Colloids and surfaces. B, Biointerfaces, 2018, May-01, Volume: 165

    Topics: Breast Neoplasms; Cell Proliferation; Cell Survival; Coumarins; Curcumin; Drug Liberation; Endocytosis; Female; Humans; Lipids; MCF-7 Cells; Nanocapsules; Serum Albumin; Thiazoles

2018
Inhibition of amyloid fibrillation of lysozyme by bisdemethoxycurcumin and diacetylbisdemethoxycurcumin.
    Biophysical chemistry, 2018, Volume: 235

    Topics: Amyloid; Animals; Benzothiazoles; Chickens; Curcumin; Diarylheptanoids; Molecular Docking Simulation; Molecular Structure; Muramidase; Particle Size; Protein Aggregates; Thiazoles

2018
Trastuzumab- and Fab' fragment-modified curcumin PEG-PLGA nanoparticles: preparation and evaluation in vitro and in vivo.
    International journal of nanomedicine, 2018, Volume: 13

    Topics: Animals; Cell Death; Cell Line, Tumor; Coumarins; Curcumin; Endocytosis; Female; Flow Cytometry; Humans; Immunoglobulin Fab Fragments; Injections, Intravenous; Mice, Inbred BALB C; Microscopy, Fluorescence; Nanoparticles; Polyesters; Polyethylene Glycols; Rats, Sprague-Dawley; Thiazoles; Tissue Distribution; Trastuzumab

2018
Fabrication, optimisation and
    Journal of microencapsulation, 2020, Volume: 37, Issue:8

    Topics: Antineoplastic Agents; Calorimetry, Differential Scanning; Carcinoma, Non-Small-Cell Lung; Cell Line, Tumor; Cell Survival; Cobalt; Curcumin; Docetaxel; Drug Delivery Systems; Drug Screening Assays, Antitumor; Hemolysis; Humans; Hydrogen-Ion Concentration; In Vitro Techniques; Lipids; Lung Neoplasms; Microspheres; Nanostructures; Particle Size; Temperature; Tetrazolium Salts; Thiazoles; X-Ray Diffraction

2020
Comparison of Virosome vs. Liposome as drug delivery vehicle using HepG2 and CaCo2 cell lines.
    Journal of microencapsulation, 2021, Volume: 38, Issue:5

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Antineoplastic Agents, Phytogenic; Caco-2 Cells; Cell Movement; Curcumin; Drug Delivery Systems; Excipients; Hep G2 Cells; Humans; Liposomes; Microbial Sensitivity Tests; Neoplasms; Nitric Oxide; Tetrazolium Salts; Thiazoles; Virosomes; Wound Healing

2021
Reversal effects of traditional Chinese herbs on multidrug resistance in cancer cells.
    Natural product research, 2011, Volume: 25, Issue:19

    Topics: Acetates; Cassia; Cell Line, Tumor; Chrysanthemum; Curcuma; Doxorubicin; Drug Resistance, Multiple; Drugs, Chinese Herbal; Humans; Ligusticum; Medicine, Chinese Traditional; Methylene Chloride; Plant Extracts; Plants, Medicinal; Salvia; Tetrazolium Salts; Thiazoles

2011
Cytotoxic constituents from the rhizomes of Curcuma zedoaria.
    TheScientificWorldJournal, 2014, Volume: 2014

    Topics: Analysis of Variance; Breast Neoplasms; Cell Proliferation; Chromatography, Thin Layer; Curcuma; Female; Human Umbilical Vein Endothelial Cells; Humans; Indonesia; Malaysia; MCF-7 Cells; Microscopy, Fluorescence; Molecular Structure; Phytotherapy; Plant Extracts; Rhizome; Tetrazolium Salts; Thiazoles

2014