Compounds > thiazoles
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thiazoles and casein kinase ii

thiazoles has been researched along with casein kinase ii in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (27.27)29.6817
2010's7 (63.64)24.3611
2020's1 (9.09)2.80

Authors

AuthorsStudies
Alonso, LG; Castaño, E; Centeno, JM; de Prat-Gay, G; García-Alai, MM; Gualfetti, P; Iacono, R; Smal, C1
Kang, J; Luan, B; Pei, G; Wu, Y; Zhang, Z1
Aci, S; Barette, C; Bisson, G; Cochet, C; Denis, JN; Einhorn, C; Einhorn, J; Florent, JC; Lafanechere, L; Laudet, B; López-Ramos, M; Mouawad, L; Moucadel, V; Prudent, R; Roy, S; Schmidt, F1
Bovée, JV; Bruijn, IH; Hogendoorn, PC; Schrage, YM; Szuhai, K; Willems, SM1
Fujii, N; Hirasawa, A; Hou, Z; Kinoshita, T; Kitaura, K; Kure, T; Misu, R; Murata, K; Nakamura, S; Nakanishi, I; Ohno, H; Oishi, S; Suzuki, Y; Takei, Y; Tsujimoto, G; Yasue, M1
Fujii, N; Honda, M; Kinoshita, T; Minamiguchi, D; Misu, R; Moriwaki, H; Nakamura, S; Nakanishi, I; Nakanishi, S; Ohno, H; Oishi, S; Okazaki, S; Shu, K1
Enkvist, E; Haljasorg, T; Lavogina, D; Mazina, O; Rahnel, H; Uri, A; Viht, K1
Enkvist, E; Manoharan, GB; Uri, A; Vahter, J; Viht, K1
Abagyan, R; Abell, C; Bestgen, B; Cochet, C; Engel, M; Filhol, O; Hartmann, RW; Kufareva, I; Le Borgne, M; Lomberget, T; Seetoh, W1
Abagyan, R; Abell, C; Bestgen, B; Cochet, C; Engel, M; Hartmann, RW; Kamal, AAM; Krimm, I; Kufareva, I; Le Borgne, M; Lomberget, T; Seetoh, WG1
Applegate, VM; Jose, J; Lindenblatt, D; Nickelsen, A; Niefind, K1

Other Studies

11 other study(ies) available for thiazoles and casein kinase ii

ArticleYear
The HPV16 E7 viral oncoprotein self-assembles into defined spherical oligomers.
    Biochemistry, 2004, Mar-30, Volume: 43, Issue:12

    Topics: Benzothiazoles; Casein Kinase II; Circular Dichroism; Congo Red; Dimerization; Fluorescent Dyes; Humans; Molecular Weight; Oncogene Proteins, Viral; Papillomaviridae; Papillomavirus E7 Proteins; Phosphorylation; Protein Binding; Protein Serine-Threonine Kinases; Protein Structure, Secondary; Solubility; Thiazoles; Virus Assembly; Zinc

2004
Beta-arrestin2 functions as a phosphorylation-regulated suppressor of UV-induced NF-kappaB activation.
    The EMBO journal, 2005, Dec-21, Volume: 24, Issue:24

    Topics: Apoptosis; Arrestins; beta-Arrestins; Binding Sites; Casein Kinase II; Cell Death; Cell Line, Tumor; Cell Nucleus; Cell Separation; DNA Fragmentation; Dose-Response Relationship, Radiation; Epidermis; Flow Cytometry; Humans; Immunoblotting; Immunoprecipitation; In Situ Nick-End Labeling; Models, Biological; Models, Statistical; NF-kappa B; Phosphorylation; Plasmids; Protein Structure, Tertiary; Receptors, G-Protein-Coupled; Reverse Transcriptase Polymerase Chain Reaction; Tetrazolium Salts; Thiazoles; Time Factors; Transfection; Ultraviolet Rays

2005
Expanding the chemical diversity of CK2 inhibitors.
    Molecular and cellular biochemistry, 2008, Volume: 316, Issue:1-2

    Topics: Biological Assay; Casein Kinase II; Cell Line, Tumor; Humans; Models, Molecular; Phthalimides; Protein Kinase Inhibitors; Recombinant Proteins; Substrate Specificity; Thiazoles; Xanthenes

2008
Kinome profiling of myxoid liposarcoma reveals NF-kappaB-pathway kinase activity and casein kinase II inhibition as a potential treatment option.
    Molecular cancer, 2010, Sep-23, Volume: 9

    Topics: Casein Kinase II; Cell Line; Cell Line, Tumor; Cell Survival; Cells, Cultured; Dasatinib; HeLa Cells; Humans; Immunoblotting; Jurkat Cells; Karyotyping; Liposarcoma, Myxoid; NF-kappa B; Oncogene Proteins, Fusion; Protein Kinase Inhibitors; Pyrimidines; Reverse Transcriptase Polymerase Chain Reaction; Thiazoles; Triazoles

2010
Structure-based design of novel potent protein kinase CK2 (CK2) inhibitors with phenyl-azole scaffolds.
    Journal of medicinal chemistry, 2012, Mar-22, Volume: 55, Issue:6

    Topics: Adenosine Triphosphate; Adenylyl Imidodiphosphate; Antineoplastic Agents; Casein Kinase II; Cell Line, Tumor; Cell Proliferation; Crystallography, X-Ray; Databases, Factual; Drug Design; Drug Screening Assays, Antitumor; Humans; Models, Molecular; Protein Binding; Small Molecule Libraries; Structure-Activity Relationship; Thiazoles

2012
Structure-activity relationship study of 4-(thiazol-5-yl)benzoic acid derivatives as potent protein kinase CK2 inhibitors.
    Bioorganic & medicinal chemistry, 2016, Mar-01, Volume: 24, Issue:5

    Topics: Benzoic Acid; Casein Kinase II; Cell Line, Tumor; Cell Proliferation; Humans; Models, Molecular; Protein Kinase Inhibitors; Structure-Activity Relationship; Thiazoles

2016
A Selective Biligand Inhibitor of CK2 Increases Caspase-3 Activity in Cancer Cells and Inhibits Platelet Aggregation.
    ChemMedChem, 2017, 10-20, Volume: 12, Issue:20

    Topics: Antineoplastic Agents; Casein Kinase II; Caspase 3; Cell Cycle Proteins; Chaperonins; Enzyme Activation; Gene Expression Regulation, Neoplastic; Glycine; HeLa Cells; Humans; Molecular Structure; Phosphorylation; Platelet Aggregation; Thiazoles

2017
Thiazole- and selenazole-comprising high-affinity inhibitors possess bright microsecond-scale photoluminescence in complex with protein kinase CK2.
    Bioorganic & medicinal chemistry, 2018, 10-01, Volume: 26, Issue:18

    Topics: Casein Kinase II; Dose-Response Relationship, Drug; Fluorescence; Fluorescence Polarization; Fluorescent Dyes; Humans; Molecular Structure; Organoselenium Compounds; Photochemical Processes; Protein Kinase Inhibitors; Structure-Activity Relationship; Thiazoles; Time Factors

2018
2-Aminothiazole Derivatives as Selective Allosteric Modulators of the Protein Kinase CK2. 2. Structure-Based Optimization and Investigation of Effects Specific to the Allosteric Mode of Action.
    Journal of medicinal chemistry, 2019, 02-28, Volume: 62, Issue:4

    Topics: Allosteric Regulation; Allosteric Site; Antineoplastic Agents; Apoptosis; Benzoates; Casein Kinase II; Cell Line, Tumor; Humans; Ligands; Molecular Docking Simulation; Molecular Structure; Naphthyridines; Phenazines; Prodrugs; Protein Binding; Protein Kinase Inhibitors; Structure-Activity Relationship; Thiazoles

2019
2-Aminothiazole Derivatives as Selective Allosteric Modulators of the Protein Kinase CK2. 1. Identification of an Allosteric Binding Site.
    Journal of medicinal chemistry, 2019, 02-28, Volume: 62, Issue:4

    Topics: Allosteric Regulation; Allosteric Site; Casein Kinase II; Humans; Kinetics; Molecular Docking Simulation; Molecular Structure; Mutation; Naphthyridines; Phenazines; Protein Binding; Protein Kinase Inhibitors; Protein Stability; Structure-Activity Relationship; Temperature; Thiazoles

2019
Structural and Mechanistic Basis of the Inhibitory Potency of Selected 2-Aminothiazole Compounds on Protein Kinase CK2.
    Journal of medicinal chemistry, 2020, 07-23, Volume: 63, Issue:14

    Topics: Binding Sites; Casein Kinase II; Crystallography, X-Ray; Enzyme Assays; Humans; Kinetics; Protein Binding; Protein Kinase Inhibitors; Thiazoles

2020