thiazoles has been researched along with cgp 52608 in 27 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 9 (33.33) | 18.2507 |
| 2000's | 15 (55.56) | 29.6817 |
| 2010's | 3 (11.11) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Carlberg, C; Kahlen, JP; Missbach, M; Schräder, M; Wiesenberg, I | 1 |
| Carlberg, C; Jagher, B; Missbach, M; Nayeri, S; Sigg, I; Wiesenberg, I | 1 |
| Tslm, ST; Wong, JT; Wong, YH | 1 |
| Carlberg, C; Chiesi, M; Missbach, M; Pignat, W; Spanka, C; Wiesenberg, I | 1 |
| Calvo, JR; García-Mauriño, S; Guerrero, JM; Harmouch, A; Rafii-El-Idrissi, M | 1 |
| Calvo, JR; Garcia-Mauriño, S; Goberna, R; Gonzalez-Haba, MG; Guerrero, JM | 1 |
| Baldwin, W; Barrett, JC; Biermann, J; Jayadev, S; Murphy, E; Petranka, J | 1 |
| Li, L; Pang, SF; Shiu, SY; Wong, JT | 1 |
| Hu, DN; Roberts, JE; Wiechmann, AF | 1 |
| Gruszka, A; Karasek, M; Kunert-Radek, J; Melen-Mucha, G; Pawlikowski, M; Winczyk, K | 1 |
| Chignell, CF; Hu, DN; Martinez, L; Roberts, JE | 1 |
| Calvo, JR; García-Mauriño, S; Guerrero, JM; Pozo, D | 1 |
| Limonta, P; Marelli, MM; Monestiroli, S; Moretti, RM; Motta, M; Polizzi, D; Pratesi, G | 1 |
| Limonta, P; Montagnani Marelli, M; Moretti, RM; Motta, M | 1 |
| Karasek, M; Pawlikowski, M; Winczyk, K | 1 |
| Dai, J; Dong, C; Hill, SM; Kiefer, TL; Lai, L; Ram, PT; Yuan, L | 1 |
| Calvo, JR; Carrillo-Vico, A; García-Mauriño, S; Guerrero, JM | 1 |
| Gruszka, A; Karasek, M; Kunert-Radek, J; Lawnicka, H; Pawlikowski, M | 1 |
| Antolin, I; Herrera, F; Martín, V; Mayo, JC; Rodriguez, C; Sainz, RM | 1 |
| Limonta, P; Montagnani Marelli, M; Moretti, RM; Motta, M; Sala, A | 1 |
| Guerrero, JM; Leon-Blanco, MM; Pozo, D; Reiter, RJ | 1 |
| Karasek, M; Kunert-Radek, J; Lawnicka, H; Pawlikowski, M; Winczyk, K | 1 |
| Acuña-Castroviejo, D; Camacho, E; Escames, G; Espinosa, A; Gallo, MA; García-Navarro, A; González-Puga, C; López, A; López, LC; López-Cantarero, M | 1 |
| Balla, A; Dunlop, DS; Javitt, DC; Lajtha, A; Nattini, ME; Sershen, H | 1 |
| Cho, WJ; Hong, S; Jung, H; Kim, EJ; Lee, M; Lee, MO; Park, HG; Park, Y; Son, HY | 1 |
| Coban, N; Erginel-Unaltuna, N; Gulec, C; Ozsait-Selcuk, B; Sirma-Ekmekci, S; Yildirim, O | 1 |
| Bhagyaraj, E; Gupta, P; Gupta, R; Kalra, R; Khatri, N; Mahajan, S; Nanduri, R; Saini, A | 1 |
27 other study(ies) available for thiazoles and cgp 52608
| Article | Year |
|---|---|
Transcriptional activation of the nuclear receptor RZR alpha by the pineal gland hormone melatonin and identification of CGP 52608 as a synthetic ligand.
Topics: Animals; Base Sequence; Binding, Competitive; Cell Line; Drosophila; Kinetics; Ligands; Melatonin; Molecular Sequence Data; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Thiazoles; Thiosemicarbazones; Transcriptional Activation; Transfection | 1995 |
Thiazolidine diones, specific ligands of the nuclear receptor retinoid Z receptor/retinoid acid receptor-related orphan receptor alpha with potent antiarthritic activity.
Topics: Acetamides; Adjuvants, Immunologic; Animals; Anti-Inflammatory Agents, Non-Steroidal; Arthritis, Experimental; Autoimmune Diseases; Ligands; Male; Melatonin; Nuclear Receptor Subfamily 1, Group F, Member 1; Rats; Rats, Inbred Lew; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Receptors, Retinoic Acid; Structure-Activity Relationship; Thiazoles; Thiosemicarbazones; Trans-Activators | 1996 |
CGP 52608-induced cyst formation in dinoflagellates: possible involvement of a nuclear receptor for melatonin.
Topics: 5-Methoxytryptamine; Animals; Dinoflagellida; Dose-Response Relationship, Drug; Endocytosis; GTP-Binding Proteins; Intercellular Signaling Peptides and Proteins; Melatonin; Peptides; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Thiazoles; Thiosemicarbazones; Transcription Factors; Transcription, Genetic; Wasp Venoms | 1996 |
Specific activation of the nuclear receptors PPARgamma and RORA by the antidiabetic thiazolidinedione BRL 49653 and the antiarthritic thiazolidinedione derivative CGP 52608.
Topics: 3T3 Cells; Animals; Arthritis, Experimental; Cell Nucleus; Dexamethasone; Hypoglycemic Agents; Insulin Resistance; Leptin; Male; Mice; Proteins; Rats; Rats, Inbred Lew; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Retinoic Acid Receptor alpha; Rosiglitazone; Thiazoles; Thiazolidinediones; Thiosemicarbazones; Transcription Factors; Triglycerides | 1998 |
Specific binding of melatonin by purified cell nuclei from spleen and thymus of the rat.
Topics: Animals; Binding, Competitive; Cell Nucleus; Iodine Radioisotopes; Kinetics; Male; Melatonin; Pineal Gland; Rats; Rats, Wistar; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Spleen; Thiazoles; Thiosemicarbazones; Thymus Gland | 1998 |
Involvement of nuclear binding sites for melatonin in the regulation of IL-2 and IL-6 production by human blood mononuclear cells.
Topics: Acetamides; Adult; Binding Sites; Cell Membrane; Cell Nucleus; Cytokines; Humans; Interleukin-2; Interleukin-6; Melatonin; Middle Aged; Monocytes; Thiazoles; Thiosemicarbazones | 1998 |
The oncostatic action of melatonin in an ovarian carcinoma cell line.
Topics: Adenocarcinoma; Antineoplastic Agents; Apoptosis; Calcium; Cell Count; Cell Cycle; Cell Division; DNA; Dose-Response Relationship, Drug; Female; Flow Cytometry; Humans; Melatonin; Ovarian Neoplasms; Signal Transduction; Thiazoles; Thiosemicarbazones; Trypan Blue; Tumor Cells, Cultured | 1999 |
Melatonin-induced stimulation of rat corpus epididymal epithelial cell proliferation.
Topics: Animals; Cell Division; Cells, Cultured; Dihydrotestosterone; DNA; Drug Antagonism; Epididymis; Epithelial Cells; Flow Cytometry; Male; Melatonin; Ploidies; Rats; Thiazoles; Thiosemicarbazones; Thymidine | 1999 |
Melatonin receptors in human uveal melanocytes and melanoma cells.
Topics: Acetamides; Blotting, Southern; Choroid Neoplasms; Dose-Response Relationship, Drug; Gene Expression; Humans; Melanocytes; Melanoma; Melatonin; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; RNA, Neoplasm; Thiazoles; Thiosemicarbazones; Tumor Cells, Cultured | 2000 |
The antiproliferative effects of melatonin on experimental pituitary and colonic tumors. Possible involvement of the putative nuclear binding site?
Topics: Animals; Cell Division; Cell Nucleus; Colonic Neoplasms; Diethylstilbestrol; Male; Melatonin; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Pituitary Neoplasms; Rats; Rats, Wistar; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Thiazoles; Thiosemicarbazones | 1999 |
Photophysical studies on melatonin and its receptor agonists.
Topics: Acetamides; Hematoporphyrins; Kynurenine; Luminescent Measurements; Melatonin; Oxygen; Phenalenes; Photochemistry; Polycyclic Compounds; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Spectrophotometry, Ultraviolet; Thiazoles; Thiosemicarbazones; Ultraviolet Rays | 2000 |
Correlation between nuclear melatonin receptor expression and enhanced cytokine production in human lymphocytic and monocytic cell lines.
Topics: Acetamides; Adjuvants, Immunologic; Cell Membrane; Cell Nucleus; DNA Primers; Humans; Interleukin-2; Interleukin-6; Jurkat Cells; Lymphocytes; Melatonin; Monocytes; Phytohemagglutinins; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetradecanoylphorbol Acetate; Thiazoles; Thiosemicarbazones; U937 Cells | 2000 |
Activation of the orphan nuclear receptor RORalpha induces growth arrest in androgen-independent DU 145 prostate cancer cells.
Topics: Animals; Antineoplastic Agents; Cell Cycle; Cell Division; Cyclin-Dependent Kinase Inhibitor p21; Cyclins; Dose-Response Relationship, Drug; Gene Expression Regulation, Neoplastic; Humans; Ligands; Male; Mice; Mice, Nude; Nuclear Receptor Subfamily 1, Group F, Member 1; Prostatic Neoplasms; Receptors, Cytoplasmic and Nuclear; Reverse Transcriptase Polymerase Chain Reaction; Thiazoles; Thiosemicarbazones; Trans-Activators; Transplantation, Heterologous; Tumor Cells, Cultured | 2001 |
Oncostatic activity of a thiazolidinedione derivative on human androgen-dependent prostate cancer cells.
Topics: Androgens; Antineoplastic Agents; Cell Cycle; Cell Division; Cyclin-Dependent Kinase Inhibitor p21; Cyclins; Humans; Male; Neoplasms, Hormone-Dependent; Nuclear Receptor Subfamily 1, Group F, Member 1; Prostatic Neoplasms; Receptors, Cytoplasmic and Nuclear; Reverse Transcriptase Polymerase Chain Reaction; Thiazoles; Thiosemicarbazones; Trans-Activators; Tumor Cells, Cultured | 2001 |
Melatonin and RZR/ROR receptor ligand CGP 52608 induce apoptosis in the murine colonic cancer.
Topics: Animals; Apoptosis; Colonic Neoplasms; Ligands; Male; Melatonin; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Thiazoles; Thiosemicarbazones | 2001 |
Involvement of the mt1 melatonin receptor in human breast cancer.
Topics: Breast Neoplasms; Carbazoles; Cell Division; Dose-Response Relationship, Drug; Humans; Immunoblotting; Luciferases; Melatonin; Nuclear Receptor Subfamily 1, Group F, Member 1; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; Recombinant Fusion Proteins; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiazoles; Thiosemicarbazones; Trans-Activators; Tumor Cells, Cultured | 2002 |
Melatonin counteracts the inhibitory effect of PGE2 on IL-2 production in human lymphocytes via its mt1 membrane receptor.
Topics: Acetamides; Cyclic AMP; Dinoprostone; Gene Expression Regulation; Humans; Interleukin-2; Lymphocytes; Melatonin; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Receptors, Melatonin; RNA, Messenger; Tetradecanoylphorbol Acetate; Thiazoles; Thiosemicarbazones | 2003 |
Melatonin inhibits growth of diethylstilbestrol-induced prolactin-secreting pituitary tumor in vitro: possible involvement of nuclear RZR/ROR receptors.
Topics: Animals; Diethylstilbestrol; Disease Models, Animal; Male; Melatonin; Nuclear Receptor Subfamily 1, Group F, Member 1; Pituitary Neoplasms; Prolactin; Rats; Rats, Inbred F344; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Thiazoles; Thiosemicarbazones; Trans-Activators | 2003 |
Cytotoxicity and oncostatic activity of the thiazolidinedione derivative CGP 52608 on central nervous system cancer cells.
Topics: Animals; Antineoplastic Agents; Apoptosis; Caspase 3; Caspases; Cell Cycle; Cell Division; Central Nervous System Neoplasms; Drug Screening Assays, Antitumor; Flow Cytometry; Humans; Mice; Oxidative Stress; PC12 Cells; Rats; Thiazoles; Thiosemicarbazones; Tumor Cells, Cultured | 2004 |
Activation of the orphan nuclear receptor RORalpha counteracts the proliferative effect of fatty acids on prostate cancer cells: crucial role of 5-lipoxygenase.
Topics: Arachidonate 5-Lipoxygenase; Arachidonic Acid; Cell Division; Humans; Hydroxyeicosatetraenoic Acids; Linoleic Acid; Male; Neoplasms, Hormone-Dependent; Nerve Tissue Proteins; Nuclear Receptor Subfamily 1, Group F, Member 1; Prostatic Neoplasms; Protein Isoforms; Receptors, Cytoplasmic and Nuclear; Reverse Transcriptase Polymerase Chain Reaction; Thiazoles; Thiosemicarbazones; Trans-Activators; Tumor Cells, Cultured | 2004 |
RNA expression of human telomerase subunits TR and TERT is differentially affected by melatonin receptor agonists in the MCF-7 tumor cell line.
Topics: Acetamides; Breast Neoplasms; Catalytic Domain; Female; Humans; Hypnotics and Sedatives; Melatonin; Receptors, Melatonin; RNA; Signal Transduction; Telomerase; Thiazoles; Thiosemicarbazones; Tumor Cells, Cultured | 2004 |
Growth-inhibitory action of melatonin and thiazolidinedione derivative CGP 52608 on murine 16/C breast cancer cells.
Topics: Adenocarcinoma; Animals; Antimetabolites, Antineoplastic; Antineoplastic Agents, Hormonal; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Melatonin; Methotrexate; Mice; Nuclear Receptor Subfamily 1, Group F, Member 2; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Statistics, Nonparametric; Thiazoles; Thiosemicarbazones | 2006 |
Cellular mechanisms involved in the melatonin inhibition of HT-29 human colon cancer cell proliferation in culture.
Topics: Cell Proliferation; Colonic Neoplasms; Glutathione; Glutathione Peroxidase; Glutathione Reductase; HT29 Cells; Humans; Inhibitory Concentration 50; Kynurenine; Melatonin; Molecular Structure; Receptors, Melatonin; Structure-Activity Relationship; Thiazoles; Thiosemicarbazones | 2007 |
GABAB/NMDA receptor interaction in the regulation of extracellular dopamine levels in rodent prefrontal cortex and striatum.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Corpus Striatum; Dopamine; Extracellular Space; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Ligands; Male; Microdialysis; Organophosphorus Compounds; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate; Thiazoles; Thiosemicarbazones | 2009 |
N-methylthioureas as new agonists of retinoic acid receptor-related orphan receptor.
Topics: Hep G2 Cells; Humans; Nuclear Receptor Subfamily 1, Group F, Member 1; Structure-Activity Relationship; Thiazoles; Thiosemicarbazones; Thiourea | 2012 |
Identification of potential target genes of ROR-alpha in THP1 and HUVEC cell lines.
Topics: Base Sequence; Cell Line; Chromatin Immunoprecipitation; Consensus Sequence; HSC70 Heat-Shock Proteins; Human Umbilical Vein Endothelial Cells; Humans; Nuclear Receptor Subfamily 1, Group F, Member 1; Osteopontin; Promoter Regions, Genetic; Protein Binding; Thiazoles; Thiosemicarbazones; Transcriptional Activation; Transcriptome | 2017 |
An Accord of Nuclear Receptor Expression in CD4
Topics: Animals; Anti-Inflammatory Agents; Antibodies; Arthritis, Experimental; Arthritis, Rheumatoid; CD4-Positive T-Lymphocytes; Collagen Type II; Cytokines; Female; Humans; Inflammation; Male; Mice; Mice, Inbred DBA; Phenylacetates; Receptors, Cytoplasmic and Nuclear; Retinoids; Synovial Fluid; Thiazoles; Thiosemicarbazones; Transcription, Genetic | 2019 |