thiazoles has been researched along with almorexant in 5 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 1 (20.00) | 29.6817 |
| 2010's | 4 (80.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Borroni, E; Knoflach, F; Malherbe, P; Pinard, E; Wettstein, JG | 1 |
| Bissantz, C; Kratzeisen, C; Malherbe, P; Marcuz, A; Roche, O; Wettstein, JG | 1 |
| Antolini, M; Corsi, M; di Fabio, R; Faedo, S; Merlo Pich, E; Perdonà, E | 1 |
| Czajkowska, B; Krzystanek, M; Lapray, D; Markowski, G; Pałasz, A; Peyron, C; Rojczyk-Gołębiewska, E; Skowronek, R; Wiaderkiewicz, R | 1 |
| Hoyer, D; Jacobson, LH | 1 |
2 review(s) available for thiazoles and almorexant
| Article | Year |
|---|---|
Dual orexin receptor antagonists - promising agents in the treatment of sleep disorders.
Topics: Acetamides; Animals; Azepines; Benzofurans; Humans; Isoquinolines; Models, Biological; Orexin Receptor Antagonists; Orexin Receptors; Piperidines; Pyrimidines; Sleep; Sleep Initiation and Maintenance Disorders; Thiazoles; Triazoles; Wakefulness | 2014 |
Orexin in sleep, addiction and more: is the perfect insomnia drug at hand?
Topics: Acetamides; Animals; Azepines; Behavior, Addictive; Benzofurans; Feeding Behavior; Humans; Intracellular Signaling Peptides and Proteins; Isoquinolines; Mice; Neuropeptides; Orexin Receptor Antagonists; Orexin Receptors; Orexins; Piperidines; Pyrimidines; Rats; Reward; Sleep; Sleep Initiation and Maintenance Disorders; Thiazoles; Triazoles | 2013 |
3 other study(ies) available for thiazoles and almorexant
| Article | Year |
|---|---|
Biochemical and electrophysiological characterization of almorexant, a dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist: comparison with selective OX1 and OX2 antagonists.
Topics: Acetamides; Animals; Evoked Potentials; Humans; Isoquinolines; Kinetics; Molecular Structure; Neurons; Orexin Receptors; Phenylurea Compounds; Pyrrolidines; Rats; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Sleep; Thiazoles | 2009 |
Mapping the binding pocket of dual antagonist almorexant to human orexin 1 and orexin 2 receptors: comparison with the selective OX1 antagonist SB-674042 and the selective OX2 antagonist N-ethyl-2-[(6-methoxy-pyridin-3-yl)-(toluene-2-sulfonyl)-amino]-N-py
Topics: Acetamides; Amino Acid Sequence; Aminopyridines; Binding Sites; Cell Line; Humans; Isoquinolines; Molecular Sequence Data; Mutagenesis, Site-Directed; Orexin Receptors; Pyrrolidines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Sequence Homology, Amino Acid; Sulfonamides; Thiazoles | 2010 |
Functional and binding kinetic studies make a distinction between OX1 and OX2 orexin receptor antagonists.
Topics: Acetamides; Animals; Benzofurans; Binding, Competitive; CHO Cells; Cricetinae; Cricetulus; Dioxanes; Humans; Isoquinolines; Kinetics; Orexin Receptors; Phenylurea Compounds; Piperidines; Protein Binding; Pyrimidines; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Thiazoles | 2012 |